Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 9

Results: 11

Cover Feature: Covalent Inhibition in Drug Discovery (ChemMedChem 9/2019).
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 888, doi. 10.1002/cmdc.201900236
By:
- Ghosh, Avick Kumar;
- Samanta, Indranil;
- Mondal, Anushree;
- Liu, Wenshe Ray
Publication type:
Article
Front Cover: Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity (ChemMedChem 9/2019).
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 887, doi. 10.1002/cmdc.201900235
By:
- Mackwitz, Marcel K. W.;
- Hesping, Eva;
- Antonova‐Koch, Yevgeniya;
- Diedrich, Daniela;
- Woldearegai, Tamirat Gebru;
- Skinner‐Adams, Tina;
- Clarke, Mary;
- Schöler, Andrea;
- Limbach, Laura;
- Kurz, Thomas;
- Winzeler, Elizabeth A.;
- Held, Jana;
- Andrews, Katherine T.;
- Hansen, Finn K.
Publication type:
Article
Sulfide Analogues of Flupirtine and Retigabine with Nanomolar KV7.2/KV7.3 Channel Opening Activity.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 952, doi. 10.1002/cmdc.201900112
By:
- Bock, Christian;
- Surur, Abdrrahman S.;
- Beirow, Kristin;
- Kindermann, Markus K.;
- Schulig, Lukas;
- Bodtke, Anja;
- Bednarski, Patrick J.;
- Link, Andreas
Publication type:
Article
Covalent Inhibition in Drug Discovery.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 889, doi. 10.1002/cmdc.201900107
By:
- Ghosh, Avick Kumar;
- Samanta, Indranil;
- Mondal, Anushree;
- Liu, Wenshe Ray
Publication type:
Article
Discovery, Optimization, and Biological Characterization of 2,3,6‐Trisubstituted Pyridine‐Containing M4 Positive Allosteric Modulators.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 943, doi. 10.1002/cmdc.201900088
By:
- Schubert, Jeffrey W.;
- Harrison, Scott T.;
- Mulhearn, James;
- Gomez, Robert;
- Tynebor, Robert;
- Jones, Kristen;
- Bunda, Jaime;
- Hanney, Barbara;
- Wai, Jenny Miu‐Chen;
- Cox, Chris;
- McCauley, John A.;
- Sanders, John M.;
- Magliaro, Brian;
- O'Brien, Julie;
- Pajkovic, Natasa;
- Huszar Agrapides, Sarah L.;
- Taylor, Anne;
- Gotter, Anthony;
- Smith, Sean M.;
- Uslaner, Jason
Publication type:
Article
Structure–Activity Relationships of 1‐Benzoylazulenes at the OX1 and OX2 Orexin Receptors.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 965, doi. 10.1002/cmdc.201900074
By:
- Turku, Ainoleena;
- Leino, Teppo O.;
- Karhu, Lasse;
- Yli‐Kauhaluoma, Jari;
- Kukkonen, Jyrki P.;
- Wallén, Erik A. A.;
- Xhaard, Henri
Publication type:
Article
Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin αVβ3.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 938, doi. 10.1002/cmdc.201900049
By:
- Raposo Moreira Dias, André;
- Bodero, Lizeth;
- Martins, Ana;
- Arosio, Daniela;
- Gazzola, Silvia;
- Belvisi, Laura;
- Pignataro, Luca;
- Steinkühler, Christian;
- Dal Corso, Alberto;
- Gennari, Cesare;
- Piarulli, Umberto
Publication type:
Article
Ionic Liquids and Salts from Ibuprofen as Promising Innovative Formulations of an Old Drug.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 907, doi. 10.1002/cmdc.201900040
By:
- Santos, Miguel M.;
- Raposo, Luís R.;
- Carrera, Gonçalo V. S. M.;
- Costa, Alexandra;
- Dionísio, Madalena;
- Baptista, Pedro V.;
- Fernandes, Alexandra R.;
- Branco, Luís C.
Publication type:
Article
Identification of Anti‐Mycobacterial Biofilm Agents Based on the 2‐Aminoimidazole Scaffold.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 927, doi. 10.1002/cmdc.201900033
By:
- Nguyen, T. Vu;
- Minrovic, Bradley M.;
- Melander, Roberta J.;
- Melander, Christian
Publication type:
Article
Radiosynthesis of (R,S)‐[18F]GE387: A Potential PET Radiotracer for Imaging Translocator Protein 18 kDa (TSPO) with Low Binding Sensitivity to the Human Gene Polymorphism rs6971.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 982, doi. 10.1002/cmdc.201900023
By:
- Qiao, Luxi;
- Fisher, Emily;
- McMurray, Lindsay;
- Milicevic Sephton, Selena;
- Hird, Matthew;
- Kuzhuppilly‐Ramakrishnan, Nisha;
- Williamson, David J.;
- Zhou, Xiouyun;
- Werry, Eryn;
- Kassiou, Michael;
- Luthra, Saijinder;
- Trigg, William;
- Aigbirhio, Franklin I.
Publication type:
Article
Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity.
Published in:
ChemMedChem, 2019, v. 14, n. 9, p. 912, doi. 10.1002/cmdc.201800808
By:
- Mackwitz, Marcel K. W.;
- Hesping, Eva;
- Antonova‐Koch, Yevgeniya;
- Diedrich, Daniela;
- Woldearegai, Tamirat Gebru;
- Skinner‐Adams, Tina;
- Clarke, Mary;
- Schöler, Andrea;
- Limbach, Laura;
- Kurz, Thomas;
- Winzeler, Elizabeth A.;
- Held, Jana;
- Andrews, Katherine T.;
- Hansen, Finn K.
Publication type:
Article

Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 9

Cover Feature: Covalent Inhibition in Drug Discovery (ChemMedChem 9/2019).

Front Cover: Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity (ChemMedChem 9/2019).

Sulfide Analogues of Flupirtine and Retigabine with Nanomolar K<sub>V</sub>7.2/K<sub>V</sub>7.3 Channel Opening Activity.

Covalent Inhibition in Drug Discovery.

Discovery, Optimization, and Biological Characterization of 2,3,6‐Trisubstituted Pyridine‐Containing M<sub>4</sub> Positive Allosteric Modulators.

Structure–Activity Relationships of 1‐Benzoylazulenes at the OX<sub>1</sub> and OX<sub>2</sub> Orexin Receptors.

Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin α<sub>V</sub>β<sub>3</sub>.

Ionic Liquids and Salts from Ibuprofen as Promising Innovative Formulations of an Old Drug.

Identification of Anti‐Mycobacterial Biofilm Agents Based on the 2‐Aminoimidazole Scaffold.

Radiosynthesis of (R,S)‐[<sup>18</sup>F]GE387: A Potential PET Radiotracer for Imaging Translocator Protein 18 kDa (TSPO) with Low Binding Sensitivity to the Human Gene Polymorphism rs6971.

Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity.