Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 19

Results: 18

Front Cover: Dinitrophenol‐Hyaluronan Conjugates as Multivalent Antibody‐Recruiting Glycopolymers for Targeted Cancer Immunotherapy (ChemMedChem 19/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2907, doi. 10.1002/cmdc.202100607

By:

Lin, Han;
Zhou, Kun;
Li, Dan;
Hong, Haofei;
Xie, Yuntian;
Gong, Liang;
Shen, Yu;
Zhou, Zhifang;
Shi, Jie;
Wu, Zhimeng

Publication type:

Article

Cover Feature: Recent Advances in Radiometals for Combined Imaging and Therapy in Cancer (ChemMedChem 19/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2908, doi. 10.1002/cmdc.202100609

By:

Herrero Álvarez, Natalia;
Bauer, David;
Hernández‐Gil, Javier;
Lewis, Jason S.

Publication type:

Article

Development of LM98, a Small‐Molecule TEAD Inhibitor Derived from Flufenamic Acid.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2982, doi. 10.1002/cmdc.202100432

By:

Mélin, Léa;
Abdullayev, Shuay;
Fnaiche, Ahmed;
Vu, Victoria;
González Suárez, Narjara;
Zeng, Hong;
Szewczyk, Magdalena M.;
Li, Fengling;
Senisterra, Guillermo;
Allali‐Hassani, Abdellah;
Chau, Irene;
Dong, Aiping;
Woo, Simon;
Annabi, Borhane;
Halabelian, Levon;
LaPlante, Steven R.;
Vedadi, Masoud;
Barsyte‐Lovejoy, Dalia;
Santhakumar, Vijayaratnam;
Gagnon, Alexandre

Publication type:

Article

Screening for New Inhibitors of Glycine Transporter 1 and 2 by Means of MS Binding Assays.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3094, doi. 10.1002/cmdc.202100408

By:

Ackermann, Thomas M.;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

N‐(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3071, doi. 10.1002/cmdc.202100405

By:

Ferlenghi, Francesca;
Mari, Michele;
Gobbi, Gabriella;
Elisi, Gian Marco;
Mor, Marco;
Rivara, Silvia;
Vacondio, Federica;
Bartolucci, Silvia;
Bedini, Annalida;
Fanini, Fabiola;
Spadoni, Gilberto

Publication type:

Article

Evaluation of 4‐(4‐Fluorobenzyl)piperazin‐1‐yl]‐Based Compounds as Competitive Tyrosinase Inhibitors Endowed with Antimelanogenic Effects.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3083, doi. 10.1002/cmdc.202100396

By:

Mirabile, Salvatore;
Vittorio, Serena;
Paola Germanò, Maria;
Adornato, Ilenia;
Ielo, Laura;
Rapisarda, Antonio;
Gitto, Rosaria;
Pintus, Francesca;
Fais, Antonella;
De Luca, Laura

Publication type:

Article

LYTACs: An Emerging Tool for the Degradation of Non‐Cytosolic Proteins.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2951, doi. 10.1002/cmdc.202100393

By:

Ramadas, Bhavana;
Kumar Pain, Pritam;
Manna, Debasish

Publication type:

Article

An Organogold Compound as Potential Antimicrobial Agent against Drug‐Resistant Bacteria: Initial Mechanistic Insights.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3060, doi. 10.1002/cmdc.202100342

By:

Chakraborty, Parichita;
Oosterhuis, Dorenda;
Bonsignore, Riccardo;
Casini, Angela;
Olinga, Peter;
Scheffers, Dirk‐Jan

Publication type:

Article

Design, Synthesis, and in vitro Evaluation of Tubulin‐Targeting Dibenzothiazines with Antiproliferative Activity as a Novel Heterocycle Building Block.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3003, doi. 10.1002/cmdc.202100383

By:

Guerra, Walter D.;
Lucena‐Agell, Daniel;
Hortigüela, Rafael;
Rossi, Roberto A.;
Fernando Díaz, J.;
Padrón, José M.;
Barolo, Silvia M.

Publication type:

Article

A Diarylpentanoid with Potential Activation of the p53 Pathway: Combination of in silico Screening Studies, Synthesis, and Biological Activity Evaluation.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2969, doi. 10.1002/cmdc.202100337

By:

Moreira, Joana;
Almeida, Joana;
Loureiro, Joana B.;
Ramos, Helena;
Palmeira, Andreia;
Pinto, Madalena M.;
Saraiva, Lucília;
Cidade, Honorina

Publication type:

Article

Autophagy‐Dependent Ferroptosis as a Therapeutic Target in Cancer.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2942, doi. 10.1002/cmdc.202100334

By:

Liu, Li;
Li, Liqi;
Li, Menghuan;
Luo, Zhong

Publication type:

Article

Dinitrophenol‐Hyaluronan Conjugates as Multivalent Antibody‐Recruiting Glycopolymers for Targeted Cancer Immunotherapy.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2960, doi. 10.1002/cmdc.202100313

By:

Lin, Han;
Zhou, Kun;
Li, Dan;
Hong, Haofei;
Xie, Yuntian;
Gong, Liang;
Shen, Yu;
Zhou, Zhifang;
Shi, Jie;
Wu, Zhimeng

Publication type:

Article

Triazolyl‐Functionalized N‐Heterocyclic Carbene Half‐Sandwich Compounds: Coordination Mode, Reactivity and in vitro Anticancer Activity.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3017, doi. 10.1002/cmdc.202100311

By:

Tong, Kelvin K. H.;
Hanif, Muhammad;
Movassaghi, Sanam;
Sullivan, Matthew P.;
Lovett, James H.;
Hummitzsch, Katja;
Söhnel, Tilo;
Jamieson, Stephen M. F.;
Bhargava, Suresh K.;
Harris, Hugh H.;
Hartinger, Christian G.

Publication type:

Article

METTL3 Inhibitors for Epitranscriptomic Modulation of Cellular Processes.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3035, doi. 10.1002/cmdc.202100291

By:

Moroz‐Omori, Elena V.;
Huang, Danzhi;
Kumar Bedi, Rajiv;
Cheriyamkunnel, Sherry J.;
Bochenkova, Elena;
Dolbois, Aymeric;
Rzeczkowski, Maciej D.;
Li, Yaozong;
Wiedmer, Lars;
Caflisch, Amedeo

Publication type:

Article

Novel Phenyl‐Based Bis‐quaternary Ammonium Compounds as Broad‐Spectrum Biocides.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2954, doi. 10.1002/cmdc.202100284

By:

Frolov, Nikita A.;
Fedoseeva, Ksenia A.;
Hansford, Karl A.;
Vereshchagin, Anatoly N.

Publication type:

Article

From Quinoline to Quinazoline‐Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3044, doi. 10.1002/cmdc.202100282

By:

Cedraro, Nicholas;
Cannalire, Rolando;
Astolfi, Andrea;
Mangiaterra, Gianmarco;
Felicetti, Tommaso;
Vaiasicca, Salvatore;
Cernicchi, Giada;
Massari, Serena;
Manfroni, Giuseppe;
Tabarrini, Oriana;
Cecchetti, Violetta;
Barreca, Maria Letizia;
Biavasco, Francesca;
Sabatini, Stefano

Publication type:

Article

Polycomb Paralog Chromodomain Inhibitors Active against Both CBX6 and CBX8**.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 3027, doi. 10.1002/cmdc.202100262

By:

Milosevich, Natalia;
Wilson, Chelsea R.;
Brown, Tyler M.;
Alpsoy, Aktan;
Wang, Sijie;
Connelly, Katelyn E.;
Sinclair, Kirsten A. D.;
Ponio, Felino R.;
Hof, Rebecca;
Dykhuizen, Emily C.;
Hof, Fraser

Publication type:

Article

Recent Advances in Radiometals for Combined Imaging and Therapy in Cancer.

Published in:

ChemMedChem, 2021, v. 16, n. 19, p. 2909, doi. 10.1002/cmdc.202100135

By:

Herrero Álvarez, Natalia;
Bauer, David;
Hernández‐Gil, Javier;
Lewis, Jason S.

Publication type:

Article