Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 16

Results: 15

Cover Feature: Design and Synthesis of Pyrophosphate‐Targeting Vancomycin Derivatives for Combating Vancomycin‐Resistant Enterococci (ChemMedChem 16/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1618, doi. 10.1002/cmdc.201800522

By:

Guan, Dongliang;
Chen, Feifei;
Faridoon;
Liu, Junjie;
Li, Jian;
Lan, Lefu;
Huang, Wei

Publication type:

Article

Front Cover: Deciphering Specificity Determinants for FR900359‐Derived Gqα Inhibitors Based on Computational and Structure–Activity Studies (ChemMedChem 16/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1617, doi. 10.1002/cmdc.201800521

By:

Reher, Raphael;
Kühl, Toni;
Annala, Suvi;
Benkel, Tobias;
Kaufmann, Desireé;
Nubbemeyer, Britta;
Odhiambo, Justin Patrick;
Heimer, Pascal;
Bäuml, Charlotte Anneke;
Kehraus, Stefan;
Crüsemann, Max;
Kostenis, Evi;
Tietze, Daniel;
König, Gabriele M.;
Imhof, Diana

Publication type:

Article

NVP‐BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1629, doi. 10.1002/cmdc.201800398

By:

Tröster, Alix;
Heinzlmeir, Stephanie;
Berger, Benedict‐Tilman;
Gande, Santosh L.;
Saxena, Krishna;
Sreeramulu, Sridhar;
Linhard, Verena;
Nasiri, Amir H.;
Bolte, Michael;
Müller, Susanne;
Kuster, Bernhard;
Médard, Guillaume;
Kudlinzki, Denis;
Schwalbe, Harald

Publication type:

Article

Automated Synthesis of (rac)‐, (R)‐, and (S)‐[18F]Epifluorohydrin and Their Application for Developing PET Radiotracers Containing a 3‐[18F]Fluoro‐2‐hydroxypropyl Moiety.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1723, doi. 10.1002/cmdc.201800359

By:

Fujinaga, Masayuki;
Ohkubo, Takayuki;
Yamasaki, Tomoteru;
Zhang, Yiding;
Mori, Wakana;
Hanyu, Masayuki;
Kumata, Katsushi;
Hatori, Akiko;
Xie, Lin;
Nengaki, Nobuki;
Zhang, Ming‐Rong

Publication type:

Article

Differentiating Antiproliferative and Chemopreventive Modes of Activity for Electron‐Deficient Aryl Isothiocyanates against Human MCF‐7 Cells.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1695, doi. 10.1002/cmdc.201800348

By:

Anderson, Ruthellen H.;
Lensing, Cody J.;
Forred, Benjamin J.;
Amolins, Michael W.;
Aegerter, Cassandra L.;
Vitiello, Peter F.;
Mays, Jared R.

Publication type:

Article

A Compact and Synthetically Accessible Fluorine‐18 Labelled Cyclooctyne Prosthetic Group for Labelling of Biomolecules by Copper‐Free Click Chemistry.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1625, doi. 10.1002/cmdc.201800334

By:

Murrell, Emily;
Kovacs, Michael S.;
Luyt, Leonard G.

Publication type:

Article

Deciphering Specificity Determinants for FR900359‐Derived Gqα Inhibitors Based on Computational and Structure–Activity Studies.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1634, doi. 10.1002/cmdc.201800304

By:

Reher, Raphael;
Kühl, Toni;
Annala, Suvi;
Benkel, Tobias;
Kaufmann, Desireé;
Nubbemeyer, Britta;
Odhiambo, Justin Patrick;
Heimer, Pascal;
Bäuml, Charlotte Anneke;
Kehraus, Stefan;
Crüsemann, Max;
Kostenis, Evi;
Tietze, Daniel;
König, Gabriele M.;
Imhof, Diana

Publication type:

Article

Tertiary‐Amine‐Based Inhibitors of the Astacin Protease Meprin α.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1619, doi. 10.1002/cmdc.201800300

By:

Tan, Kathrin;
Jäger, Christian;
Schlenzig, Dagmar;
Schilling, Stephan;
Buchholz, Mirko;
Ramsbeck, Daniel

Publication type:

Article

A Minimalist Approach to the Design of Complexity‐Enriched Bioactive Small Molecules: Discovery of Phenanthrenoid Mimics as Antiproliferative Agents.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1732, doi. 10.1002/cmdc.201800295

By:

Alonso, Fernando;
Quezada, María Josefina;
Gola, Gabriel F.;
Richmond, Victoria;
Cabrera, Gabriela M.;
Barquero, Andrea A.;
Ramírez, Javier A.

Publication type:

Article

Methinylogation Approach in Chiral Pharmacophore Design: from Alkynyl‐ to Allenyl‐carbinol Warheads against Tumor Cells.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1711, doi. 10.1002/cmdc.201800284

By:

Listunov, Dymytrii;
Joly, Etienne;
Duhayon, Carine;
Saffon‐Merceron, Nathalie;
Fabing, Isabelle;
Génisson, Yves;
Maraval, Valérie;
Chauvin, Remi

Publication type:

Article

Hydroxypyridonecarboxylic Acids as Inhibitors of Human Cytomegalovirus pUL89 Endonuclease.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1658, doi. 10.1002/cmdc.201800283

By:

Kankanala, Jayakanth;
Wang, Yan;
Geraghty, Robert J.;
Wang, Zhengqiang

Publication type:

Article

Design and Synthesis of Pyrophosphate‐Targeting Vancomycin Derivatives for Combating Vancomycin‐Resistant Enterococci.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1644, doi. 10.1002/cmdc.201800252

By:

Guan, Dongliang;
Chen, Feifei;
Faridoon;
Liu, Junjie;
Li, Jian;
Lan, Lefu;
Huang, Wei

Publication type:

Article

Structure‐Based Design of a Monosaccharide Ligand Targeting Galectin‐8.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1664, doi. 10.1002/cmdc.201800224

By:

Bohari, Mohammad H.;
Yu, Xing;
Kishor, Chandan;
Patel, Brijesh;
Go, Rob Marc;
Eslampanah Seyedi, Hadieh A.;
Vinik, Yaron;
Grice, I. Darren;
Zick, Yehiel;
Blanchard, Helen

Publication type:

Article

Development of Potent Pyrazolopyrimidinone‐Based WEE1 Inhibitors with Limited Single‐Agent Cytotoxicity for Cancer Therapy.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1681, doi. 10.1002/cmdc.201800188

By:

Matheson, Christopher J.;
Casalvieri, Kimberly A.;
Backos, Donald S.;
Reigan, Philip

Publication type:

Article

Design, Synthesis, Biological Activity, and Structural Analysis of Lactam‐Constrained PTPRJ Agonist Peptides.

Published in:

ChemMedChem, 2018, v. 13, n. 16, p. 1673, doi. 10.1002/cmdc.201800147

By:

Sala, Marina;
Spensiero, Antonia;
Scala, Maria Carmina;
Pepe, Giacomo;
Bilotta, Anna;
Paduano, Francesco;
D'Agostino, Sabrina;
Lanzillotta, Delia;
Bertamino, Alessia;
Novellino, Ettore;
Trapasso, Francesco;
Gomez‐Monterrey, Isabel M.;
Campiglia, Pietro

Publication type:

Article

Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 16

Cover Feature: Design and Synthesis of Pyrophosphate‐Targeting Vancomycin Derivatives for Combating Vancomycin‐Resistant Enterococci (ChemMedChem 16/2018).

Front Cover: Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies (ChemMedChem 16/2018).

NVP‐BHG712: Effects of Regioisomers on the Affinity and Selectivity toward the EPHrin Family.

Automated Synthesis of (rac)‐, (R)‐, and (S)‐[<sup>18</sup>F]Epifluorohydrin and Their Application for Developing PET Radiotracers Containing a 3‐[<sup>18</sup>F]Fluoro‐2‐hydroxypropyl Moiety.

Differentiating Antiproliferative and Chemopreventive Modes of Activity for Electron‐Deficient Aryl Isothiocyanates against Human MCF‐7 Cells.

A Compact and Synthetically Accessible Fluorine‐18 Labelled Cyclooctyne Prosthetic Group for Labelling of Biomolecules by Copper‐Free Click Chemistry.

Deciphering Specificity Determinants for FR900359‐Derived G<sub>q</sub>α Inhibitors Based on Computational and Structure–Activity Studies.

Tertiary‐Amine‐Based Inhibitors of the Astacin Protease Meprin α.

A Minimalist Approach to the Design of Complexity‐Enriched Bioactive Small Molecules: Discovery of Phenanthrenoid Mimics as Antiproliferative Agents.

Methinylogation Approach in Chiral Pharmacophore Design: from Alkynyl‐ to Allenyl‐carbinol Warheads against Tumor Cells.

Hydroxypyridonecarboxylic Acids as Inhibitors of Human Cytomegalovirus pUL89 Endonuclease.

Design and Synthesis of Pyrophosphate‐Targeting Vancomycin Derivatives for Combating Vancomycin‐Resistant Enterococci.

Structure‐Based Design of a Monosaccharide Ligand Targeting Galectin‐8.

Development of Potent Pyrazolopyrimidinone‐Based WEE1 Inhibitors with Limited Single‐Agent Cytotoxicity for Cancer Therapy.

Design, Synthesis, Biological Activity, and Structural Analysis of Lactam‐Constrained PTPRJ Agonist Peptides.