Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 18

Results: 10

Rational Design, Development, and Stability Assessment of a Macrocyclic Four-Hydroxamate-Bearing Bifunctional Chelating Agent for <sup>89</sup>Zr.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1555, doi. 10.1002/cmdc.201700377

By:

Seibold, Uwe;
Wängler, Björn;
Wängler, Carmen

Publication type:

Article

Reducing the Flexibility of Type II Dehydroquinase for Inhibition: A Fragment-Based Approach and Molecular Dynamics Study.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1512, doi. 10.1002/cmdc.201700396

By:

Peón, Antonio;
Robles, Adrián;
Blanco, Beatriz;
Convertino, Marino;
Thompson, Paul;
Hawkins, Alastair R.;
Caflisch, Amedeo;
González‐Bello, Concepción

Publication type:

Article

Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1542, doi. 10.1002/cmdc.201700340

By:

Pirali, Tracey;
Ciraolo, Elisa;
Aprile, Silvio;
Massarotti, Alberto;
Berndt, Alex;
Griglio, Alessia;
Serafini, Marta;
Mercalli, Valentina;
Landoni, Clarissa;
Campa, Carlo Cosimo;
Margaria, Jean Piero;
Silva, Rangel L.;
Grosa, Giorgio;
Sorba, Giovanni;
Williams, Roger;
Hirsch, Emilio;
Tron, Gian Cesare

Publication type:

Article

Characterization of Small-Molecule Scaffolds That Bind to the Shigella Type III Secretion System Protein IpaD.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1534, doi. 10.1002/cmdc.201700348

By:

Dey, Supratim;
Anbanandam, Asokan;
Mumford, Ben E.;
De Guzman, Roberto N.

Publication type:

Article

Front Cover: Targeting of a Helix-Loop-Helix Transcriptional Regulator by a Short Helical Peptide (ChemMedChem 18/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1480, doi. 10.1002/cmdc.201700537

By:

Roschger, Cornelia;
Neukirchen, Saskia;
Elsässer, Brigitta;
Schubert, Mario;
Maeding, Nicole;
Verwanger, Thomas;
Krammer, Barbara;
Cabrele, Chiara

Publication type:

Article

Silicon Phthalocyanines Axially Disubstituted with Erlotinib toward Small-Molecular-Target-Based Photodynamic Therapy.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1504, doi. 10.1002/cmdc.201700384

By:

Chen, Juan‐Juan;
Huang, Yi‐Zhen;
Song, Mei‐Ru;
Zhang, Zhi‐Hong;
Xue, Jin‐Ping

Publication type:

Article

Application of the Pentafluorosulfanyl Group as a Bioisosteric Replacement.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1481, doi. 10.1002/cmdc.201700356

By:

Sowaileh, Munia F.;
Hazlitt, Robert A.;
Colby, David A.

Publication type:

Article

Structure-Guided Design of Peptides as Tools to Probe the Protein-Protein Interaction between Cullin-2 and Elongin BC Substrate Adaptor in Cullin RING E3 Ubiquitin Ligases.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1491, doi. 10.1002/cmdc.201700359

By:

Cardote, Teresa A. F.;
Ciulli, Alessio

Publication type:

Article

Targeting of a Helix-Loop-Helix Transcriptional Regulator by a Short Helical Peptide.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1497, doi. 10.1002/cmdc.201700305

By:

Roschger, Cornelia;
Neukirchen, Saskia;
Elsässer, Brigitta;
Schubert, Mario;
Maeding, Nicole;
Verwanger, Thomas;
Krammer, Barbara;
Cabrele, Chiara

Publication type:

Article

Design and Synthesis of 4-Alkylidene-β-lactams: Benzyl- and Phenethyl-carbamates as Key Fragments to Switch on Antibacterial Activity.

Published in:

ChemMedChem, 2017, v. 12, n. 18, p. 1525, doi. 10.1002/cmdc.201700307

By:

Giacomini, Daria;
Martelli, Giulia;
Piccichè, Miriam;
Calaresu, Enrico;
Cocuzza, Clementina Elvezia;
Musumeci, Rosario

Publication type:

Article