Works matching IS 18607179 AND DT 2019 AND VI 14 AND IP 14

Results: 10

Front Cover: Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes (ChemMedChem 14/2019).

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1304, doi. 10.1002/cmdc.201900400

By:

Kallen, Joerg;
Izaac, Aude;
Chau, Suzanne;
Wirth, Emmanuelle;
Schoepfer, Joseph;
Mah, Robert;
Schlapbach, Achim;
Stutz, Stefan;
Vaupel, Andrea;
Guagnano, Vito;
Masuya, Keiichi;
Stachyra, Therese‐Marie;
Salem, Bahaa;
Chene, Patrick;
Gessier, Francois;
Holzer, Philipp;
Furet, Pascal

Publication type:

Article

The Design of Potent, Selective and Drug‐Like RGD αvβ1 Small‐Molecule Inhibitors Derived from non‐RGD α4β1 Antagonists.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1315, doi. 10.1002/cmdc.201900359

By:

Hatley, Richard J. D.;
Barrett, Tim N.;
Slack, Robert J.;
Watson, Morag E.;
Baillache, Daniel J.;
Gruszka, Anna;
Washio, Yoshiaki;
Rowedder, James E.;
Pogány, Peter;
Pal, Sandeep;
Macdonald, Simon J. F.

Publication type:

Article

Experimental and Computational Evaluation of Piperonylic Acid Derived Hydrazones Bearing Isatin Moieties as Dual Inhibitors of Cholinesterases and Monoamine Oxidases.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1359, doi. 10.1002/cmdc.201900277

By:

Vishnu, M. S.;
Pavankumar, V.;
Kumar, Sandeep;
Raja, A. Senthil

Publication type:

Article

Substituted Aminoacetamides as Novel Leads for Malaria Treatment.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1329, doi. 10.1002/cmdc.201900329

By:

Norcross, Neil R.;
Wilson, Caroline;
Baragaña, Beatriz;
Hallyburton, Irene;
Osuna‐Cabello, Maria;
Norval, Suzanne;
Riley, Jennifer;
Fletcher, Daniel;
Sinden, Robert;
Delves, Michael;
Ruecker, Andrea;
Duffy, Sandra;
Meister, Stephan;
Antonova‐Koch, Yevgeniya;
Crespo, Benigno;
de Cózar, Cristina;
Sanz, Laura M.;
Gamo, Francisco Javier;
Avery, Vicky M.;
Frearson, Julie A.

Publication type:

Article

Fragment Growing to Design Optimized Inhibitors for Human Blood Group B Galactosyltransferase (GTB).

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1336, doi. 10.1002/cmdc.201900296

By:

Strecker, Claas;
Peters, Hannelore;
Hackl, Thomas;
Peters, Thomas;
Meyer, Bernd

Publication type:

Article

Computer‐Assisted Selective Optimization of Side‐Activities—from Cinalukast to a PPARα Modulator.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1343, doi. 10.1002/cmdc.201900286

By:

Pollinger, Julius;
Schierle, Simone;
Neumann, Sebastian;
Ohrndorf, Julia;
Kaiser, Astrid;
Merk, Daniel

Publication type:

Article

Novel BQCA‐ and TBPB‐Derived M<sub>1</sub> Receptor Hybrid Ligands: Orthosteric Carbachol Differentially Regulates Partial Agonism.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1349, doi. 10.1002/cmdc.201900283

By:

Schramm, Simon;
Agnetta, Luca;
Bermudez, Marcel;
Gerwe, Hubert;
Irmen, Matthias;
Holze, Janine;
Littmann, Timo;
Wolber, Gerhard;
Tränkle, Christian;
Decker, Michael

Publication type:

Article

Small‐Molecule Activators of Glucose‐6‐phosphate Dehydrogenase (G6PD) Bridging the Dimer Interface.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1321, doi. 10.1002/cmdc.201900341

By:

Raub, Andrew G.;
Hwang, Sunhee;
Horikoshi, Naoki;
Cunningham, Anna D.;
Rahighi, Simin;
Wakatsuki, Soichi;
Mochly‐Rosen, Daria

Publication type:

Article

Combining 1,3‐Ditriazolylbenzene and Quinoline to Discover a New G‐Quadruplex‐Interactive Small Molecule Active against Cancer Stem‐Like Cells.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1325, doi. 10.1002/cmdc.201900243

By:

Mendes, Eduarda;
Cadoni, Enrico;
Carneiro, Filipa;
Afonso, Marta B.;
Brito, Hugo;
Lavrado, João;
dos Santos, Daniel J. V. A.;
Vítor, Jorge B.;
Neidle, Stephen;
Rodrigues, Cecília M. P.;
Paulo, Alexandra

Publication type:

Article

Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes.

Published in:

ChemMedChem, 2019, v. 14, n. 14, p. 1305, doi. 10.1002/cmdc.201900201

By:

Kallen, Joerg;
Izaac, Aude;
Chau, Suzanne;
Wirth, Emmanuelle;
Schoepfer, Joseph;
Mah, Robert;
Schlapbach, Achim;
Stutz, Stefan;
Vaupel, Andrea;
Guagnano, Vito;
Masuya, Keiichi;
Stachyra, Therese‐Marie;
Salem, Bahaa;
Chene, Patrick;
Gessier, Francois;
Holzer, Philipp;
Furet, Pascal

Publication type:

Article