Works matching IS 18607179 AND DT 2025 AND VI 20 AND IP 6

Results: 22

Cover Feature: Improving Affinity while Reducing Kidney Uptake of CXCR4‐Targeting Radioligands Derived from the Endogenous Antagonist EPI‐X4 (ChemMedChem 6/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202580604

By:

Gaonkar, Raghuvir H.;
Bailly, Thibaud;
Millul, Jacopo;
Mansi, Rosalba;
Harms, Mirja;
Münch, Jan;
Fani, Melpomeni

Publication type:

Article

Front Cover: Beyond the Toll‐Like Receptor 4. Structure‐Dependent Lipopolysaccharide Recognition Systems: How far are we? (ChemMedChem 6/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202580601

By:

De Chiara, Stefania;
De Simone Carone, Luca;
Cirella, Roberta;
Andretta, Emanuela;
Silipo, Alba;
Molinaro, Antonio;
Mercogliano, Marcello;
Di Lorenzo, Flaviana

Publication type:

Article

CORRIGENDUM: α‐Triazolylboronic Acids: A Novel Scaffold to Target FLT3 in AML.

Published in:: ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400982
Publication type:: Article

Isopeptidic Desferrioxamine Analogues: The Role of Hydroxamate Spacing for Chelation of Zr<sup>4+</sup>.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400890

By:

Outzen, Lasse;
Ludolfs, Darius;
Irl, Maximilian;
Kossatz, Susanne;
Maison, Wolfgang

Publication type:

Article

Autophagy‐Mediated Targeted Protein Degradation.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400866

By:

Shao, Jinning;
Xie, Shangzhi;
Hong, Shurui;
Qian, Linghui

Publication type:

Article

Investigating the C2 Modulation of the Imidazo[1,2‐a]pyrazine‐Based Hit Compound CTN1122: Synthesis, in vitro Antileishmanial Activity, Cytotoxicity and Casein Kinase 1 Inhibition.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400862

By:

Tisseur, Lhana;
Cojean, Sandrine;
Gassama, Khadidiatou;
Logé, Cédric;
Pagniez, Fabrice;
Cavé, Christian;
Bernadat, Guillaume;
Loiseau, Philippe M.;
Bach, Stéphane;
Thiéfaine, Jérôme;
Picot, Carine;
Tomasoni, Christophe;
Leclercq, Olivier;
Baratte, Blandine;
Robert, Thomas;
Le Pape, Patrice;
Rachidi, Najma;
Bazin, Marc‐Antoine;
Marchand, Pascal

Publication type:

Article

Design and Synthesis of Unsymmetric Benzils, Quinoxalines, and Evaluations of their Anticancer Activities against Human Non‐Small Lung Cancer Cells.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400847

By:

Hsu, Ping‐Chih;
Hsu, Yu‐Hsin;
Chang, Chuan‐Hsin;
Shih, Tzenge‐Lien

Publication type:

Article

The Evaluation of Glyceryl C3‐Azolyl‐Thiogalactosides as Galectin‐1 and Galectin‐3 Ligands.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400826

By:

Prouza, Vít;
Zýka, Jakub;
Kozák, Jaroslav;
Magdolenová, Alžbeta;
Pohl, Radek;
Parkan, Kamil

Publication type:

Article

4‐Aza Cyclopentenone Prostaglandin Analogues: Synthesis and NF‐κB Inhibitory Activities.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400823

By:

Doherty, William;
Conway, Lorna;
Leveau, Brian;
Giulia Nacca, Francesca;
Chiappa, Lucia;
Riccio, Anna;
Roberts, Stanley M.;
Gabriella Santoro, M.;
Evans, Paul

Publication type:

Article

Coordination Compounds as Antivirals against Neglected Tropical Diseases.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400799

By:

Rezende, Wallace S.;
Neto, Antonio Marçal;
Corbi, Juliano J.;
Corbi, Pedro P.;
de Paiva, Raphael E. F.;
Bergamini, Fernando R. G.

Publication type:

Article

Synthesis of New Enantiopure Aminoalcohol Fluorenes as Promising Antimalarial Compounds.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400790

By:

Tisnerat, Camille;
Schneider, Jérémy;
Mustière, Romain;
Herrero, Aurélie;
Momha, René;
Damiani, Céline;
Agnamey, Patrice;
Totet, Anne;
Marchivie, Mathieu;
Guillon, Jean;
Dassonville‐Klimpt, Alexandra;
Sonnet, Pascal

Publication type:

Article

Oligomerization of 33‐mer Gliadin Peptides: Supramolecular Assemblies in Celiac Disease.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400789

By:

Dodero, Verónica I.;
Herrera, María G.

Publication type:

Article

Beyond the Toll‐Like Receptor 4. Structure‐Dependent Lipopolysaccharide Recognition Systems: How far are we?

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400780

By:

De Chiara, Stefania;
De Simone Carone, Luca;
Cirella, Roberta;
Andretta, Emanuela;
Silipo, Alba;
Molinaro, Antonio;
Mercogliano, Marcello;
Di Lorenzo, Flaviana

Publication type:

Article

Improving Affinity while Reducing Kidney Uptake of CXCR4‐Targeting Radioligands Derived from the Endogenous Antagonist EPI‐X4.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400773

By:

Gaonkar, Raghuvir H.;
Bailly, Thibaud;
Millul, Jacopo;
Mansi, Rosalba;
Harms, Mirja;
Münch, Jan;
Fani, Melpomeni

Publication type:

Article

Synthesis of 1,2,3‐Triazole‐Methyl‐Menadione Derivatives: Evaluation of Electrochemical and Antiparasitic Properties against two Blood‐Dwelling Parasites.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400731

By:

Dupouy, Baptiste;
Karpstein, Tanja;
Häberli, Cécile;
Cal, Monica;
Rottmann, Matthias;
Mäser, Pascal;
Keiser, Jennifer;
Elhabiri, Mourad;
Davioud‐Charvet, Elisabeth

Publication type:

Article

Crystal Structure of Ritonavir Polymorphs I and II Revisited with the Application of NMR Crystallography.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400709

By:

Szeleszczuk, Łukasz;
Gubica, Tomasz;
Maciej Pisklak, Dariusz

Publication type:

Article

Insight into Stabilization of G‐Quadruplex in c‐MYC Region with Phenanthroimidazoisoindol‐Acrylates and their Binding Behaviour towards Human Serum Albumin.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400705

By:

Thakur, Rekha;
Luxami, Vijay;
Paul, Kamaldeep

Publication type:

Article

Structure‐Based Virtual Screening and Biological Characterization of Novel BACE‐1 and Amyloid‐β Aggregation Inhibitors.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400685

By:

Sharma, Ankita;
Nayak, Madhusmita;
Thakur, Shikha;
Jadhav, Hemant R.;
Bharate, Sandip B.

Publication type:

Article

Inflammaging and Immunosenescence in the Post‐COVID Era: Small Molecules, Big Challenges.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400672

By:

Francavilla, Fabio;
Intranuovo, Francesca;
La Spada, Gabriella;
Lacivita, Enza;
Catto, Marco;
Graps, Elisabetta Anna;
Altomare, Cosimo Damiano

Publication type:

Article

Third‐Generation CD73 Inhibitors Based on a 4,6‐Disubstituted‐2‐Thiopyridine Scaffold.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400662

By:

Grosjean, Félix;
Shaldaeva, Maria;
Cros‐Perrial, Emeline;
Rodriguez, Céline;
Ghoteimi, Rayane;
Lebrun, Aurélien;
Gao, Zhan‐Guo;
Uttaro, Jean‐Pierre;
Mathé, Christophe;
Jacobson, Kenneth A.;
Petter Jordheim, Lars;
Ménétrier‐Caux, Christine;
Chaloin, Laurent;
Peyrottes, Suzanne

Publication type:

Article

Current Approaches and Strategies Applied in First‐in‐class Drug Discovery.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400639

By:

Mohammed, Idrees;
Sagurthi, Someswar Rao

Publication type:

Article

Discovery of Novel Pyrido[2,3‐b]Pyrazine Human Cytomegalovirus Polymerase Inhibitors with Broad Spectrum Antiherpetic Activity and Reduced hERG Inhibition.

Published in:

ChemMedChem, 2025, v. 20, n. 6, p. 1, doi. 10.1002/cmdc.202400629

By:

Bai, Bing;
Srinivas Kandadai, Appan;
Hena, Mostofa;
Belovodskiy, Alexandr;
Shen, John;
Houghton, Michael;
Nieman, James A.

Publication type:

Article