Works matching IS 18607179 AND DT 2025 AND VI 20 AND IP 4

Results: 18

Highlights from the Lowlands: Early Career Researchers Shine at Medicinal Chemistry Frontiers 2024.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400853

By:

McKenna, Sean M.;
Borsari, Chiara;
Chin Chan, Sean;
Donckele, Etienne J.;
Faucher, Franco F.;
Grenier‐Davies, Melissa C.;
Haranahalli, Krupanandan;
Matagne, Brieuc;
Monastyrskyi, Andrii;
Petracca, Rita

Publication type:

Article

Cover Feature: Design, Synthesis, and Anti‐Prostate Cancer Potential of 2‐(4‐Nitrobenzyl) Malonates In Vitro and DAL Acute Oral Toxicity Assessment In Vivo (ChemMedChem 4/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202580402

By:

Hassan Ganesh, Bharathi;
Aruchamy, Baladhandapani;
Mudradi, Srikrishna;
Mohanty, Sarthak;
Padinjarathil, Himabindu;
Carradori, Simone;
Ramani, Prasanna

Publication type:

Article

Front Cover: [18F]NP3‐627, a Candidate PET Imaging Agent Targeting the NLRP3 Inflammasome in the Central Nervous System (ChemMedChem 4/2025).

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400816

By:

Whitehead, David M.;
Fischer, Christian;
Briard, Emmanuelle;
Farady, Christopher J.;
Graveleau, Nadège;
Karrer, Joel;
Kaupmann, Klemens;
Lapointe, Guillaume;
Mackay, Angela;
Reichert, Lisa;
Wright, Michael;
Mu, Linjing;
Auberson, Yves P.

Publication type:

Article

Tumor Microenvironment‐Responsive Multinucleated Nanocomplexes Loaded with Carbon Dots for Combined Photothermal/Chemodynamic Therapy of Breast Cancer.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400983

By:

Zhu, Zihan;
Zhang, Yan;
He, Cui;
Jin, Yimin;
Bian, Wei;
Tang, Xinjing;
Wang, Jing

Publication type:

Article

[18F]NP3‐627, a Candidate PET Imaging Agent Targeting the NLRP3 Inflammasome in the Central Nervous System.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400816

By:

Whitehead, David M.;
Fischer, Christian;
Briard, Emmanuelle;
Farady, Christopher J.;
Graveleau, Nadège;
Karrer, Joel;
Kaupmann, Klemens;
Lapointe, Guillaume;
Mackay, Angela;
Reichert, Lisa;
Wright, Michael;
Mu, Linjing;
Auberson, Yves P.

Publication type:

Article

Styrylchromones: Biological Activities and Structure‐Activity Relationship.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400782

By:

Lucas, Mariana;
Freitas, Marisa;
Silva, Artur M. S.;
Fernandes, Eduarda;
Ribeiro, Daniela

Publication type:

Article

MuDRA‐Based Virtual Screening of Terpenes for Anti‐Leishmania Infantum Activity: In Vitro Validation and Mechanistic Insights from Molecular Docking.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400743

By:

Barros de Menezes, Renata Priscila;
Ferreira de Sousa, Natália;
Herrera‐Acevedo, Chonny;
Santos Aquino de Araújo, Rodrigo;
Durand Trigueiro Lira, Nikole;
Fechine Tavares, Josean;
Jorge Kato, Massuo;
Alex da Rocha Coelho, Francisco;
Sousa dos Santos, Airton Lucas;
Antonio da Franca Rodrigues, Klinger;
Bezerra Mendonça‐Júnior, Francisco Jaime;
Scotti, Luciana;
Tullius Scotti, Marcus

Publication type:

Article

Ac34deoGlcNAz: A Selective Probe for Identifying O‐GlcNAc‐Modified Proteins in Prostate Cancer.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400716

By:

Xu, Guoliang;
Zhu, Jiangtao;
Wang, Xihao;
Liu, Pengyue;
Yan, Yongjun;
Li, Xiaodong;
Wang, Lianqu;
Wang, Jiajia

Publication type:

Article

Targeting N‐Methyl‐lysine Histone Demethylase KDM4 in Cancer: Natural Products Inhibitors as a Driving Force for Epigenetic Drug Discovery.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400682

By:

Cursaro, Ilaria;
Milioni, Leonardo;
Eslami, Kourosh;
Sirous, Hajar;
Carullo, Gabriele;
Gemma, Sandra;
Butini, Stefania;
Campiani, Giuseppe

Publication type:

Article

Characterization of Opioid Agonist Morphine Derivatives with Emphasis on Medicinal Chemistry.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400654

By:

Malik, Alaa;
Hosztafi, Sándor;
Vincze, Anna;
Marton, András;
Kraszni, Márta;
Balogh, György T.;
Noszál, Béla;
Mazák, Károly

Publication type:

Article

Synthesis and Evaluation of Fluorinated Piperazine‐Hydroxyethylamine Analogues as Potential Antiplasmodial Candidates.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400616

By:

Upadhyay, Charu;
Bhattacharya, Shreya;
Kumar, Sumit;
Vashisht, Kapil;
Zhang, Xujie;
Gagnon, Dominic;
Singh, Pooja;
Zhan, Peng;
Richard, Dave;
Rathi, Brijesh;
Prasad Singh, Agam;
Singh, Priyamvada

Publication type:

Article

Progress of Photoantibiotics in Overcoming Antibiotic Resistance.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400613

By:

Bhunia, Supriya;
Box, Sk Majid;
Bera, Satyajit;
Dolai, Anirban;
Samanta, Subhas

Publication type:

Article

Emerging Trends in Quinoxaline‐Based Analogs as Protein Kinase Inhibitors: Structural Developments and SAR Insights.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400592

By:

Shivani;
Mahajan, Amol T.;
Chaudhary, Sandeep

Publication type:

Article

Synthesis of 1,10‐Phenanthroline‐2,9‐bistriazoles: Evaluation as G‐Quadruplex Binders and Anti‐Tumor Activity.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400591

By:

Figueiredo, Joana;
Carreira‐Barral, Israel;
Lourenço, Pedro;
Miranda, André;
Lopes‐Nunes, Jéssica;
Quesada, Roberto;
Laranjo, Mafalda;
Mergny, Jean‐Louis;
Cruz, Carla

Publication type:

Article

Exploring C2 and N6 Substituent Effects on Truncated 4′‐Thioadenosine Derivatives as Dual A2A and A3 Adenosine Receptor Ligands.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400575

By:

Naik, Siddhi D.;
Kim, Minjae;
Choi, Jiyoung;
Kim, Gibae;
Woo Kim, Seung;
Aswar, Vikas R.;
Tripathi, Sushil K.;
Gaikwad, Vidyasagar;
Yu, Jinha;
Shin Jeong, Lak

Publication type:

Article

Bushy‐Tailed Multicationic Quaternary Phosphonium Compounds: Potent Amphiphilic Disinfectants with Promising Therapeutic Indices.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400546

By:

Rachii, Diana;
Bezold, Elise L.;
Wuest, William M.;
Minbiole, Kevin P. C.

Publication type:

Article

Development of Small Molecular Hyper‐activators of Human Caseinolytic Peptidase P (hClpP) with a [1,8]‐naphthyridinone Scaffold as Novel Anti‐cancer Agents.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400528

By:

Fu, Yuantao;
Yuan, Yinan;
Tan, Rongliang;
Jiang, Jinxin;
Li, Zhilong;
Li, Tong;
Xie, Guangjun;
Xiao, Yibei;
Sun, Haiying

Publication type:

Article

Design, Synthesis, and Anti‐Prostate Cancer Potential of 2‐(4‐Nitrobenzyl) Malonates In Vitro and DAL Acute Oral Toxicity Assessment In Vivo.

Published in:

ChemMedChem, 2025, v. 20, n. 4, p. 1, doi. 10.1002/cmdc.202400371

By:

Hassan Ganesh, Bharathi;
Aruchamy, Baladhandapani;
Mudradi, Srikrishna;
Mohanty, Sarthak;
Padinjarathil, Himabindu;
Carradori, Simone;
Ramani, Prasanna

Publication type:

Article

Works matching IS 18607179 AND DT 2025 AND VI 20 AND IP 4

Highlights from the Lowlands: Early Career Researchers Shine at Medicinal Chemistry Frontiers 2024.

Cover Feature: Design, Synthesis, and Anti‐Prostate Cancer Potential of 2‐(4‐Nitrobenzyl) Malonates In Vitro and DAL Acute Oral Toxicity Assessment In Vivo (ChemMedChem 4/2025).

Front Cover: [<sup>18</sup>F]NP3‐627, a Candidate PET Imaging Agent Targeting the NLRP3 Inflammasome in the Central Nervous System (ChemMedChem 4/2025).

Tumor Microenvironment‐Responsive Multinucleated Nanocomplexes Loaded with Carbon Dots for Combined Photothermal/Chemodynamic Therapy of Breast Cancer.

[<sup>18</sup>F]NP3‐627, a Candidate PET Imaging Agent Targeting the NLRP3 Inflammasome in the Central Nervous System.

Styrylchromones: Biological Activities and Structure‐Activity Relationship.

MuDRA‐Based Virtual Screening of Terpenes for Anti‐Leishmania Infantum Activity: In Vitro Validation and Mechanistic Insights from Molecular Docking.

Ac<sub>3</sub>4deoGlcNAz: A Selective Probe for Identifying O‐GlcNAc‐Modified Proteins in Prostate Cancer.

Targeting N‐Methyl‐lysine Histone Demethylase KDM4 in Cancer: Natural Products Inhibitors as a Driving Force for Epigenetic Drug Discovery.

Characterization of Opioid Agonist Morphine Derivatives with Emphasis on Medicinal Chemistry.

Synthesis and Evaluation of Fluorinated Piperazine‐Hydroxyethylamine Analogues as Potential Antiplasmodial Candidates.

Progress of Photoantibiotics in Overcoming Antibiotic Resistance.

Emerging Trends in Quinoxaline‐Based Analogs as Protein Kinase Inhibitors: Structural Developments and SAR Insights.

Synthesis of 1,10‐Phenanthroline‐2,9‐bistriazoles: Evaluation as G‐Quadruplex Binders and Anti‐Tumor Activity.

Exploring C2 and N<sup>6</sup> Substituent Effects on Truncated 4′‐Thioadenosine Derivatives as Dual A<sub>2A</sub> and A<sub>3</sub> Adenosine Receptor Ligands.

Bushy‐Tailed Multicationic Quaternary Phosphonium Compounds: Potent Amphiphilic Disinfectants with Promising Therapeutic Indices.

Development of Small Molecular Hyper‐activators of Human Caseinolytic Peptidase P (hClpP) with a [1,8]‐naphthyridinone Scaffold as Novel Anti‐cancer Agents.

Design, Synthesis, and Anti‐Prostate Cancer Potential of 2‐(4‐Nitrobenzyl) Malonates In Vitro and DAL Acute Oral Toxicity Assessment In Vivo.