Works matching AU Cassels, Bruce

Results: 37

Evaluation of benzyltetrahydroisoquinolines as ligands for neuronal nicotinic acetylcholine receptors.

Published in:

2005

By:

Exley, Richard;
Iturriaga-V&ásquez, Patricio;
Lukas, Ronald J.;
Sher, Emanuele;
Cassels, Bruce K.;
Bermudez, Isabel;
Iturriaga-Vásquez, Patricio

Publication type:

journal article

4-Bromo-2,5-dimethoxyphenethylamine (2C-B) and structurally related phenylethylamines are potent 5-HT2A receptor antagonists in Xenopus laevis oocytes.

Published in:

British Journal of Pharmacology, 2004, v. 141, n. 7, p. 1167, doi. 10.1038/sj.bjp.0705722

By:

Villalobos, Claudio A.;
Bull, Paulina;
Sáez, Patricio;
Cassels, Bruce K.;
Huidobro-Toro, J. Pablo

Publication type:

Article

Differences in potency and efficacy of a series of phenylisopropylamine/phenylethylamine pairs at 5-HT[sub 2A] and 5-HT[sub 2C] receptors.

Published in:

British Journal of Pharmacology, 2002, v. 136, n. 4, p. 510

By:

Villalobos, Claudio;
Moya, Pablo R.;
Cassels, Bruce K.;
Huidobro-Toro, J, Pablo;
Acuña-Castillo, Claudio;
Sáez, Patricio

Publication type:

Article

Boldine inhibits the alveolar bone resorption during ligature-induced periodontitis by modulating the Th17/Treg imbalance.

Published in:

2021

By:

Cafferata, Emilio A.;
Castro‐Saavedra, Sebastián;
Fuentes‐Barros, Gonzalo;
Melgar‐Rodríguez, Samanta;
Rivera, Felipe;
Carvajal, Paola;
Hernández, Marcela;
Cortés, Bastián I.;
Cortez, Cristian;
Cassels, Bruce K.;
Vernal, Rolando;
Castro-Saavedra, Sebastián;
Fuentes-Barros, Gonzalo;
Melgar-Rodríguez, Samanta

Publication type:

journal article

Dibenzofuran annulated 1-azepines: Synthesis and cytotoxicity.

Published in:

Synthetic Communications, 2020, v. 50, n. 3, p. 438, doi. 10.1080/00397911.2019.1703001

By:

Yempala, Thirumal;
Babu, Tomer;
Gibson, Dan;
Cassels, Bruce K.

Publication type:

Article

Simple and efficient synthesis of various dibenzofuran carbaldehydes.

Published in:

Synthetic Communications, 2016, v. 46, n. 23, p. 1909, doi. 10.1080/00397911.2016.1235201

By:

Yempala, Thirumal;
Cassels, Bruce K.

Publication type:

Article

Functional roles of T3.37 and S5.46 in the activation mechanism of the dopamine D1 receptor.

Published in:

Journal of Molecular Modeling, 2017, v. 23, n. 4, p. 1, doi. 10.1007/s00894-017-3313-0

By:

Hugo, Estefanía A.;
Cassels, Bruce K.;
Fierro, Angélica

Publication type:

Article

Why is quercetin a better antioxidant than taxifolin? Theoretical study of mechanisms involving activated forms.

Published in:

Journal of Molecular Modeling, 2013, v. 19, n. 5, p. 2165, doi. 10.1007/s00894-012-1732-5

By:

Osorio, Edison;
Pérez, Edwin;
Areche, Carlos;
Ruiz, Lina;
Cassels, Bruce;
Flórez, Elizabeth;
Tiznado, William

Publication type:

Article

Targeting Sentinel Proteins and Extrasynaptic Glutamate Receptors: a Therapeutic Strategy for Preventing the Effects Elicited by Perinatal Asphyxia?

Published in:

Neurotoxicity Research, 2018, v. 33, n. 2, p. 461, doi. 10.1007/s12640-017-9795-9

By:

Herrera-Marschitz, Mario;
Perez-Lobos, Ronald;
Lespay-Rebolledo, Carolyne;
Tapia-Bustos, Andrea;
Casanova-Ortiz, Emmanuel;
Morales, Paola;
Valdes, Jose-Luis;
Bustamante, Diego;
Cassels, Bruce K.

Publication type:

Article

Neurochemical and Behavioural Characterisation of Alkoxyamphetamine Derivatives in Rats.

Published in:

Neurotoxicity Research, 2006, v. 10, n. 1, p. 11, doi. 10.1007/BF03033330

By:

Romero, Cesar A.;
Bustamante, Diego A.;
Zapata-Torres, Gerald;
Goiny, Michel;
Cassels, Bruce;
Herrera-Marschitz, Mario

Publication type:

Article

Telomerase Inhibition by a New Synthetic Derivative of the Aporphine Alkaloid Boldine.

Published in:

International Journal of Molecular Sciences, 2018, v. 19, n. 4, p. 1239, doi. 10.3390/ijms19041239

By:

Noureini, Sakineh Kazemi;
Kheirabadi, Mitra;
Masoumi, Fatima;
Khosrogerdi, Farve;
Zarei, Younes;
Suárez-Rozas, Cristian;
Salas-Norambuena, Julio;
Cassels, Bruce Kennedy

Publication type:

Article

Molecular dynamics simulation of halogen bonding mimics experimental data for cathepsin L inhibition.

Published in:

Journal of Computer-Aided Molecular Design, 2015, v. 29, n. 1, p. 37, doi. 10.1007/s10822-014-9802-7

By:

Celis-Barros, Cristian;
Saavedra-Rivas, Leslie;
Salgado, J.;
Cassels, Bruce;
Zapata-Torres, Gerald

Publication type:

Article

Distinguishing rotamers in N-trifluoroacetyl-3-benzazepine derivatives.

Published in:

Magnetic Resonance in Chemistry, 2016, v. 54, n. 7, p. 597, doi. 10.1002/mrc.4406

By:

Acevedo‐Fuentes, Williams A.;
Cassels, Bruce K.

Publication type:

Article

Complete 1H and 13C NMR spectral assignment of hydrogenated oxoisoaporphine derivatives.

Published in:

Magnetic Resonance in Chemistry, 2003, v. 41, n. 7, p. 545, doi. 10.1002/mrc.1205

By:

Eduardo Sobarzo-Sánchez;
Bruce K. Cassels;
Luis Castedo

Publication type:

Article

Complete structural and spectral assignment of oxoisoaporphines by HMQC and HMBC experiments.

Published in:

Magnetic Resonance in Chemistry, 2003, v. 41, n. 4, p. 296, doi. 10.1002/mrc.1177

By:

Eduardo Sobarzo-Sánchez;
Bruce K. Cassels;
Carolina Jullian;
Luis Castedo

Publication type:

Article

Amphetamine Derivatives as Monoamine Oxidase Inhibitors.

Published in:

Frontiers in Pharmacology, 2020, p. 1, doi. 10.3389/fphar.2019.01590

By:

Reyes-Parada, Miguel;
Iturriaga-Vasquez, Patricio;
Cassels, Bruce K.

Publication type:

Article

Cathodic behavior of 4,5-dimethoxy-2-nitroamphetamine.

Published in:

Electroanalysis, 1992, v. 4, n. 5, p. 555, doi. 10.1002/elan.1140040508

By:

Squella, J. A.;
Pezzani, M.;
Cassels, Bruce K.;
Aillon-Torres, Milton;
Rezende, Marcos C.;
Nuñez-Vergara, L. J.

Publication type:

Article

Varenicline and cytisine: two nicotinic acetylcholine receptor ligands reduce ethanol intake in University of Chile bibulous rats.

Published in:

Psychopharmacology, 2013, v. 227, n. 2, p. 287, doi. 10.1007/s00213-013-2974-3

By:

Sotomayor-Zárate, Ramón;
Gysling, Katia;
Busto, Usoa;
Cassels, Bruce;
Tampier, Lutske;
Quintanilla, María

Publication type:

Article

Synthesis, scope, H and C spectral assignments of isomeric dibenzofuran carboxaldehydes.

Published in:

Research on Chemical Intermediates, 2017, v. 43, n. 3, p. 1291, doi. 10.1007/s11164-016-2698-1

By:

Yempala, Thirumal;
Cassels, Bruce

Publication type:

Article

5-HT2 receptor binding, functional activity and selectivity in N-benzyltryptamines.

Published in:

PLoS ONE, 2019, v. 14, n. 01, p. 1, doi. 10.1371/journal.pone.0209804

By:

Toro-Sazo, Miguel;
Brea, José;
Loza, María I.;
Cimadevila, Marta;
Cassels, Bruce K.

Publication type:

Article

Inhibitory effect of boldine on fish oil oxidation.

Published in:

Journal of the American Oil Chemists' Society (JAOCS), 1991, v. 68, n. 12, p. 935, doi. 10.1007/BF02657538

By:

Valenzuela, Alfonso;
Nieto, Susana;
Cassels, Bruce;
Speisky, Hernan

Publication type:

Article

A Novel Route to 5,7-Dimethoxy-6-hydroxyflavone.

Published in:

Synthetic Communications, 1999, v. 29, n. 5, p. 815, doi. 10.1080/00397919908086038

By:

Osorio-olivares, Mauricio;
Cassels, Bruce K.;
Sepúlveda-Boza, Silvia;
Rezende, Marcos Caroli

Publication type:

Article

Total Synthesis of Annofolin.

Published in:

Synthetic Communications, 1999, v. 29, n. 5, p. 809, doi. 10.1080/00397919908086037

By:

Vallejos, Gabriel;
Cassels, Bruce K.;
Rezende, Marcos Caroli;
Sepulveda, Silvia

Publication type:

Article

The Regioselective Bromination of 4,4-Dimethyl-5,8-Dihydroxy-4 H -Naphthalen-1-One.

Published in:

Synthetic Communications, 1998, v. 28, n. 23, p. 4365, doi. 10.1080/00397919808004471

By:

Mejías, Lorenzo;
Sepúlveda, Silvia;
Araya, Ramiro;
Cassels, Bruce K.;
CaroliRezende, Marcos

Publication type:

Article

The Preparation of Potentially Psychoactive β-Alkoxyphenethylamines.

Published in:

Synthetic Communications, 1995, v. 25, n. 8, p. 1239, doi. 10.1080/00397919508012687

By:

Torres, Milton Aillón.;
Cassels, Bruce;
Rezende, Macros C.

Publication type:

Article

Some Fluoro and Nitro Analogues of Hallucinogenic Amphetamines.

Published in:

Synthetic Communications, 1994, v. 24, n. 3, p. 417, doi. 10.1080/00397919408011201

By:

Jara, Aida Neira;
Torres, Milton Aillon;
Cassels, Bruce Kennedy;
Rezende, Marcos Caroli

Publication type:

Article

Topical anti-inflammatory activity of quillaic acid from Quillaja saponaria Mol. and some derivatives.

Published in:

Journal of Pharmacy & Pharmacology, 2011, v. 63, n. 5, p. 718, doi. 10.1111/j.2042-7158.2011.01263.x

By:

Rodríguez-Díaz, Maité;
Delporte, Carla;
Cartagena, Carlos;
Cassels, Bruce K.;
González, Patricia;
Silva, Ximena;
León, Fredy;
Wessjohann, Ludger A.

Publication type:

Article

Monoamine Oxidase Inhibitory Properties of Optical Isomers and N -substituted Derivatives of 4-methylthioamphetamine.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2003, v. 18, n. 4, p. 339, doi. 10.1080/1475636031000118437

By:

Hurtado-Guzmán, Claudio;
Fierro, Angélica;
Iturriaga-Vásquez, Patricio;
Sepúlveda-Boza, Silvia;
Cassels, Bruce K.;
Reyes-Parada, Miguel

Publication type:

Article

(R)-Salsolinol, a product of ethanol metabolism, stereospecifically induces behavioral sensitization and leads to excessive alcohol intake.

Published in:

2016

By:

Quintanilla, María Elena;
Rivera‐Meza, Mario;
Berríos‐Cárcamo, Pablo;
Cassels, Bruce K.;
Herrera‐Marschitz, Mario;
Israel, Yedy;
Quintanilla, María Elena;
Rivera-Meza, Mario;
Berríos-Cárcamo, Pablo;
Herrera-Marschitz, Mario

Publication type:

journal article

Iron Chelators and Antioxidants Regenerate Neuritic Tree and Nigrostriatal Fibers of MPP+/MPTP-Lesioned Dopaminergic Neurons.

Published in:

PLoS ONE, 2015, v. 10, n. 12, p. 1, doi. 10.1371/journal.pone.0144848

By:

Aguirre, Pabla;
Mena, Natalia P.;
Carrasco, Carlos M.;
Muñoz, Yorka;
Pérez-Henríquez, Patricio;
Morales, Rodrigo A.;
Cassels, Bruce K.;
Méndez-Gálvez, Carolina;
García-Beltrán, Olimpo;
González-Billault, Christian;
Núñez, Marco T.

Publication type:

Article

Analysis of 25 C NBOMe in Seized Blotters by HPTLC and GC-MS.

Published in:

Journal of Chromatographic Science, 2016, v. 54, n. 7, p. 1153, doi. 10.1093/chromsci/bmw095

By:

Duffau, Boris;
Camargo, Cristian;
Kogan, Marcelo;
Fuentes, Edwar;
Cassels, Bruce Kennedy

Publication type:

Article

Coumarin-Based Fluorescent Probes for Dual Recognition of Copper(II) and Iron(III) Ions and Their Application in Bio-Imaging.

Published in:

Sensors (14248220), 2014, v. 14, n. 1, p. 1358, doi. 10.3390/s140101358

By:

García-Beltrán, Olimpo;
Cassels, Bruce K.;
Pérez, Claudio;
Mena, Natalia;
Núñez, Marco T.;
Martínez, Natalia P.;
Pavez, Paulina;
Aliaga, Margarita E.

Publication type:

Article

Aromatic Bromination Abolishes the Psychomotor Features and Pro-social Responses of MDMA ("Ecstasy") in Rats and Preserves Affinity for the Serotonin Transporter (SERT).

Published in:

Frontiers in Pharmacology, 2019, p. N.PAG, doi. 10.3389/fphar.2019.00157

By:

Sáez-Briones, Patricio;
Castro-Castillo, Vicente;
Díaz-Véliz, Gabriela;
Valladares, Luis;
Barra, Rafael;
Hernández, Alejandro;
Cassels, Bruce K.

Publication type:

Article

Theoretical insights into the regioselectivity of a Pictet-Spengler reaction: Transition state structures leading to salsolinol and isosalsolinol.

Published in:

Journal of Physical Organic Chemistry, 2017, v. 30, n. 8, p. n/a, doi. 10.1002/poc.3666

By:

Almodovar, Iriux;
Rezende, Marcos Caroli;
Cassels, Bruce K.;
García‐Arriagada, Macarena

Publication type:

Article

Nucleophilic reactivity of biothiols toward coumarin-based derivatives containing a chalcone moiety Nucleophilic reactivity of biothiols toward coumarin-based derivatives containing a chalcone moiety.

Published in:

Journal of Physical Organic Chemistry, 2012, v. 25, n. 11, p. 946, doi. 10.1002/poc.2975

By:

García‐Beltrán, Olimpo;
González, Christopher;
Pérez, Edwin G.;
Cassels, Bruce K.;
Santos, José G.;
Millán, Daniela;
Mena, Natalia;
Pavez, Paulina;
Aliaga, Margarita E.

Publication type:

Article

NEW HETEROCYCLIC SKELETONS DERIVED FROM THE APORPHINE ALKALOID BOLDINE.

Published in:

Synthetic Communications, 2002, v. 32, n. 23, p. 3687, doi. 10.1081/SCC-120014990

By:

Sobarzo-Sánchez, Eduardo;
Jullian, Carolina;
Cassels, Bruce K.;
Saitz, Claudio

Publication type:

Article

S-OXIDATION PRODUCTS OF ALKYLTHIOAMPHETAMINES.

Published in:

Synthetic Communications, 2002, v. 32, n. 17, p. 2741, doi. 10.1081/SCC-120006041

By:

Rezende, Marcos Caroli;
Núñez, Christián;
Sepúlveda-Boza, Silvia;
Cassels, Bruce K.;
Guzmán, Claudio Hurtado

Publication type:

Article

Works matching AU Cassels, Bruce

Evaluation of benzyltetrahydroisoquinolines as ligands for neuronal nicotinic acetylcholine receptors.

4-Bromo-2,5-dimethoxyphenethylamine (2C-B) and structurally related phenylethylamines are potent 5-HT<sub>2A</sub> receptor antagonists in Xenopus laevis oocytes.

Differences in potency and efficacy of a series of phenylisopropylamine/phenylethylamine pairs at 5-HT[sub 2A] and 5-HT[sub 2C] receptors.

Boldine inhibits the alveolar bone resorption during ligature-induced periodontitis by modulating the Th17/Treg imbalance.

Dibenzofuran annulated 1-azepines: Synthesis and cytotoxicity.

Simple and efficient synthesis of various dibenzofuran carbaldehydes.

Functional roles of T3.37 and S5.46 in the activation mechanism of the dopamine D1 receptor.

Why is quercetin a better antioxidant than taxifolin? Theoretical study of mechanisms involving activated forms.

Targeting Sentinel Proteins and Extrasynaptic Glutamate Receptors: a Therapeutic Strategy for Preventing the Effects Elicited by Perinatal Asphyxia?

Neurochemical and Behavioural Characterisation of Alkoxyamphetamine Derivatives in Rats.

Telomerase Inhibition by a New Synthetic Derivative of the Aporphine Alkaloid Boldine.

Molecular dynamics simulation of halogen bonding mimics experimental data for cathepsin L inhibition.

Distinguishing rotamers in N-trifluoroacetyl-3-benzazepine derivatives.

Complete <sup>1</sup>H and <sup>13</sup>C NMR spectral assignment of hydrogenated oxoisoaporphine derivatives.

Complete structural and spectral assignment of oxoisoaporphines by HMQC and HMBC experiments.

Amphetamine Derivatives as Monoamine Oxidase Inhibitors.

Cathodic behavior of 4,5-dimethoxy-2-nitroamphetamine.

Varenicline and cytisine: two nicotinic acetylcholine receptor ligands reduce ethanol intake in University of Chile bibulous rats.

Synthesis, scope, H and C spectral assignments of isomeric dibenzofuran carboxaldehydes.

5-HT<sub>2</sub> receptor binding, functional activity and selectivity in N-benzyltryptamines.

Inhibitory effect of boldine on fish oil oxidation.

A Novel Route to 5,7-Dimethoxy-6-hydroxyflavone.

Total Synthesis of Annofolin.

The Regioselective Bromination of 4,4-Dimethyl-5,8-Dihydroxy-4 H -Naphthalen-1-One.

The Preparation of Potentially Psychoactive β-Alkoxyphenethylamines.

Some Fluoro and Nitro Analogues of Hallucinogenic Amphetamines.

Topical anti-inflammatory activity of quillaic acid from Quillaja saponaria Mol. and some derivatives.

Monoamine Oxidase Inhibitory Properties of Optical Isomers and N -substituted Derivatives of 4-methylthioamphetamine.

(R)-Salsolinol, a product of ethanol metabolism, stereospecifically induces behavioral sensitization and leads to excessive alcohol intake.

Iron Chelators and Antioxidants Regenerate Neuritic Tree and Nigrostriatal Fibers of MPP+/MPTP-Lesioned Dopaminergic Neurons.

Analysis of 25 C NBOMe in Seized Blotters by HPTLC and GC-MS.

Coumarin-Based Fluorescent Probes for Dual Recognition of Copper(II) and Iron(III) Ions and Their Application in Bio-Imaging.

Aromatic Bromination Abolishes the Psychomotor Features and Pro-social Responses of MDMA ("Ecstasy") in Rats and Preserves Affinity for the Serotonin Transporter (SERT).

Theoretical insights into the regioselectivity of a Pictet-Spengler reaction: Transition state structures leading to salsolinol and isosalsolinol.

Nucleophilic reactivity of biothiols toward coumarin-based derivatives containing a chalcone moiety Nucleophilic reactivity of biothiols toward coumarin-based derivatives containing a chalcone moiety.

NEW HETEROCYCLIC SKELETONS DERIVED FROM THE APORPHINE ALKALOID BOLDINE.

S-OXIDATION PRODUCTS OF ALKYLTHIOAMPHETAMINES.