Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 4

Results: 13

New Insight into the Structure-Activity Relationships of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitors UCPH-101 and UCPH-102.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 382, doi. 10.1002/cmdc.201500525

By:

Hansen, Stinne W.;
Erichsen, Mette N.;
Huynh, Tri H. V.;
Ruiz, Josep A.;
Haym, Isabell;
Bjørn‐Yoshimoto, Walden E.;
Abrahamsen, Bjarke;
Hansen, Jeanette;
Storgaard, Morten;
Eriksen, Anette L.;
Jensen, Anders A.;
Bunch, Lennart

Publication type:

Article

Bioavailability Studies and in vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH-102.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 403, doi. 10.1002/cmdc.201500527

By:

Haym, Isabell;
Huynh, Tri H. V.;
Hansen, Stinne W.;
Pedersen, Martin H. F.;
Ruiz, Josep A.;
Erichsen, Mette N.;
Gynther, Mikko;
Bjørn‐Yoshimoto, Walden E.;
Abrahamsen, Bjarke;
Bastlund, Jesper F.;
Bundgaard, Christoffer;
Eriksen, Anette L.;
Jensen, Anders A.;
Bunch, Lennart

Publication type:

Article

Cover Picture: Antivirulence Isoquinolone Mannosides: Optimization of the Biaryl Aglycone for FimH Lectin Binding Affinity and Efficacy in the Treatment of Chronic UTI (ChemMedChem 4/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 351, doi. 10.1002/cmdc.201600045

By:

Jarvis, Cassie;
Han, Zhenfu;
Kalas, Vasilios;
Klein, Roger;
Pinkner, Jerome S.;
Ford, Bradley;
Binkley, Jana;
Cusumano, Corinne K.;
Cusumano, Zachary;
Mydock‐McGrane, Laurel;
Hultgren, Scott J.;
Janetka, James W.

Publication type:

Article

Inside Cover: Screening, Synthesis, and In Vitro Evaluation of Vinyl Sulfones as Inhibitors of Complement-Dependent Cytotoxicity in Neuromyelitis Optica (ChemMedChem 4/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 352, doi. 10.1002/cmdc.201600046

By:

Ju, Eun Ji;
Yeon, Seul Ki;
Park, Jong‐Hyun;
Cheon, So Young;
Choi, Ji Won;
Ha, Taehwan;
Jang, Bo Ko;
Kim, Siwon;
Kang, Yong Gu;
Hwang, Hayoung;
Cho, Sung Jin;
Cheong, Eunji;
Bahn, Yong Sun;
Pae, Ae Nim;
Kim, Sung Min;
Park, Ki Duk

Publication type:

Article

Back Cover: EPR Studies of V-ATPase with Spin-Labeled Inhibitors DCC and Archazolid: Interaction Dynamics with Proton Translocating Subunit c (ChemMedChem 4/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 444, doi. 10.1002/cmdc.201600047

By:

Gölz, Jan Philipp;
Bockelmann, Svenja;
Mayer, Kerstin;
Steinhoff, Heinz‐Jürgen;
Wieczorek, Helmut;
Huss, Markus;
Klare, Johann P.;
Menche, Dirk

Publication type:

Article

Screening, Synthesis, and In Vitro Evaluation of Vinyl Sulfones as Inhibitors of Complement-Dependent Cytotoxicity in Neuromyelitis Optica.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 377, doi. 10.1002/cmdc.201500546

By:

Ju, Eun Ji;
Yeon, Seul Ki;
Park, Jong‐Hyun;
Cheon, So Young;
Choi, Ji Won;
Ha, Taehwan;
Jang, Bo Ko;
Kim, Siwon;
Kang, Yong Gu;
Hwang, Hayoung;
Cho, Sung Jin;
Cheong, Eunji;
Bahn, Yong Sun;
Pae, Ae Nim;
Kim, Sung Min;
Park, Ki Duk

Publication type:

Article

Broadly Neutralizing Antibody-Guided Carbohydrate-Based HIV Vaccine Design: Challenges and Opportunities.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 357, doi. 10.1002/cmdc.201500498

By:

Liu, Chang‐Cheng;
Zheng, Xiu‐Jing;
Ye, Xin‐Shan

Publication type:

Article

ω-Imidazolyl- and ω-Tetrazolylalkylcarbamates as Inhibitors of Fatty Acid Amide Hydrolase: Biological Activity and in vitro Metabolic Stability.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 429, doi. 10.1002/cmdc.201500445

By:

Terwege, Tobias;
Hanekamp, Walburga;
Garzinsky, David;
König, Simone;
Koch, Oliver;
Lehr, Matthias

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 4/2016.

Published in:: ChemMedChem, 2016, v. 11, n. 4, p. 353, doi. 10.1002/cmdc.201680413
Publication type:: Article

A Potent and Selective P-gp Modulator for Altering Multidrug Resistance Due to Pump Overexpression.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 374, doi. 10.1002/cmdc.201500538

By:

Guglielmo, Stefano;
Contino, Marialessandra;
Lazzarato, Loretta;
Perrone, Maria Grazia;
Blangetti, Marco;
Fruttero, Roberta;
Colabufo, Nicola Antonio

Publication type:

Article

Antivirulence Isoquinolone Mannosides: Optimization of the Biaryl Aglycone for FimH Lectin Binding Affinity and Efficacy in the Treatment of Chronic UTI.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 367, doi. 10.1002/cmdc.201600006

By:

Jarvis, Cassie;
Han, Zhenfu;
Kalas, Vasilios;
Klein, Roger;
Pinkner, Jerome S.;
Ford, Bradley;
Binkley, Jana;
Cusumano, Corinne K.;
Cusumano, Zachary;
Mydock‐McGrane, Laurel;
Hultgren, Scott J.;
Janetka, James W.

Publication type:

Article

Application of Site-Specific Spin Labeling for NMR Detecting Inhibitor-Induced Conformational Change of HIV-1 Reverse Transcriptase.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 363, doi. 10.1002/cmdc.201500554

By:

Seetaha, Supaporn;
Yagi‐Utsumi, Maho;
Yamaguchi, Takumi;
Ishii, Kentaro;
Hannongbua, Supa;
Choowongkomon, Kiattawee;
Kato, Koichi

Publication type:

Article

EPR Studies of V-ATPase with Spin-Labeled Inhibitors DCC and Archazolid: Interaction Dynamics with Proton Translocating Subunit c.

Published in:

ChemMedChem, 2016, v. 11, n. 4, p. 420, doi. 10.1002/cmdc.201500500

By:

Gölz, Jan Philipp;
Bockelmann, Svenja;
Mayer, Kerstin;
Steinhoff, Heinz‐Jürgen;
Wieczorek, Helmut;
Huss, Markus;
Klare, Johann P.;
Menche, Dirk

Publication type:

Article