Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 3

Results: 21

On the Metabolically Active Form of Metaglidasen: Improved Synthesis and Investigation of Its Peculiar Activity on Peroxisome Proliferator-Activated Receptors and Skeletal Muscles.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 555, doi. 10.1002/cmdc.201402462

By:

Laghezza, Antonio;
Montanari, Roberta;
Lavecchia, Antonio;
Piemontese, Luca;
Pochetti, Giorgio;
Iacobazzi, Vito;
Infantino, Vittoria;
Capelli, Davide;
De Bellis, Michela;
Liantonio, Antonella;
Pierno, Sabata;
Tortorella, Paolo;
Conte Camerino, Diana;
Loiodice, Fulvio

Publication type:

Article

Synthesis and Biological Evaluation of Ferrocenylquinoline as a Potential Antileishmanial Agent.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 546, doi. 10.1002/cmdc.201402537

By:

Yousuf, Md;
Mukherjee, Debarati;
Pal, Abhishek;
Dey, Somaditya;
Mandal, Supratim;
Pal, Chiranjib;
Adhikari, Susanta

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 3/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 3, p. 436, doi. 10.1002/cmdc.201580313
Publication type:: Article

Synthesis, Bioactivity, Docking and Molecular Dynamics Studies of Furan-Based Peptides as 20S Proteasome Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 498, doi. 10.1002/cmdc.201402484

By:

Sun, Qi;
Xu, Bo;
Niu, Yan;
Xu, Fengrong;
Liang, Lei;
Wang, Chao;
Yu, Jiapei;
Yan, Gang;
Wang, Wei;
Jin, Hongwei;
Xu, Ping

Publication type:

Article

Evaluation of tert-Butyl Isosteres: Case Studies of Physicochemical and Pharmacokinetic Properties, Efficacies, and Activities.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 461, doi. 10.1002/cmdc.201402502

By:

Westphal, Matthias V.;
Wolfstädter, Bernd T.;
Plancher, Jean‐Marc;
Gatfield, John;
Carreira, Erick M.

Publication type:

Article

Ligand-Biased and Probe-Dependent Modulation of Chemokine Receptor CXCR3 Signaling by Negative Allosteric Modulators.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 566, doi. 10.1002/cmdc.201402507

By:

Bernat, Viachaslau;
Brox, Regine;
Heinrich, Markus R.;
Auberson, Yves P.;
Tschammer, Nuska

Publication type:

Article

Design, Synthesis, and Biological Evaluation of Simplified Side Chain Hybrids of the Potent Actin Binding Polyketides Rhizopodin and Bistramide.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 470, doi. 10.1002/cmdc.201402508

By:

Herkommer, Daniel;
Dreisigacker, Sandra;
Sergeev, Galina;
Sasse, Florenz;
Gohlke, Holger;
Menche, Dirk

Publication type:

Article

Screening and In Vitro Testing of Antifolate Inhibitors of Human Cytosolic Serine Hydroxymethyltransferase.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 490, doi. 10.1002/cmdc.201500028

By:

Paiardini, Alessandro;
Fiascarelli, Alessio;
Rinaldo, Serena;
Daidone, Frederick;
Giardina, Giorgio;
Koes, David R.;
Parroni, Alessia;
Montini, Giulia;
Marani, Marina;
Paone, Alessio;
McDermott, Lee A.;
Contestabile, Roberto;
Cutruzzolà, Francesca

Publication type:

Article

Cover Picture: Merging Allosteric and Active Site Binding Motifs: De novo Generation of Target Selectivity and Potency via Natural-Product-Derived Fragments (ChemMedChem 3/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 425, doi. 10.1002/cmdc.201590003

By:

Lanz, Jan;
Riedl, Rainer

Publication type:

Article

Inside Cover: Evaluation of tert-Butyl Isosteres: Case Studies of Physicochemical and Pharmacokinetic Properties, Efficacies, and Activities (ChemMedChem 3/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 426, doi. 10.1002/cmdc.201590004

By:

Westphal, Matthias V.;
Wolfstädter, Bernd T.;
Plancher, Jean‐Marc;
Gatfield, John;
Carreira, Erick M.

Publication type:

Article

Graphical Abstract: ChemMedChem 3/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 3, p. 427, doi. 10.1002/cmdc.201590005
Publication type:: Article

Back Cover: Rational Design, Synthesis, and Biological Evaluation of Lactam-Bridged Gramicidin A Analogues: Discovery of a Low-Hemolytic Antibacterial Peptide (ChemMedChem 3/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 584, doi. 10.1002/cmdc.201590006

By:

Mao, Ji;
Kuranaga, Takefumi;
Hamamoto, Hiroshi;
Sekimizu, Kazuhisa;
Inoue, Masayuki

Publication type:

Article

Novel Tacrine-Grafted Ugi Adducts as Multipotent Anti-Alzheimer Drugs: A Synthetic Renewal in Tacrine-Ferulic Acid Hybrids.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 523, doi. 10.1002/cmdc.201402409

By:

Benchekroun, Mohamed;
Bartolini, Manuela;
Egea, Javier;
Romero, Alejandro;
Soriano, Elena;
Pudlo, Marc;
Luzet, Vincent;
Andrisano, Vincenza;
Jimeno, María‐Luisa;
López, Manuela G.;
Wehle, Sarah;
Gharbi, Tijani;
Refouvelet, Bernard;
de Andrés, Lucía;
Herrera‐Arozamena, Clara;
Monti, Barbara;
Bolognesi, Maria Laura;
Rodríguez‐Franco, María Isabel;
Decker, Michael;
Marco‐Contelles, José

Publication type:

Article

Rational Design, Synthesis, and Biological Evaluation of Lactam-Bridged Gramicidin A Analogues: Discovery of a Low-Hemolytic Antibacterial Peptide.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 540, doi. 10.1002/cmdc.201402473

By:

Mao, Ji;
Kuranaga, Takefumi;
Hamamoto, Hiroshi;
Sekimizu, Kazuhisa;
Inoue, Masayuki

Publication type:

Article

Computer-Guided Design, Synthesis, and Biological Evaluation of Quinoxalinebisarylureas as FLT3 Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 511, doi. 10.1002/cmdc.201402477

By:

Göring, Stefan;
Bensinger, Dennis;
Naumann, Eva C.;
Schmidt, Boris

Publication type:

Article

Merging Allosteric and Active Site Binding Motifs: De novo Generation of Target Selectivity and Potency via Natural-Product-Derived Fragments.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 451, doi. 10.1002/cmdc.201402478

By:

Lanz, Jan;
Riedl, Rainer

Publication type:

Article

Inhibitors of Molecular Chaperones as Therapeutic Agents. Edited by Timothy D. Machajewski and Zhenhai Gao.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 581, doi. 10.1002/cmdc.201402540

By:

Kitson, Russell R. A.

Publication type:

Article

Drug Discovery Summit: 11<sup>th</sup> Swiss Course on Medicinal Chemistry.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 575, doi. 10.1002/cmdc.201402543

By:

Frei, Priska;
Navarra, Giulio;
Sager, Christoph P.;
Silbermann, Marleen;
Varga, Norbert;
Wamhoff, Eike‐Christian

Publication type:

Article

Macrocycles in Drug Discovery. Edited by Jeremy I. Levin.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 580, doi. 10.1002/cmdc.201500013

By:

Kihlberg, Jan

Publication type:

Article

Preclinical Characterization of Acyl Sulfonimidamides: Potential Carboxylic Acid Bioisosteres with Tunable Properties.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 455, doi. 10.1002/cmdc.201402497

By:

Borhade, Sanjay R.;
Svensson, Richard;
Brandt, Peter;
Artursson, Per;
Arvidsson, Per I.;
Sandström, Anja

Publication type:

Article

Natural Products as Zinc-Dependent Histone Deacetylase Inhibitors.

Published in:

ChemMedChem, 2015, v. 10, n. 3, p. 441, doi. 10.1002/cmdc.201402460

By:

Tan, Shuai;
Liu, Zhao‐Peng

Publication type:

Article