Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 22


Results: 8
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    Trifluoromethyl Dihydrothiazine‐Based β‐Secretase (BACE1) Inhibitors with Robust Central β‐Amyloid Reduction and Minimal Covalent Binding Burden.

    Published in:
    ChemMedChem, 2019, v. 14, n. 22, p. 1894, doi. 10.1002/cmdc.201900478
    By:
    • Anan, Kosuke;
    • Iso, Yasuyoshi;
    • Oguma, Takuya;
    • Nakahara, Kenji;
    • Suzuki, Shinji;
    • Yamamoto, Takahiko;
    • Matsuoka, Eriko;
    • Ito, Hisanori;
    • Sakaguchi, Gaku;
    • Ando, Shigeru;
    • Morimoto, Kenji;
    • Kanegawa, Naoki;
    • Kido, Yasuto;
    • Kawachi, Tomoyuki;
    • Fukushima, Tamio;
    • Teisman, Ard;
    • Urmaliya, Vijay;
    • Dhuyvetter, Deborah;
    • Borghys, Herman;
    • Austin, Nigel
    Publication type:
    Article
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    Design and Synthesis of Conformationally Constrained RORγt Inverse Agonists.

    Published in:
    ChemMedChem, 2019, v. 14, n. 22, p. 1917, doi. 10.1002/cmdc.201900416
    By:
    • Sato, Ayumu;
    • Fukase, Yoshiyuki;
    • Kono, Mitsunori;
    • Ochida, Atsuko;
    • Oda, Tsuneo;
    • Sasaki, Yusuke;
    • Ishii, Naoki;
    • Tomata, Yoshihide;
    • Fukumoto, Shoji;
    • Imai, Yumi N.;
    • Uga, Keiko;
    • Shibata, Akira;
    • Yamasaki, Masashi;
    • Nakagawa, Hideyuki;
    • Shirasaki, Mikio;
    • Skene, Robert;
    • Hoffman, Isaac;
    • Sang, Bi‐Ching;
    • Snell, Gyorgy;
    • Shirai, Junya
    Publication type:
    Article
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