Works matching DE "BINDING sites"


Results: 5000
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    Discovery of 1‐(Cyclopropylmethyl)‐2‐(Dibenzo[b,d]Thiophen‐2‐yl)‐1H‐Benzo[d]Imidazole‐5‐Carboxylic Acid as Orally Bioavailable EP4 Receptor Antagonist.

    Published in:
    Chemical Biology & Drug Design, 2025, v. 105, n. 6, p. 1, doi. 10.1111/cbdd.70132
    By:
    • Kumar, Sanjay;
    • Chakraborty, Rajib;
    • Roy, Chandreyee;
    • Basu, Sohini;
    • Hajra, Arun K.;
    • Sen, Priyam;
    • Paul, Debajyoti;
    • Phukan, Karabi;
    • Roy, Subhasis;
    • Bera, Rammohan;
    • Mondal, Trisha;
    • Chakraborty, Sabyasachi;
    • Banerjee, Manish;
    • Mondal, Susanta K.;
    • Das, Sonali;
    • Malik, Pradip;
    • De Mandal, Surajit;
    • Subudhi, Enketeswara;
    • Kundu, Mrinalkanti
    Publication type:
    Article
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    In Vitro and In Silico Assessments of Curcuminoids and Turmerones from Curcuma longa as Novel Inhibitors of Leishmania infantum Arginase.

    Published in:
    Pharmaceuticals (14248247), 2025, v. 18, n. 6, p. 851, doi. 10.3390/ph18060851
    By:
    • Spíndola, Flora F. S.;
    • Pinheiro, Anderson S.;
    • Mpalantinos, Maria Athana;
    • Silva, Jefferson R. A.;
    • Neto, Walter S. M. F.;
    • Conceição, Raissa A.;
    • Barreto, Eduarda M.;
    • Abrahim-Vieira, Barbara A.;
    • Rodrigues, Carlos R.;
    • Souza, Alessandra M. T.;
    • Nico, Dirlei;
    • Amaral, Ana Claudia F.;
    • Garcia, Andreza R.;
    • Rodrigues, Igor A.
    Publication type:
    Article
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    Transcriptional Dysregulation in NIPBL and Cohesin Mutant Human Cells.

    Published in:
    PLoS Biology, 2009, v. 7, n. 5, p. 1, doi. 10.1371/journal.pbio.1000119
    By:
    • Jinglan Liu;
    • Zhe Zhang;
    • Bando, Masashige;
    • Itoh, Takehiko;
    • Deardorff, Matthew A.;
    • Clark, Dinah;
    • Kaur, Maninder;
    • Tandy, Stephany;
    • Kondoh, Tatsuro;
    • Rappaport, Eric;
    • Spinner, Nancy B.;
    • Vega, Hugo;
    • Jackson, Laird G.;
    • Shirahige, Katsuhiko;
    • Krantz, Ian D.
    Publication type:
    Article
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    The Active Site of a Carbohydrate Esterase Displays Divergent Catalytic and Noncatalytic Binding Functions.

    Published in:
    PLoS Biology, 2009, v. 7, n. 3, p. e1000071, doi. 10.1371/journal.pbio.1000071
    By:
    • Montanier, Cedric;
    • Money, Victoria A.;
    • Pires, Virginia M. R.;
    • Flint, James E.;
    • Pinheiro, Benedita A.;
    • Goyal, Arun;
    • Prates, José A. M.;
    • Izumi, Atsushi;
    • Stålbrand, Henrik;
    • Morland, Carl;
    • Cartmell, Alan;
    • Kolenova, Katarina;
    • Topakas, Evangelos;
    • Dodson, Eleanor J.;
    • Bolam, David N.;
    • Davies, Gideon J.;
    • Fontes, Carlos M. G. A.;
    • Gilbert, Harry J.
    Publication type:
    Article
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    The Influence of Catalysis on Mad2 Activation Dynamics.

    Published in:
    PLoS Biology, 2009, v. 7, n. 1, p. e1000010, doi. 10.1371/journal.pbio.1000010
    By:
    • Simonetta, Marco;
    • Manzoni, Romilde;
    • Mosca, Roberto;
    • Mapelli, Marina;
    • Massimiliano, Lucia;
    • Vink, Martin;
    • Novak, Bela;
    • Musacchio, Andrea;
    • Ciliberto, Andrea
    Publication type:
    Article
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    The Ticket to Transport.

    Published in:
    PLoS Biology, 2008, v. 6, n. 6, p. e144, doi. 10.1371/journal.pbio.0060144
    By:
    • Hoff, Mary
    Publication type:
    Article
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