Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 21

Results: 13

Front Cover: Synthesis of L‐[5‐11C]Leucine and L‐α‐[5‐11C]Methylleucine via Pd0‐mediated 11C‐Methylation and Microfluidic Hydrogenation: Potentiality of Leucine PET Probes for Tumor Imaging (ChemMedChem 21/2021)

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3236, doi. 10.1002/cmdc.202100672

By:

Takatani, Shuhei;
Tahara, Tsuyoshi;
Tsuji, Mieko;
Ozaki, Daiki;
Shibata, Nina;
Hashizume, Yoshinobu;
Suzuki, Masaaki;
Onoe, Hirotaka;
Watanabe, Yasuyoshi;
Doi, Hisashi

Publication type:

Article

A Patent Review on the Current Developments of Benzoxazoles in Drug Discovery.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3237, doi. 10.1002/cmdc.202100370

By:

Wong, Xi Khai;
Yeong, Keng Yoon

Publication type:

Article

Synthesis, Biological Evaluation, and Computational Analysis of Biaryl Side‐Chain Analogs of Solithromycin.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3368, doi. 10.1002/cmdc.202100435

By:

Daher, Samer S.;
Lee, Miseon;
Jin, Xiao;
Teijaro, Christiana N.;
Wheeler, Steven E.;
Jacobson, Marlene A.;
Buttaro, Bettina;
Andrade, Rodrigo B.

Publication type:

Article

Inhibitors of Human Divalent Metal Transporters DMT1 (SLC11A2) and ZIP8 (SLC39A8) from a GDB‐17 Fragment Library.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3306, doi. 10.1002/cmdc.202100467

By:

Pujol‐Giménez, Jonai;
Poirier, Marion;
Bühlmann, Sven;
Schuppisser, Céline;
Bhardwaj, Rajesh;
Awale, Mahendra;
Visini, Ricardo;
Javor, Sacha;
Hediger, Matthias A.;
Reymond, Jean‐Louis

Publication type:

Article

25CN‐NBOH: A Selective Agonist for in vitro and in vivo Investigations of the Serotonin 2A Receptor.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3263, doi. 10.1002/cmdc.202100395

By:

Märcher Rørsted, Emil;
Jensen, Anders A.;
Kristensen, Jesper L.

Publication type:

Article

Exploration of Pyrazolo[1,5‐a]pyrimidines as Membrane‐Bound Pyrophosphatase Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3360, doi. 10.1002/cmdc.202100392

By:

Johansson, Niklas G.;
Dreano, Loïc;
Vidilaseris, Keni;
Khattab, Ayman;
Liu, Jianing;
Lasbleiz, Arthur;
Ribeiro, Orquidea;
Kiriazis, Alexandros;
Boije af Gennäs, Gustav;
Meri, Seppo;
Goldman, Adrian;
Yli‐Kauhaluoma, Jari;
Xhaard, Henri

Publication type:

Article

Rational Design of Potent Inhibitors of a Metallohydrolase Using a Fragment‐Based Approach.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3342, doi. 10.1002/cmdc.202100486

By:

Feder, Daniel;
Mohd‐Pahmi, Siti H.;
Hussein, Waleed M.;
Guddat, Luke W.;
McGeary, Ross P.;
Schenk, Gerhard

Publication type:

Article

Structure‐Activity Relationship Explorations and Discovery of a Potent Antagonist for the Free Fatty Acid Receptor 2.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3326, doi. 10.1002/cmdc.202100356

By:

Højgaard Hansen, Anders;
Christensen, Henriette B.;
Pandey, Sunil K.;
Sergeev, Eugenia;
Valentini, Alice;
Dunlop, Julia;
Dedeo, Domonkos;
Fratta, Simone;
Hudson, Brian D.;
Milligan, Graeme;
Ulven, Trond;
Rexen Ulven, Elisabeth

Publication type:

Article

Stimulation of Ca2+‐ATPase Transport Activity by a Small‐Molecule Drug.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3293, doi. 10.1002/cmdc.202100350

By:

Sordi, Giacomo;
Goti, Andrea;
Young, Howard S.;
Palchetti, Ilaria;
Tadini‐Buoninsegni, Francesco

Publication type:

Article

Investigation of the Effects and Mechanisms of Anticancer Action of a Ru(II)‐Arene Iminophosphorane Compound in Triple Negative Breast Cancer Cells.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3280, doi. 10.1002/cmdc.202100325

By:

Nayeem, Nazia;
Yeasmin, Arefa;
Cobos, Samantha N.;
Younes, Ali;
Hubbard, Karen;
Contel, Maria

Publication type:

Article

Homarine Alkyl Ester Derivatives as Promising Acetylcholinesterase Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3315, doi. 10.1002/cmdc.202100265

By:

João, Karen G.;
Videira, Romeu A.;
Paiva‐Martins, Fátima;
Valentão, Patrícia;
Pereira, David M.;
Andrade, Paula B.

Publication type:

Article

Synthesis of L‐[5‐11C]Leucine and L‐α‐[5‐11C]Methylleucine via Pd0‐mediated 11C‐Methylation and Microfluidic Hydrogenation: Potentiality of Leucine PET Probes for Tumor Imaging

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3271, doi. 10.1002/cmdc.202100255

By:

Takatani, Shuhei;
Tahara, Tsuyoshi;
Tsuji, Mieko;
Ozaki, Daiki;
Shibata, Nina;
Hashizume, Yoshinobu;
Suzuki, Masaaki;
Onoe, Hirotaka;
Watanabe, Yasuyoshi;
Doi, Hisashi

Publication type:

Article

Chalcone‐Supported Cardiac Mesoderm Induction in Human Pluripotent Stem Cells for Heart Muscle Engineering.

Published in:

ChemMedChem, 2021, v. 16, n. 21, p. 3300, doi. 10.1002/cmdc.202100222

By:

Raad, Farah S.;
Khan, Taukeer A.;
Esser, Tilman U.;
Hudson, James E.;
Seth, Bhakti Irene;
Fujita, Buntaro;
Gandamala, Ravi;
Tietze, Lutz F.;
Zimmermann, Wolfram

Publication type:

Article

Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 21

Front Cover: Synthesis of L‐[5‐<sup>11</sup>C]Leucine and L‐α‐[5‐<sup>11</sup>C]Methylleucine via Pd<sup>0</sup>‐mediated <sup>11</sup>C‐Methylation and Microfluidic Hydrogenation: Potentiality of Leucine PET Probes for Tumor Imaging (ChemMedChem 21/2021)

A Patent Review on the Current Developments of Benzoxazoles in Drug Discovery.

Synthesis, Biological Evaluation, and Computational Analysis of Biaryl Side‐Chain Analogs of Solithromycin.

Inhibitors of Human Divalent Metal Transporters DMT1 (SLC11A2) and ZIP8 (SLC39A8) from a GDB‐17 Fragment Library.

25CN‐NBOH: A Selective Agonist for in vitro and in vivo Investigations of the Serotonin 2A Receptor.

Exploration of Pyrazolo[1,5‐a]pyrimidines as Membrane‐Bound Pyrophosphatase Inhibitors.

Rational Design of Potent Inhibitors of a Metallohydrolase Using a Fragment‐Based Approach.

Structure‐Activity Relationship Explorations and Discovery of a Potent Antagonist for the Free Fatty Acid Receptor 2.

Stimulation of Ca<sup>2+</sup>‐ATPase Transport Activity by a Small‐Molecule Drug.

Investigation of the Effects and Mechanisms of Anticancer Action of a Ru(II)‐Arene Iminophosphorane Compound in Triple Negative Breast Cancer Cells.

Homarine Alkyl Ester Derivatives as Promising Acetylcholinesterase Inhibitors.

Synthesis of L‐[5‐<sup>11</sup>C]Leucine and L‐α‐[5‐<sup>11</sup>C]Methylleucine via Pd<sup>0</sup>‐mediated <sup>11</sup>C‐Methylation and Microfluidic Hydrogenation: Potentiality of Leucine PET Probes for Tumor Imaging

Chalcone‐Supported Cardiac Mesoderm Induction in Human Pluripotent Stem Cells for Heart Muscle Engineering.