Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 16

Results: 22

Identification of Transthyretin Fibril Formation Inhibitors Using Structure-Based Virtual Screening.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1327, doi. 10.1002/cmdc.201700051

By:

Ortore, Gabriella;
Martinelli, Adriano

Publication type:

Article

Investigating Structural Requirements for the Antiproliferative Activity of Biphenyl Nicotinamides.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1380, doi. 10.1002/cmdc.201700365

By:

Majellaro, Maria;
Stefanachi, Angela;
Tardia, Piero;
Vicenti, Chiara;
Boccarelli, Angelina;
Pannunzio, Alessandra;
Campanella, Federica;
Coluccia, Mauro;
Denora, Nunzio;
Leonetti, Francesco;
de Candia, Modesto;
Altomare, Cosimo Damiano;
Cellamare, Saverio

Publication type:

Article

Discovery of wtRET and V804MRET Inhibitors: From Hit to Lead.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1390, doi. 10.1002/cmdc.201700243

By:

Mologni, Luca;
Dalla Via, Martina;
Chilin, Adriana;
Palumbo, Manlio;
Marzaro, Giovanni

Publication type:

Article

Cannabinoid Type 1 Receptor (CB1) Ligands with Therapeutic Potential for Withdrawal Syndrome in Chemical Dependents of Cannabis sativa.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1408, doi. 10.1002/cmdc.201700129

By:

Ferreira, Jaderson V.;
Chaves, Gisele A.;
Marino, Bianca L. B.;
Sousa, Kessia P. A.;
Souza, Lucilene R.;
Brito, Maiara F. B.;
Teixeira, Hueldem R. C.;
da Silva, Carlos H. T. P.;
Santos, Cleydson B. R.;
Hage‐Melim, Lorane I. S.

Publication type:

Article

Identification of Breast Cancer Inhibitors Specific for G Protein-Coupled Estrogen Receptor (GPER)-Expressing Cells.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1279, doi. 10.1002/cmdc.201700145

By:

Aiello, Francesca;
Carullo, Gabriele;
Giordano, Francesca;
Spina, Elena;
Nigro, Alessandra;
Garofalo, Antonio;
Tassini, Sabrina;
Costantino, Gabriele;
Vincetti, Paolo;
Bruno, Agostino;
Radi, Marco

Publication type:

Article

Novel, Selective, and Developable Dopamine D3 Antagonists with a Modified 'Amino' Region.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1254, doi. 10.1002/cmdc.201700148

By:

Micheli, Fabrizio

Publication type:

Article

A Molecular Dynamics-Shared Pharmacophore Approach to Boost Early-Enrichment Virtual Screening: A Case Study on Peroxisome Proliferator-Activated Receptor α.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1399, doi. 10.1002/cmdc.201600526

By:

Perricone, Ugo;
Wieder, Marcus;
Seidel, Thomas;
Langer, Thierry;
Padova, Alessandro;
Almerico, Anna Maria;
Tutone, Marco

Publication type:

Article

Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1349, doi. 10.1002/cmdc.201700282

By:

Pisani, Leonardo;
Catto, Marco;
De Palma, Annalisa;
Farina, Roberta;
Cellamare, Saverio;
Altomare, Cosimo D.

Publication type:

Article

Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1293, doi. 10.1002/cmdc.201700286

By:

Felicetti, Tommaso;
Cannalire, Rolando;
Burali, Maria Sole;
Massari, Serena;
Manfroni, Giuseppe;
Barreca, Maria Letizia;
Tabarrini, Oriana;
Schindler, Bryan D.;
Sabatini, Stefano;
Kaatz, Glenn W.;
Cecchetti, Violetta

Publication type:

Article

Identification of α7 Nicotinic Acetylcholine Receptor Silent Agonists Based on the Spirocyclic Quinuclidine-Δ2-Isoxazoline Scaffold: Synthesis and Electrophysiological Evaluation.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1335, doi. 10.1002/cmdc.201700162

By:

Quadri, Marta;
Matera, Carlo;
Silnović, Almin;
Pismataro, Maria Chiara;
Horenstein, Nicole A.;
Stokes, Clare;
Papke, Roger L.;
Dallanoce, Clelia

Publication type:

Article

Cover Picture: Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues (ChemMedChem 16/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1224, doi. 10.1002/cmdc.201700470

By:

Felicetti, Tommaso;
Cannalire, Rolando;
Burali, Maria Sole;
Massari, Serena;
Manfroni, Giuseppe;
Barreca, Maria Letizia;
Tabarrini, Oriana;
Schindler, Bryan D.;
Sabatini, Stefano;
Kaatz, Glenn W.;
Cecchetti, Violetta

Publication type:

Article

Inside Cover: 2,6-Difluorobenzamide Inhibitors of Bacterial Cell Division Protein FtsZ: Design, Synthesis, and Structure-Activity Relationships (ChemMedChem 16/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1225, doi. 10.1002/cmdc.201700471

By:

Straniero, Valentina;
Zanotto, Carlo;
Straniero, Letizia;
Casiraghi, Andrea;
Duga, Stefano;
Radaelli, Antonia;
De Giuli Morghen, Carlo;
Valoti, Ermanno

Publication type:

Article

Back Cover: Identification of α7 Nicotinic Acetylcholine Receptor Silent Agonists Based on the Spirocyclic Quinuclidine-Δ2-Isoxazoline Scaffold: Synthesis and Electrophysiological Evaluation (ChemMedChem 16/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1417, doi. 10.1002/cmdc.201700472

By:

Quadri, Marta;
Matera, Carlo;
Silnović, Almin;
Pismataro, Maria Chiara;
Horenstein, Nicole A.;
Stokes, Clare;
Papke, Roger L.;
Dallanoce, Clelia

Publication type:

Article

Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1359, doi. 10.1002/cmdc.201700040

By:

Madia, Valentina Noemi;
Benedetti, Rosaria;
Barreca, Maria Letizia;
Ngo, Liza;
Pescatori, Luca;
Messore, Antonella;
Pupo, Giovanni;
Saccoliti, Francesco;
Valente, Sergio;
Mai, Antonello;
Scipione, Luigi;
Zheng, Yujun George;
Tintori, Cristina;
Botta, Maurizio;
Cecchetti, Violetta;
Altucci, Lucia;
Di Santo, Roberto;
Costi, Roberta

Publication type:

Article

Structure-Activity Relationship Studies on 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Multidrug Resistance Reversers.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1369, doi. 10.1002/cmdc.201700239

By:

Teodori, Elisabetta;
Dei, Silvia;
Bartolucci, Gianluca;
Perrone, Maria Grazia;
Manetti, Dina;
Romanelli, Maria Novella;
Contino, Marialessandra;
Colabufo, Nicola Antonio

Publication type:

Article

A Small-Molecule Inhibitor of Prion Replication and Mutant Prion Protein Toxicity.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1286, doi. 10.1002/cmdc.201700302

By:

Massignan, Tania;
Sangiovanni, Valeria;
Biggi, Silvia;
Stincardini, Claudia;
Elezgarai, Saioa R.;
Maietta, Giulia;
Andreev, Ivan A.;
Ratmanova, Nina K.;
Belov, Dmitry S.;
Lukyanenko, Evgeny R.;
Belov, Grigory M.;
Barreca, Maria Letizia;
Altieri, Andrea;
Kurkin, Alexander V.;
Biasini, Emiliano

Publication type:

Article

Repurposing of Human Kinase Inhibitors in Neglected Protozoan Diseases.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1235, doi. 10.1002/cmdc.201700259

By:

Dichiara, Maria;
Marrazzo, Agostino;
Prezzavento, Orazio;
Collina, Simona;
Rescifina, Antonio;
Amata, Emanuele

Publication type:

Article

Bridging Pharmaceutical Chemistry with Drug and Nanoparticle Targeting to Investigate the Role of the 18-kDa Translocator Protein TSPO.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1261, doi. 10.1002/cmdc.201700322

By:

Iacobazzi, Rosa Maria;
Lopalco, Antonio;
Cutrignelli, Annalisa;
Laquintana, Valentino;
Lopedota, Angela;
Franco, Massimo;
Denora, Nunzio

Publication type:

Article

Comparison of the Human A2A Adenosine Receptor Recognition by Adenosine and Inosine: New Insight from Supervised Molecular Dynamics Simulations.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1319, doi. 10.1002/cmdc.201700200

By:

Deganutti, Giuseppe;
Welihinda, Ajith;
Moro, Stefano

Publication type:

Article

2,6-Difluorobenzamide Inhibitors of Bacterial Cell Division Protein FtsZ: Design, Synthesis, and Structure-Activity Relationships.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1303, doi. 10.1002/cmdc.201700201

By:

Straniero, Valentina;
Zanotto, Carlo;
Straniero, Letizia;
Casiraghi, Andrea;
Duga, Stefano;
Radaelli, Antonia;
De Giuli Morghen, Carlo;
Valoti, Ermanno

Publication type:

Article

The XXIV National Meeting in Medicinal Chemistry (NMMC 2016) in Perugia, Italy.

Published in:

2017

By:

Cecchetti, Violetta;
Natalini, Benedetto

Publication type:

Editorial

Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N, N-Dialkyl-2-arylindol-3-ylglyoxylamides.

Published in:

ChemMedChem, 2017, v. 12, n. 16, p. 1275, doi. 10.1002/cmdc.201700220

By:

Costa, Barbara;
Taliani, Sabrina;
Da Pozzo, Eleonora;
Barresi, Elisabetta;
Robello, Marco;
Cavallini, Chiara;
Cosconati, Sandro;
Da Settimo, Federico;
Novellino, Ettore;
Martini, Claudia

Publication type:

Article

Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 16

Identification of Transthyretin Fibril Formation Inhibitors Using Structure-Based Virtual Screening.

Investigating Structural Requirements for the Antiproliferative Activity of Biphenyl Nicotinamides.

Discovery of <sup>wt</sup>RET and <sup>V804M</sup>RET Inhibitors: From Hit to Lead.

Cannabinoid Type 1 Receptor (CB1) Ligands with Therapeutic Potential for Withdrawal Syndrome in Chemical Dependents of Cannabis sativa.

Identification of Breast Cancer Inhibitors Specific for G Protein-Coupled Estrogen Receptor (GPER)-Expressing Cells.

Novel, Selective, and Developable Dopamine D<sub>3</sub> Antagonists with a Modified 'Amino' Region.

A Molecular Dynamics-Shared Pharmacophore Approach to Boost Early-Enrichment Virtual Screening: A Case Study on Peroxisome Proliferator-Activated Receptor α.

Discovery of Potent Dual Binding Site Acetylcholinesterase Inhibitors via Homo- and Heterodimerization of Coumarin-Based Moieties.

Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues.

Identification of α7 Nicotinic Acetylcholine Receptor Silent Agonists Based on the Spirocyclic Quinuclidine-Δ<sup>2</sup>-Isoxazoline Scaffold: Synthesis and Electrophysiological Evaluation.

Cover Picture: Searching for Novel Inhibitors of the S. aureus NorA Efflux Pump: Synthesis and Biological Evaluation of the 3-Phenyl-1,4-benzothiazine Analogues (ChemMedChem 16/2017).

Inside Cover: 2,6-Difluorobenzamide Inhibitors of Bacterial Cell Division Protein FtsZ: Design, Synthesis, and Structure-Activity Relationships (ChemMedChem 16/2017).

Back Cover: Identification of α7 Nicotinic Acetylcholine Receptor Silent Agonists Based on the Spirocyclic Quinuclidine-Δ<sup>2</sup>-Isoxazoline Scaffold: Synthesis and Electrophysiological Evaluation (ChemMedChem 16/2017).

Structure-Activity Relationships on Cinnamoyl Derivatives as Inhibitors of p300 Histone Acetyltransferase.

Structure-Activity Relationship Studies on 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline Derivatives as Multidrug Resistance Reversers.

A Small-Molecule Inhibitor of Prion Replication and Mutant Prion Protein Toxicity.

Repurposing of Human Kinase Inhibitors in Neglected Protozoan Diseases.

Bridging Pharmaceutical Chemistry with Drug and Nanoparticle Targeting to Investigate the Role of the 18-kDa Translocator Protein TSPO.

Comparison of the Human A<sub>2A</sub> Adenosine Receptor Recognition by Adenosine and Inosine: New Insight from Supervised Molecular Dynamics Simulations.

2,6-Difluorobenzamide Inhibitors of Bacterial Cell Division Protein FtsZ: Design, Synthesis, and Structure-Activity Relationships.

The XXIV National Meeting in Medicinal Chemistry (NMMC 2016) in Perugia, Italy.

Residence Time, a New parameter to Predict Neurosteroidogenic Efficacy of Translocator Protein (TSPO) Ligands: the Case Study of N, N-Dialkyl-2-arylindol-3-ylglyoxylamides.