Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 22

Results: 11

C2-Modified Sparteine Derivatives Are a New Class of Potentially Long-Acting Sodium Channel Blockers.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1819, doi. 10.1002/cmdc.201700568

By:

Gawali, Vaibhavkumar S.;
Simeonov, Svilen;
Drescher, Martina;
Knott, Thomas;
Scheel, Olaf;
Kudolo, John;
Kählig, Hanspeter;
Hochenegg, Ulla;
Roller, Alexander;
Todt, Hannes;
Maulide, Nuno

Publication type:

Article

Heme Oxygenase Database (HemeOxDB) and QSAR Analysis of Isoform 1 Inhibitors.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1873, doi. 10.1002/cmdc.201700321

By:

Amata, Emanuele;
Marrazzo, Agostino;
Dichiara, Maria;
Modica, Maria N.;
Salerno, Loredana;
Prezzavento, Orazio;
Nastasi, Giovanni;
Rescifina, Antonio;
Romeo, Giuseppe;
Pittalà, Valeria

Publication type:

Article

Sugar-Coated Nanobullet: Growth Inhibition of Cancer Cells Induced by Metformin-Loaded Glyconanoparticles.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1823, doi. 10.1002/cmdc.201700583

By:

Qian, Ruo‐Can;
Lv, Jian;
Li, Hao‐Wen;
Long, Yi‐Tao

Publication type:

Article

Synthesis and Determination of Lipophilicity, Anticonvulsant Activity, and Preliminary Safety of 3-Substituted and 3-Unsubstituted N-[(4-Arylpiperazin-1-yl)alkyl]pyrrolidine-2,5-dione Derivatives.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1848, doi. 10.1002/cmdc.201700539

By:

Rybka, Sabina;
Obniska, Jolanta;
Żmudzki, Paweł;
Koczurkiewicz, Paulina;
Wójcik‐Pszczoła, Katarzyna;
Pękala, Elżbieta;
Bryła, Adrian;
Rapacz, Anna

Publication type:

Article

Potent Pyrimidine and Pyrrolopyrimidine Inhibitors of Testis-Specific Serine/Threonine Kinase 2 (TSSK2).

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1857, doi. 10.1002/cmdc.201700503

By:

Hawkinson, Jon E.;
Sinville, Rondedrick;
Mudaliar, Deepti;
Shetty, Jagathpala;
Ward, Timothy;
Herr, John C.;
Georg, Gunda I.

Publication type:

Article

Synthesis and in vitro Biological Evaluation of Ferrocenyl Side-Chain-Functionalized Paclitaxel Derivatives.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1882, doi. 10.1002/cmdc.201700576

By:

Plażuk, Damian;
Wieczorek, Anna;
Ciszewski, Wojciech M.;
Kowalczyk, Karolina;
Błauż, Andrzej;
Pawlędzio, Sylwia;
Makal, Anna;
Eurtivong, Chatchakorn;
Arabshahi, Homayon J.;
Reynisson, Jóhannes;
Hartinger, Christian G.;
Rychlik, Błażej

Publication type:

Article

Minor Structural Variations of Small Molecules Tune Regulatory Activities toward Pathological Factors in Alzheimer's Disease.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1828, doi. 10.1002/cmdc.201700456

By:

Beck, Michael W.;
Derrick, Jeffrey S.;
Suh, Jong‐Min;
Kim, Mingeun;
Korshavn, Kyle J.;
Kerr, Richard A.;
Cho, Woo Jong;
Larsen, Scott D.;
Ruotolo, Brandon T.;
Ramamoorthy, Ayyalusamy;
Lim, Mi Hee

Publication type:

Article

Front Cover: Minor Structural Variations of Small Molecules Tune Regulatory Activities toward Pathological Factors in Alzheimer's Disease (ChemMedChem 22/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1818, doi. 10.1002/cmdc.201700711

By:

Beck, Michael W.;
Derrick, Jeffrey S.;
Suh, Jong‐Min;
Kim, Mingeun;
Korshavn, Kyle J.;
Kerr, Richard A.;
Cho, Woo Jong;
Larsen, Scott D.;
Ruotolo, Brandon T.;
Ramamoorthy, Ayyalusamy;
Lim, Mi Hee

Publication type:

Article

Computational Macrocyclization: From de novo Macrocycle Generation to Binding Affinity Estimation.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1866, doi. 10.1002/cmdc.201700478

By:

Wagner, Vincent;
Jantz, Linda;
Briem, Hans;
Sommer, Kai;
Rarey, Matthias;
Christ, Clara D.

Publication type:

Article

Structure-Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1893, doi. 10.1002/cmdc.201700427

By:

Franchini, Silvia;
Sorbi, Claudia;
Battisti, Umberto Maria;
Tait, Annalisa;
Bencheva, Leda Ivanova;
Cichero, Elena;
Fossa, Paola;
Cilia, Antonio;
Prezzavento, Orazio;
Ronsisvalle, Simone;
Aricò, Giuseppina;
Benassi, Luisa;
Vaschieri, Cristina;
Azzoni, Paola;
Magnoni, Cristina;
Brasili, Livio

Publication type:

Article

Functional N-Formyl Peptide Receptor 2 (FPR2) Antagonists Based on the Ureidopropanamide Scaffold Have Potential To Protect Against Inflammation-Associated Oxidative Stress.

Published in:

ChemMedChem, 2017, v. 12, n. 22, p. 1839, doi. 10.1002/cmdc.201700429

By:

Stama, Madia L.;
Lacivita, Enza;
Kirpotina, Liliya N.;
Niso, Mauro;
Perrone, Roberto;
Schepetkin, Igor A.;
Quinn, Mark T.;
Leopoldo, Marcello

Publication type:

Article