Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 4

Results: 15

Front Cover: A Single Second Shell Amino Acid Determines Affinity and Kinetics of Linagliptin Binding to Type 4 Dipeptidyl Peptidase and Fibroblast Activation Protein (ChemMedChem 4/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 599, doi. 10.1002/cmdc.202100054

By:

Schnapp, Gisela;
Hoevels, Yvette;
Bakker, Remko A.;
Schreiner, Patrick;
Klein, Thomas;
Nar, Herbert

Publication type:

Article

Corrigendum: Kiss1R Identification and Biodistribution Analysis Employing a Western Ligand Blot and Ligand‐Derivative Stain with a FITC‐Kisspeptin Derivative.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 725, doi. 10.1002/cmdc.202000990

By:

Hasegawa, Koki;
Maedomari, Rika;
Sato, Younosuke;
Gotoh, Kumiko;
Kudoh, Shinji;
Kojima, Akihiro;
Okada, Seiji;
Ito, Takaaki

Publication type:

Article

Targeting the CRD F‐face of Human Galectin‐3 and Allosterically Modulating Glycan Binding by Angiostatic PTX008 and a Structurally Optimized Derivative.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 713, doi. 10.1002/cmdc.202000742

By:

Miller, Michelle C.;
Zheng, Yi;
Suylen, Dennis;
Ippel, Hans;
Cañada, F. Javier;
Berbís, M. Alvaro;
Jiménez‐Barbero, Jesús;
Tai, Guihua;
Gabius, Hans‐Joachim;
Mayo, Kevin H.

Publication type:

Article

Development of the First Potential Nonpeptidic Positron Emission Tomography Tracer for the Imaging of CCR2 Receptors.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 640, doi. 10.1002/cmdc.202000728

By:

Wagner, Stefan;
Moura Gatti, Fernando;
Silva, Daniel G.;
Ortiz Zacarias, Natalia V.;
Zweemer, Annelien J. M.;
Hermann, Sven;
De Maria, Monica;
Koch, Michael;
Weiss, Christina;
Schepmann, Dirk;
Heitman, Laura H.;
Tschammer, Nuska;
Kopka, Klaus;
Junker, Anna

Publication type:

Article

Withdrawal: K.T. Wanner et al. "MS‐based screening of small amino acid derived oxime libraries for hGAT3 inhibitors".

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 724, doi. 10.1002/cmdc.202000720

By:

Andreß, Janina C.;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

Highly Phototoxic Transplatin‐Modified Distyryl‐BODIPY Photosensitizers for Photodynamic Therapy.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 694, doi. 10.1002/cmdc.202000702

By:

Padrutt, Roxane;
Babu, Vipin;
Klingler, Simon;
Kalt, Martina;
Schumer, Frank;
Anania, Maria I.;
Schneider, Lukas;
Spingler, Bernhard

Publication type:

Article

Evaluation of the Toxicity of Two Electron‐Deficient Half‐Sandwich Complexes against Human Lymphocytes from Healthy Individuals.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 624, doi. 10.1002/cmdc.202000672

By:

Habas, Khaled;
Soldevila‐Barreda, Joan J.;
Azmanova, Maria;
Rafols, Laia;
Pitto‐Barry, Anaïs;
Anderson, Diana;
Barry, Nicolas P. E.

Publication type:

Article

Novel Phenylmethylenecyclohexenone Derivatives as Potent TrxR Inhibitors Display High Antiproliferative Activity and Induce ROS, Apoptosis, and DNA Damage.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 702, doi. 10.1002/cmdc.202000660

By:

Wang, Xiaomei;
Qian, Jianqiang;
Zhu, Peng;
Hua, Rong;
Liu, Ji;
Hang, Jiaying;
Meng, Chi;
Shan, Wenpei;
Miao, Jiefei;
Ling, Yong

Publication type:

Article

Recent Advances in the Discovery of Multitargeted Tyrosine Kinase Inhibitors as Anticancer Agents.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 600, doi. 10.1002/cmdc.202000658

By:

Guo, Ting;
Ma, Shutao

Publication type:

Article

A Novel Hybrid of Chloroquine and Primaquine Linked by Gold(I): Multitarget and Multiphase Antiplasmodial Agent.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 662, doi. 10.1002/cmdc.202000653

By:

Souza Pereira, Caroline;
Costa Quadros, Helenita;
Magalhaes Moreira, Diogo Rodrigo;
Castro, William;
Santos De Deus Da Silva, Romulo Ivisson;
Botelho Pereira Soares, Milena;
Fontinha, Diana;
Prudêncio, Miguel;
Schmitz, Vinicius;
Dos Santos, Hélio F.;
Gendrot, Mathieu;
Fonta, Isabelle;
Mosnier, Joel;
Pradines, Bruno;
Navarro, Maribel

Publication type:

Article

Puzzling Out the Colchicine Biosynthetic Pathway.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 621, doi. 10.1002/cmdc.202000633

By:

Stander, Emily A.;
Papon, Nicolas;
Courdavault, Vincent

Publication type:

Article

Benzimidazole and Benzoxazole Zinc Chelators as Inhibitors of Metallo‐β‐Lactamase NDM‐1.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 654, doi. 10.1002/cmdc.202000607

By:

Jackson, Abigail C.;
Pinter, Tyler B. J.;
Talley, Daniel C.;
Baker‐Agha, Adnan;
Patel, Dhruvil;
Smith, Paul J.;
Franz, Katherine J.

Publication type:

Article

A Single Second Shell Amino Acid Determines Affinity and Kinetics of Linagliptin Binding to Type 4 Dipeptidyl Peptidase and Fibroblast Activation Protein.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 630, doi. 10.1002/cmdc.202000591

By:

Schnapp, Gisela;
Hoevels, Yvette;
Bakker, Remko A.;
Schreiner, Patrick;
Klein, Thomas;
Nar, Herbert

Publication type:

Article

Red Emissive Carbon Dots Prepared from Polymers as an Efficient Nanocarrier for Coptisine Delivery in vivo and in vitro.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 646, doi. 10.1002/cmdc.202000420

By:

Ren, Wei;
Nan, Fuchun;
Li, Shumu;
Yang, Sijin;
Ge, Jiechao;
Zhao, Zhenwen

Publication type:

Article

Structure‐Activity Studies of Truncated Latrunculin Analogues with Antimalarial Activity.

Published in:

ChemMedChem, 2021, v. 16, n. 4, p. 679, doi. 10.1002/cmdc.202000399

By:

Varghese, Swapna;
Rahmani, Raphaël;
Drew, Damien R.;
Beeson, James G.;
Baum, Jake;
Smith, Brian J.;
Baell, Jonathan B.

Publication type:

Article