Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 23

Results: 15

Cover Feature: Mapping the Pathway and Dynamics of Bestatin Inhibition of the Plasmodium falciparum M1 Aminopeptidase PfA‐M1 (ChemMedChem 23/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2465, doi. 10.1002/cmdc.201800741

By:

Yang, Wei;
Riley, Blake T.;
Lei, Xiangyun;
Porebski, Benjamin T.;
Kass, Itamar;
Buckle, Ashley M.;
McGowan, Sheena

Publication type:

Article

Front Cover: Identification of Pyrrolidine‐3‐acetic Acid Derived Oximes as Potent Inhibitors of γ‐Aminobutyric Acid Transporter 1 through Library Screening with MS Binding Assays (ChemMedChem 23/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2464, doi. 10.1002/cmdc.201800740

By:

Huber, Simone K.;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

Antimicrobial and Antibiofilm Activity of Disubstituted Bis‐benzimidazolium Salts.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2567, doi. 10.1002/cmdc.201800639

By:

Tessier, Jérémie;
Lecluse, Margaux;
Gravel, Julien;
Schmitzer, Andreea‐Ruxandra

Publication type:

Article

<sup>18</sup>F‐Labeled Derivatives of Irbesartan for Angiotensin II Receptor PET Imaging.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2546, doi. 10.1002/cmdc.201800638

By:

Hoffmann, Matthias;
Chen, Xinyu;
Hirano, Mitsuru;
Arimitsu, Kenji;
Kimura, Hiroyuki;
Higuchi, Takahiro;
Decker, Michael

Publication type:

Article

In silico Screening and Evaluation of Plasmodium falciparum Protein Kinase 5 (PK5) Inhibitors.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2479, doi. 10.1002/cmdc.201800625

By:

Eubanks, Amber L.;
Perkins, Marisha M.;
Sylvester, Kayla;
Ganley, Jack G.;
Posfai, Dora;
Sanschargrin, Paul C.;
Hong, Jiyong;
Sliz, Piotr;
Derbyshire, Emily R.

Publication type:

Article

Antibody Fragment and Affibody ImmunoPET Imaging Agents: Radiolabelling Strategies and Applications.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2466, doi. 10.1002/cmdc.201800624

By:

Fu, Ruisi;
Carroll, Laurence;
Yahioglu, Gokhan;
Aboagye, Eric O.;
Miller, Philip W.

Publication type:

Article

In vitro Anti‐atherogenic Properties of N‐Heterocyclic Carbene Aurate(I) Compounds.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2484, doi. 10.1002/cmdc.201800601

By:

Sioriki, Eleni;
Lordan, Ronan;
Nahra, Fady;
van Hecke, Kristof;
Zabetakis, Ioannis;
Nolan, Steven P.

Publication type:

Article

Elucidating the Catalytic Power of Glutamate Racemase by Investigating a Series of Covalent Inhibitors.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2514, doi. 10.1002/cmdc.201800592

By:

Vance, Nicholas R.;
Witkin, Katie R.;
Rooney, Patrick W.;
Li, Yalan;
Pope, Marshall;
Spies, M. Ashley

Publication type:

Article

Orally Effective Aminoalkyl 10H‐Indolo[3,2‐b]quinoline‐11‐carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2581, doi. 10.1002/cmdc.201800579

By:

Mudududdla, Ramesh;
Mohanakrishnan, Dinesh;
Bharate, Sonali S.;
Vishwakarma, Ram A.;
Sahal, Dinkar;
Bharate, Sandip B.

Publication type:

Article

Identification and Biological Evaluation of Novel Type II B‐Raf<sup>V600E</sup> Inhibitors.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2558, doi. 10.1002/cmdc.201800574

By:

Wang, Peng‐Fei;
Wang, Ze‐Feng;
Qiu, Han‐Yue;
Huang, Yue;
Hu, Hui‐Min;
Wang, Zhong‐Chang;
Zhu, Hai‐Liang

Publication type:

Article

Replacement of the Benzylpiperidine Moiety with Fluorinated Phenylalkyl Side Chains for the Development of GluN2B Receptor Ligands.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2522, doi. 10.1002/cmdc.201800566

By:

Thum, Simone;
Schepmann, Dirk;
Kalinin, Dmitrii V.;
Ametamey, Simon M.;
Wünsch, Bernhard

Publication type:

Article

Mapping the Pathway and Dynamics of Bestatin Inhibition of the Plasmodium falciparum M1 Aminopeptidase PfA‐M1.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2504, doi. 10.1002/cmdc.201800563

By:

Yang, Wei;
Riley, Blake T.;
Lei, Xiangyun;
Porebski, Benjamin T.;
Kass, Itamar;
Buckle, Ashley M.;
McGowan, Sheena

Publication type:

Article

Identification of Pyrrolidine‐3‐acetic Acid Derived Oximes as Potent Inhibitors of γ‐Aminobutyric Acid Transporter 1 through Library Screening with MS Binding Assays.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2488, doi. 10.1002/cmdc.201800556

By:

Huber, Simone K.;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

Selective Optimization of Pranlukast to Farnesoid X Receptor Modulators.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2530, doi. 10.1002/cmdc.201800549

By:

Schierle, Simone;
Schmidt, Jurema;
Kaiser, Astrid;
Merk, Daniel

Publication type:

Article

Gram‐Positive and Gram‐Negative Antibiotic Activity of Asymmetric and Monomeric Robenidine Analogues.

Published in:

ChemMedChem, 2018, v. 13, n. 23, p. 2573, doi. 10.1002/cmdc.201800463

By:

Russell, Cecilia C.;
Stevens, Andrew;
Pi, Hongfei;
Khazandi, Manouchehr;
Ogunniyi, Abiodun D.;
Young, Kelly A.;
Baker, Jennifer R.;
McCluskey, Siobhann N.;
Page, Stephen W.;
Trott, Darren J.;
McCluskey, Adam

Publication type:

Article