Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 24

Results: 9

Carbazole Aminoalcohols Induce Antiproliferation and Apoptosis of Human Tumor Cells by Inhibiting Topoisomerase I.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2675, doi. 10.1002/cmdc.201600391

By:

Wang, Weisi;
Sun, Xiao;
Sun, Deheng;
Li, Shizhu;
Yu, Yang;
Yang, Tingyuan;
Yao, Junmin;
Chen, Zhuo;
Duan, Liping

Publication type:

Article

Discovery of a Novel Scaffold as an Indoleamine 2,3-Dioxygenase 1 (IDO1) Inhibitor Based on the Pyrrolopiperazinone Alkaloid, Longamide B.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2682, doi. 10.1002/cmdc.201600446

By:

Shiokawa, Zenyu;
Kashiwabara, Emi;
Yoshidome, Daisuke;
Fukase, Koichi;
Inuki, Shinsuke;
Fujimoto, Yukari

Publication type:

Article

Targeting Cancer Cells with a Bisphosphonate Prodrug.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2656, doi. 10.1002/cmdc.201600465

By:

Matsumoto, Kenji;
Hayashi, Kosuke;
Murata‐Hirai, Kaoru;
Iwasaki, Masashi;
Okamura, Haruki;
Minato, Nagahiro;
Morita, Craig T.;
Tanaka, Yoshimasa

Publication type:

Article

A Quinacrine Analogue Selective Against Gastric Cancer Cells: Insight from Biochemical and Biophysical Studies.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2703, doi. 10.1002/cmdc.201600477

By:

Gomes, Ana;
Fernandes, Iva;
Teixeira, Cátia;
Mateus, Nuno;
Sottomayor, M. J.;
Gomes, Paula

Publication type:

Article

From Type I to Type II: Design, Synthesis, and Characterization of Potent Pyrazin-2-ones as DFG-Out Inhibitors of PDGFRβ.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2664, doi. 10.1002/cmdc.201600494

By:

Bethke, Eugen;
Pinchuk, Boris;
Renn, Christian;
Witt, Lydia;
Schlosser, Joachim;
Peifer, Christian

Publication type:

Article

Monoamine Oxidase Inhibitory Activity: Methyl- versus Chlorochalcone Derivatives.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2649, doi. 10.1002/cmdc.201600497

By:

Mathew, Bijo;
Uçar, Gülberk;
Mathew, Githa Elizabeth;
Mathew, Sincy;
Kalatharakkal Purapurath, Praseedha;
Moolayil, Fasil;
Mohan, Smrithy;
Varghese Gupta, Sheeba

Publication type:

Article

Synthesis and Biological Evaluation of New Triazolo- and Imidazolopyridine RORγt Inverse Agonists.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2640, doi. 10.1002/cmdc.201600500

By:

Hintermann, Samuel;
Guntermann, Christine;
Mattes, Henri;
Carcache, David A.;
Wagner, Juergen;
Vulpetti, Anna;
Billich, Andreas;
Dawson, Janet;
Kaupmann, Klemens;
Kallen, Joerg;
Stringer, Rowan;
Orain, David

Publication type:

Article

Activity of Fluorine-Containing Analogues of WC-9 and Structurally Related Analogues against Two Intracellular Parasites: Trypanosoma cruzi and Toxoplasma gondii.

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2690, doi. 10.1002/cmdc.201600505

By:

Chao, María N.;
Li, Catherine;
Storey, Melissa;
Falcone, Bruno N.;
Szajnman, Sergio H.;
Bonesi, Sergio M.;
Docampo, Roberto;
Moreno, Silvia N. J.;
Rodriguez, Juan B.

Publication type:

Article

Cover Picture: Targeting Cancer Cells with a Bisphosphonate Prodrug (ChemMedChem 24/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 24, p. 2639, doi. 10.1002/cmdc.201600605

By:

Matsumoto, Kenji;
Hayashi, Kosuke;
Murata‐Hirai, Kaoru;
Iwasaki, Masashi;
Okamura, Haruki;
Minato, Nagahiro;
Morita, Craig T.;
Tanaka, Yoshimasa

Publication type:

Article