Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 2

Results: 16

Cover Feature: Peptide‐Mimicking Poly(2‐oxazoline)s Displaying Potent Antimicrobial Properties (2/2021)

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 302, doi. 10.1002/cmdc.202000989

By:

Zhou, Min;
Jiang, Weinan;
Xie, Jiayang;
Zhang, Wenjing;
Ji, Zhemin;
Zou, Jingcheng;
Cong, Zihao;
Xiao, Ximian;
Gu, Jiawei;
Liu, Runhui

Publication type:

Article

Front Cover: Structure‐Activity Relationships of Benzamides and Isoindolines Designed as SARS‐CoV Protease Inhibitors Effective against SARS‐CoV‐2 (2/2021)

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 301, doi. 10.1002/cmdc.202000987

By:

Welker, Armin;
Kersten, Christian;
Müller, Christin;
Madhugiri, Ramakanth;
Zimmer, Collin;
Müller, Patrick;
Zimmermann, Robert;
Hammerschmidt, Stefan;
Maus, Hannah;
Ziebuhr, John;
Sotriffer, Christoph;
Schirmeister, Tanja

Publication type:

Article

The Effects of the Alkaloid Tambjamine J on Mice Implanted with Sarcoma 180 Tumor Cells.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 420, doi. 10.1002/cmdc.202000387

By:

A. Barros-Nepomuceno, Francisco Washington;
de Araújo Viana, Daniel;
Pascoalino Pinheiro, Daniel;
Evangelista de Oliveira, Fátima de Cássia;
Magalhães Ferreira, Jamile;
de Queiroz, Maria Goretti R.;
Xinghua Ma;
Coêlho Cavalcanti, Bruno;
Pessoa, Claudia;
Banwell, Martin G.

Publication type:

Article

Evaluation of a Platinum-Acridine Anticancer Agent and Its Liposomal Formulation in an in vivo Model of Lung Adenocarcinoma.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 412, doi. 10.1002/cmdc.202000637

By:

Song Ding;
Hackett, Christopher L.;
Fang Liu;
Hackett, Ryan G.;
Bierbach, Ulrich

Publication type:

Article

BODIPY-Based Photosensitizers as Potential Anticancer and Antibacterial Agents: Role of the Positive Charge and the Heavy Atom Effect.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 399, doi. 10.1002/cmdc.202000529

By:

Piskorz, Jaroslaw;
Porolnik, Weronika;
Kucinska, Malgorzata;
Dlugaszewska, Jolanta;
Murias, Marek;
Mielcarek, Jadwiga

Publication type:

Article

Synthesis and Structure-Activity Relationships of 3-Arylisoquinolone Analogues as Highly Specific hCES2A Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 388, doi. 10.1002/cmdc.202000581

By:

Yitian Zhao;
Yuan Xiong;
Sanfeng Dong;
Xiaoqing Guan;
Yunqing Song;
Yanqing Yang;
Kun Zou;
Zhao Li;
Yong Zhang;
Shengquan Fang;
Bo Li;
Weiliang Zhu;
Kaixian Chen;
Qi Jia;
Guangbo Ge

Publication type:

Article

Small-Molecule Inhibition of the uPAR·uPA Interaction by Conformational Selection.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 377, doi. 10.1002/cmdc.202000558

By:

Xu, David;
Bum-Erdene, Khuchtumur;
Leth, Julie M.;
Ghozayel, Mona K.;
Ploug, Michael;
Meroueh, Samy O.

Publication type:

Article

Gramicidin-S-Inspired Cyclopeptidomimetics as Potent Membrane-Active Bactericidal Agents with Therapeutic Potential.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 368, doi. 10.1002/cmdc.202000568

By:

Chengfei Hu;
Quan Wen;
Shuhui Huang;
Saisai Xie;
Yuanying Fang;
Yi Jin;
Campagne, Rémy;
Alezra, Valérie;
Miclet, Emeric;
Jinhua Zhu;
Yang Wan

Publication type:

Article

Effect of Secondary Structure and Side Chain Length of Hydrophobic Amino Acid Residues on the Antimicrobial Activity and Toxicity of 14-Residue-Long de novo AMPs.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 355, doi. 10.1002/cmdc.202000550

By:

Pandit, Gopal;
Chowdhury, Nabarupa;
Mohid, Sk. Abdul;
Bidkar, Anil P.;
Bhunia, Anirban;
Chatterjee, Sunanda

Publication type:

Article

Structure-Activity Relationships of Benzamides and Isoindolines Designed as SARS-CoV Protease Inhibitors Effective against SARS-CoV-2.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 340, doi. 10.1002/cmdc.202000548

By:

Welker, Armin;
Kersten, Christian;
Müller, Christin;
Madhugiri, Ramakanth;
Zimmer, Collin;
Müller, Patrick;
Zimmermann, Robert;
Hammerschmidt, Stefan;
Maus, Hannah;
Ziebuhr, John;
Sotriffer, Christoph;
Schirmeister, Tanja

Publication type:

Article

An Advanced Apralog with Increased in vitro and in vivo Activity toward Gram-negative Pathogens and Reduced ex vivo Cochleotoxicity.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 335, doi. 10.1002/cmdc.202000726

By:

Sonousi, Amr;
Quirke, Jonathan C. K.;
Waduge, Prabuddha;
Janusic, Tanja;
Gysin, Marina;
Haldimann, Klara;
Shan Xu;
Hobbie, Sven N.;
Su-Hua Sha;
Schacht, Jochen;
Chow, Christine S.;
Vasella, Andrea;
Böttger, Erik C.;
Crich, David

Publication type:

Article

Design and Synthesis of Fused Pyridine Building Blocks for Automated Library Generation.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 328, doi. 10.1002/cmdc.202000852

By:

Mora-Radó, Helena;
Czechtizky, Werngard;
Méndez, María;
Harrity, Joseph P. A.

Publication type:

Article

Further SAR on the (Phenylsulfonyl)piperazine Scaffold as Inhibitors of the Aedes aegypti Kir1 (AeKir) Channel and Larvicides.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 319, doi. 10.1002/cmdc.202000598

By:

Aretz, Christopher D.;
Kharade, Sujay V.;
Chronister, Keagan;
Trigueros, Renata Rusconi;
Rodriguez, Erick J. Martinez;
Piermarini, Peter M.;
Denton, Jerod S.;
Hopkins, Corey R.

Publication type:

Article

PROTAC Compatibilities, Degrading Cell-Surface Receptors, and the Sticky Problem of Finding a Molecular Glue.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 316, doi. 10.1002/cmdc.202000683

By:

Conghe Tian;
Burgess, Kevin

Publication type:

Article

Peptide-Mimicking Poly(2-oxazoline)s Displaying Potent Antimicrobial Properties.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 309, doi. 10.1002/cmdc.202000530

By:

Min Zhou;
Weinan Jiang;
Jiayang Xie;
Wenjing Zhang;
Zhemin Ji;
Jingcheng Zou;
Zihao Cong;
Ximian Xiao;
Jiawei Gu;
Runhui Liu

Publication type:

Article

2020 Italian Special Anniversary Collection: Celebrating NMMC 2019 and 40 Years of the DCF-SCI.

Published in:

ChemMedChem, 2021, v. 16, n. 2, p. 303, doi. 10.1002/cmdc.202000926

By:

Carini, Marina;
De Amici, Marco

Publication type:

Article