Works matching IS 18607179 AND DT 2024 AND VI 19 AND IP 24

Results: 27

Leveraging Natural Product‐Inspired Antifungals to Investigate the Mechanism of Action of Peniciaculin A.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400500
By:
- Wilt, Ingrid K.;
- Demeritte, Adrian R.;
- Kim, Alexander T.;
- Wang, Weiwei;
- Wuest, William M.
Publication type:
Article
Cover Feature: Phosphate‐Containing Glycolipids: A Review on Synthesis and Bioactivity (ChemMedChem 24/2024).
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202482402
By:
- Pinheiro, Luís;
- Freitas, Marisa;
- Branco, Paula S.
Publication type:
Article
Front Cover: Cholinesterase Inhibitory Activity and Molecular Docking Studies of Isocryptolepine‐Triazole Adducts (ChemMedChem 24/2024).
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202482401
By:
- Tummatorn, Jumreang;
- Meewan, Ittipat;
- Khunnawutmanotham, Nisachon;
- Chimnoi, Nitirat;
- Suwanwong, Nutchapong;
- Rodphon, Warabhorn;
- Thongsornkleeb, Charnsak;
- Yang, Jingyue;
- Ruchirawat, Somsak
Publication type:
Article
Medicinal Chemistry in Bosnia and Herzegovina ‐ Past, Present and Perspectives**.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400669
By:
- Kondža, Martin
Publication type:
Article
Structural Basis for Inhibition of the SARS‐CoV‐2 nsp16 by Substrate‐Based Dual Site Inhibitors.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400618
By:
- Kalnins, Gints;
- Rudusa, Laura;
- Bula, Anna L.;
- Zelencova‐Gopejenko, Diana;
- Bobileva, Olga;
- Sisovs, Mihails;
- Tars, Kaspars;
- Jirgensons, Aigars;
- Jaudzems, Kristaps;
- Bobrovs, Raitis
Publication type:
Article
Two‐Step Synthesis of Enantiomerically Pure Morphans from (R)‐Carvone.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400596
By:
- Costanzo, Giuliana;
- Cosentino, Giuseppe;
- Pasquinucci, Lorella;
- Amata, Emanuele;
- Schepmann, Dirk;
- Wünsch, Bernhard
Publication type:
Article
Lactam Truncation Yields a Dihydroquinazolinone Scaffold with Potent Antimalarial Activity that Targets PfATP4.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400549
By:
- Ashton, Trent D.;
- Calic, Petar P. S.;
- Dans, Madeline G.;
- Kang Ooi, Zi;
- Zhou, Qingmiao;
- Loi, Katie;
- Jarman, Kate E.;
- Palandri, Josephine;
- Qiu, Deyun;
- Lehane, Adele M.;
- Maity, Bikash;
- De, Nirupam;
- Famodimu, Mufuliat T.;
- Delves, Michael J.;
- Mao, Emma Y.;
- Gancheva, Maria R.;
- Wilson, Danny W.;
- Chowdury, Mrittika;
- de Koning‐Ward, Tania F.;
- Baud, Delphine
Publication type:
Article
Serum Circulating mRNA Panel for the Early Detection of Gastric Cancer: A Potential Biomarker Test.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400523
By:
- Peng, Xinyu;
- Teng, Xiaoyan;
- Ma, Qian;
- Han, Da
Publication type:
Article
Crystallographic and Selectivity Studies on the Approved HIF Prolyl Hydroxylase Inhibitors Desidustat and Enarodustat.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400504
By:
- Corner, Thomas P.;
- Salah, Eidarus;
- Tumber, Anthony;
- Kaur, Samanpreet;
- Nakashima, Yu;
- Allen, Mark D.;
- Schnaubelt, Lara I.;
- Fiorini, Giorgia;
- Brewitz, Lennart;
- Schofield, Christopher J.
Publication type:
Article
Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400601
By:
- Kilbile, Jaydeo T.;
- Sapkal, Suryakant B.;
- Renzi, Gioele;
- D'Agostino, Ilaria;
- Boudjelal, Mohamed;
- Tamboli, Yasinalli;
- Cutarella, Luigi;
- Mori, Mattia;
- Sgambellone, Silvia;
- Villano, Serafina;
- Marri, Silvia;
- Lucarini, Laura;
- Carradori, Simone;
- Carta, Fabrizio;
- Supuran, Claudiu T.
Publication type:
Article
In Vitro and In Vivo Biological Evaluation of Novel 1,4‐Naphthoquinone Derivatives as Potential Anticancer Agents.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400495
By:
- Ravichandiran, Palanisamy;
- Martyna, Aleksandra;
- Kochanowicz, Elżbieta;
- Maroli, Nikhil;
- Kubiński, Konrad;
- Masłyk, Maciej;
- Boguszewska‐Czubara, Anna;
- Ramesh, Thiyagarajan
Publication type:
Article
Discovery of Palindrome Dual PPARγ‐GPR40 Agonists for Treating Type 2 Diabetes.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400492
By:
- Rodríguez‐Luévano, Ana;
- Almanza‐Pérez, Julio C.;
- Ortiz‐Andrade, Rolffy;
- Lara‐González, Samuel;
- Santillán, Rosa;
- Navarrete‐Vázquez, Gabriel;
- Giacoman‐Martínez, Abraham;
- Lazzarini‐Lechuga, Roberto C.;
- Bautista, Elihú;
- Hidalgo‐Figueroa, Sergio
Publication type:
Article
Tumor‐Associated Carbohydrate Antigen 19–9 (CA 19–9), a Promising Target for Antibody‐Based Detection, Diagnosis, and Immunotherapy of Cancer.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400491
By:
- Nakisa, Athar;
- Sempere, Lorenzo F.;
- Chen, Xi;
- Qu, Linda T.;
- Woldring, Daniel;
- Crawford, Howard C.;
- Huang, Xuefei
Publication type:
Article
Phenotypic‐Based Discovery and Exploration of a Resorufin Scaffold with Activity against Mycobacterium tuberculosis.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400482
By:
- Tran, Eric;
- Cheung, Chen‐Yi;
- Li, Lucy;
- Carter, Glen P.;
- Gable, Robert W.;
- West, Nicholas P.;
- Kaur, Amandeep;
- Gee, Yi Sing;
- Cook, Gregory M.;
- Baell, Jonathan B.;
- Jörg, Manuela
Publication type:
Article
Bacterial Secondary Metabolites Embedded in Producer Cell Membranes and Antibiotics Targeting Their Biosynthesis.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400469
By:
- Xia, Zhao;
- Xiang, Hao;
- Shi, Yi‐Ming
Publication type:
Article
Discovery of KW0113 as a First and Effective PROTAC Degrader of DNMT1 Protein.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400467
By:
- Wang, Huihui;
- Wang, Zhaoliang;
- Hu, Linghao;
- Yang, Bingjie;
- Zong, Liangyi;
- Xu, Dounan;
- Yu, Bo;
- Kong, Xiangqian;
- Wang, Mingliang
Publication type:
Article
Fluorescence‐Based HTS Assays for Ion Channel Modulation in Drug Discovery Pipelines.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400383
By:
- Voldřich, Jan;
- Matoušová, Marika;
- Šmídková, Markéta;
- Mertlíková‐Kaiserová, Helena
Publication type:
Article
Two Step One‐Pot Synthesis of 7‐Azaindole Linked 1,2,3‐Triazole Hybrids: In‐Vitro and In‐Silico Antimicrobial Evaluation.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400451
By:
- Sharma, Kanika;
- Lal, Bajrang;
- Kumar Tittal, Ram;
- Lal, Kashmiri;
- Vats, Lalit;
- Vikas D, Ghule
Publication type:
Article
How to Find a Fragment: Methods for Screening and Validation in Fragment‐Based Drug Discovery.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400342
By:
- Kirkman, Tim;
- dos Santos Silva, Catharina;
- Tosin, Manuela;
- Bertacine Dias, Marcio Vinicius
Publication type:
Article
Evaluation of a Radioiodinated G‐Quadruplex Binder in Cervical Cancer Models.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400438
By:
- Cristina Oliveira, Maria;
- Campello, Maria Paula Cabral;
- Gano, Lurdes;
- Raposinho, Paula;
- Belchior, Ana;
- Mendes, Edgar;
- Silva, Catarina D.;
- Lopes‐Nunes, Jéssica;
- Cruz, Carla;
- Paulo, António
Publication type:
Article
The Investigation of Hsp90C‐Terminal Inhibitors Containing Amide Bioisosteres.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400418
By:
- Amatya, Eva;
- Subramanian, Chitra;
- Long, Reagan;
- McNamara, Kelli;
- Cohen, Mark S.;
- Blagg, Brian S. J.
Publication type:
Article
Substrate‐Based Ligand Design for Phenazine Biosynthesis Enzyme PhzF.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400466
By:
- Baumgarten, Janosch;
- Schneider, Philipp;
- Thiemann, Marie;
- Zimmermann, Moritz;
- Diederich, Christina;
- Blankenfeldt, Wulf;
- Kunick, Conrad
Publication type:
Article
Cyclodextrin Dimers Functionalized with Biotin as Nanocapsules for Active Doxorubicin Delivery Against MCF‐7 Breast Cell Line.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400368
By:
- Bognanni, Noemi;
- Scuderi, Chiara;
- Giglio, Valentina;
- Spiteri, Fabio;
- La Piana, Luana;
- Condorelli, Daniele;
- Barresi, Vincenza;
- Vecchio, Graziella
Publication type:
Article
Cholinesterase Inhibitory Activity and Molecular Docking Studies of Isocryptolepine‐Triazole Adducts.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400447
By:
- Tummatorn, Jumreang;
- Meewan, Ittipat;
- Khunnawutmanotham, Nisachon;
- Chimnoi, Nitirat;
- Suwanwong, Nutchapong;
- Rodphon, Warabhorn;
- Thongsornkleeb, Charnsak;
- Yang, Jingyue;
- Ruchirawat, Somsak
Publication type:
Article
Phosphate‐Containing Glycolipids: A Review on Synthesis and Bioactivity.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400315
By:
- Pinheiro, Luís;
- Freitas, Marisa;
- Branco, Paula S.
Publication type:
Article
Development of Integrin Targeting Chimeras (ITACs) for the Lysosomal Degradation of Extracellular Proteins.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202300643
By:
- Zhou, Yaxian;
- Liao, Yaxian;
- Zhao, Yuan;
- Tang, Weiping
Publication type:
Article
Flavonol‐Ruthenium Complexes as Antioxidant and Anticancer Agents.
Published in:
ChemMedChem, 2024, v. 19, n. 24, p. 1, doi. 10.1002/cmdc.202400313
By:
- Wu, Ting‐Wei;
- Chu, Yi‐Cheng;
- Chang, Chuan‐Hsin;
- Hsieh, Yu‐Hui;
- Tang, Mei‐Hsin;
- Hsu, Pei‐Hsuan;
- Wu, Hsin‐Ying;
- Chen, Jih‐Jung;
- Shih, Tzenge‐Lien
Publication type:
Article