Works by Katzenellenbogen, John

Results: 100
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    Hormone–PAMAM Dendrimer Conjugates: Polymer Dynamics and Tether Structure Affect Ligand Access to ReceptorsWe are grateful for support of this research through grants from the National Institutes of Health (PHS 5R37 DK15556). We thank Kathryn Carlson for determining the receptor binding affinities. NMR spectra were obtained in the Varian Oxford Instrument Center for Excellence in NMR Laboratory. Funding for this instrumentation was provided in part by the W. M. Keck Foundation, the National Institutes of Health (PHS 1 S10 RR104444-01), and the National Science Foundation (NSF CHE 96-10502). Mass spectra were obtained on instruments supported by grants from the National Institute of General Medical Sciences (GM 27029), the National Institutes of Health (RR 01575), and the National Science Foundation (PCM 8121494). PAMAM=poly(amide)polyamine.

    Published in:
    Angewandte Chemie, 2006, v. 118, n. 43, p. 7401, doi. 10.1002/ange.200601923
    By:
    • Sung Hoon Kim;
    • John A. Katzenellenbogen
    Publication type:
    Article
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    Non-nuclear estrogen receptor alpha signaling promotes cardiovascular protection but not uterine or breast cancer growth in mice.

    Published in:
    2010
    By:
    • Chambliss, Ken L.;
    • Qian Wu;
    • Oltmann, Sarah;
    • Konaniah, Eddy S.;
    • Umetani, Michihisa;
    • Korach, Kenneth S.;
    • Thomas, Gail D.;
    • Mineo, Chieko;
    • Yuhanna, Ivan S.;
    • Sung Hoon Kim;
    • Madak-Erdogan, Zeynep;
    • Maggi, Adriana;
    • Dineen, Sean P.;
    • Roland, Christina L.;
    • Hui, David Y.;
    • Brekken, Rolf A.;
    • Katzenellenbogen, John A.;
    • Katzenellenbogen, Benita S.;
    • Shaul, Philip W.;
    • Wu, Qian
    Publication type:
    journal article
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    Optimization of the preparation of fluorine-18-labeled steroid receptor ligands 16alpha-[<sup>18</sup>F]fluoroestradiol (FES), [<sup>18</sup>F]fluoro furanyl norprogesterone (FFNP), and 16beta-[<sup>18</sup>F]fluoro-5alpha-dihydrotestosterone (FDHT) as radiopharmaceuticals

    Published in:
    Journal of Labelled Compounds & Radiopharmaceuticals, 2014, v. 57, n. 5, p. 371, doi. 10.1002/jlcr.3191
    By:
    • Zhou, Dong;
    • Lin, Mai;
    • Yasui, Norio;
    • Al ‐ Qahtani, Mohammed H.;
    • Dence, Carmen S.;
    • Schwarz, Sally;
    • Katzenellenbogen, John A.
    Publication type:
    Article
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    Predominant Role of Nuclear Versus Membrane Estrogen Receptor α in Arterial Protection: Implications for Estrogen Receptor α Modulation in Cardiovascular Prevention/Safety.

    Published in:
    2018
    By:
    • Guivarc'h, Emmanuel;
    • Buscato, Mélissa;
    • Guihot, Anne-Laure;
    • Favre, Julie;
    • Vessières, Emilie;
    • Grimaud, Linda;
    • Wakim, Jamal;
    • Melhem, Nada-Joe;
    • Zahreddine, Rana;
    • Adlanmerini, Marine;
    • Loufrani, Laurent;
    • Knauf, Claude;
    • Katzenellenbogen, John A.;
    • Katzenellenbogen, Benita S.;
    • Foidart, Jean-Michel;
    • Gourdy, Pierre;
    • Lenfant, Françoise;
    • Arnal, Jean-François;
    • Henrion, Daniel;
    • Fontaine, Coralie
    Publication type:
    journal article
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    PLASMIN-ACTIVATED ANTICANCER PRODRUGS.

    Published in:
    Annals of the New York Academy of Sciences, 1982, v. 397, n. 1, p. 324, doi. 10.1111/j.1749-6632.1982.tb43455.x
    By:
    • Weber, Michael J.;
    • Chakravarty, Prasun K.;
    • Bruesch, Margaret R.;
    • Johnson, Gail L.;
    • Katzenellenbogen, John A.;
    • Carl, Philip L.
    Publication type:
    Article
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    PI3K inhibition results in enhanced estrogen receptor function and dependence in hormone receptor–positive breast cancer.

    Published in:
    Science Translational Medicine, 2015, v. 7, n. 283, p. 1, doi. 10.1126/scitranslmed.aaa4442
    By:
    • Bosch, Ana;
    • Zhiqiang Li;
    • Bergamaschi, Anna;
    • Ellis, Haley;
    • Toska, Eneda;
    • Prat, Aleix;
    • Tao, Jessica J.;
    • Spratt, Daniel E.;
    • Viola-Villegas, Nerissa T.;
    • Castel, Pau;
    • Minuesa, Gerard;
    • Morse, Natasha;
    • Rodón, Jordi;
    • Ibrahim, Yasir;
    • Cortes, Javier;
    • Perez-Garcia, Jose;
    • Galvan, Patricia;
    • Grueso, Judit;
    • Guzman, Marta;
    • Katzenellenbogen, John A.
    Publication type:
    Article
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    Endothelial ERα promotes glucose tolerance by enhancing endothelial insulin transport to skeletal muscle.

    Published in:
    Nature Communications, 2023, v. 14, n. 1, p. 1, doi. 10.1038/s41467-023-40562-w
    By:
    • Sacharidou, Anastasia;
    • Chambliss, Ken;
    • Peng, Jun;
    • Barrera, Jose;
    • Tanigaki, Keiji;
    • Luby-Phelps, Katherine;
    • Özdemir, İpek;
    • Khan, Sohaib;
    • Sirsi, Shashank R.;
    • Kim, Sung Hoon;
    • Katzenellenbogen, Benita S.;
    • Katzenellenbogen, John A.;
    • Kanchwala, Mohammed;
    • Sathe, Adwait A.;
    • Lemoff, Andrew;
    • Xing, Chao;
    • Hoyt, Kenneth;
    • Mineo, Chieko;
    • Shaul, Philip W.
    Publication type:
    Article
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    Dietary licorice root supplementation reduces diet-induced weight gain, lipid deposition, and hepatic steatosis in ovariectomized mice without stimulating reproductive tissues and mammary gland.

    Published in:
    Molecular Nutrition & Food Research, 2016, v. 60, n. 2, p. 369, doi. 10.1002/mnfr.201500445
    By:
    • Madak‐Erdogan, Zeynep;
    • Gong, Ping;
    • Zhao, Yiru Chen;
    • Xu, Liwen;
    • Wrobel, Kinga U.;
    • Hartman, James A.;
    • Wang, Michelle;
    • Cam, Anthony;
    • Iwaniec, Urszula T.;
    • Turner, Russell T.;
    • Twaddle, Nathan C.;
    • Doerge, Daniel R.;
    • Khan, Ikhlas A.;
    • Katzenellenbogen, John A.;
    • Katzenellenbogen, Benita S.;
    • Helferich, William G.
    Publication type:
    Article
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    Reprogramming of endothelial gene expression by tamoxifen inhibits angiogenesis and ERα-negative tumor growth.

    Published in:
    Theranostics, 2024, v. 14, n. 1, p. 249, doi. 10.7150/thno.87306
    By:
    • Fébrissy, Chanaëlle;
    • Adlanmerini, Marine;
    • Péqueux, Christel;
    • Boudou, Frédéric;
    • Buscato, Mélissa;
    • Gargaros, Adrien;
    • Gilardi-Bresson, Silveric;
    • Boriak, Khrystyna;
    • Laurell, Henrik;
    • Fontaine, Coralie;
    • Katzenellenbogen, Benita S.;
    • Katzenellenbogen, John A.;
    • Guillermet-Guibert, Julie;
    • Arnal, Jean-François;
    • Metivier, Raphaël;
    • Lenfant, Françoise
    Publication type:
    Article
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    Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.

    Published in:
    ChemMedChem, 2016, v. 11, n. 16, p. 1752, doi. 10.1002/cmdc.201600140
    By:
    • Granchi, Carlotta;
    • Lapillo, Margherita;
    • Spena, Concetta Russo;
    • Rizzolio, Flavio;
    • Tuccinardi, Tiziano;
    • Martin, Teresa A.;
    • Carlson, Kathryn E.;
    • Katzenellenbogen, John A.;
    • Minutolo, Filippo
    Publication type:
    Article
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    Development of Selective Estrogen Receptor Modulator (SERM)-Like Activity Through an Indirect Mechanism of Estrogen Receptor Antagonism: Defining the Binding Mode of 7-Oxabicyclo[2.2.1]hept-5-ene Scaffold Core Ligands.

    Published in:
    ChemMedChem, 2012, v. 7, n. 6, p. 1094, doi. 10.1002/cmdc.201200048
    By:
    • Zheng, Yangfan;
    • Zhu, Manghong;
    • Srinivasan, Sathish;
    • Nwachukwu, Jerome C.;
    • Cavett, Valerie;
    • Min, Jian;
    • Carlson, Kathryn E.;
    • Wang, Pengcheng;
    • Dong, Chune;
    • Katzenellenbogen, John A.;
    • Nettles, Kendall W.;
    • Zhou, Hai-Bing
    Publication type:
    Article
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