Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 16

Results: 26

Serpin A1 C-Terminal Peptides as Collagen Turnover Modulators.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1850, doi. 10.1002/cmdc.201500472

By:

Pascarella, Simona;
Tiberi, Caterina;
Sabatino, Giuseppina;
Nuti, Francesca;
Papini, Anna Maria;
Giovannelli, Lisa;
Rovero, Paolo

Publication type:

Article

Reactivity, Selectivity, and Reaction Mechanisms of Aminoguanidine, Hydralazine, Pyridoxamine, and Carnosine as Sequestering Agents of Reactive Carbonyl Species: A Comparative Study.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1778, doi. 10.1002/cmdc.201500552

By:

Colzani, Mara;
De Maddis, Danilo;
Casali, Gaia;
Carini, Marina;
Vistoli, Giulio;
Aldini, Giancarlo

Publication type:

Article

Enhanced Efficacy of Artemisinin Loaded in Transferrin-Conjugated Liposomes versus Stealth Liposomes against HCT-8 Colon Cancer Cells.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1745, doi. 10.1002/cmdc.201500586

By:

Leto, Isabella;
Coronnello, Marcella;
Righeschi, Chiara;
Bergonzi, Maria Camilla;
Mini, Enrico;
Bilia, Anna Rita

Publication type:

Article

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A2A Adenosine Receptor.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1829, doi. 10.1002/cmdc.201500595

By:

Thomas, Ajiroghene;
Buccioni, Michela;
Dal Ben, Diego;
Lambertucci, Catia;
Marucci, Gabriella;
Santinelli, Claudia;
Spinaci, Andrea;
Kachler, Sonja;
Klotz, Karl‐Norbert;
Volpini, Rosaria

Publication type:

Article

In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1812, doi. 10.1002/cmdc.201500596

By:

Bruno, Elvira;
Buemi, Maria R.;
De Luca, Laura;
Ferro, Stefania;
Monforte, Anna‐Maria;
Supuran, Claudiu T.;
Vullo, Daniela;
De Sarro, Giovambattista;
Russo, Emilio;
Gitto, Rosaria

Publication type:

Article

Cationic Supramolecular Vesicular Aggregates for Pulmonary Tissue Selective Delivery in Anticancer Therapy.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1734, doi. 10.1002/cmdc.201600070

By:

Licciardi, Mariano;
Paolino, Donatella;
Mauro, Nicolò;
Cosco, Donato;
Giammona, Gaetano;
Fresta, Massimo;
Cavallaro, Gennara;
Celia, Christian

Publication type:

Article

Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1709, doi. 10.1002/cmdc.201600015

By:

Corona, Angela;
Desantis, Jenny;
Massari, Serena;
Distinto, Simona;
Masaoka, Takashi;
Sabatini, Stefano;
Esposito, Francesca;
Manfroni, Giuseppe;
Maccioni, Elias;
Cecchetti, Violetta;
Pannecouque, Christophe;
Le Grice, Stuart F. J.;
Tramontano, Enzo;
Tabarrini, Oriana

Publication type:

Article

A Series of COX-2 Inhibitors Endowed with NO-Releasing Properties: Synthesis, Biological Evaluation, and Docking Analysis.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1804, doi. 10.1002/cmdc.201600086

By:

Consalvi, Sara;
Poce, Giovanna;
Ragno, Rino;
Sabatino, Manuela;
La Motta, Concettina;
Sartini, Stefania;
Calderone, Vincenzo;
Martelli, Alma;
Ghelardini, Carla;
Di Cesare Mannelli, Lorenzo;
Biava, Mariangela

Publication type:

Article

A Novel Class of Dopamine D4 Receptor Ligands Bearing an Imidazoline Nucleus.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1819, doi. 10.1002/cmdc.201600022

By:

Mammoli, Valerio;
Bonifazi, Alessandro;
Dal Ben, Diego;
Giannella, Mario;
Giorgioni, Gianfabio;
Piergentili, Alessandro;
Pigini, Maria;
Quaglia, Wilma;
Thomas, Ajiroghene;
Newman, Amy H.;
Ferré, Sergi;
Sanchez‐Soto, Marta;
Keck, Thomas M.;
Del Bello, Fabio

Publication type:

Article

Design, Synthesis, and Evaluation of Acrylamide Derivatives as Direct NLRP3 Inflammasome Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1790, doi. 10.1002/cmdc.201600055

By:

Cocco, Mattia;
Miglio, Gianluca;
Giorgis, Marta;
Garella, Davide;
Marini, Elisabetta;
Costale, Annalisa;
Regazzoni, Luca;
Vistoli, Giulio;
Orioli, Marica;
Massulaha‐Ahmed, Raïhane;
Détraz‐Durieux, Isabelle;
Groslambert, Marine;
Py, Bénédicte F.;
Bertinaria, Massimo

Publication type:

Article

Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position 9.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1856, doi. 10.1002/cmdc.201500607

By:

Merlino, Francesco;
Brancaccio, Diego;
Yousif, Ali M.;
Piras, Linda;
Campiglia, Pietro;
Gomez‐Monterrey, Isabel;
Santicioli, Paolo;
Meini, Stefania;
Maggi, Carlo A.;
Novellino, Ettore;
Carotenuto, Alfonso;
Grieco, Paolo

Publication type:

Article

Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1770, doi. 10.1002/cmdc.201600078

By:

Gobbi, Silvia;
Hu, Qingzhong;
Zimmer, Christina;
Belluti, Federica;
Rampa, Angela;
Hartmann, Rolf W.;
Bisi, Alessandra

Publication type:

Article

Albumin Nanoparticles for Brain Delivery: A Comparison of Chemical versus Thermal Methods and in vivo Behavior.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1840, doi. 10.1002/cmdc.201600080

By:

Bergonzi, Maria C.;
Guccione, Clizia;
Grossi, Cristina;
Piazzini, Vieri;
Torracchi, Andrea;
Luccarini, Ilaria;
Casamenti, Fiorella;
Bilia, Anna R.

Publication type:

Article

Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1721, doi. 10.1002/cmdc.201600053

By:

Rocca, Roberta;
Costa, Giosuè;
Artese, Anna;
Parrotta, Lucia;
Ortuso, Francesco;
Maccioni, Elias;
Pinato, Odra;
Greco, Maria Laura;
Sissi, Claudia;
Alcaro, Stefano;
Distinto, Simona;
Moraca, Federica

Publication type:

Article

Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1865, doi. 10.1002/cmdc.201600092

By:

Ortore, Gabriella;
Orlandini, Elisabetta;
Braca, Alessandra;
Ciccone, Lidia;
Rossello, Armando;
Martinelli, Adriano;
Nencetti, Susanna

Publication type:

Article

Synthesis and Biological Evaluation of N2-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1705, doi. 10.1002/cmdc.201600108

By:

Cortese, Daniela;
Chegaev, Konstantin;
Guglielmo, Stefano;
Wang, Lan Z.;
Golding, Bernard T.;
Cano, Céline;
Fruttero, Roberta

Publication type:

Article

TRPV1-FAAH-COX: The Couples Game in Pain Treatment.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1686, doi. 10.1002/cmdc.201600111

By:

Aiello, Francesca;
Carullo, Gabriele;
Badolato, Mariateresa;
Brizzi, Antonella

Publication type:

Article

Molecular Basis for Differential Recognition of G-Quadruplex versus Double-Helix DNA by Bis-Phenanthroline Metal Complexes.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1762, doi. 10.1002/cmdc.201600129

By:

Rigo, Riccardo;
Bianco, Sara;
Musetti, Caterina;
Palumbo, Manlio;
Sissi, Claudia

Publication type:

Article

Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1752, doi. 10.1002/cmdc.201600140

By:

Granchi, Carlotta;
Lapillo, Margherita;
Spena, Concetta Russo;
Rizzolio, Flavio;
Tuccinardi, Tiziano;
Martin, Teresa A.;
Carlson, Kathryn E.;
Katzenellenbogen, John A.;
Minutolo, Filippo

Publication type:

Article

Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1695, doi. 10.1002/cmdc.201600204

By:

Maccallini, Cristina;
Di Matteo, Mauro;
Vullo, Daniela;
Ammazzalorso, Alessandra;
Carradori, Simone;
De Filippis, Barbara;
Fantacuzzi, Marialuigia;
Giampietro, Letizia;
Pandolfi, Assunta;
Supuran, Claudiu T.;
Amoroso, Rosa

Publication type:

Article

3-Arylidene- N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor Activity.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1700, doi. 10.1002/cmdc.201600225

By:

Musso, Loana;
Cincinelli, Raffaella;
Zuco, Valentina;
De Cesare, Michelandrea;
Zunino, Franco;
Fallacara, Anna Lucia;
Botta, Maurizio;
Dallavalle, Sabrina

Publication type:

Article

Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1680, doi. 10.1002/cmdc.201600272

By:

Milite, Ciro;
Feoli, Alessandra;
Viviano, Monica;
Rescigno, Donatella;
Mai, Antonello;
Castellano, Sabrina;
Sbardella, Gianluca

Publication type:

Article

The 23rd National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015).

Published in:

2016

By:

Campiglia, Pietro;
Sbardella, Gianluca

Publication type:

Editorial

Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1669, doi. 10.1002/cmdc.201600392

By:

Corona, Angela;
Desantis, Jenny;
Massari, Serena;
Distinto, Simona;
Masaoka, Takashi;
Sabatini, Stefano;
Esposito, Francesca;
Manfroni, Giuseppe;
Maccioni, Elias;
Cecchetti, Violetta;
Pannecouque, Christophe;
Le Grice, Stuart F. J.;
Tramontano, Enzo;
Tabarrini, Oriana

Publication type:

Article

Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016).

Published in:

ChemMedChem, 2016, v. 11, n. 16, p. 1875, doi. 10.1002/cmdc.201600393

By:

Rocca, Roberta;
Costa, Giosuè;
Artese, Anna;
Parrotta, Lucia;
Ortuso, Francesco;
Maccioni, Elias;
Pinato, Odra;
Greco, Maria Laura;
Sissi, Claudia;
Alcaro, Stefano;
Distinto, Simona;
Moraca, Federica

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 16/2016.

Published in:: ChemMedChem, 2016, v. 11, n. 16, p. 1676, doi. 10.1002/cmdc.201681613
Publication type:: Article

Works matching IS 18607179 AND DT 2016 AND VI 11 AND IP 16

Serpin A1 C-Terminal Peptides as Collagen Turnover Modulators.

Reactivity, Selectivity, and Reaction Mechanisms of Aminoguanidine, Hydralazine, Pyridoxamine, and Carnosine as Sequestering Agents of Reactive Carbonyl Species: A Comparative Study.

Enhanced Efficacy of Artemisinin Loaded in Transferrin-Conjugated Liposomes versus Stealth Liposomes against HCT-8 Colon Cancer Cells.

The Length and Flexibility of the 2-Substituent of 9-Ethyladenine Derivatives Modulate Affinity and Selectivity for the Human A<sub>2A</sub> Adenosine Receptor.

In Vivo Evaluation of Selective Carbonic Anhydrase Inhibitors as Potential Anticonvulsant Agents.

Cationic Supramolecular Vesicular Aggregates for Pulmonary Tissue Selective Delivery in Anticancer Therapy.

Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors.

A Series of COX-2 Inhibitors Endowed with NO-Releasing Properties: Synthesis, Biological Evaluation, and Docking Analysis.

A Novel Class of Dopamine D<sub>4</sub> Receptor Ligands Bearing an Imidazoline Nucleus.

Design, Synthesis, and Evaluation of Acrylamide Derivatives as Direct NLRP3 Inflammasome Inhibitors.

Structure-Activity Study of the Peptides P5U and Urantide by the Development of Analogues Containing Uncoded Amino Acids at Position 9.

Targeting Steroidogenic Cytochromes P450 (CYPs) with 6-Substituted 1-Imidazolylmethylxanthones.

Albumin Nanoparticles for Brain Delivery: A Comparison of Chemical versus Thermal Methods and in vivo Behavior.

Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement.

Targeting Different Transthyretin Binding Sites with Unusual Natural Compounds.

Synthesis and Biological Evaluation of N<sup>2</sup>-Substituted 2,4-Diamino-6-cyclohexylmethoxy-5-nitrosopyrimidines and Related 5-Cyano-NNO-azoxy Derivatives as Cyclin-Dependent Kinase 2 (CDK2) Inhibitors.

TRPV1-FAAH-COX: The Couples Game in Pain Treatment.

Molecular Basis for Differential Recognition of G-Quadruplex versus Double-Helix DNA by Bis-Phenanthroline Metal Complexes.

Cyclic Ketoximes as Estrogen Receptor β Selective Agonists.

Indazole, Pyrazole, and Oxazole Derivatives Targeting Nitric Oxide Synthases and Carbonic Anhydrases.

3-Arylidene- N-hydroxyoxindoles: A New Class of Compounds Endowed with Antitumor Activity.

Progress in the Development of Lysine Methyltransferase SETD8 Inhibitors.

The 23<sup>rd</sup> National Meeting of the Medicinal Chemistry Division of the Italian Chemical Society (DCF-SCI) in Salerno (NMMC 2015).

Cover Picture: Studies on Cycloheptathiophene-3-carboxamide Derivatives as Allosteric HIV-1 Ribonuclease H Inhibitors (ChemMedChem 16/2016).

Back Cover: Hit Identification of a Novel Dual Binder for h-telo/c-myc G-Quadruplex by a Combination of Pharmacophore Structure-Based Virtual Screening and Docking Refinement (ChemMedChem 16/2016).

Spotlights on our sister journals: ChemMedChem 16/2016.