Works matching IS 18607179 AND DT 2021 AND VI 16 AND IP 1

Results: 26

Cover Feature: Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar‐Based Molecules that Target Bacterial Glucosyltransferase (ChemMedChem 1/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 3, doi. 10.1002/cmdc.202000959

By:

Hartman, Alwin M.;
Jumde, Varsha R.;
Elgaher, Walid A. M.;
Te Poele, Evelien M.;
Dijkhuizen, Lubbert;
Hirsch, Anna K. H.

Publication type:

Article

Cover Feature: Broad‐Spectrum Antifungal Agents: Fluorinated Aryl‐ and Heteroaryl‐Substituted Hydrazones (ChemMedChem 1/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 2, doi. 10.1002/cmdc.202000958

By:

Thamban Chandrika, Nishad;
Dennis, Emily K.;
Brubaker, Katelyn R.;
Kwiatkowski, Stefan;
Watt, David S.;
Garneau‐Tsodikova, Sylvie

Publication type:

Article

Front Cover: Fabulous at Fifteen! (ChemMedChem 1/2021).

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 1, doi. 10.1002/cmdc.202000957

By:

Peralta, David

Publication type:

Article

Fabulous at Fifteen!

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 4, doi. 10.1002/cmdc.202000955

By:

Peralta, David

Publication type:

Article

François Diederich – In Memoriam**.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 11, doi. 10.1002/cmdc.202000920

By:

Hof, Fraser;
Hirsch, Anna K. H.

Publication type:

Article

Therapeutic Strategies To Counteract Antibiotic Resistance in MRSA Biofilm‐Associated Infections.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 65, doi. 10.1002/cmdc.202000677

By:

Cascioferro, Stella;
Carbone, Daniela;
Parrino, Barbara;
Pecoraro, Camilla;
Giovannetti, Elisa;
Cirrincione, Girolamo;
Diana, Patrizia

Publication type:

Article

N‐Phenyl‐1,2,3,4‐tetrahydroisoquinoline: An Alternative Scaffold for the Design of 17β‐Hydroxysteroid Dehydrogenase 1 Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 259, doi. 10.1002/cmdc.202000762

By:

Mottinelli, Marco;
Sinreih, Maša;
Rižner, Tea L.;
Leese, Mathew P.;
Potter, Barry V. L.

Publication type:

Article

Broad‐Spectrum Antifungal Agents: Fluorinated Aryl‐ and Heteroaryl‐Substituted Hydrazones.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 124, doi. 10.1002/cmdc.202000626

By:

Thamban Chandrika, Nishad;
Dennis, Emily K.;
Brubaker, Katelyn R.;
Kwiatkowski, Stefan;
Watt, David S.;
Garneau‐Tsodikova, Sylvie

Publication type:

Article

Two Methods, One Goal: Structural Differences between Cocrystallization and Crystal Soaking to Discover Ligand Binding Poses.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 292, doi. 10.1002/cmdc.202000565

By:

Wienen‐Schmidt, Barbara;
Oebbeke, Matthias;
Ngo, Khang;
Heine, Andreas;
Klebe, Gerhard

Publication type:

Article

Development of Novel 4‐Arylpyridin‐2‐one and 6‐Arylpyrimidin‐4‐one Positive Allosteric Modulators of the M<sub>1</sub> Muscarinic Acetylcholine Receptor.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 216, doi. 10.1002/cmdc.202000540

By:

Jörg, Manuela;
Khajehali, Elham;
Westhuizen, Emma T.;
C. Choy, K. H.;
Shackleford, David M.;
Tobin, Andrew B.;
Sexton, Patrick M.;
Valant, Celine;
Capuano, Ben;
Christopoulos, Arthur;
Scammells, Peter J.

Publication type:

Article

A Structure−Activity Relationship Study of Novel Hydroxamic Acid Inhibitors around the S1 Subsite of Human Aminopeptidase N.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 234, doi. 10.1002/cmdc.202000527

By:

Lee, Jisook;
Drinkwater, Nyssa;
McGowan, Sheena;
Scammells, Peter

Publication type:

Article

Potency and Selectivity Optimization of Tryptophanol‐Derived Oxazoloisoindolinones: Novel p53 Activators in Human Colorectal Cancer.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 250, doi. 10.1002/cmdc.202000522

By:

Barcherini, Valentina;
Almeida, Joana;
Lopes, Elizabeth A.;
Wang, Mi;
Magalhães e Silva, Diogo;
Mori, Mattia;
Wang, Shaomeng;
Saraiva, Lucília;
Santos, Maria M. M.

Publication type:

Article

Shuttling of Peptide‐Drug Conjugates by G Protein‐Coupled Receptors Is Significantly Improved by Pulsed Application.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 164, doi. 10.1002/cmdc.202000490

By:

Ziffert, Isabelle;
Kaiser, Anette;
Hoppenz, Paul;
Mörl, Karin;
Beck‐Sickinger, Annette G.

Publication type:

Article

Turning Donepezil into a Multi‐Target‐Directed Ligand through a Merging Strategy.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 187, doi. 10.1002/cmdc.202000484

By:

Perone, Rosaria;
Albertini, Claudia;
Uliassi, Elisa;
Di Pietri, Flaminia;
Sena Murteira Pinheiro, Pedro;
Petralla, Sabrina;
Rizzardi, Nicola;
Fato, Romana;
Pulkrabkova, Lenka;
Soukup, Ondrej;
Tramarin, Anna;
Bartolini, Manuela;
Bolognesi, Maria Laura

Publication type:

Article

Glycoconjugated Metal Complexes as Cancer Diagnostic and Therapeutic Agents.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 30, doi. 10.1002/cmdc.202000456

By:

Bononi, Giulia;
Iacopini, Dalila;
Cicio, Gaspare;
Di Pietro, Sebastiano;
Granchi, Carlotta;
Di Bussolo, Valeria;
Minutolo, Filippo

Publication type:

Article

7‐Amidocoumarins as Multitarget Agents against Neurodegenerative Diseases: Substitution Pattern Modulation.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 179, doi. 10.1002/cmdc.202000454

By:

Rodríguez‐Enríquez, Fernanda;
Viña, Dolores;
Uriarte, Eugenio;
Laguna, Reyes;
Matos, Maria J.

Publication type:

Article

Allosteric Molecular Switches in Metabotropic Glutamate Receptors.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 81, doi. 10.1002/cmdc.202000444

By:

Orgován, Zoltán;
Ferenczy, György G.;
Keserű, György M.

Publication type:

Article

Solid‐Phase Protein Modifications: Towards Precision Protein Hybrids for Biological Applications.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 94, doi. 10.1002/cmdc.202000412

By:

Kuan, Seah Ling;
Raabe, Marco

Publication type:

Article

HIV‐1 Envelope Spike MPER: From a Vaccine Target to a New Druggable Pocket for Novel and Effective Fusion Inhibitors.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 105, doi. 10.1002/cmdc.202000411

By:

Luque, Francisco Javier;
Camarasa, María‐José

Publication type:

Article

Radiolabelled CCK<sub>2</sub>R Antagonists Containing PEG Linkers: Design, Synthesis and Evaluation.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 155, doi. 10.1002/cmdc.202000392

By:

Novak, Doroteja;
Tomašič, Tihomir;
Krošelj, Marko;
Javornik, Uroš;
Plavec, Janez;
Anderluh, Marko;
Kolenc Peitl, Petra

Publication type:

Article

Effective Oral Administration of an Antitumorigenic Nanoformulated Titanium Complex.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 108, doi. 10.1002/cmdc.202000384

By:

Nahari, Gilad;
Braitbard, Ori;
Larush, Liraz;
Hochman, Jacob;
Tshuva, Edit Y.

Publication type:

Article

MS Binding Assays for Glycine Transporter 2 (GlyT2) Employing Org25543 as Reporter Ligand.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 199, doi. 10.1002/cmdc.202000342

By:

Ackermann, Thomas M.;
Allmendinger, Lars;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

The Triazole Ring as a Privileged Scaffold for Putative Antifungals: Synthesis and Evaluation of a Series of New Analogues.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 134, doi. 10.1002/cmdc.202000312

By:

Zoidis, Grigoris;
Kritsi, Eftichia;
Lecinska, Paulina;
Ivanov, Marija;
Zoumpoulakis, Panagiotis;
Sokovic, Marina;
Catto, Marco

Publication type:

Article

Differentiation of Cancer Stem Cells by Using Synthetic Small Molecules: Toward New Therapeutic Strategies against Therapy Resistance.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 14, doi. 10.1002/cmdc.202000251

By:

Maucort, Chloé;
Di Giorgio, Audrey;
Azoulay, Stéphane;
Duca, Maria

Publication type:

Article

Potential Dental Biofilm Inhibitors: Dynamic Combinatorial Chemistry Affords Sugar‐Based Molecules that Target Bacterial Glucosyltransferase.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 113, doi. 10.1002/cmdc.202000222

By:

Hartman, Alwin M.;
Jumde, Varsha R.;
Elgaher, Walid A. M.;
Te Poele, Evelien M.;
Dijkhuizen, Lubbert;
Hirsch, Anna K. H.

Publication type:

Article

Synthesis and Biological Evaluation of Endocannabinoid Uptake Inhibitors Derived from WOBE437.

Published in:

ChemMedChem, 2021, v. 16, n. 1, p. 145, doi. 10.1002/cmdc.202000153

By:

Mäder, Patrick;
Bartholomäus, Ruben;
Nicolussi, Simon;
Baumann, Alice;
Weis, Melanie;
Chicca, Andrea;
Rau, Mark;
Simão, Ana Catarina;
Gertsch, Jürg;
Altmann, Karl‐Heinz

Publication type:

Article