Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 2

Results: 11

Front Cover: [<italic>Carboxyl</italic>‐<sup>11</sup>C]Labelling of Four High‐Affinity cPLA2α Inhibitors and Their Evaluation as Radioligands in Mice by Positron Emission Tomography (ChemMedChem 2/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 127, doi. 10.1002/cmdc.201800029

By:

Fisher, Martin J.;
McMurray, Lindsay;
Lu, Shuiyu;
Morse, Cheryl L.;
Liow, Jeih‐San;
Zoghbi, Sami S.;
Kowalski, Aneta;
Tye, George L.;
Innis, Robert B.;
Aigbirhio, Franklin I.;
Pike, Victor W.

Publication type:

Article

Corrigendum: Inhibitor Selectivity for Cyclin‐Dependent Kinase 7: A Structural, Thermodynamic, and Modelling Study.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 207, doi. 10.1002/cmdc.201700826

By:

Hazel, Pascale;
Kroll, Sebastian H. B.;
Bondke, Alexander;
Barbazanges, Marion;
Patel, Hetal;
Fuchter, Matthew J.;
Coombes, R. Charles;
Ali, Simak;
Barrett, Anthony G. M.;
Freemont, Paul S.

Publication type:

Article

Monosaccharide Derivatives with Low‐Nanomolar Lectin Affinity and High Selectivity Based on Combined Fluorine–Amide, Phenyl–Arginine, Sulfur–π, and Halogen Bond Interactions.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 133, doi. 10.1002/cmdc.201700744

By:

Zetterberg, Fredrik R.;
Peterson, Kristoffer;
Johnsson, Richard E.;
Brimert, Thomas;
Håkansson, Maria;
Logan, Derek T.;
Leffler, Hakon;
Nilsson, Ulf J.

Publication type:

Article

Inhibitors against Fungal Cell Wall Remodeling Enzymes.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 128, doi. 10.1002/cmdc.201700720

By:

Delso, Ignacio;
Valero‐Gonzalez, Jessika;
Gomollón‐Bel, Fernando;
Castro‐López, Jorge;
Fang, Wenxia;
Navratilova, Iva;
van Aalten, Daan M. F.;
Tejero, Tomás;
Merino, Pedro;
Hurtado‐Guerrero, Ramon

Publication type:

Article

Synthesis of α‐Branched Acyclic Nucleoside Phosphonates as Potential Inhibitors of Bacterial Adenylate Cyclases.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 199, doi. 10.1002/cmdc.201700715

By:

Frydrych, Jan;
Skácel, Jan;
Šmídková, Markéta;
Mertlíková‐Kaiserová, Helena;
Dračínský, Martin;
Gnanasekaran, Ramachandran;
Lepšík, Martin;
Soto‐Velasquez, Monica;
Watts, Val J.;
Janeba, Zlatko

Publication type:

Article

[<italic>Carboxyl</italic>‐<sup>11</sup>C]Labelling of Four High‐Affinity cPLA2α Inhibitors and Their Evaluation as Radioligands in Mice by Positron Emission Tomography.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 138, doi. 10.1002/cmdc.201700697

By:

Fisher, Martin J.;
McMurray, Lindsay;
Lu, Shuiyu;
Morse, Cheryl L.;
Liow, Jeih‐San;
Zoghbi, Sami S.;
Kowalski, Aneta;
Tye, George L.;
Innis, Robert B.;
Aigbirhio, Franklin I.;
Pike, Victor W.

Publication type:

Article

A Novel Prodrug of a γ‐Glutamylcyclotransferase Inhibitor Suppresses Cancer Cell Proliferation in vitro and Inhibits Tumor Growth in a Xenograft Mouse Model of Prostate Cancer.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 155, doi. 10.1002/cmdc.201700660

By:

Ii, Hiromi;
Yoshiya, Taku;
Nakata, Susumu;
Taniguchi, Keiko;
Hidaka, Koushi;
Tsuda, Shugo;
Mochizuki, Masayoshi;
Nishiuchi, Yuji;
Tsuda, Yuko;
Ito, Kosei;
Kageyama, Susumu;
Yoshiki, Tatsuhiro

Publication type:

Article

Anticancer Properties of Halogenated Pyrrolo[3,2‐<italic>d</italic>]pyrimidines with Decreased Toxicity via N5 Substitution.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 178, doi. 10.1002/cmdc.201700641

By:

Cawrse, Brian M.;
Lapidus, Rena S.;
Cooper, Brandon;
Choi, Eun Yong;
Seley‐Radtke, Katherine L.

Publication type:

Article

Synthetic Indolactam V Analogues as Inhibitors of PAR2‐Induced Calcium Mobilization in Triple‐Negative Breast Cancer Cells.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 147, doi. 10.1002/cmdc.201700640

By:

Stein, Jan;
Stahn, Sonja;
Neudörfl, Jörg‐M.;
Sperlich, Julia;
Schmalz, Hans‐Günther;
Teusch, Nicole

Publication type:

Article

Discovery and Mechanistic Elucidation of a Class of Protein Disulfide Isomerase Inhibitors for the Treatment of Glioblastoma.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 164, doi. 10.1002/cmdc.201700629

By:

Kyani, Anahita;
Tamura, Shuzo;
Yang, Suhui;
Shergalis, Andrea;
Samanta, Soma;
Kuang, Yuting;
Ljungman, Mats;
Neamati, Nouri

Publication type:

Article

Synthesis and Evaluation of <italic>N</italic>‐Phenylpyrrolamides as DNA Gyrase B Inhibitors.

Published in:

ChemMedChem, 2018, v. 13, n. 2, p. 186, doi. 10.1002/cmdc.201700549

By:

Durcik, Martina;
Tammela, Päivi;
Barančoková, Michaela;
Tomašič, Tihomir;
Ilaš, Janez;
Kikelj, Danijel;
Zidar, Nace

Publication type:

Article