Works by Angeli, Andrea

Results: 182

Hitting Two Birds With One Stone: Dual Modulation of Brain Carbonic Anhydrases and Histone Deacetylases Boosts Memory Consolidation.

Published in:

Archiv der Pharmazie, 2025, v. 358, n. 6, p. 1, doi. 10.1002/ardp.70020

By:

Costa, Alessia;
Bozdag, Murat;
Renzi, Gioele;
Rani, Barbara;
Passani, Maria Beatrice;
Angeli, Andrea;
Provensi, Gustavo;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Discovery of a new potent oxindole multi-kinase inhibitor among a series of designed 3-alkenyl-oxindoles with ancillary carbonic anhydrase inhibitory activity as antiproliferative agents.

Published in:

BMC Chemistry, 2023, v. 17, n. 1, p. 1, doi. 10.1186/s13065-023-00994-3

By:

Ismail, Rania S. M.;
El Kerdawy, Ahmed M.;
Soliman, Dalia H.;
Georgey, Hanan H.;
Abdel Gawad, Nagwa M.;
Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Phenols from Origanum dictamnus L. and Thymus vulgaris L. and their activity against Malassezia globosa carbonic anhydrase.

Published in:

Natural Product Research, 2022, v. 36, n. 6, p. 1558, doi. 10.1080/14786419.2021.1880406

By:

Paloukopoulou, Charikleia;
Govari, Sofia;
Soulioti, Athina;
Stefanis, Ilias;
Angeli, Andrea;
Matheeussen, An;
Capasso, Clemente;
Cos, Paul;
Supuran, Claudiu T.;
Karioti, Anastasia

Publication type:

Article

Two Photographs.

Published in:

disClosure, 2011, v. 20, p. 102

By:

Angeli, Andrea

Publication type:

Article

Seven Photographs.

Published in:

disClosure, 2011, v. 20, p. 72

By:

Angeli, Andrea

Publication type:

Article

Calixarenes Incorporating Sulfonamide Moieties: Versatile Ligands for Carbonic Anhydrases Inhibition.

Published in:

Chemistry - A European Journal, 2022, v. 28, n. 6, p. 1, doi. 10.1002/chem.202103527

By:

Sbravati, Davide;
Bonardi, Alessandro;
Bua, Silvia;
Angeli, Andrea;
Ferraroni, Marta;
Nocentini, Alessio;
Casnati, Alessandro;
Gratteri, Paola;
Sansone, Francesco;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of Schistosoma mansoni carbonic anhydrase by the antiparasitic drug clorsulon: X‐ray crystallographic and in vitro studies.

Published in:

Acta Crystallographica: Section D, Structural Biology, 2022, v. 78, n. 3, p. 321, doi. 10.1107/S2059798322000079

By:

Ferraroni, Marta;
Angeli, Andrea;
Carradori, Simone;
Supuran, Claudiu T.

Publication type:

Article

Carbonic Anhydrases: Versatile and Useful Biocatalysts in Chemistry and Biochemistry.

Published in:

Catalysts (2073-4344), 2020, v. 10, n. 9, p. 1008, doi. 10.3390/catal10091008

By:

Angeli, Andrea;
Carta, Fabrizio;
Supuran, Claudiu T.

Publication type:

Article

Investigation on Human Carbonic Anhydrase IX and XII Inhibitory Activity and A549 Antiproliferative Activity of a New Class of Coumarinamides.

Published in:

Pharmaceuticals (14248247), 2025, v. 18, n. 3, p. 372, doi. 10.3390/ph18030372

By:

Moi, Davide;
Carradori, Simone;
Gallorini, Marialucia;
Mencarelli, Noemi;
Deplano, Alberto;
Angeli, Andrea;
Vittorio, Serena;
Supuran, Claudiu T.;
Onnis, Valentina

Publication type:

Article

Azobenzenesulfonamide Carbonic Anhydrase Inhibitors as New Weapons to Fight Helicobacter pylori : Synthesis, Bioactivity Evaluation, In Vivo Toxicity, and Computational Studies.

Published in:

Pharmaceuticals (14248247), 2024, v. 17, n. 8, p. 1027, doi. 10.3390/ph17081027

By:

Giampietro, Letizia;
Marinacci, Beatrice;
Della Valle, Alice;
D'Agostino, Ilaria;
Lauro, Aldo;
Mori, Mattia;
Carradori, Simone;
Ammazzalorso, Alessandra;
De Filippis, Barbara;
Maccallini, Cristina;
Angeli, Andrea;
Capasso, Clemente;
Francati, Santolo;
Mollica, Adriano;
Grande, Rossella;
Supuran, Claudiu T.

Publication type:

Article

Pyrazolo[4,3-c]pyridine Sulfonamides as Carbonic Anhydrase Inhibitors: Synthesis, Biological and In Silico Studies.

Published in:

Pharmaceuticals (14248247), 2022, v. 15, n. 3, p. 316, doi. 10.3390/ph15030316

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Lichitsky, Boris;
Komogortsev, Andrey;
Pinteala, Mariana;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

New Sulfanilamide Derivatives Incorporating Heterocyclic Carboxamide Moieties as Carbonic Anhydrase Inhibitors.

Published in:

Pharmaceuticals (14248247), 2021, v. 14, n. 8, p. 828, doi. 10.3390/ph14080828

By:

Angeli, Andrea;
Kartsev, Victor;
Petrou, Anthi;
Pinteala, Mariana;
Vydzhak, Roman M.;
Panchishin, Svitlana Y.;
Brovarets, Volodymyr;
De Luca, Viviana;
Capasso, Clemente;
Geronikaki, Athina;
Supuran, Claudiu T.

Publication type:

Article

Species-Specific Secondary Metabolites from Primula veris subsp. veris Obtained In Vitro Adventitious Root Cultures: An Alternative for Sustainable Production.

Published in:

Sustainability (2071-1050), 2023, v. 15, n. 3, p. 2452, doi. 10.3390/su15032452

By:

Sarropoulou, Virginia;
Sarrou, Eirini;
Angeli, Andrea;
Martens, Stefan;
Maloupa, Eleni;
Grigoriadou, Katerina

Publication type:

Article

An insight into the last 5-year patents on Porphyromonas gingivalis and Streptococcus mutans, the pivotal pathogens in the oral cavity.

Published in:

Expert Opinion on Therapeutic Patents, 2024, v. 34, n. 6, p. 433, doi. 10.1080/13543776.2024.2349739

By:

Bernardoni, Bianca Laura;
D'Agostino, Ilaria;
La Motta, Concettina;
Angeli, Andrea

Publication type:

Article

Proteasome inhibitors as anticancer agents.

Published in:

Expert Opinion on Therapeutic Patents, 2023, v. 33, n. 11, p. 775, doi. 10.1080/13543776.2023.2272648

By:

Gazzaroli, Giorgia;
Angeli, Andrea;
Giacomini, Arianna;
Ronca, Roberto

Publication type:

Article

Prostaglandin receptor agonists as antiglaucoma agents (a patent review 2013 – 2018).

Published in:

Expert Opinion on Therapeutic Patents, 2019, v. 29, n. 10, p. 793, doi. 10.1080/13543776.2019.1661992

By:

Angeli, Andrea;
Supuran, Claudiu T

Publication type:

Article

Treatment of sleep apnea with a combination of a carbonic anhydrase inhibitor and an aldosterone antagonist: a patent evaluation of CA2958110 and IN6616DEN2012.

Published in:

Expert Opinion on Therapeutic Patents, 2018, v. 28, n. 10, p. 723, doi. 10.1080/13543776.2018.1497160

By:

Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Metabolite profiling of wines made from disease-tolerant varieties.

Published in:

European Food Research & Technology, 2019, v. 245, n. 9, p. 2039, doi. 10.1007/s00217-019-03314-z

By:

Ruocco, Silvia;
Perenzoni, Daniele;
Angeli, Andrea;
Stefanini, Marco;
Rühl, Ernst;
Patz, Claus-Dieter;
Mattivi, Fulvio;
Rauhut, Doris;
Vrhovsek, Urska

Publication type:

Article

Propolis Hydroalcoholic Extracts: Biochemical Characterization and Antifungal Efficacy.

Published in:

Horticulturae, 2025, v. 11, n. 2, p. 122, doi. 10.3390/horticulturae11020122

By:

Sadallah, Abderraouf;
Aprea, Eugenio;
Cignola, Rudy;
Caratti, Andrea;
Cordero, Chiara;
Angeli, Andrea;
Martens, Stefan;
Di Francesco, Alessandra

Publication type:

Article

Crystal structure and chemical inhibition of essential schistosome host-interactive virulence factor carbonic anhydrase SmCA.

Published in:

Communications Biology, 2019, v. 2, n. 1, p. N.PAG, doi. 10.1038/s42003-019-0578-0

By:

Da'dara, Akram A.;
Angeli, Andrea;
Ferraroni, Marta;
Supuran, Claudiu T.;
Skelly, Patrick J.

Publication type:

Article

2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2270183

By:

Sequeira, Lisa;
Distinto, Simona;
Meleddu, Rita;
Gaspari, Marco;
Angeli, Andrea;
Cottiglia, Filippo;
Secci, Daniela;
Onali, Alessia;
Sanna, Erica;
Borges, Fernanda;
Uriarte, Eugenio;
Alcaro, Stefano;
Supuran, Claudiu T.;
Maccioni, Elias

Publication type:

Article

Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2203389

By:

Shaldam, Moataz A.;
Almahli, Hadia;
Angeli, Andrea;
Badi, Rehab Mustafa;
Khaleel, Eman F.;
Zain-Alabdeen, Abdelrahman I.;
Elsayed, Zainab M.;
Elkaeed, Eslam B.;
Salem, Rofaida;
Supuran, Claudiu T.;
Eldehna, Wagdy M.;
Tawfik, Haytham O.

Publication type:

Article

Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2201402

By:

Fantacuzzi, Marialuigia;
D'Agostino, Ilaria;
Carradori, Simone;
Liguori, Francesco;
Carta, Fabrizio;
Agamennone, Mariangela;
Angeli, Andrea;
Sannio, Filomena;
Docquier, Jean-Denis;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2191165

By:

Astrain-Redin, Nora;
Paoletti, Niccolò;
Plano, Daniel;
Bonardi, Alessandro;
Gratteri, Paola;
Angeli, Andrea;
Sanmartin, Carmen;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2185760

By:

Mahammad Ghouse, Shaik;
Bahatam, Kavyaraj;
Angeli, Andrea;
Pawar, Gaurav;
Chinchilli, Krishna Kartheek;
Yaddanapudi, Venkata Madhavi;
Mohammed, Arifuddin;
Supuran, Claudiu T.;
Nanduri, Srinivas

Publication type:

Article

Cloning, characterization, and inhibition of the novel β-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2184299

By:

Haapanen, Susanna;
Angeli, Andrea;
Tolvanen, Martti;
Emameh, Reza Zolfaghari;
Supuran, Claudiu T.;
Parkkila, Seppo

Publication type:

Article

Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2178430

By:

Angeli, Andrea;
Ferraroni, Marta;
Bonardi, Alessandro;
Supuran, Claudiu T.;
Nocentini, Alessio

Publication type:

Article

Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2023, v. 38, n. 1, p. 1, doi. 10.1080/14756366.2023.2166503

By:

Angeli, Andrea;
Supuran, Claudiu T.

Publication type:

Article

Selective inhibition of carbonic anhydrase IX by sulphonylated 1,2,3-triazole incorporated benzenesulphonamides capable of inducing apoptosis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1454, doi. 10.1080/14756366.2022.2077333

By:

Siwach, Kiran;
Kumar, Amit;
Panchal, Harish;
Kumar, Rajiv;
Bhardwaj, Jitender Kumar;
Angeli, Andrea;
Supuran, Claudiu T.;
Sharma, Pawan K.

Publication type:

Article

Heterologous expression and biochemical characterisation of the recombinant β-carbonic anhydrase (MpaCA) from the warm-blooded vertebrate pathogen malassezia pachydermatis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 62, doi. 10.1080/14756366.2021.1994559

By:

De Luca, Viviana;
Angeli, Andrea;
Mazzone, Valeria;
Adelfio, Claudia;
Carginale, Vincenzo;
Scaloni, Andrea;
Carta, Fabrizio;
Selleri, Silvia;
Supuran, Claudiu T.;
Capasso, Clemente

Publication type:

Article

Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 857, doi. 10.1080/14756366.2022.2051023

By:

Sharonova, Tatiana;
Zhmurov, Petr;
Kalinin, Stanislav;
Nocentini, Alessio;
Angeli, Andrea;
Ferraroni, Marta;
Korsakov, Mikhail;
Supuran, Claudiu T.;
Krasavin, Mikhail

Publication type:

Article

Development of Praziquantel sulphonamide derivatives as antischistosomal drugs.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 1479, doi. 10.1080/14756366.2022.2078970

By:

Angeli, Andrea;
Ferraroni, Marta;
Carta, Fabrizio;
Häberli, Cécile;
Keiser, Jennifer;
Costantino, Gabriele;
Supuran, Claudiu T.

Publication type:

Article

Dependence on linkers' flexibility designed for benzenesulfonamides targeting discovery of novel hCA IX inhibitors as potent anticancer agents.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2765, doi. 10.1080/14756366.2022.2130285

By:

Tawfik, Haytham O.;
Belal, Amany;
Abourehab, Mohammed A. S.;
Angeli, Andrea;
Bonardi, Alessandro;
Supuran, Claudiu T.;
El-Hamamsy, Mervat H.

Publication type:

Article

Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 986, doi. 10.1080/14756366.2022.2055009

By:

D'Agostino, Ilaria;
Mathew, Githa Elizabeth;
Angelini, Paola;
Venanzoni, Roberto;
Flores, Giancarlo Angeles;
Angeli, Andrea;
Carradori, Simone;
Marinacci, Beatrice;
Menghini, Luigi;
Abdelgawad, Mohamed A.;
Ghoneim, Mohammed M.;
Mathew, Bijo;
Supuran, Claudiu T.

Publication type:

Article

Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic anhydrase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 2786, doi. 10.1080/14756366.2022.2131780

By:

Angeli, Andrea;
Urbański, Linda J.;
Capasso, Clemente;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological studies.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2022, v. 37, n. 1, p. 994, doi. 10.1080/14756366.2022.2055553

By:

Nada, Hossam;
Elkamhawy, Ahmed;
Abdellattif, Magda H.;
Angeli, Andrea;
Chang Hoon Lee;
Supuran, Claudiu T.;
Kyeong Lee

Publication type:

Article

Carbonic anhydrase activation profile of indole-based derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 1783, doi. 10.1080/14756366.2021.1959573

By:

Barresi, Elisabetta;
Ravichandran, Rahul;
Germelli, Lorenzo;
Angeli, Andrea;
Baglini, Emma;
Salerno, Silvia;
Marini, Anna Maria;
Costa, Barbara;
Da Pozzo, Eleonora;
Martini, Claudia;
Da Settimo, Federico;
Supuran, Claudiu;
Cosconati, Sandro;
Taliani, Sabrina

Publication type:

Article

Activation of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with amines and amino acids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 758, doi. 10.1080/14756366.2021.1897802

By:

Angeli, Andrea;
Urbański, Linda J.;
Hytönen, Vesa P.;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 685, doi. 10.1080/14756366.2021.1887171

By:

Meleddu, Rita;
Deplano, Serenella;
Maccioni, Elias;
Ortuso, Francesco;
Cottiglia, Filippo;
Secci, Daniela;
Onali, Alessia;
Sanna, Erica;
Angeli, Andrea;
Angius, Rossella;
Alcaro, Stefano;
Supuran, Claudiu T.;
Distinto, Simona

Publication type:

Article

Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 561, doi. 10.1080/14756366.2021.1882453

By:

Nocentini, Alessio;
Angeli, Andrea;
Carta, Fabrizio;
Winum, Jean-Yves;
Zalubovskis, Raivis;
Carradori, Simone;
Capasso, Clemente;
Donald, William A.;
Supuran, Claudiu T.

Publication type:

Article

Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2021, v. 36, n. 1, p. 330, doi. 10.1080/14756366.2020.1863958

By:

Urbański, Linda J.;
Angeli, Andrea;
Hytönen, Vesa P.;
Di Fiore, Anna;
De Simone, Giuseppina;
Parkkila, Seppo;
Supuran, Claudiu T.

Publication type:

Article

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1891, doi. 10.1080/14756366.2020.1828401

By:

Guglielmi, Paolo;
Rotondi, Giulia;
Secci, Daniela;
Angeli, Andrea;
Chimenti, Paola;
Nocentini, Alessio;
Bonardi, Alessandro;
Gratteri, Paola;
Carradori, Simone;
Supuran, Claudiu T.

Publication type:

Article

Sulphonamide inhibition profile of Staphylococcus aureus β-carbonic anhydrase.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1834, doi. 10.1080/14756366.2020.1826942

By:

Urbanski, Linda J.;
Bua, Silvia;
Angeli, Andrea;
Kuuslahti, Marianne;
Hytönen, Vesa. P.;
Supuran, Claudiu T.;
Parkkila, Seppo

Publication type:

Article

Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1442, doi. 10.1080/14756366.2020.1786821

By:

Mancuso, Francesca;
De Luca, Laura;
Angeli, Andrea;
Del Prete, Sonia;
Capasso, Clemente;
Supuran, Claudiu T.;
Gitto, Rosaria

Publication type:

Article

Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase from Trichomonas vaginalis.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1292, doi. 10.1080/14756366.2020.1774572

By:

Urbański, Linda J.;
Di Fiore, Anna;
Azizi, Latifeh;
Hytönen, Vesa P.;
Kuuslahti, Marianne;
Buonanno, Martina;
Monti, Simona M.;
Angeli, Andrea;
Zolfaghari Emameh, Reza;
Supuran, Claudiu T.;
De Simone, Giuseppina;
Parkkila, Seppo

Publication type:

Article

Preparation, carbonic anhydrase enzyme inhibition and antioxidant activity of novel 7-amino-3,4-dihydroquinolin-2(1H)-one derivatives incorporating mono or dipeptide moiety.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1021, doi. 10.1080/14756366.2020.1751620

By:

Küçükbay, Hasan;
Gönül, Zeynep;
Küçükbay, F. Zehra;
Angeli, Andrea;
Bartolucci, Gianluca;
Supuran, Claudiu T.

Publication type:

Article

Synthesis and carbonic anhydrase activating properties of a series of 2-amino-imidazolines structurally related to clonidine<sup>1</sup>.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 1003, doi. 10.1080/14756366.2020.1749602

By:

Chiaramonte, Niccolò;
Maach, Soumia;
Biliotti, Caterina;
Angeli, Andrea;
Bartolucci, Gianluca;
Braconi, Laura;
Dei, Silvia;
Teodori, Elisabetta;
Supuran, Claudiu T.;
Romanelli, Maria Novella

Publication type:

Article

1,2,4-Triazole-based anticonvulsant agents with additional ROS scavenging activity are effective in a model of pharmacoresistant epilepsy.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 993, doi. 10.1080/14756366.2020.1748026

By:

Kaproń, Barbara;
Czarnomysy, Robert;
Wysokiński, Mariusz;
Andrys, Rudolf;
Musilek, Kamil;
Angeli, Andrea;
Supuran, Claudiu T.;
Plech, Tomasz

Publication type:

Article

Activation studies of the β-carbonic anhydrases from Malassezia restricta with amines and amino acids.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 824, doi. 10.1080/14756366.2020.1743284

By:

Angeli, Andrea;
Prete, Sonia Del;
Ghobril, Cynthia;
Hitce, Julien;
Clavaud, Cécile;
Marrat, Xavier;
Donald, William A.;
Capasso, Clemente;
Supuran, Claudiu T.

Publication type:

Article

Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation.

Published in:

Journal of Enzyme Inhibition & Medicinal Chemistry, 2020, v. 35, n. 1, p. 539, doi. 10.1080/14756366.2020.1713114

By:

Fois, Benedetta;
Distinto, Simona;
Meleddu, Rita;
Deplano, Serenella;
Maccioni, Elias;
Floris, Costantino;
Rosa, Antonella;
Nieddu, Mariella;
Caboni, Pierluigi;
Sissi, Claudia;
Angeli, Andrea;
Supuran, Claudiu T.;
Cottiglia, Filippo

Publication type:

Article