Works matching IS 18607179 AND DT 2018 AND VI 13 AND IP 15

Results: 15

Cover Feature: Development of Novel Inhibitors for Histone Methyltransferase SET7/9 based on Cyproheptadine (ChemMedChem 15/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1489, doi. 10.1002/cmdc.201800495

By:

Hirano, Tomoya;
Fujiwara, Takashi;
Niwa, Hideaki;
Hirano, Michitake;
Ohira, Kasumi;
Okazaki, Yusuke;
Sato, Shin;
Umehara, Takashi;
Maemoto, Yuki;
Ito, Akihiro;
Yoshida, Minoru;
Kagechika, Hiroyuki

Publication type:

Article

Front Cover: Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of Schistosomiasis (ChemMedChem 15/2018).

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1488, doi. 10.1002/cmdc.201800494

By:

Bayer, Theresa;
Chakrabarti, Alokta;
Lancelot, Julien;
Shaik, Tajith B.;
Hausmann, Kristin;
Melesina, Jelena;
Schmidtkunz, Karin;
Marek, Martin;
Erdmann, Frank;
Schmidt, Matthias;
Robaa, Dina;
Romier, Christophe;
Pierce, Raymond J.;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

Effect of Acylation on the Antimicrobial Activity of Temporin B Analogues.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1549, doi. 10.1002/cmdc.201800289

By:

Avitabile, Concetta;
D'Andrea, Luca Domenico;
D'Aversa, Elisabetta;
Milani, Roberta;
Gambari, Roberto;
Romanelli, Alessandra

Publication type:

Article

1,2,3‐Triazolium‐Based Cationic Amphipathic Peptoid Oligomers Mimicking Antimicrobial Helical Peptides.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1513, doi. 10.1002/cmdc.201800273

By:

Shyam, Radhe;
Charbonnel, Nicolas;
Job, Aurélie;
Blavignac, Christelle;
Forestier, Christiane;
Taillefumier, Claude;
Faure, Sophie

Publication type:

Article

Efficient Synthesis of Immunomodulatory Drug Analogues Enables Exploration of Structure–Degradation Relationships.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1508, doi. 10.1002/cmdc.201800271

By:

Burslem, George M.;
Ottis, Philipp;
Jaime‐Figueroa, Saul;
Morgan, Alicia;
Cromm, Philipp M.;
Toure, Momar;
Crews, Craig M.

Publication type:

Article

Recent Advances in the Development of Indazole‐based Anticancer Agents.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1490, doi. 10.1002/cmdc.201800253

By:

Dong, Jinyun;
Zhang, Qijing;
Wang, Zengtao;
Huang, Guang;
Li, Shaoshun

Publication type:

Article

PET Imaging of T Cells: Target Identification and Feasibility Assessment.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1566, doi. 10.1002/cmdc.201800241

By:

Auberson, Yves P.;
Briard, Emmanuelle;
Rudolph, Bettina;
Kaupmann, Klemens;
Smith, Paul;
Oberhauser, Berndt

Publication type:

Article

Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of Schistosomiasis.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1517, doi. 10.1002/cmdc.201800238

By:

Bayer, Theresa;
Chakrabarti, Alokta;
Lancelot, Julien;
Shaik, Tajith B.;
Hausmann, Kristin;
Melesina, Jelena;
Schmidtkunz, Karin;
Marek, Martin;
Erdmann, Frank;
Schmidt, Matthias;
Robaa, Dina;
Romier, Christophe;
Pierce, Raymond J.;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

Development of Novel Inhibitors for Histone Methyltransferase SET7/9 based on Cyproheptadine.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1530, doi. 10.1002/cmdc.201800233

By:

Hirano, Tomoya;
Fujiwara, Takashi;
Niwa, Hideaki;
Hirano, Michitake;
Ohira, Kasumi;
Okazaki, Yusuke;
Sato, Shin;
Umehara, Takashi;
Maemoto, Yuki;
Ito, Akihiro;
Yoshida, Minoru;
Kagechika, Hiroyuki

Publication type:

Article

Understanding the Rate‐Limiting Step of Glycogenolysis by Using QM/MM Calculations on Human Glycogen Phosphorylase.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1608, doi. 10.1002/cmdc.201800218

By:

Brás, Natércia F.;
Fernandes, Pedro A.;
Ramos, Maria J.

Publication type:

Article

Synthesis and Pharmacological Evaluation of Enantiomerically Pure GluN2B Selective NMDA Receptor Antagonists.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1580, doi. 10.1002/cmdc.201800214

By:

Börgel, Frederik;
Szermerski, Marina;
Schreiber, Julian A.;
Temme, Louisa;
Strutz‐Seebohm, Nathalie;
Lehmkuhl, Kirstin;
Schepmann, Dirk;
Ametamey, Simon M.;
Seebohm, Guiscard;
Schmidt, Thomas J.;
Wünsch, Bernhard

Publication type:

Article

Targeting Serotonin 2A and Adrenergic α<sub>1</sub> Receptors for Ocular Antihypertensive Agents: Discovery of 3,4‐Dihydropyrazino[1,2‐b]indazol‐1(2H)‐one Derivatives.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1597, doi. 10.1002/cmdc.201800199

By:

Furlotti, Guido;
Alisi, Maria Alessandra;
Cazzolla, Nicola;
Ceccacci, Francesca;
Garrone, Beatrice;
Gasperi, Tecla;
La Bella, Angela;
Leonelli, Francesca;
Loreto, Maria Antonietta;
Magarò, Gabriele;
Mangano, Giorgina;
Bettolo, Rinaldo Marini;
Masini, Emanuela;
Miceli, Martina;
Migneco, Luisa Maria;
Vitiello, Marco

Publication type:

Article

A New Class of 1‐Aryl‐5,6‐dihydropyrrolo[2,1‐a]isoquinoline Derivatives as Reversers of P‐Glycoprotein‐Mediated Multidrug Resistance in Tumor Cells.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1588, doi. 10.1002/cmdc.201800177

By:

Nevskaya, Alisa A.;
Matveeva, Maria D.;
Borisova, Tatiana N.;
Niso, Mauro;
Colabufo, Nicola A.;
Boccarelli, Angelina;
Purgatorio, Rosa;
de Candia, Modesto;
Cellamare, Saverio;
Voskressensky, Leonid G.;
Altomare, Cosimo D.

Publication type:

Article

Structure‐Based Design of a Eukaryote‐Selective Antiprotozoal Fluorinated Aminoglycoside.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1541, doi. 10.1002/cmdc.201800166

By:

Kanazawa, Hiroki;
Saavedra, Oscar M.;
Maianti, Juan Pablo;
Young, Simon A.;
Izquierdo, Luis;
Smith, Terry K.;
Hanessian, Stephen;
Kondo, Jiro

Publication type:

Article

Cyclic Hexapeptide Mimics of the LEDGF Integrase Recognition Loop in Complex with HIV‐1 Integrase.

Published in:

ChemMedChem, 2018, v. 13, n. 15, p. 1555, doi. 10.1002/cmdc.201800129

By:

Northfield, Susan E.;
Wielens, Jerome;
Headey, Stephen J.;
Williams‐Noonan, Billy J.;
Mulcair, Mark;
Scanlon, Martin J.;
Parker, Michael W.;
Thompson, Philip E.;
Chalmers, David K.

Publication type:

Article