Works matching IS 18607179 AND DT 2020 AND VI 15 AND IP 7

Results: 12

Elucidation of an Allosteric Mode of Action for a Thienopyrazole RORγt Inverse Agonist.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 561, doi. 10.1002/cmdc.202000044
By:
- Vries, Rens M. J. M.;
- Doveston, Richard G.;
- Meijer, Femke A.;
- Brunsveld, Luc
Publication type:
Article
Shape Similarity by Fractal Dimensionality: An Application in the de novo Design of (−)‐Englerin A Mimetics.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 566, doi. 10.1002/cmdc.202000017
By:
- Friedrich, Lukas;
- Byrne, Ryan;
- Treder, Aaron;
- Singh, Inderjeet;
- Bauer, Christoph;
- Gudermann, Thomas;
- Mederos y Schnitzler, Michael;
- Storch, Ursula;
- Schneider, Gisbert
Publication type:
Article
Design, Synthesis, and Dual Evaluation of Quinoline and Quinolinium Iodide Salt Derivatives as Potential Anticancer and Antibacterial Agents.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 600, doi. 10.1002/cmdc.202000002
By:
- Jin, Guofan;
- Xiao, Fuyan;
- Li, Zhenwang;
- Qi, Xueyong;
- Zhao, Lei;
- Sun, Xianyu
Publication type:
Article
Tranylcypromine‐Based LSD1 Inhibitors: Structure‐Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 643, doi. 10.1002/cmdc.201900730
By:
- Fioravanti, Rossella;
- Romanelli, Annalisa;
- Mautone, Nicola;
- Di Bello, Elisabetta;
- Rovere, Annarita;
- Corinti, Davide;
- Zwergel, Clemens;
- Valente, Sergio;
- Rotili, Dante;
- Botrugno, Oronza A.;
- Dessanti, Paola;
- Vultaggio, Stefania;
- Vianello, Paola;
- Cappa, Anna;
- Binda, Claudia;
- Mattevi, Andrea;
- Minucci, Saverio;
- Mercurio, Ciro;
- Varasi, Mario;
- Mai, Antonello
Publication type:
Article
Covalent Complex of DNA and Bacterial Topoisomerase: Implications in Antibacterial Drug Development.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 623, doi. 10.1002/cmdc.201900721
By:
- Tiwari, Purushottam B.;
- Chapagain, Prem P.;
- Seddek, Ahmed;
- Annamalai, Thirunavukkarasu;
- Üren, Aykut;
- Tse‐Dinh, Yuk‐Ching
Publication type:
Article
Comparative in vitro Studies of the Topoisomerase I Inhibition and Anticancer Activities of Metallated N‐Confused Porphyrins and Metallated Porphyrins.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 632, doi. 10.1002/cmdc.201900633
By:
- Halder, Nyancy;
- Dzhemileva, Lilya U.;
- Ramazanov, Ilfir R.;
- D'yakonov, Vladimir A.;
- Dzhemilev, Usein M.;
- Rath, Harapriya
Publication type:
Article
Synthesis, Molecular Docking, and Preliminary Evaluation of 2‐(1,2,3‐Triazoyl)benzaldehydes As Multifunctional Agents for the Treatment of Alzheimer's Disease.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 610, doi. 10.1002/cmdc.201900622
By:
- Costa, Gabriel P.;
- Baldinotti, Rodolfo S. M.;
- Fronza, Mariana G.;
- Nascimento, José Edmilson R.;
- Dias, Ítalo F. C.;
- Sonego, Mariana Souza;
- Seixas, Fabiana Kömmling;
- Collares, Tiago;
- Perin, Gelson;
- Jacob, Raquel G.;
- Savegnago, Lucielli;
- Alves, Diego
Publication type:
Article
A Comparative Study of in vitro Assays for Predicting the Nonspecific Binding of PET Imaging Agents in vivo.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 585, doi. 10.1002/cmdc.201900608
By:
- Gobbi, Luca;
- Mercier, Joël;
- Bang‐Andersen, Benny;
- Nicolas, Jean‐Marie;
- Reilly, John;
- Wagner, Björn;
- Whitehead, David;
- Briard, Emmanuelle;
- Maguire, R. Paul;
- Borroni, Edilio;
- Auberson, Yves P.
Publication type:
Article
Biodegradable Periodic Mesoporous Organosilica (BPMO) Loaded with Daunorubicin: A Promising Nanoparticle‐Based Anticancer Drug.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 593, doi. 10.1002/cmdc.201900595
By:
- Mai, Ngoc Xuan Dat;
- Birault, Albane;
- Matsumoto, Kotaro;
- Ta, Hanh Kieu Thi;
- Intasa‐ard, Soontaree Grace;
- Morrison, Kendall;
- Thang, Phan Bach;
- Doan, Tan Le Hoang;
- Tamanoi, Fuyuhiko
Publication type:
Article
Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors.
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 571, doi. 10.1002/cmdc.201900583
By:
- Kalinin, Dmitrii V.;
- Jana, Sunit K.;
- Pfafenrot, Maxim;
- Chakrabarti, Alokta;
- Melesina, Jelena;
- Shaik, Tajith B.;
- Lancelot, Julien;
- Pierce, Raymond J.;
- Sippl, Wolfgang;
- Romier, Christophe;
- Jung, Manfred;
- Holl, Ralph
Publication type:
Article
Cover Feature: A Comparative Study of in vitro Assays for Predicting the Nonspecific Binding of PET Imaging Agents in vivo (ChemMedChem 7/2020).
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 560, doi. 10.1002/cmdc.201000140
By:
- Gobbi, Luca;
- Mercier, Joël;
- Bang‐Andersen, Benny;
- Nicolas, Jean‐Marie;
- Reilly, John;
- Wagner, Björn;
- Whitehead, David;
- Briard, Emmanuelle;
- Maguire, R. Paul;
- Borroni, Edilio;
- Auberson, Yves P.
Publication type:
Article
Front Cover: Structure‐Based Design, Synthesis, and Biological Evaluation of Triazole‐Based smHDAC8 Inhibitors (ChemMedChem 7/2020).
Published in:
ChemMedChem, 2020, v. 15, n. 7, p. 559, doi. 10.1002/cmdc.201000139
By:
- Kalinin, Dmitrii V.;
- Jana, Sunit K.;
- Pfafenrot, Maxim;
- Chakrabarti, Alokta;
- Melesina, Jelena;
- Shaik, Tajith B.;
- Lancelot, Julien;
- Pierce, Raymond J.;
- Sippl, Wolfgang;
- Romier, Christophe;
- Jung, Manfred;
- Holl, Ralph
Publication type:
Article