Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 20

Results: 14

2-Amino[1,2,4]triazolo[1,5 -c]quinazolines and Derived Novel Heterocycles: Syntheses and Structure-Activity Relationships of Potent Adenosine Receptor Antagonists.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2272, doi. 10.1002/cmdc.201600255

By:

Burbiel, Joachim C.;
Ghattas, Wadih;
Küppers, Petra;
Köse, Meryem;
Lacher, Svenja;
Herzner, Anna‐Maria;
Kombu, Rajan Subramanian;
Akkinepally, Raghuram Rao;
Hockemeyer, Jörg;
Müller, Christa E.

Publication type:

Article

Microwave-Assisted Syntheses of Benzimidazole-Containing Selenadiazole Derivatives That Induce Cell-Cycle Arrest and Apoptosis in Human Breast Cancer Cells by Activation of the ROS/AKT Pathway.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2339, doi. 10.1002/cmdc.201600261

By:

Liang, Yuanwei;
Zhou, Yangliang;
Deng, Shulin;
Chen, Tianfeng

Publication type:

Article

Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2261, doi. 10.1002/cmdc.201600276

By:

Siebeneicher, Holger;
Cleve, Arwed;
Rehwinkel, Hartmut;
Neuhaus, Roland;
Heisler, Iring;
Müller, Thomas;
Bauser, Marcus;
Buchmann, Bernd

Publication type:

Article

Oral Administration of Peptide-Based Drugs: Beyond Lipinski's Rule.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2245, doi. 10.1002/cmdc.201600288

By:

Santos, Gabriela B.;
Ganesan, A.;
Emery, Flavio S.

Publication type:

Article

Development of Tetrachlorophthalimides as Liver X Receptor β (LXRβ)-Selective Agonists.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2347, doi. 10.1002/cmdc.201600305

By:

Nomura, Sayaka;
Endo‐Umeda, Kaori;
Makishima, Makoto;
Hashimoto, Yuichi;
Ishikawa, Minoru

Publication type:

Article

Bacterial Cell Growth Inhibitors Targeting Undecaprenyl Diphosphate Synthase and Undecaprenyl Diphosphate Phosphatase.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2311, doi. 10.1002/cmdc.201600342

By:

Wang, Yang;
Desai, Janish;
Zhang, Yonghui;
Malwal, Satish R.;
Shin, Christopher J.;
Feng, Xinxin;
Sun, Hong;
Liu, Guizhi;
Guo, Rey‐Ting;
Oldfield, Eric

Publication type:

Article

Discovery of α-Substituted Imidazole-4-acetic Acid Analogues as a Novel Class of ρ<sub>1</sub> γ-Aminobutyric Acid Type A Receptor Antagonists with Effect on Retinal Vascular Tone.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2299, doi. 10.1002/cmdc.201600356

By:

Krall, Jacob;
Brygger, Benjamin M.;
Sigurðardóttir, Sara B.;
Ng, Clarissa K. L.;
Bundgaard, Christoffer;
Kehler, Jan;
Nielsen, Birgitte;
Bek, Toke;
Jensen, Anders A.;
Frølund, Bente

Publication type:

Article

Chromones: A Promising Ring System for New Anti-inflammatory Drugs.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2252, doi. 10.1002/cmdc.201600359

By:

Silva, Carlos F. M.;
Pinto, Diana C. G. A.;
Silva, Artur M. S.

Publication type:

Article

Identification and Structure-Activity Relationship Studies of Small-Molecule Inhibitors of the Methyllysine Reader Protein Spindlin1.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2327, doi. 10.1002/cmdc.201600362

By:

Robaa, Dina;
Wagner, Tobias;
Luise, Chiara;
Carlino, Luca;
McMillan, Joel;
Flaig, Ralf;
Schüle, Roland;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

A Triazinone Derivative Inhibits HIV-1 Replication by Interfering with Reverse Transcriptase Activity.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2320, doi. 10.1002/cmdc.201600375

By:

Urano, Emiko;
Miyauchi, Kosuke;
Kojima, Yoko;
Hamatake, Makiko;
Ablan, Sherimay D.;
Fudo, Satoshi;
Freed, Eric O.;
Hoshino, Tyuji;
Komano, Jun

Publication type:

Article

The Versatile 2-Substituted Imidazoline Nucleus as a Structural Motif of Ligands Directed to the Serotonin 5-HT<sub>1A</sub> Receptor.

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2287, doi. 10.1002/cmdc.201600383

By:

Del Bello, Fabio;
Cilia, Antonio;
Carrieri, Antonio;
Fasano, Domenico Claudio;
Ghelardini, Carla;
Di Cesare Mannelli, Lorenzo;
Micheli, Laura;
Santini, Carlo;
Diamanti, Eleonora;
Giannella, Mario;
Giorgioni, Gianfabio;
Mammoli, Valerio;
Paoletti, Corinne Dalila;
Petrelli, Riccardo;
Piergentili, Alessandro;
Quaglia, Wilma;
Pigini, Maria

Publication type:

Article

Cover Picture: Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY-876 (ChemMedChem 20/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2240, doi. 10.1002/cmdc.201600503

By:

Siebeneicher, Holger;
Cleve, Arwed;
Rehwinkel, Hartmut;
Neuhaus, Roland;
Heisler, Iring;
Müller, Thomas;
Bauser, Marcus;
Buchmann, Bernd

Publication type:

Article

Back Cover: 2-Amino[1,2,4]triazolo[1,5 -c]quinazolines and Derived Novel Heterocycles: Syntheses and Structure-Activity Relationships of Potent Adenosine Receptor Antagonists (ChemMedChem 20/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 20, p. 2361, doi. 10.1002/cmdc.201600504

By:

Burbiel, Joachim C.;
Ghattas, Wadih;
Küppers, Petra;
Köse, Meryem;
Lacher, Svenja;
Herzner, Anna‐Maria;
Kombu, Rajan Subramanian;
Akkinepally, Raghuram Rao;
Hockemeyer, Jörg;
Müller, Christa E.

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 20/2016.

Published in:: ChemMedChem, 2016, v. 11, n. 20, p. 2241, doi. 10.1002/cmdc.201682013
Publication type:: Article