Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 5

Results: 23

Can Silicon Make an Excellent Drug Even Better? An in vitro and in vivo Head-to-Head Comparison between Loperamide and Its Silicon Analogue Sila-Loperamide.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 911, doi. 10.1002/cmdc.201500040

By:

Geyer, Marcel;
Wellner, Eric;
Jurva, Ulrik;
Saloman, Sebastian;
Armstrong, Duncan;
Tacke, Reinhold

Publication type:

Article

New Approaches in the Design and Development of Cannabinoid Receptor Ligands: Multifunctional and Bivalent Compounds.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 773, doi. 10.1002/cmdc.201500041

By:

Nimczick, Martin;
Decker, Michael

Publication type:

Article

A Chemical Chaperone-Based Drug Candidate is Effective in a Mouse Model of Amyotrophic Lateral Sclerosis (ALS).

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 850, doi. 10.1002/cmdc.201500045

By:

Getter, Tamar;
Zaks, Ilana;
Barhum, Yael;
Ben‐Zur, Tali;
Böselt, Sebastian;
Gregoire, Simpson;
Viskind, Olga;
Shani, Tom;
Gottlieb, Hugo;
Green, Omer;
Shubely, Moran;
Senderowitz, Hanoch;
Israelson, Adrian;
Kwon, Inchan;
Petri, Susanne;
Offen, Daniel;
Gruzman, Arie

Publication type:

Article

Exploiting the Lactose-GM<sub>3</sub> Interaction for Drug Delivery.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 792, doi. 10.1002/cmdc.201500046

By:

Murthy, Raghavendra Vasudeva;
Bavireddi, Harikrishna;
Gade, Madhuri;
Kikkeri, Raghavendra

Publication type:

Article

Ion Channel Drug Discovery. Edited by Brian Cox and Martin Gosling.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 925, doi. 10.1002/cmdc.201500062

By:

Brown, Alan D.

Publication type:

Article

Bis(benzoyloxybenzyl)-Di PPro Nucleoside Diphosphates of Anti-HIV Active Nucleoside Analogues.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 891, doi. 10.1002/cmdc.201500063

By:

Weinschenk, Lina;
Gollnest, Tristan;
Schols, Dominique;
Balzarini, Jan;
Meier, Chris

Publication type:

Article

Indolo[3,2- c]quinoline G-Quadruplex Stabilizers: a Structural Analysis of Binding to the Human Telomeric G-Quadruplex.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 836, doi. 10.1002/cmdc.201500067

By:

Lavrado, João;
Ohnmacht, Stephan A.;
Correia, Isabel;
Leitão, Clara;
Pisco, Sílvia;
Gunaratnam, Mekala;
Moreira, Rui;
Neidle, Stephen;
Santos, Daniel J. V. A. dos;
Paulo, Alexandra

Publication type:

Article

Benzo[ b]tryptanthrin Inhibits MDR1, Topoisomerase Activity, and Reverses Adriamycin Resistance in Breast Cancer Cells.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 827, doi. 10.1002/cmdc.201500068

By:

Jun, Kyu‐Yeon;
Park, So‐Eun;
Liang, Jing Lu;
Jahng, Yurngdong;
Kwon, Youngjoo

Publication type:

Article

Targeting the Erythrocytic and Liver Stages of Malaria Parasites with s-Triazine-Based Hybrids.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 883, doi. 10.1002/cmdc.201500011

By:

Rodrigues, Catarina A. B.;
Frade, Raquel F. M.;
Albuquerque, Inês S.;
Perry, Maria J.;
Gut, Jiri;
Machado, Marta;
Rosenthal, Philip J.;
Prudêncio, Miguel;
Afonso, Carlos A. M.;
Moreira, Rui

Publication type:

Article

Structure-Based Design of Drugs and Other Bioactive Molecules. Edited by Arun K. Ghosh and Sandra Gemma.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 926, doi. 10.1002/cmdc.201500105

By:

Stocks, Michael

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 5/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 5, p. 768, doi. 10.1002/cmdc.201580513
Publication type:: Article

Platinum(II) as Bifunctional Linker in Antibody-Drug Conjugate Formation: Coupling of a 4-Nitrobenzo-2-oxa-1,3-diazole Fluorophore to Trastuzumab as a Model.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 797, doi. 10.1002/cmdc.201402496

By:

Waalboer, Dennis C. J.;
Muns, Joey A.;
Sijbrandi, Niels J.;
Schasfoort, Richard B. M.;
Haselberg, Rob;
Somsen, Govert W.;
Houthoff, Hendrik‐Jan;
van Dongen, Guus A. M. S.

Publication type:

Article

Controlling Toxicity of Peptide-Drug Conjugates by Different Chemical Linker Structures.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 804, doi. 10.1002/cmdc.201402514

By:

Böhme, David;
Beck‐Sickinger, Annette G.

Publication type:

Article

Investigation of Structure-Activity Relationships of Synthetic Anti-Gonadotropin Releasing Hormone Vaccine Candidates.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 901, doi. 10.1002/cmdc.201500036

By:

Chang, Chenghung;
Varamini, Pegah;
Giddam, Ashwini Kumar;
Mansfeld, Friederike M.;
D'Occhio, Michael J.;
Toth, Istvan

Publication type:

Article

Selective Inhibitors of the Protein Tyrosine Phosphatase SHP2 Block Cellular Motility and Growth of Cancer Cells in vitro and in vivo.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 815, doi. 10.1002/cmdc.201500015

By:

Grosskopf, Stefanie;
Eckert, Chris;
Arkona, Christoph;
Radetzki, Silke;
Böhm, Kerstin;
Heinemann, Udo;
Wolber, Gerhard;
von Kries, Jens‐Peter;
Birchmeier, Walter;
Rademann, Jörg

Publication type:

Article

Cover Picture: Selective Inhibitors of the Protein Tyrosine Phosphatase SHP2 Block Cellular Motility and Growth of Cancer Cells in vitro and in vivo (ChemMedChem 5/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 757, doi. 10.1002/cmdc.201590011

By:

Grosskopf, Stefanie;
Eckert, Chris;
Arkona, Christoph;
Radetzki, Silke;
Böhm, Kerstin;
Heinemann, Udo;
Wolber, Gerhard;
von Kries, Jens‐Peter;
Birchmeier, Walter;
Rademann, Jörg

Publication type:

Article

Inside Cover: Novel 1,4-Substituted-1,2,3-Triazoles as Antitubercular Agents (ChemMedChem 5/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 758, doi. 10.1002/cmdc.201590012

By:

Altimari, Jarrad M.;
Hockey, Samantha C.;
Boshoff, Helena I.;
Sajid, Andaleeb;
Henderson, Luke C.

Publication type:

Article

Graphical Abstract: ChemMedChem 5/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 5, p. 759, doi. 10.1002/cmdc.201590013
Publication type:: Article

Back Cover: New Approaches in the Design and Development of Cannabinoid Receptor Ligands: Multifunctional and Bivalent Compounds (ChemMedChem 5/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 932, doi. 10.1002/cmdc.201590014

By:

Nimczick, Martin;
Decker, Michael

Publication type:

Article

Novel 1,4-Substituted-1,2,3-Triazoles as Antitubercular Agents.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 787, doi. 10.1002/cmdc.201500051

By:

Altimari, Jarrad M.;
Hockey, Samantha C.;
Boshoff, Helena I.;
Sajid, Andaleeb;
Henderson, Luke C.

Publication type:

Article

Indanones As High-Potency Reversible Inhibitors of Monoamine Oxidase.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 862, doi. 10.1002/cmdc.201500059

By:

Mostert, Samantha;
Petzer, Anél;
Petzer, Jacobus P.

Publication type:

Article

Development of Urea and Thiourea Kynurenamine Derivatives: Synthesis, Molecular Modeling, and Biological Evaluation as Nitric Oxide Synthase Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 874, doi. 10.1002/cmdc.201500007

By:

Chayah, Mariem;
Carrión, M. Dora;
Gallo, Miguel A.;
Jiménez, Rosario;
Duarte, Juan;
Camacho, M. Encarnación

Publication type:

Article

Antibiotics: Current Innovations and Future Trends. Edited by Sergio Sánchez and Arnold L. Demain.

Published in:

ChemMedChem, 2015, v. 10, n. 5, p. 925, doi. 10.1002/cmdc.201500099

By:

Schofield, Christopher

Publication type:

Article