Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 2

Results: 9

A Multi‐step Virtual Screening Protocol for the Identification of Novel Non‐acidic Microsomal Prostaglandin E<sub>2</sub> Synthase‐1 (mPGES‐1) Inhibitors.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 273, doi. 10.1002/cmdc.201800701

By:

Shekfeh, Suhaib;
Çalışkan, Burcu;
Fischer, Katrin;
Yalçın, Tansu;
Garscha, Ulrike;
Werz, Oliver;
Banoglu, Erden

Publication type:

Article

Front Cover: Identifying Lysophosphatidic Acid Acyltransferase β (LPAAT‐β) as the Target of a Nanomolar Angiogenesis Inhibitor from a Phenotypic Screen Using the Polypharmacology Browser PPB2 (ChemMedChem 2/2019).

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 189, doi. 10.1002/cmdc.201900013

By:

Poirier, Marion;
Awale, Mahendra;
Roelli, Matthias A.;
Giuffredi, Guy T.;
Ruddigkeit, Lars;
Evensen, Lasse;
Stooss, Amandine;
Calarco, Serafina;
Lorens, James B.;
Charles, Roch‐Philippe;
Reymond, Jean‐Louis

Publication type:

Article

Discovery of Affinity‐Based Probes for Btk Occupancy Assays.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 217, doi. 10.1002/cmdc.201800714

By:

Qiu, Hui;
Caldwell, Richard;
Liu‐Bujalski, Lesley;
Goutopoulos, Andreas;
Jones, Reinaldo;
Potnick, Justin;
Sherer, Brian;
Bender, Andrew;
Grenningloh, Roland;
Xu, Daigen;
Gardberg, Anna;
Mochalkin, Igor;
Johnson, Theresa;
Viacava Follis, Ariele;
Head, Jared;
Morandi, Federica

Publication type:

Article

Assembly of Fully Substituted 2H‐Indazoles Catalyzed by Cu<sub>2</sub>O Rhombic Dodecahedra and Evaluation of Anticancer Activity.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 262, doi. 10.1002/cmdc.201800707

By:

Panchangam, Rajeeva Lochana;
Manickam, Venkatraman;
Chanda, Kaushik

Publication type:

Article

Synthesis of Modified RGD‐Based Peptides and Their in vitro Activity.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 282, doi. 10.1002/cmdc.201800704

By:

Hamdan, Fatima;
Bigdeli, Zahra;
Asghari, S. Mohsen;
Sadremomtaz, Afsaneh;
Balalaie, Saeed

Publication type:

Article

The Role of the Phosphorus Atom in Drug Design.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 190, doi. 10.1002/cmdc.201800693

By:

Rodriguez, Juan B.;
Gallo‐Rodriguez, Carola

Publication type:

Article

A Scaffold‐Hopping Strategy toward the Identification of Inhibitors of Cyclin G Associated Kinase.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 237, doi. 10.1002/cmdc.201800690

By:

Wouters, Randy;
Tian, Junjun;
Herdewijn, Piet;
De Jonghe, Steven

Publication type:

Article

Carborane‐Based Analogues of 5‐Lipoxygenase Inhibitors Co‐inhibit Heat Shock Protein 90 in HCT116 Cells.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 255, doi. 10.1002/cmdc.201800651

By:

Kuhnert, Robert;
Sárosi, Menyhárt‐Botond;
George, Sven;
Lönnecke, Peter;
Hofmann, Bettina;
Steinhilber, Dieter;
Steinmann, Sara;
Schneider‐Stock, Regine;
Murganić, Blagoje;
Mijatović, Sanja;
Maksimović‐Ivanić, Danijela;
Hey‐Hawkins, Evamarie

Publication type:

Article

Identifying Lysophosphatidic Acid Acyltransferase β (LPAAT‐β) as the Target of a Nanomolar Angiogenesis Inhibitor from a Phenotypic Screen Using the Polypharmacology Browser PPB2.

Published in:

ChemMedChem, 2019, v. 14, n. 2, p. 224, doi. 10.1002/cmdc.201800554

By:

Poirier, Marion;
Awale, Mahendra;
Roelli, Matthias A.;
Giuffredi, Guy T.;
Ruddigkeit, Lars;
Evensen, Lasse;
Stooss, Amandine;
Calarco, Serafina;
Lorens, James B.;
Charles, Roch‐Philippe;
Reymond, Jean‐Louis

Publication type:

Article