Works matching IS 18607179 AND DT 2017 AND VI 12 AND IP 12

Results: 19

Nucleic Acid Templated Reactions for Chemical Biology.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 872, doi. 10.1002/cmdc.201700266

By:

Di Pisa, Margherita;
Seitz, Oliver

Publication type:

Article

Targeting DNA-Dependent Protein Kinase for Cancer Therapy.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 895, doi. 10.1002/cmdc.201700143

By:

Harnor, Suzannah J.;
Brennan, Alfie;
Cano, Céline

Publication type:

Article

Target Deconvolution Efforts on Wnt Pathway Screen Reveal Dual Modulation of Oxidative Phosphorylation and SERCA2.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 917, doi. 10.1002/cmdc.201700028

By:

Casás‐Selves, Matias;
Zhang, Andrew X.;
Dowling, James E.;
Hallén, Stefan;
Kawatkar, Aarti;
Pace, Nicholas J.;
Denz, Christopher R.;
Pontz, Timothy;
Garahdaghi, Farzin;
Cao, Qing;
Sabirsh, Alan;
Thakur, Kumar;
O'Connell, Nichole;
Hu, Jun;
Cornella‐Taracido, Iván;
Weerapana, Eranthie;
Zinda, Michael;
Goodnow, Robert A.;
Castaldi, M. Paola

Publication type:

Article

The 52<sup>nd</sup> International Conference on Medicinal Chemistry (RICT 2016) of the French Medicinal Chemistry Society (SCT) Held in Caen (Normandy).

Published in:

2017

By:

Sapi, Janos;
Van Hijfte, Luc;
Dallemagne, Patrick

Publication type:

Editorial

Lanthanide Complexes in Molecular Magnetic Resonance Imaging and Theranostics.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 883, doi. 10.1002/cmdc.201700210

By:

Lacerda, Sara;
Tóth, Éva

Publication type:

Article

Synthesis and Antiproliferative Effect of Ethyl 4-[4-(4-Substituted Piperidin-1-yl)]benzylpyrrolo[1,2- a]quinoxalinecarboxylate Derivatives on Human Leukemia Cells.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 940, doi. 10.1002/cmdc.201700049

By:

Desplat, Vanessa;
Vincenzi, Marian;
Lucas, Romain;
Moreau, Stéphane;
Savrimoutou, Solène;
Rubio, Sandra;
Pinaud, Noël;
Bigat, David;
Enriquez, Elodie;
Marchivie, Mathieu;
Routier, Sylvain;
Sonnet, Pascal;
Rossi, Filomena;
Ronga, Luisa;
Guillon, Jean

Publication type:

Article

1,2,4-Triazole-3-thione Compounds as Inhibitors of Dizinc Metallo-β-lactamases.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 972, doi. 10.1002/cmdc.201700186

By:

Sevaille, Laurent;
Gavara, Laurent;
Bebrone, Carine;
De Luca, Filomena;
Nauton, Lionel;
Achard, Maud;
Mercuri, Paola;
Tanfoni, Silvia;
Borgianni, Luisa;
Guyon, Carole;
Lonjon, Pauline;
Turan‐Zitouni, Gülhan;
Dzieciolowski, Julia;
Becker, Katja;
Bénard, Lionel;
Condon, Ciaran;
Maillard, Ludovic;
Martinez, Jean;
Frère, Jean‐Marie;
Dideberg, Otto

Publication type:

Article

Physiochemical Tuning of Potent Escherichia coli Anti-Adhesives by Microencapsulation and Methylene Homologation.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 986, doi. 10.1002/cmdc.201700061

By:

Alvarez Dorta, Dimitri;
Chalopin, Thibaut;
Sivignon, Adeline;
de Ruyck, Jérôme;
Dumych, Tetiana I.;
Bilyy, Rostyslav O.;
Deniaud, David;
Barnich, Nicolas;
Bouckaert, Julie;
Gouin, Sébastien G.

Publication type:

Article

Molecular Features of the YAP Inhibitor Verteporfin: Synthesis of Hexasubstituted Dipyrrins as Potential Inhibitors of YAP/TAZ, the Downstream Effectors of the Hippo Pathway.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 954, doi. 10.1002/cmdc.201700063

By:

Gibault, Floriane;
Bailly, Fabrice;
Corvaisier, Matthieu;
Coevoet, Mathilde;
Huet, Guillemette;
Melnyk, Patricia;
Cotelle, Philippe

Publication type:

Article

Chemoproteomics-Aided Medicinal Chemistry for the Discovery of EPHA2 Inhibitors.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 999, doi. 10.1002/cmdc.201700217

By:

Heinzlmeir, Stephanie;
Lohse, Jonas;
Treiber, Tobias;
Kudlinzki, Denis;
Linhard, Verena;
Gande, Santosh Lakshmi;
Sreeramulu, Sridhar;
Saxena, Krishna;
Liu, Xiaofeng;
Wilhelm, Mathias;
Schwalbe, Harald;
Kuster, Bernhard;
Médard, Guillaume

Publication type:

Article

Identifying Protein Allosteric Transitions for Drug Discovery with 1D NMR.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 901, doi. 10.1002/cmdc.201700064

By:

Krimm, Isabelle

Publication type:

Article

Inside Cover: Lanthanide Complexes in Molecular Magnetic Resonance Imaging and Theranostics (ChemMedChem 12/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 861, doi. 10.1002/cmdc.201700342

By:

Lacerda, Sara;
Tóth, Éva

Publication type:

Article

Back Cover: Benzylphenylpyrrolizinones with Anti-amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment (ChemMedChem 12/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 1012, doi. 10.1002/cmdc.201700343

By:

Jourdan, Jean‐Pierre;
Since, Marc;
El Kihel, Laïla;
Lecoutey, Cédric;
Corvaisier, Sophie;
Legay, Rémi;
Sopková‐de Oliveira Santos, Jana;
Cresteil, Thierry;
Malzert‐Fréon, Aurélie;
Rochais, Christophe;
Dallemagne, Patrick

Publication type:

Article

Cover Picture: Target Deconvolution Efforts on Wnt Pathway Screen Reveal Dual Modulation of Oxidative Phosphorylation and SERCA2 (ChemMedChem 12/2017).

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 860, doi. 10.1002/cmdc.201700341

By:

Casás‐Selves, Matias;
Zhang, Andrew X.;
Dowling, James E.;
Hallén, Stefan;
Kawatkar, Aarti;
Pace, Nicholas J.;
Denz, Christopher R.;
Pontz, Timothy;
Garahdaghi, Farzin;
Cao, Qing;
Sabirsh, Alan;
Thakur, Kumar;
O'Connell, Nichole;
Hu, Jun;
Cornella‐Taracido, Iván;
Weerapana, Eranthie;
Zinda, Michael;
Goodnow, Robert A.;
Castaldi, M. Paola

Publication type:

Article

1,3,5-Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu<sub>2/3</sub> Receptors.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 905, doi. 10.1002/cmdc.201700101

By:

Van Gool, Michiel;
Alonso De Diego, Sergio A.;
Delgado, Oscar;
Trabanco, Andrés A.;
Jourdan, Fabrice;
Macdonald, Gregor J.;
Somers, Marijke;
Ver Donck, Luc

Publication type:

Article

Rational Design and Synthesis of 1-(Arylideneamino)-4-aryl-1 H-imidazole-2-amine Derivatives as Antiplatelet Agents.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 962, doi. 10.1002/cmdc.201700123

By:

Amidi, Salimeh;
Esfahanizadeh, Marjan;
Tabib, Kimia;
Soleimani, Zohreh;
Kobarfard, Farzad

Publication type:

Article

Benzylphenylpyrrolizinones with Anti-amyloid and Radical Scavenging Effects, Potentially Useful in Alzheimer's Disease Treatment.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 913, doi. 10.1002/cmdc.201700102

By:

Jourdan, Jean‐Pierre;
Since, Marc;
El Kihel, Laïla;
Lecoutey, Cédric;
Corvaisier, Sophie;
Legay, Rémi;
Sopková‐de Oliveira Santos, Jana;
Cresteil, Thierry;
Malzert‐Fréon, Aurélie;
Rochais, Christophe;
Dallemagne, Patrick

Publication type:

Article

A Time-Resolved FRET Cell-Based Binding Assay for the Apelin Receptor.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 925, doi. 10.1002/cmdc.201700106

By:

Valencia, Christel;
Dujet, Céline;
Margathe, Jean‐François;
Iturrioz, Xavier;
Roux, Thomas;
Trinquet, Eric;
Villa, Pascal;
Hibert, Marcel;
Dupuis, Elodie;
Llorens‐Cortes, Catherine;
Bonnet, Dominique

Publication type:

Article

Structure-Based Design and Synthesis of Harmine Derivatives with Different Selectivity Profiles in Kinase versus Monoamine Oxidase Inhibition.

Published in:

ChemMedChem, 2017, v. 12, n. 12, p. 932, doi. 10.1002/cmdc.201600539

By:

Bálint, Balázs;
Wéber, Csaba;
Cruzalegui, Francisco;
Burbridge, Mike;
Kotschy, Andras

Publication type:

Article