Works about RADIOLIGAND assay

Results: 976

Making Competitive Binding Assay Theory Interesting in an Undergraduate Endocrinology Lab.

Published in:

Bioscene, 2007, v. 33, n. 4, p. 6

By:

Eichinger, Mark R.

Publication type:

Article

Serum hyaluronic acid levels do not explain morning stiffness in patients with fibromyalgia.

Published in:

2010

By:

Jong-Sun Kim;
Shin-Seok Lee;
Tae-Jong Kim;
Yong-Wook Park

Publication type:

Report

Ictal SPECT in neocortical epilepsies: clinical usefulness and factors affecting the pattern of hyperperfusion.

Published in:

Neuroradiology, 2006, v. 48, n. 9, p. 678, doi. 10.1007/s00234-006-0106-z

By:

Lee, Sang Kun;
Lee, Seo-Young;
Yun, Chang-Ho;
Lee, Ho-Young;
Lee, Jae-Sung;
Lee, Dong-Soo

Publication type:

Article

Selection and characterization of DNA aptamers with binding selectivity to Campylobacter jejuni using whole-cell SELEX.

Published in:

Applied Microbiology & Biotechnology, 2010, v. 87, n. 6, p. 2323, doi. 10.1007/s00253-010-2728-7

By:

Dwivedi, Hari;
Smiley, R.;
Jaykus, Lee-Ann

Publication type:

Article

Receptor-binding specificity of the human parainfluenza virus type 1 hemagglutinin–neuraminidase glycoprotein.

Published in:

Glycobiology, 2012, v. 22, n. 2, p. 174, doi. 10.1093/glycob/cwr112

By:

Alymova, Irina V;
Portner, Allen;
Mishin, Vasiliy P;
McCullers, Jonathan A;
Freiden, Pamela;
Taylor, Garry L

Publication type:

Article

Application of nano-baskets in preconcentration of tetrahedral oxoanions in the produced water of oil wells.

Published in:

Supramolecular Chemistry, 2012, v. 24, n. 12, p. 859, doi. 10.1080/10610278.2012.732225

By:

Mokhtari, Bahram;
Pourabdollah, Kobra

Publication type:

Article

CHRONIC EXPOSURE TO DIFFERENT AMBIENT TEMPERATURES AFFECTS b-AR PROFILE AND HEART RESPONSIVENESS TO ISOPROTERENOL AND CALCIUM.

Published in:

Israel Journal of Zoology, 2003, v. 49, n. 2/3, p. 219, doi. 10.1560/DTRB-NLUJ-0EMP-N0K4

By:

Arieli, Yehuda;
Kaspler, Pavel;
Horowitz, Michal

Publication type:

Article

Exploring the K+ binding site and its coupling to transport in the neurotransmitter: sodium symporter LeuT.

Published in:

eLife, 2024, p. 1, doi. 10.7554/eLife.87985

By:

Schmidt, Solveig G.;
Nygaard, Andreas;
Mindell, Joseph A.;
Loland, Claus J.

Publication type:

Article

THE FUCUS (PHAEOPHYCEAE) SPERM RECEPTOR FOR EGGS. II. ISOLATION OF A BINDING PROTEIN WHICH PARTIALLY ACTIVATES EGGS.

Published in:

Journal of Phycology, 1995, v. 31, n. 4, p. 592, doi. 10.1111/j.1529-8817.1995.tb02555.x

By:

Wright, Philip J.;
Callow, James A.;
Green, Jonathan R.

Publication type:

Article

THE FUCUS (PHAEOPHYCEAE) SPERM RECEPTOR FOR EGGS. I. DEVELOPMENT AND CHARACTERISTICS OF A BINDING ASSAY.

Published in:

Journal of Phycology, 1995, v. 31, n. 4, p. 584, doi. 10.1111/j.1529-8817.1995.tb02554.x

By:

Wright, Philip J.;
Green, Jonathan R.;
Callow, James A.

Publication type:

Article

DREADD agonist compound 21 causes acute diuresis in wild-type mice.

Published in:

Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1471059

By:

MacIver, Bryce;
Wu, Ali;
Hill, Warren G.;
Yu, Weiqun

Publication type:

Article

SAL0114: a novel deuterated dextromethorphan-bupropion combination with improved antidepressant efficacy and safety profile.

Published in:

Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1464564

By:

Xiao, Ying;
Hu, Xuefeng;
Xing, Wei;
Yan, Jie;
Wang, Ruhuan;
Li, Xiaoqing;
Li, Jiahuan;
Zhang, Zhixin;
Sun, Jingchao;
Wu, Junjun

Publication type:

Article

SAL0114: a novel deuterated dextromethorphan-bupropion combination with improved antidepressant efficacy and safety profile.

Published in:

Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1464564

By:

Ying Xiao;
Xuefeng Hu;
Wei Xing;
Jie Yan;
Ruhuan Wang;
Xiaoqing Li;
Jiahuan Li;
Zhixin Zhang;
Jingchao Sun;
Junjun Wu

Publication type:

Article

SAL0114: a novel deuterated dextromethorphan-bupropion combination with improved antidepressant efficacy and safety profile.

Published in:

Frontiers in Pharmacology, 2024, p. 1, doi. 10.3389/fphar.2024.1464564

By:

Ying Xiao;
Xuefeng Hu;
Wei Xing;
Jie Yan;
Ruhuan Wang;
Xiaoqing Li;
Jiahuan Li;
Zhixin Zhang;
Jingchao Sun;
Junjun Wu

Publication type:

Article

Empagliflozin, a novel selective sodium glucose cotransporter-2 (SGLT-2) inhibitor: characterisation and comparison with other SGLT-2 inhibitors.

Published in:

Diabetes, Obesity & Metabolism, 2012, v. 14, n. 1, p. 83, doi. 10.1111/j.1463-1326.2011.01517.x

By:

Grempler, R.;
Thomas, L.;
Eckhardt, M.;
Himmelsbach, F.;
Sauer, A.;
Sharp, D. E.;
Bakker, R. A.;
Mark, M.;
Klein, T.;
Eickelmann, P.

Publication type:

Article

Use of the H3 receptor antagonist radioligand [3H]-A-349821 to reveal in vivo receptor occupancy of cognition enhancing H3 receptor antagonists.

Published in:

2009

By:

Miller, T. R.;
Milicic, I.;
Bauch, J.;
Du, J.;
Surber, B.;
Browman, K. E.;
Marsh, K.;
Cowart, M.;
Brioni, J. D.;
Esbenshade, T. A.

Publication type:

journal article

In vitro and in vivo characterization of A-796260: a selective cannabinoid CB2 receptor agonist exhibiting analgesic activity in rodent pain models.

Published in:

2008

By:

Yao, B. B.;
Hsieh, G. C.;
Frost, J. M.;
Fan, Y.;
Garrison, T. R.;
Daza, A. V.;
Grayson, G. K.;
Zhu, C. Z.;
Pai, M.;
Chandran, P.;
Salyers, A. K.;
Wensink, E. J.;
Honore, P.;
Sullivan, J. P.;
Dart, M. J.;
Meyer, M. D.

Publication type:

journal article

Characterization of 4-(2-hydroxyphenyl)-1-[2'-[N-(2''-pyridinyl)-p-fluorobenzamido]ethyl]piperazine (p-DMPPF) as a new potent 5-HT1A antagonist.

Published in:

2007

By:

Defraiteur, C.;
Plenevaux, A.;
Scuvée-Moreau, J.;
Rouchet, N.;
Goblet, D.;
Luxen, A.;
Seutin, V.;
Scuvée-Moreau, J

Publication type:

journal article

Meta-analysis of cannabinoid ligand binding affinity and receptor distribution: interspecies differences.

Published in:

British Journal of Pharmacology, 2007, v. 152, n. 5, p. 583, doi. 10.1038/sj.bjp.0707399

By:

McPartland, J. M.;
Glass, M.;
Pertwee, R. G.

Publication type:

Article

Agonist potency at P2X7 receptors is modulated by structurally diverse lipids.

Published in:

British Journal of Pharmacology, 2007, v. 152, n. 4, p. 523, doi. 10.1038/sj.bjp.0707417

By:

Michel, A. D.;
Fonfria, E.

Publication type:

Article

Thermodynamic analysis of ligands at cholecystokinin CCK2 receptors in rat cerebral cortex.

Published in:

British Journal of Pharmacology, 2007, v. 151, n. 8, p. 1352, doi. 10.1038/sj.bjp.0707355

By:

Harper, E. A.;
Roberts, S. P.;
Kalindjian, S. B.

Publication type:

Article

A 17beta-derivative of allopregnanolone is a neurosteroid antagonist at a cerebellar subpopulation of GABA A receptors with nanomolar affinity.

Published in:

2007

By:

Maksay, G.;
Fodor, L.;
Bíró, T.;
Avlonitis, N;
Calogeropoulou, T;
Bíró, T

Publication type:

journal article

Achieving signalling selectivity of ligands for the corticotropin-releasing factor type 1 receptor by modifying the agonist's signalling domain.

Published in:

British Journal of Pharmacology, 2007, v. 151, n. 6, p. 851, doi. 10.1038/sj.bjp.0707293

By:

Beyermann, M.;
Heinrich, N.;
Fechner, K.;
Furkert, J.;
Zhang, W.;
Kraetke, O.;
Bienert, M.;
Berger, H.

Publication type:

Article

Correlation of apparent affinity values from H3-receptor binding assays with apparent affinity (pKapp) and intrinsic activity (α) from functional bioassays.

Published in:

British Journal of Pharmacology, 2007, v. 151, n. 1, p. 128, doi. 10.1038/sj.bjp.0707174

By:

Harper, E. A.;
Shankley, N. P.;
Black, J. W.

Publication type:

Article

Comparative antagonist pharmacology at the native mouse bradykinin B2 receptor: radioligand binding and smooth muscle contractility studies.

Published in:

British Journal of Pharmacology, 2007, v. 150, n. 3, p. 313, doi. 10.1038/sj.bjp.0706995

By:

Meini, S.;
Cucchi, P.;
Bellucci, F.;
Catalani, C.;
Giuliani, S.;
Santicioli, P.;
Maggi, C. A.

Publication type:

Article

Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand.

Published in:

British Journal of Pharmacology, 2006, v. 148, n. 5, p. 657, doi. 10.1038/sj.bjp.0706752

By:

Witte, David G.;
Bei Yao, Betty;
Miller, Thomas R.;
Carr, Tracy L.;
Cassar, Steven;
Sharma, Rahul;
Faghih, Ramin;
Surber, Bruce W;
Esbenshade, Timothy A.;
Hancock, Arthur A.;
Krueger, Kathleen M.

Publication type:

Article

[32P]2-iodo-N6-methyl-(N)-methanocarba-2'-deoxyadenosine-3',5'-bisphosphate ([32P]MRS2500), a novel radioligand for quantification of native P2Y1 receptors.

Published in:

2006

By:

Houston, Dayle;
Ohno, Michihiro;
Nicholas, Robert A.;
Jacobson, Kenneth A.;
Harden, T. Kendall

Publication type:

journal article

Allosteric modulation, thermodynamics and binding to wild-type and mutant (T277A) adenosine A1 receptors of LUF5831, a novel nonadenosine-like agonist.

Published in:

2006

By:

Heitman, Laura H.;
Mulder-Krieger, Thea;
Spanjersberg, Ronald F.;
von Frijtag Drabbe Künzel, Jacobien K.;
Dalpiaz, Alessandro;
IJzerman, Adriaan P.;
von Frijtag Drabbe Künzel, Jacobien K

Publication type:

journal article

RO1138452 and RO3244794: characterization of structurally distinct, potent and selective IP (prostacyclin) receptor antagonists.

Published in:

British Journal of Pharmacology, 2006, v. 147, n. 3, p. 335, doi. 10.1038/sj.bjp.0706554

By:

Bley, Keith R.;
Bhattacharya, Anindya;
Daniels, Don V.;
Gever, Joel;
Jahangir, Alam;
O'Yang, Counde;
Smith, Steven;
Srinivasan, Dinesh;
Ford, Anthony P. D. W.;
Jett, Mary-Frances

Publication type:

Article

Efficacy in CB1 receptor-mediated signal transduction.

Published in:

2004

By:

Howlett, Allyn C.

Publication type:

journal article

Cannabinoid CB1 receptor-mediated modulation of evoked dopamine release and of adenylyl cyclase activity in the human neocortex.

Published in:

2004

By:

Steffens, M.;
Engler, C.;
Zentner, J.;
Feuerstein, T.J.

Publication type:

journal article

Alpha-1 adrenoceptors: evaluation of receptor subtype-binding kinetics in intact arterial tissues and comparison with membrane binding.

Published in:

British Journal of Pharmacology, 2004, v. 141, n. 3, p. 468, doi. 10.1038/sj.bjp.0705627

By:

Tanaka, Takashi;
Zhang, Li;
Suzuki, Fumiko;
Muramatsu, Ikunobu

Publication type:

Article

Endosome sorting of ß2-adrenoceptors is GRK5 independent.

Published in:

British Journal of Pharmacology, 2004, v. 141, n. 2, p. 277, doi. 10.1038/sj.bjp.0705504

By:

Millman, Ellen E.;
Rosenfeld, Jennifer L.;
Vaughan, David J.;
Nguyen, Jacqueline;
WenPing Dai, Jacqueline;
Alpizar-Foster, Estrella;
Clark, Richard B.;
Knoll, Brian J.;
Moore, Robert H.

Publication type:

Article

Oleamide is a selective endogenous agonist of rat and human CB1 cannabinoid receptors.

Published in:

2004

By:

Leggett, James D.;
Aspley, S.;
Beckett, S. R. G.;
D'Antona, A. M.;
Kendall, D. A.

Publication type:

journal article

Characterisation of the binding of [3H]-SB-674042, a novel nonpeptide antagonist, to the human orexin-1 receptor.

Published in:

British Journal of Pharmacology, 2004, v. 141, n. 2, p. 340, doi. 10.1038/sj.bjp.0705610

By:

Langmead, Christopher J.;
Jerman, Jeffrey C.;
Brough, Stephen J.;
Scott, Claire;
Porter, Rod A.;
Herdon, Hugh J.

Publication type:

Article

Anandamide and vanilloid TRPV1 receptors.

Published in:

2003

By:

Ross, Ruth A.

Publication type:

journal article

Pharmacological characterization of a 7-benzylidenenaltrexone-preferring opioid receptor in porcine ileal submucosa.

Published in:

2003

By:

Townsend IV, De Wayne;
Brown, David R.;
Townsend, De Wayne 4th

Publication type:

journal article

PROLONGED TREATMENT OF NATIVE OR MUTANT (T343K) D[2SHORT] DOPAMINE RECEPTORS WITH THE INVERSE AGONIST HALOPERIDOL RESULTS IN AN INCREASE IN RECEPTOR DENSITY.

Published in:

British Journal of Pharmacology, 2003, v. 140, p. 68P

By:

Gardner, B.;
Franks, D. J.;
Strange, P. G.

Publication type:

Article

THE SELECTIVITY OF Β-BLOCKERS FOR THE HUMAN Β1- AND Β2- ADRENOCEPTORS.

Published in:

British Journal of Pharmacology, 2003, v. 140, p. 70P

By:

Baker, J. G.;
Hall, I. P.;
Hill, S. J.

Publication type:

Article

EFFECT OF SODIUM IONS ON LIGAND BINDING TO THE D[2SHORT] DOPAMINE RECEPTOR.

Published in:

British Journal of Pharmacology, 2003, v. 140, p. 69P

By:

Vivo, M.;
Strange, P. G.

Publication type:

Article

CHARACTERIZATION OF [³H]-ZM 241385 BINDING IN WILDTYPE AND A[sub2A] KNOCKOUT MOUSE BRAIN.

Published in:

British Journal of Pharmacology, 2003, v. 140, p. 58P

By:

Kelly, M. D. W.;
Ledent, C.;
Kitchen, I.;
Hourani, S. M. O.

Publication type:

Article

ABEA-BY630 IS A FLUORESCENT AGONIST AT A[SUB2B] ADENOSINE RECEPTORS IN HUMAN PROSTATIC STROMAL CELLS.

Published in:

British Journal of Pharmacology, 2003, v. 140, p. 16P

By:

Cordeaux, Y.;
Middleton, R. J.;
Myatt, A.;
Kellam, B.;
Hill, S. J.

Publication type:

Article

Pharmacological comparison of the alternatively spliced short and long CCK[sub2] receptors.

Published in:

British Journal of Pharmacology, 2003, v. 140, n. 1, p. 218, doi. 10.1038/sj.bjp.0705423

By:

Morton, M.F.;
Harper, E.A.;
Tavares, I.A.;
Shankley, N.P.

Publication type:

Article

Castration decreases amylase release associated with muscarinic acetylcholine receptor downregulation in rat parotid gland.

Published in:

British Journal of Pharmacology, 2003, v. 139, n. 2, p. 399, doi. 10.1038/sj.bjp.0705260

By:

Busch, Lucila;
Borda, Enri

Publication type:

Article

Pharmacology and direct visualisation of BODIPY-TMR-CGP: a long-acting fluorescent Β2-adrenoceptor agonist.

Published in:

British Journal of Pharmacology, 2003, v. 139, n. 2, p. 232, doi. 10.1038/sj.bjp.0705287

By:

Baker, Jillian G.;
Hall, Ian P.;
Hill, Stephen J.

Publication type:

Article

A COMPARISON OF THE BINDING AFFINITIES OF ENDOTHELIN (ET) RECEPTOR ANTAGONISTS AT RECOMBINANT AND NATIVE ETA RECEPTORS.

Published in:: British Journal of Pharmacology, 2002, v. 137, p. 80
Publication type:: Article

BINDING OF THE A2A ADENOSINE RECEPTOR ANTAGONIST RADIOLIGAND [3H]-ZM241385 TO PARTICULATE PREPARATIONS FROM THE PORCINE PUTAMEN AND NUCLEUS ACCUMBENS.

Published in:: British Journal of Pharmacology, 2002, v. 137, p. 79
Publication type:: Article

RADIOSYNTHESIS AND IN VIVO BIODISTRIBUTION OF [18F]-BIG ET-1, A POTENTIAL PET RADIOLIGAND FOR THE STUDY OF ENZYME CONVERSION OF BIG ET-1 TO ET-1.

Published in:: British Journal of Pharmacology, 2002, v. 137, p. 46
Publication type:: Article

Studies of GABA[subB] receptors labelled with [[sup3]H]-CGP62349 in hippocampus resected from patients with temporal lobe epilepsy.

Published in:

British Journal of Pharmacology, 2002, v. 136, n. 8, p. 1099, doi. 10.1038/sj.bjp.0704812

By:

Princivalle, A.P.;
Duncan, J.S.;
Thom, M.;
Bowery, N.G.

Publication type:

Article

Method development, validation, and impurity measurement of β-estradiol from radiolabeled [131I] β-estradiol using radio-high-performance liquid chromatography for radioligand of saturation binding assay.

Published in:

Journal of Advanced Pharmaceutical Technology & Research, 2023, v. 14, n. 2, p. 105, doi. 10.4103/japtr.japtr_624_22

By:

Daruwati, Isti;
Gwiharto, Abednego Kristande;
Wongso, Hendris;
Achmad, Tri Hanggono;
Syaifudin, Mukh;
Muchtaridi, Muchtaridi

Publication type:

Article