Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 21

Results: 10

Front Cover: Discovery of Vilaprisan (BAY 1002670): A Highly Potent and Selective Progesterone Receptor Modulator Optimized for Gynecologic Therapies (ChemMedChem 21/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2250, doi. 10.1002/cmdc.201800681

By:

Möller, Carsten;
Bone, Wilhelm;
Cleve, Arwed;
Klar, Ulrich;
Rotgeri, Andrea;
Rottmann, Antje;
Schultze‐Mosgau, Marcus‐Hillert;
Wagenfeld, Andrea;
Schwede, Wolfgang

Publication type:

Article

In Vivo Anticancer Activity of a Nontoxic Inert Phenolato Titanium Complex: High Efficacy on Solid Tumors Alone and Combined with Platinum Drugs.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2290, doi. 10.1002/cmdc.201800551

By:

Ganot, Nitzan;
Briaitbard, Ori;
Gammal, Asaad;
Tam, Joseph;
Hochman, Jacob;
Tshuva, Edit Y.

Publication type:

Article

Synthesis, Antiviral Activity, and Structure–Activity Relationship of 1,3‐Benzodioxolyl Pyrrole‐Based Entry Inhibitors Targeting the Phe43 Cavity in HIV‐1 gp120.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2332, doi. 10.1002/cmdc.201800534

By:

Curreli, Francesca;
Belov, Dmitry S.;
Ahmed, Shahad;
Ramesh, Ranjith R.;
Kurkin, Alexander V.;
Altieri, Andrea;
Debnath, Asim K.

Publication type:

Article

Ectonucleotidase Inhibitory and Redox Activity of Imidazole‐Based Organic Salts and Ionic Liquids.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2297, doi. 10.1002/cmdc.201800520

By:

Boldescu, Veaceslav;
Sucman, Natalia;
Hassan, Sidra;
Iqbal, Jamshed;
Neamtu, Mariana;
Lecka, Joanna;
Sévigny, Jean;
Prodius, Denis;
Macaev, Fliur

Publication type:

Article

Disaccharide‐Based Anionic Amphiphiles as Potent Inhibitors of Lipopolysaccharide‐Induced Inflammation.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2317, doi. 10.1002/cmdc.201800505

By:

Borio, Alessio;
Holgado, Aurora;
Garate, Jose Antonio;
Beyaert, Rudi;
Heine, Holger;
Zamyatina, Alla

Publication type:

Article

Symmetrical Diamidates as a Class of Phosphate Prodrugs to Deliver the 5′‐Monophosphate Forms of Anticancer Nucleoside Analogues.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2305, doi. 10.1002/cmdc.201800504

By:

Slusarczyk, Magdalena;
Ferrari, Valentina;
Serpi, Michaela;
Gönczy, Blanka;
Balzarini, Jan;
McGuigan, Christopher

Publication type:

Article

Discovery of Vilaprisan (BAY 1002670): A Highly Potent and Selective Progesterone Receptor Modulator Optimized for Gynecologic Therapies.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2271, doi. 10.1002/cmdc.201800487

By:

Möller, Carsten;
Bone, Wilhelm;
Cleve, Arwed;
Klar, Ulrich;
Rotgeri, Andrea;
Rottmann, Antje;
Schultze‐Mosgau, Marcus‐Hillert;
Wagenfeld, Andrea;
Schwede, Wolfgang

Publication type:

Article

An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2251, doi. 10.1002/cmdc.201800447

By:

Fortunato, Serena;
Bononi, Giulia;
Granchi, Carlotta;
Minutolo, Filippo

Publication type:

Article

Design and Synthesis of Bioisosteres of Acylhydrazones as Stable Inhibitors of the Aspartic Protease Endothiapepsin.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2266, doi. 10.1002/cmdc.201800446

By:

Jumde, Varsha R.;
Mondal, Milon;
Gierse, Robin M.;
Unver, M. Yagiz;
Magari, Francesca;
van Lier, Roos C. W.;
Heine, Andreas;
Klebe, Gerhard;
Hirsch, Anna K. H.

Publication type:

Article

MetScore: Site of Metabolism Prediction Beyond Cytochrome P450 Enzymes.

Published in:

ChemMedChem, 2018, v. 13, n. 21, p. 2281, doi. 10.1002/cmdc.201800309

By:

Finkelmann, Arndt R.;
Goldmann, Daria;
Schneider, Gisbert;
Göller, Andreas H.

Publication type:

Article