Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 4

Results: 13

Front Cover: Helenalin Analogues Targeting NF‐κB p65: Thiol Reactivity and Cellular Potency Studies of Varied Electrophiles (ChemMedChem 4/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 288, doi. 10.1002/cmdc.201800079

By:

Widen, John C.;
Kempema, Aaron M.;
Baur, Jordan W.;
Skopec, Hannah M.;
Edwards, Jacob T.;
Brown, Tenley J.;
Brown, Dennis A.;
Meece, Frederick A.;
Harki, Daniel A.

Publication type:

Article

Discovery of Novel Muscarinic Receptor Modulators by Integrating a Natural Product Framework and a Bioactive Molecule.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 384, doi. 10.1002/cmdc.201800001

By:

Varkhedkar, Rajesh;
Dogra, Shalini;
Tiwari, Divya;
Hussain, Yusuf;
Yadav, Prem Narayan;
Pandey, Ganesh

Publication type:

Article

<bold>Cannabinoid Pharmacology, Volume 80 of Advances in Pharmacology</bold>. Edited by David Kendall and Stephen Alexander.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 398, doi. 10.1002/cmdc.201700827

By:

Decker, Michael

Publication type:

Article

Value Creation in the Pharmaceutical Industry — The Critical Path to Innovation. Edited by Alexander Schuhmacher, Markus Hinder and Oliver Gassmann.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 397, doi. 10.1002/cmdc.201700797

By:

Auriel, Daniel

Publication type:

Article

<bold>Successful Drug Discovery, Volume 2</bold>. Edited by János Fischer and Wayne E. Childers.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 396, doi. 10.1002/cmdc.201700775

By:

Gabriel, Tobias

Publication type:

Article

Interactions between Clinically Used Bisphosphonates and Bone Mineral: from Coordination Chemistry to Biomedical Applications and Beyond.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 289, doi. 10.1002/cmdc.201700769

By:

Gałęzowska, Joanna

Publication type:

Article

Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 321, doi. 10.1002/cmdc.201700758

By:

Ouvry, Gilles;
Atrux‐Tallau, Nicolas;
Bihl, Franck;
Bondu, Aline;
Bouix‐Peter, Claire;
Carlavan, Isabelle;
Christin, Olivier;
Cuadrado, Marie‐Josée;
Defoin‐Platel, Claire;
Deret, Sophie;
Duvert, Denis;
Feret, Christophe;
Forissier, Mathieu;
Fournier, Jean‐François;
Froude, David;
Hacini‐Rachinel, Fériel;
Harris, Craig Steven;
Hervouet, Catherine;
Huguet, Hélène;
Lafitte, Guillaume

Publication type:

Article

Helenalin Analogues Targeting NF‐κB p65: Thiol Reactivity and Cellular Potency Studies of Varied Electrophiles.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 303, doi. 10.1002/cmdc.201700752

By:

Widen, John C.;
Kempema, Aaron M.;
Baur, Jordan W.;
Skopec, Hannah M.;
Edwards, Jacob T.;
Brown, Tenley J.;
Brown, Dennis A.;
Meece, Frederick A.;
Harki, Daniel A.

Publication type:

Article

In Vitro Photodynamic Activity of N‐Methylated and N‐Oxidised Tripyridyl Porphyrins with Long Alkyl Chains and Their Inhibitory Activity in Sphingolipid Metabolism.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 360, doi. 10.1002/cmdc.201700748

By:

Jelovica, Mateo;
Grbčić, Petra;
Mušković, Martina;
Sedić, Mirela;
Pavelić, Sandra Kraljević;
Lončarić, Martin;
Malatesti, Nela

Publication type:

Article

Design, Synthesis and Evaluation of Oxazaborine Inhibitors of the NLRP3 Inflammasome.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 312, doi. 10.1002/cmdc.201700731

By:

Baldwin, Alex G.;
Tapia, Victor S.;
Swanton, Tessa;
White, Claire S.;
Beswick, James A.;
Brough, David;
Freeman, Sally

Publication type:

Article

Achieving Biocompatible SABRE: An in vitro Cytotoxicity Study.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 352, doi. 10.1002/cmdc.201700725

By:

Manoharan, Anand;
Rayner, Peter J.;
Iali, Wissam;
Burns, Michael J.;
Perry, V. Hugh;
Duckett, Simon B.

Publication type:

Article

<italic>N</italic>‐Benzyl Substitution of Polyhydroxypyrrolidines: The Way to Selective Inhibitors of Golgi α‐Mannosidase II.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 373, doi. 10.1002/cmdc.201700607

By:

Šesták, Sergej;
Bella, Maroš;
Klunda, Tomáš;
Gurská, Soňa;
Džubák, Petr;
Wöls, Florian;
Wilson, Iain B. H.;
Sladek, Vladimir;
Hajdúch, Marián;
Poláková, Monika;
Kóňa, Juraj

Publication type:

Article

Synthesis of N‐Substituted Iminosugar Derivatives and Evaluation of Their Immunosuppressive Activities.

Published in:

ChemMedChem, 2018, v. 13, n. 4, p. 338, doi. 10.1002/cmdc.201700706

By:

Lv, Zhuo;
Song, Chengcheng;
Niu, Youhong;
Li, Qin;
Ye, Xin‐Shan

Publication type:

Article