Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 18

Results: 16

Hedgehog Proteins Consume Steroidal CYP17A1 Antagonists: Potential Therapeutic Significance in Advanced Prostate Cancer.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1983, doi. 10.1002/cmdc.201600238

By:

Bordeau, Brandon M.;
Ciulla, Daniel A.;
Callahan, Brian P.

Publication type:

Article

Chemical Platform for the Preparation of Synthetic Orally Active Peptidomimetics with Hemoregulating Activity.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1974, doi. 10.1002/cmdc.201600157

By:

Deigin, Vladislav;
Ksenofontova, Olga;
Khrushchev, Alexey;
Yatskin, Oleg;
Goryacheva, Alexandra;
Ivanov, Vadim

Publication type:

Article

Virtual Screening of Small Drug-Like Compounds Stimulating the Enzymatic Activity of Kallikrein-Related Peptidase 3 (KLK3).

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2043, doi. 10.1002/cmdc.201600181

By:

Ylikangas, Henna;
Mattsson, Johanna M.;
Stenman, Ulf‐Håkan;
Koistinen, Hannu;
Poso, Antti;
Lahtela‐Kakkonen, Maija

Publication type:

Article

Covalent Inhibition of HIV-1 Integrase by N-Succinimidyl Peptides.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1987, doi. 10.1002/cmdc.201600190

By:

Chandra, Koushik;
Das, Priyadip;
Mamidi, Samarasimhareddy;
Hurevich, Mattan;
Iosub‐Amir, Anat;
Metanis, Norman;
Reches, Meital;
Friedler, Assaf

Publication type:

Article

4-Biphenylalanine- and 3-Phenyltyrosine-Derived Hydroxamic Acids as Inhibitors of the JumonjiC-Domain-Containing Histone Demethylase KDM4A.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2063, doi. 10.1002/cmdc.201600218

By:

Morera, Ludovica;
Roatsch, Martin;
Fürst, Michael C. D.;
Hoffmann, Inga;
Senger, Johanna;
Hau, Mirjam;
Franz, Henriette;
Schüle, Roland;
Heinrich, Markus R.;
Jung, Manfred

Publication type:

Article

Multicomponent Petasis-borono Mannich Preparation of Alkylaminophenols and Antimicrobial Activity Studies.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2015, doi. 10.1002/cmdc.201600244

By:

Neto, Íris;
Andrade, Joana;
Fernandes, A. S.;
Pinto Reis, Catarina;
Salunke, Jagadish K.;
Priimagi, Arri;
Candeias, Nuno R.;
Rijo, Patrícia

Publication type:

Article

Targeting an Aromatic Hotspot in Plasmodium falciparum 1-Deoxy- d-xylulose-5-phosphate Reductoisomerase with β-Arylpropyl Analogues of Fosmidomycin.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2024, doi. 10.1002/cmdc.201600249

By:

Sooriyaarachchi, Sanjeewani;
Chofor, René;
Risseeuw, Martijn D. P.;
Bergfors, Terese;
Pouyez, Jenny;
Dowd, Cynthia S.;
Maes, Louis;
Wouters, Johan;
Jones, T. Alwyn;
Van Calenbergh, Serge;
Mowbray, Sherry L.

Publication type:

Article

Clickable 4-Oxo-β-lactam-Based Selective Probing for Human Neutrophil Elastase Related Proteomes.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2037, doi. 10.1002/cmdc.201600258

By:

Ruivo, Eduardo F. P.;
Gonçalves, Lídia M.;
Carvalho, Luís A. R.;
Guedes, Rita C.;
Hofbauer, Stefan;
Brito, José A.;
Archer, Margarida;
Moreira, Rui;
Lucas, Susana D.

Publication type:

Article

2-Anilino-3-Aroylquinolines as Potent Tubulin Polymerization Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2050, doi. 10.1002/cmdc.201600259

By:

Srikanth, P. S.;
Nayak, V. Lakshma;
Suresh Babu, Korrapati;
Kumar, G. Bharath;
Ravikumar, A.;
Kamal, Ahmed

Publication type:

Article

Identification of Highly Potent Protein Kinase C-Related Kinase 1 Inhibitors by Virtual Screening, Binding Free Energy Rescoring, and in vitro Testing.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2084, doi. 10.1002/cmdc.201600284

By:

Slynko, Inna;
Schmidtkunz, Karin;
Rumpf, Tobias;
Klaeger, Susan;
Heinzlmeir, Stephanie;
Najar, Abdulkarim;
Metzger, Eric;
Kuster, Bernhard;
Schüle, Roland;
Jung, Manfred;
Sippl, Wolfgang

Publication type:

Article

Discovery and Characterization of ACT-451840: an Antimalarial Drug with a Novel Mechanism of Action.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1995, doi. 10.1002/cmdc.201600298

By:

Boss, Christoph;
Aissaoui, Hamed;
Amaral, Nathalie;
Bauer, Aude;
Bazire, Stephanie;
Binkert, Christoph;
Brun, Reto;
Bürki, Cédric;
Ciana, Claire‐Lise;
Corminboeuf, Olivier;
Delahaye, Stephane;
Dollinger, Claire;
Fischli, Christoph;
Fischli, Walter;
Flock, Alexandre;
Frantz, Marie‐Céline;
Girault, Malory;
Grisostomi, Corinna;
Friedli, Astrid;
Heidmann, Bibia

Publication type:

Article

Near-Infrared Intraoperative Chemiluminescence Imaging.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1978, doi. 10.1002/cmdc.201600301

By:

Büchel, Gabriel E.;
Carney, Brandon;
Shaffer, Travis M.;
Tang, Jun;
Austin, Christine;
Arora, Manish;
Zeglis, Brian M.;
Grimm, Jan;
Eppinger, Jörg;
Reiner, Thomas

Publication type:

Article

Corrigendum: Amphiphilic Bicyclic Peptides as Cellular Delivery Agents.

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2095, doi. 10.1002/cmdc.201600431

By:

Oh, Donghoon;
Darwish, Shaban Anwar;
Shirazi, Amir Nasrolahi;
Tiwari, Rakesh Kumar;
Parang, Keykavous

Publication type:

Article

Cover Picture: Covalent Inhibition of HIV-1 Integrase by N-Succinimidyl Peptides (ChemMedChem 18/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 1969, doi. 10.1002/cmdc.201600435

By:

Chandra, Koushik;
Das, Priyadip;
Mamidi, Samarasimhareddy;
Hurevich, Mattan;
Iosub‐Amir, Anat;
Metanis, Norman;
Reches, Meital;
Friedler, Assaf

Publication type:

Article

Back Cover: Discovery and Characterization of ACT-451840: an Antimalarial Drug with a Novel Mechanism of Action (ChemMedChem 18/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 18, p. 2096, doi. 10.1002/cmdc.201600436

By:

Boss, Christoph;
Aissaoui, Hamed;
Amaral, Nathalie;
Bauer, Aude;
Bazire, Stephanie;
Binkert, Christoph;
Brun, Reto;
Bürki, Cédric;
Ciana, Claire‐Lise;
Corminboeuf, Olivier;
Delahaye, Stephane;
Dollinger, Claire;
Fischli, Christoph;
Fischli, Walter;
Flock, Alexandre;
Frantz, Marie‐Céline;
Girault, Malory;
Grisostomi, Corinna;
Friedli, Astrid;
Heidmann, Bibia

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 18/2016.

Published in:: ChemMedChem, 2016, v. 11, n. 18, p. 1970, doi. 10.1002/cmdc.201681813
Publication type:: Article