Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 4

Results: 20

Synthesis and In Vitro Antiproliferative Activity of Amido and Amino Analogues of the Marine Alkaloid Isogranulatimide.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 607, doi. 10.1002/cmdc.201500025

By:

Lavrard, Hubert;
Salvetti, Béatrice;
Mathieu, Véronique;
Rodriguez, Frédéric;
Kiss, Robert;
Delfourne, Evelyne

Publication type:

Article

Fluorine in Drug Design: A Case Study with Fluoroanisoles.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 715, doi. 10.1002/cmdc.201402555

By:

Xing, Li;
Blakemore, David C.;
Narayanan, Arjun;
Unwalla, Ray;
Lovering, Frank;
Denny, R. Aldrin;
Zhou, Huanyu;
Bunnage, Mark E.

Publication type:

Article

Pharmacophore-Based Design of Novel Oxadiazoles as Selective Sphingosine-1-phosphate (S1P) Receptor Agonists with in vivo Efficacy.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 688, doi. 10.1002/cmdc.201402557

By:

Quattropani, Anna;
Sauer, Wolfgang H. B.;
Crosignani, Stefano;
Dorbais, Jerome;
Gerber, Patrick;
Gonzalez, Jerome;
Marin, Delphine;
Muzerelle, Mathilde;
Beltran, Fanny;
Nichols, Anthony;
Georgi, Katrin;
Schneider, Manfred;
Vitte, Pierre‐Alain;
Eligert, Valerie;
Novo‐Perez, Laurence;
Hantson, Jennifer;
Nock, Sebastien;
Carboni, Susanna;
de Souza, Adriano Luis Soares;
Arrighi, Jean‐François

Publication type:

Article

P2-Quinazolinones and Bis-Macrocycles as New Templates for Next-Generation Hepatitis C Virus NS3/4a Protease Inhibitors: Discovery of MK-2748 and MK-6325.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 727, doi. 10.1002/cmdc.201402558

By:

Rudd, Michael T.;
Butcher, John W.;
Nguyen, Kevin T.;
McIntyre, Charles J.;
Romano, Joseph J.;
Gilbert, Kevin F.;
Bush, Kimberly J.;
Liverton, Nigel J.;
Holloway, M. Katharine;
Harper, Steven;
Ferrara, Marco;
DiFilippo, Marcello;
Summa, Vincenzo;
Swestock, John;
Fritzen, Jeff;
Carroll, Steven S.;
Burlein, Christine;
DiMuzio, Jillian M.;
Gates, Adam;
Graham, Donald J.

Publication type:

Article

The Predicted Ensemble of Low-Energy Conformations of Human Somatostatin Receptor Subtype 5 and the Binding of Antagonists.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 650, doi. 10.1002/cmdc.201500023

By:

Dong, Sijia S.;
Abrol, Ravinder;
Goddard, William A.

Publication type:

Article

Selective Inhibitors of Glutathione Transferase P1 with Trioxane Structure as Anticancer Agents.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 629, doi. 10.1002/cmdc.201402553

By:

Bräutigam, Maria;
Teusch, Nicole;
Schenk, Tobias;
Sheikh, Miriam;
Aricioglu, Rocky Z.;
Borowski, Swantje H.;
Neudörfl, Jörg‐Martin;
Baumann, Ulrich;
Griesbeck, Axel G.;
Pietsch, Markus

Publication type:

Article

Inhibition of Neuroinflammation by Synthetic Androstene Derivatives Incorporating Amino Acid Methyl Esters on Activated BV-2 Microglia.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 610, doi. 10.1002/cmdc.201500027

By:

Wu, Jing;
Du, Juanjuan;
Gu, Ruinan;
Zhang, Li;
Zhen, Xuechu;
Li, Yuanchao;
Chen, Hongli;
Jiang, Biao;
Zheng, Longtai

Publication type:

Article

Cover Picture: Design and Synthesis of a MAO-B-Selectively Activated Prodrug Based on MPTP: A Mitochondria-Targeting Chemotherapeutic Agent for Treatment of Human Malignant Gliomas (ChemMedChem 4/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 585, doi. 10.1002/cmdc.201590007

By:

Sharpe, Martyn A.;
Han, Junyan;
Baskin, Alexandra M.;
Baskin, David S.

Publication type:

Article

Inside Cover: Looking for Efficient G-Quadruplex Ligands: Evidence for Selective Stabilizing Properties and Telomere Damage by Drug-Like Molecules (ChemMedChem 4/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 586, doi. 10.1002/cmdc.201590008

By:

Pagano, Bruno;
Amato, Jussara;
Iaccarino, Nunzia;
Cingolani, Chiara;
Zizza, Pasquale;
Biroccio, Annamaria;
Novellino, Ettore;
Randazzo, Antonio

Publication type:

Article

Graphical Abstract: ChemMedChem 4/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 4, p. 587, doi. 10.1002/cmdc.201590009
Publication type:: Article

In Vivo Targeting through Click Chemistry.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 617, doi. 10.1002/cmdc.201402527

By:

Brudno, Yevgeny;
Desai, Rajiv M.;
Kwee, Brian J.;
Joshi, Neel S.;
Aizenberg, Michael;
Mooney, David J.

Publication type:

Article

Functionalization of Fluorinated Benzenesulfonamides and Their Inhibitory Properties toward Carbonic Anhydrases.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 662, doi. 10.1002/cmdc.201402490

By:

Dudutienė, Virginija;
Zubrienė, Asta;
Smirnov, Alexey;
Timm, David D.;
Smirnovienė, Joana;
Kazokaitė, Justina;
Michailovienė, Vilma;
Zakšauskas, Audrius;
Manakova, Elena;
Gražulis, Saulius;
Matulis, Daumantas

Publication type:

Article

Scaffold Identification of a New Class of Potent and Selective BCRP Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 742, doi. 10.1002/cmdc.201402498

By:

Marighetti, Federico;
Steggemann, Kerstin;
Karbaum, Maria;
Wiese, Michael

Publication type:

Article

Design and Synthesis of a MAO-B-Selectively Activated Prodrug Based on MPTP: A Mitochondria-Targeting Chemotherapeutic Agent for Treatment of Human Malignant Gliomas.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 621, doi. 10.1002/cmdc.201402562

By:

Sharpe, Martyn A.;
Han, Junyan;
Baskin, Alexandra M.;
Baskin, David S.

Publication type:

Article

Bioisosteric Matrices for Ligands of Serotonin Receptors.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 601, doi. 10.1002/cmdc.201402563

By:

Warszycki, Dawid;
Mordalski, Stefan;
Staroń, Jakub;
Bojarski, Andrzej J.

Publication type:

Article

Back Cover: Selective Inhibitors of Glutathione Transferase P1 with Trioxane Structure as Anticancer Agents (ChemMedChem 4/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 756, doi. 10.1002/cmdc.201590010

By:

Bräutigam, Maria;
Teusch, Nicole;
Schenk, Tobias;
Sheikh, Miriam;
Aricioglu, Rocky Z.;
Borowski, Swantje H.;
Neudörfl, Jörg‐Martin;
Baumann, Ulrich;
Griesbeck, Axel G.;
Pietsch, Markus

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 4/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 4, p. 596, doi. 10.1002/cmdc.201580413
Publication type:: Article

Corrigendum: Design, Synthesis, and Structure-Activity Relationships of 3,4,5-Trisubstituted 4,5-Dihydro-1,2,4-oxadiazoles as TGR5 Agonists.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 593, doi. 10.1002/cmdc.201500054

By:

Zhu, Junjie;
Ye, Yangliang;
Ning, Mengmeng;
Mándi, Attila;
Feng, Ying;
Zou, Qingan;
Kurtán, Tibor;
Leng, Ying;
Shen, Jianhua

Publication type:

Article

Suppression of Problematic Compound Oligomerization by Cosolubilization of Nondetergent Sulfobetaines.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 736, doi. 10.1002/cmdc.201500057

By:

Mizukoshi, Yumiko;
Takeuchi, Koh;
Arutaki, Misa;
Takizawa, Takeshi;
Hanzawa, Hiroyuki;
Takahashi, Hideo;
Shimada, Ichio

Publication type:

Article

Looking for Efficient G-Quadruplex Ligands: Evidence for Selective Stabilizing Properties and Telomere Damage by Drug-Like Molecules.

Published in:

ChemMedChem, 2015, v. 10, n. 4, p. 640, doi. 10.1002/cmdc.201402552

By:

Pagano, Bruno;
Amato, Jussara;
Iaccarino, Nunzia;
Cingolani, Chiara;
Zizza, Pasquale;
Biroccio, Annamaria;
Novellino, Ettore;
Randazzo, Antonio

Publication type:

Article