Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 3

Results: 11

Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 197, doi. 10.1002/cmdc.201600467

By:

Orain, David;
Tasdelen, Engin;
Haessig, Samuel;
Koller, Manuel;
Picard, Anne;
Dubois, Celine;
Lingenhoehl, Kurt;
Desrayaud, Sandrine;
Floersheim, Phillip;
Carcache, David;
Urwyler, Stephan;
Kallen, Joerg;
Mattes, Henri

Publication type:

Article

A Multi-Mitochondrial Anticancer Agent that Selectively Kills Cancer Cells and Overcomes Drug Resistance.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 250, doi. 10.1002/cmdc.201600538

By:

Peng, Yong Bo;
Zhao, Zi Long;
Liu, Teng;
Xie, Guo Jian;
Jin, Cheng;
Deng, Tang Gang;
Sun, Yang;
Li, Xiong;
Hu, Xiao Xiao;
Zhang, Xiao Bing;
Ye, Mao;
Tan, Wei Hong

Publication type:

Article

Metal NHC Complexes with Naphthalimide Ligands as DNA-Interacting Antiproliferative Agents.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 214, doi. 10.1002/cmdc.201600557

By:

Streciwilk, Wojciech;
Terenzi, Alessio;
Misgeld, Rainer;
Frias, Corazon;
Jones, Peter G.;
Prokop, Aram;
Keppler, Bernhard K.;
Ott, Ingo

Publication type:

Article

Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide⋅⋅⋅Heteroarene π-Stacking Interactions and Chalcogen Bonding in the S3 Pocket.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 257, doi. 10.1002/cmdc.201600563

By:

Giroud, Maude;
Ivkovic, Jakov;
Martignoni, Mara;
Fleuti, Marianne;
Trapp, Nils;
Haap, Wolfgang;
Kuglstatter, Andreas;
Benz, Jörg;
Kuhn, Bernd;
Schirmeister, Tanja;
Diederich, François

Publication type:

Article

Induced Europium Circularly Polarized Luminescence Monitors Reversible Drug Binding to Native α<sub>1</sub>-Acid Glycoprotein.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 271, doi. 10.1002/cmdc.201600571

By:

Jennings, Laura;
Waters, Ryan S.;
Pal, Robert;
Parker, David

Publication type:

Article

Phosphatase-Stable Phosphoamino Acid Mimetics That Enhance Binding Affinities with the Polo-Box Domain of Polo-like Kinase 1.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 202, doi. 10.1002/cmdc.201600574

By:

Hymel, David;
Burke, Terrence R.

Publication type:

Article

Discovery of Macrocyclic Pyrimidines as MerTK-Specific Inhibitors.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 207, doi. 10.1002/cmdc.201600589

By:

McIver, Andrew L.;
Zhang, Weihe;
Liu, Qingyang;
Jiang, Xinpeng;
Stashko, Michael A.;
Nichols, James;
Miley, Michael J.;
Norris‐Drouin, Jacqueline;
Machius, Mischa;
DeRyckere, Deborah;
Wood, Edgar;
Graham, Douglas K.;
Earp, H. Shelton;
Kireev, Dmitri;
Frye, Stephen V.;
Wang, Xiaodong

Publication type:

Article

Selenophenes: Introducing a New Element into the Core of Non-Steroidal Estrogen Receptor Ligands.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 235, doi. 10.1002/cmdc.201600593

By:

Zhang, Silong;
Wang, Zhiyong;
Hu, Zhiye;
Li, Changhao;
Tang, Chu;
Carlson, Kathryn E.;
Luo, Junjie;
Dong, Chune;
Katzenellenbogen, John A.;
Huang, Jian;
Zhou, Hai‐Bing

Publication type:

Article

Synthesis of Novel Hybrids of Thymoquinone and Artemisinin with High Activity and Selectivity Against Colon Cancer.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 226, doi. 10.1002/cmdc.201600594

By:

Fröhlich, Tony;
Ndreshkjana, Benardina;
Muenzner, Julienne K.;
Reiter, Christoph;
Hofmeister, Elisabeth;
Mederer, Sandra;
Fatfat, Maamoun;
El‐Baba, Chirine;
Gali‐Muhtasib, Hala;
Schneider‐Stock, Regine;
Tsogoeva, Svetlana B.

Publication type:

Article

Cover Picture: Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist (ChemMedChem 3/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 196, doi. 10.1002/cmdc.201600627

By:

Orain, David;
Tasdelen, Engin;
Haessig, Samuel;
Koller, Manuel;
Picard, Anne;
Dubois, Celine;
Lingenhoehl, Kurt;
Desrayaud, Sandrine;
Floersheim, Phillip;
Carcache, David;
Urwyler, Stephan;
Kallen, Joerg;
Mattes, Henri

Publication type:

Article

Corrigendum: Phosphatase-Stable Phosphoamino Acid Mimetics That Enhance Binding Affinities with the Polo-Box Domain of Polo-like Kinase 1.

Published in:

ChemMedChem, 2017, v. 12, n. 3, p. 278, doi. 10.1002/cmdc.201700019

By:

Hymel, David;
Burke, Terrence R.

Publication type:

Article