Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 13

Results: 12

Thiazole-Based σ<sub>1</sub> Receptor Ligands: Diversity by Late-Stage C−H Arylation of Thiazoles, Structure-Affinity and Selectivity Relationships, and Molecular Interactions.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1070, doi. 10.1002/cmdc.201700166

By:

Kokornaczyk, Artur K.;
Schepmann, Dirk;
Yamaguchi, Junichiro;
Itami, Kenichiro;
Laurini, Erik;
Fermeglia, Maurizio;
Pricl, Sabrina;
Wünsch, Bernhard

Publication type:

Article

CarbORev-5901: The First Carborane-Based Inhibitor of the 5-Lipoxygenase Pathway.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1081, doi. 10.1002/cmdc.201700309

By:

Kuhnert, Robert;
Sárosi, Menyhárt‐Botond;
George, Sven;
Lönnecke, Peter;
Hofmann, Bettina;
Steinhilber, Dieter;
Murganic, Blagoje;
Mijatovic, Sanja;
Maksimovic‐Ivanic, Danijela;
Hey‐Hawkins, Evamarie

Publication type:

Article

Small Molecule Medicinal Chemistry: Strategies and Technologies. Edited by Werngard Czechtizky and Peter Hamley.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1101, doi. 10.1002/cmdc.201700060

By:

Klein, Christian

Publication type:

Article

Synthesis and Biological Evaluation of Glycyrrhetic Acid Derivatives as Potential VEGFR2 Inhibitors.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1087, doi. 10.1002/cmdc.201700271

By:

Yan, Tian‐Long;
Bai, Li‐Fei;
Zhu, Hai‐Liang;
Zhang, Wei‐Ming;
Lv, Peng‐Cheng

Publication type:

Article

Structural States of RORγt: X-ray Elucidation of Molecular Mechanisms and Binding Interactions for Natural and Synthetic Compounds.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1014, doi. 10.1002/cmdc.201700278

By:

Kallen, Joerg;
Izaac, Aude;
Be, Celine;
Arista, Luca;
Orain, David;
Kaupmann, Klemens;
Guntermann, Christine;
Hoegenauer, Klemens;
Hintermann, Samuel

Publication type:

Article

Synthesis, ADMET Properties, and Biological Evaluation of Benzothiazole Compounds Targeting Chemokine Receptor 2 (CXCR2).

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1045, doi. 10.1002/cmdc.201700229

By:

Mehanna, Wesam E.;
Lu, Tiangong;
Debnath, Bikash;
Lasheen, Deena S.;
Serya, Rabah A. T.;
Abouzid, Khaled A.;
Neamati, Nouri

Publication type:

Article

Design, Synthesis, and Structure-Activity Relationship Analysis of Thiazolo[3,2- a]pyrimidine Derivatives with Anti-inflammatory Activity in Acute Lung Injury.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1022, doi. 10.1002/cmdc.201700175

By:

Chen, Lingfeng;
Jin, Yiyi;
Fu, Weitao;
Xiao, Siyang;
Feng, Chen;
Fang, Bo;
Gu, Yugui;
Li, Chenglong;
Zhao, Yunjie;
Liu, Zhiguo;
Liang, Guang

Publication type:

Article

Cover Picture: Design, Synthesis, and Structure-Activity Relationship Analysis of Thiazolo[3,2- a]pyrimidine Derivatives with Anti-inflammatory Activity in Acute Lung Injury (ChemMedChem 13/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1013, doi. 10.1002/cmdc.201700367

By:

Chen, Lingfeng;
Jin, Yiyi;
Fu, Weitao;
Xiao, Siyang;
Feng, Chen;
Fang, Bo;
Gu, Yugui;
Li, Chenglong;
Zhao, Yunjie;
Liu, Zhiguo;
Liang, Guang

Publication type:

Article

Synthesis, DNA Cleavage Activity, Cytotoxicity, Acetylcholinesterase Inhibition, and Acute Murine Toxicity of Redox-Active Ruthenium(II) Polypyridyl Complexes.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1055, doi. 10.1002/cmdc.201700240

By:

Alatrash, Nagham;
Narh, Eugenia S.;
Yadav, Abhishek;
Kim, Mahn‐Jong;
Janaratne, Thamara;
Gabriel, James;
MacDonnell, Frederick M.

Publication type:

Article

Attrition in the Pharmaceutical Industry - Reasons, Implications, and Pathways Forward. Edited by Alexander Alex, C. John Harris, Dennis A. Smith.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1097, doi. 10.1002/cmdc.201600621

By:

Pellicciari, Roberto

Publication type:

Article

Synthesis and Antineoplastic Evaluation of Mitochondrial Complex II (Succinate Dehydrogenase) Inhibitors Derived from Atpenin A5.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1033, doi. 10.1002/cmdc.201700196

By:

Wang, Hezhen;
Huwaimel, Bader;
Verma, Kshitij;
Miller, James;
Germain, Todd M.;
Kinarivala, Nihar;
Pappas, Dimitri;
Brookes, Paul S.;
Trippier, Paul C.

Publication type:

Article

Synthetic Methods in Drug Discovery, Volumes 1+2. Edited by David C. Blakemore, Paul M. Doyle and Yvette M. Fobian.

Published in:

ChemMedChem, 2017, v. 12, n. 13, p. 1099, doi. 10.1002/cmdc.201600641

By:

Sbardella, Gianluca

Publication type:

Article