Works matching IS 18607179 AND DT 2025 AND VI 20 AND IP 9

Results: 21

Fast Release of Carboxylic Acid inside Cells.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202500056

By:

Moser, Pascal;
Zelli, Renaud;
dos Santos, Leandro J.;
Henry, Mickaël;
Sanchez‐Garcia, Kevin;
Caspar, Yvan;
Marro, Florian C.;
Chovelon, Benoit;
Saez Cabodevilla, Jaione;
de Choudens, Sandrine Ollagnier;
Faudry, Eric;
Wong, Yung‐Sing

Publication type:

Article

Front Cover: Novel Sulfonamide‐Sydnone Hybrids: Complementary Insight into Anti‐Inflammatory Action, Anti‐SARS‐CoV‐2 Activity, Human Serum Albumin Interaction, and in silico Analysis (ChemMedChem 9/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202580901

By:

Resendes Barbosa, Igor;
Alves Amorim, Mayara;
de Souza Oliveira, Vitor Hélio;
André, Eunice;
Pereira Guedes, Guilherme;
Augusto Chaves, Otávio;
Serpa, Carlos;
Fintelman‐Rodrigues, Natalia;
Sacramento, Carolina Q.;
Moreno L. Souza, Thiago;
Sant'Anna, Carlos Mauricio R.;
Echevarria, Aurea

Publication type:

Article

Design and Synthesis of Tetrahydropyrrolo[3,4‐c]Pyrazole Sigma‐1 Receptor Ligands.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202401015

By:

Cosentino, Giuseppe;
Dichiara, Maria;
Costanzo, Giuliana;
Coco, Alessandro;
Pasquinucci, Lorella;
Marrazzo, Agostino;
Rescifina, Antonio;
Amata, Emanuele

Publication type:

Article

Lamellarin D Acts as an Inhibitor of Type I Collagen Production.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202401001

By:

Okuno, Daisuke;
Sakamoto, Noriho;
Hayashi, Hideki;
Fukuda, Tsutomu;
Akiyama, Yoshiko;
Iketani, Chiaki;
Murakami, Ritsuko;
Tokito, Takatomo;
Miyamura, Takuto;
Yura, Hirokazu;
Kido, Takashi;
Ishimoto, Hiroshi;
Takemoto, Shinnosuke;
Takazono, Takahiro;
Nishino, Tomoya;
Ishimatsu, Yuji;
Ishihara, Jun;
Takeda, Kohsuke;
Tanaka, Yoshimasa;
Mukae, Hiroshi

Publication type:

Article

Synthesis and Antibacterial Properties of 3‐Amino‐β‐Lactams Bearing a Heteroatom‐Containing C4 Substituent.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400994

By:

Bredael, Kato;
Vanhecke, Fien;
Vandenheede, Emma;
Stevens, Christian V.;
Gobec, Stanislav;
D'hooghe, Matthias

Publication type:

Article

Molecular Engineering of Cordycepin Derivatives for Enhanced Biological Activity and Stability.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400979

By:

Gu, Yiming;
Yu, Wei;
Li, Xiang;
Fan, Yingjie;
Liu, Yanan;
Tummatorn, Jumreang;
Jiang, Siyu;
Yang, Jingyue

Publication type:

Article

Analogues of Natural Macarangin B Display Potent Antiviral Activity and Better Metabolic Stability.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400978

By:

Jézéquel, Gwenaëlle;
Fargier, Jules;
Bigay, Joëlle;
Polidori, Joël;
Geslin, Justine;
Hue, Nathalie;
El Kalamouni, Chaker;
Desrat, Sandy;
Roussi, Fanny

Publication type:

Article

Systematic Review on 1,2,3‐Oxadiazoles, 1,2,4‐Oxadiazoles, and 1,2,5‐Oxadiazoles in the Antimycobacterial Drug Discovery.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400971

By:

Kučerová‐Chlupáčová, Marta

Publication type:

Article

Structure‐Atropisomer Stability Relationship in Selective MCL‐1 Inhibitors.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400970

By:

Sipos, Szabolcs;
Balazs, Barbara;
Gati, Tamas;
Csékei, Márton;
Kováacs, Mihály;
Szlavik, Zoltan;
Paczal, Attila;
Bálint, Balázs;
Murray, James B.;
Davidson, James;
Hubbard, Roderick E.;
Le Toumelin‐Braizat, Gaëtane;
Maragno, Ana Leticia;
Geneste, Olivier;
Stirling, András;
Kotschy, András

Publication type:

Article

β‐Glucuronidase‐Responsive Albumin‐Binding Prodrug of Colchicine‐Site Binders for Selective Cancer Therapy.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400969

By:

Bordes, Alexandra;
Opalinski, Isabelle;
Thoreau, Fabien;
Provot, Olivier;
Hamze, Abdallah;
Alami, Mouad;
Papot, Sébastien

Publication type:

Article

Discovery of CCR8 Antagonist IDOR‐1136‐5177 for the Treatment of Cancer.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400968

By:

Diethelm, Stefan;
Remeň, Luboš;
Aissaoui, Hamed;
Leroy, Cédric;
Chavanton‐Arpel, Alexia;
Docci, Luca;
Seeland, Swen;
Lehembre, François;
Corminboeuf, Olivier

Publication type:

Article

GDF15 Analogues Acting as GFRAL Ligands.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400961

By:

Di Santo, Andrea;
Tarchi, Livio;
Villa, Gianluca;
Castellini, Giovanni;
Ricca, Valdo;
Squecco, Roberta;
Papini, Anna Maria;
Real‐Fernandez, Feliciana;
Rovero, Paolo

Publication type:

Article

Metal‐Catalyzed Cross‐Coupling for the Synthesis of β‐Lactam Drugs and Related Chemical Probes.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400960

By:

Bresson, Jules;
Burke, Katie;
Ethève‐Quelquejeu, Mélanie;
Iannazzo, Laura;
Cariou, Kevin

Publication type:

Article

Synthesis and Bio‐Evaluation of Quaternized Fused‐β‐Carbolines as Anti‐MRSA Agents.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400955

By:

Vutla, Adilakshmi;
Saxena, Deepanshi;
Maitra, Rahul;
Chopra, Sidharth;
Batra, Sanjay

Publication type:

Article

Advances in Lipid Nanoparticle‐Based Disease Treatment.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400938

By:

Zhou, Yujie;
Ge, Qiqi;
Wang, Xin;
Wang, Yuhui;
Sun, Qianqian;
Wang, Jianhao;
Yang, Tie;
Wang, Cheng

Publication type:

Article

Addressing Data Point Homogeneity and Annotation Challenges to Enhance Data‐Driven Approaches: The S. aureus NorA Efflux Pump Case Study.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400927

By:

Astolfi, Andrea;
Cernicchi, Giada;
Primavera, Erika;
Rocchi, Marco;
Manfroni, Giuseppe;
Sabatini, Stefano;
Letizia Barreca, Maria

Publication type:

Article

Machine Learning‐Driven Discovery of Structurally Related Natural Products as Activators of the Cardiac Calcium Pump SERCA2a.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400913

By:

Cruz‐Cortés, Carlos;
Fernández‐de Gortari, Eli;
Aguayo‐Ortiz, Rodrigo;
Šeflová, Jaroslava;
Ard, Adam;
Clasby, Martin;
Anumonwo, Justus;
Michel Espinoza‐Fonseca, L.

Publication type:

Article

Diversity‐Oriented Synthesis and Antibiofilm Evaluation of Furan‐2‐Carboxamides.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400879

By:

Muñoz‐Estrada, Ana C.;
Tovar‐Roman, Cesar E.;
García‐Mejía, Carlos D.;
García‐Contreras, Rodolfo;
Hernández‐Vázquez, Eduardo

Publication type:

Article

Design and Synthesis of <sup>68</sup>Ga‐Labeled Peptide‐Based Heterodimers for Dual Targeting of NTS<sub>1</sub> and GRPR.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400843

By:

Bodin, Sacha;
Previti, Santo;
Jestin, Emmanuelle;
Rémond, Emmanuelle;
Vimont, Delphine;
Lamare, Frédéric;
Ait‐Arsa, Imade;
Hindié, Elif;
Cavelier, Florine;
Morgat, Clément

Publication type:

Article

An Effective Reaction‐Based Virtual Screening Method to Discover New CDK8 Ligands.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400825

By:

Chen, Wei;
Fang, Hanlin;
He, Huan;
Ping, Jing;
Ge, Jianxin

Publication type:

Article

Novel Sulfonamide‐Sydnone Hybrids: Complementary Insight into Anti‐Inflammatory Action, Anti‐SARS‐CoV‐2 Activity, Human Serum Albumin Interaction, and in silico Analysis.

Published in:

ChemMedChem, 2025, v. 20, n. 9, p. 1, doi. 10.1002/cmdc.202400697

By:

Resendes Barbosa, Igor;
Alves Amorim, Mayara;
de Souza Oliveira, Vitor Hélio;
André, Eunice;
Pereira Guedes, Guilherme;
Augusto Chaves, Otávio;
Serpa, Carlos;
Fintelman‐Rodrigues, Natalia;
Sacramento, Carolina Q.;
Moreno L. Souza, Thiago;
Sant'Anna, Carlos Mauricio R.;
Echevarria, Aurea

Publication type:

Article