Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 10

Results: 23

Investigating the Selectivity of Metalloenzyme Inhibitors in the Presence of Competing Metalloproteins.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1733, doi. 10.1002/cmdc.201500293

By:

Chen, Yao;
Cohen, Seth M.

Publication type:

Article

Membrane-Active Small Molecules: Designs Inspired by Antimicrobial Peptides.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1606, doi. 10.1002/cmdc.201500299

By:

Ghosh, Chandradhish;
Haldar, Jayanta

Publication type:

Article

Thermodynamics and Kinetics of Drug Binding. Edited by György M. Keseru and David C. Swinney.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1764, doi. 10.1002/cmdc.201500364

By:

Geschwindner, Stefan

Publication type:

Article

Discovery of Novel, Potent, and Specific Cell-Death Inducers in the Jurkat Acute Lymphoblastic Leukemia Cell Line.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1700, doi. 10.1002/cmdc.201500245

By:

Carosati, Emanuele;
van den Höfel, Natascha;
Reif, Manuela;
Randazzo, Giuseppe Marco;
Stanitzki, Bettina;
Stevens, Julia;
Gabbert, Helmut E.;
Cruciani, Gabriele;
Mannhold, Raimund;
Mahotka, Csaba

Publication type:

Article

(−)-Tarchonanthuslactone: Design of New Analogues, Evaluation of their Antiproliferative Activity on Cancer Cell Lines, and Preliminary Mechanistic Studies.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1687, doi. 10.1002/cmdc.201500246

By:

Toneto Novaes, Luiz Fernando;
Martins Avila, Carolina;
Pelizzaro‐Rocha, Karin Juliane;
Vendramini‐Costa, Débora Barbosa;
Pereira Dias, Marina;
Barbosa Trivella, Daniela Barreto;
Ernesto de Carvalho, João;
Ferreira‐Halder, Carmen Veríssima;
Pilli, Ronaldo Aloise

Publication type:

Article

A Bisbenzamidine Phosphonate as a Janus-faced Inhibitor for Trypsin-like Serine Proteases.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1641, doi. 10.1002/cmdc.201500319

By:

Häußler, Daniela;
Scheidt, Tamara;
Stirnberg, Marit;
Steinmetzer, Torsten;
Gütschow, Michael

Publication type:

Article

Cover Picture: Synthesis and Evaluation of Novel Acyclic Nucleoside Phosphonates as Inhibitors of Plasmodium falciparum and Human 6-Oxopurine Phosphoribosyltransferases (ChemMedChem 10/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1589, doi. 10.1002/cmdc.201500388

By:

Kaiser, Martin M.;
Hocková, Dana;
Wang, Tzu‐Hsuan;
Dračínský, Martin;
Poštová‐Slavětínská, Lenka;
Procházková, Eliška;
Edstein, Michael D.;
Chavchich, Marina;
Keough, Dianne T.;
Guddat, Luke W.;
Janeba, Zlatko

Publication type:

Article

Inside Cover: Synthesis of 2-[18F]Fluoro-2-deoxyisosorbide 5-mononitrate and Assessment of Its in vivo Biodistribution as Determined by Dynamic Positron Emission Tomography (PET) (ChemMedChem 10/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1590, doi. 10.1002/cmdc.201500389

By:

Santschi, Nico;
Wagner, Stefan;
Daniliuc, Constantin;
Hermann, Sven;
Schäfers, Michael;
Gilmour, Ryan

Publication type:

Article

Phage Selection of Bicyclic Peptide Ligands of the Notch1 Receptor.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1754, doi. 10.1002/cmdc.201500261

By:

Urech‐Varenne, Charlotte;
Radtke, Freddy;
Heinis, Christian

Publication type:

Article

Graphical Abstract: ChemMedChem 10/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 10, p. 1591, doi. 10.1002/cmdc.201581011
Publication type:: Article

Spotlights on our sister journals: ChemMedChem 10/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 10, p. 1600, doi. 10.1002/cmdc.201581013
Publication type:: Article

Discovery, Synthesis, and Optimization of Diarylisoxazole-3-carboxamides as Potent Inhibitors of the Mitochondrial Permeability Transition Pore.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1655, doi. 10.1002/cmdc.201500284

By:

Roy, Sudeshna;
Šileikytė, Justina;
Schiavone, Marco;
Neuenswander, Benjamin;
Argenton, Francesco;
Aubé, Jeffrey;
Hedrick, Michael P.;
Chung, Thomas D. Y.;
Forte, Michael A.;
Bernardi, Paolo;
Schoenen, Frank J.

Publication type:

Article

Design, Synthesis, and Evaluation of an 18F-Labeled Radiotracer Based on Celecoxib-NBD for Positron Emission Tomography (PET) Imaging of Cyclooxygenase-2 (COX-2).

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1635, doi. 10.1002/cmdc.201500287

By:

Kaur, Jatinder;
Tietz, Ole;
Bhardwaj, Atul;
Marshall, Alison;
Way, Jenilee;
Wuest, Melinda;
Wuest, Frank

Publication type:

Article

Successful Drug Discovery. Edited by Janos Fischer.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1762, doi. 10.1002/cmdc.201500351

By:

Gabriel, Tobias

Publication type:

Article

Pyrazolopyrimidines: Potent Inhibitors Targeting the Capsid of Rhino- and Enteroviruses.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1629, doi. 10.1002/cmdc.201500304

By:

Makarov, Vadim A.;
Braun, Heike;
Richter, Martina;
Riabova, Olga B.;
Kirchmair, Johannes;
Kazakova, Elena S.;
Seidel, Nora;
Wutzler, Peter;
Schmidtke, Michaela

Publication type:

Article

Synthesis and Evaluation of Novel Acyclic Nucleoside Phosphonates as Inhibitors of Plasmodium falciparum and Human 6-Oxopurine Phosphoribosyltransferases.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1707, doi. 10.1002/cmdc.201500322

By:

Kaiser, Martin M.;
Hocková, Dana;
Wang, Tzu‐Hsuan;
Dračínský, Martin;
Poštová‐Slavětínská, Lenka;
Procházková, Eliška;
Edstein, Michael D.;
Chavchich, Marina;
Keough, Dianne T.;
Guddat, Luke W.;
Janeba, Zlatko

Publication type:

Article

Antitargets and Drug Safety. Edited by László Urbán, Vinod F. Patel, and Roy J. Vaz.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1763, doi. 10.1002/cmdc.201500324

By:

Schmidt, Friedemann

Publication type:

Article

Back Cover: Lipopeptide Nanoparticles: Development of Vaccines against Hookworm Parasite (ChemMedChem 10/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1768, doi. 10.1002/cmdc.201500390

By:

Fuaad, Abdullah A. H. Ahmad;
Pearson, Mark S.;
Pickering, Darren A.;
Becker, Luke;
Zhao, Guangzu;
Loukas, Alex C.;
Skwarczynski, Mariusz;
Toth, Istvan

Publication type:

Article

Potent Synergy between Spirocyclic Pyrrolidinoindolinones and Fluconazole against Candida albicans.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1672, doi. 10.1002/cmdc.201500271

By:

Premachandra, Ilandari Dewage Udara Anulal;
Scott, Kevin A.;
Shen, Chengtian;
Wang, Fuqiang;
Lane, Shelley;
Liu, Haoping;
Van Vranken, David L.

Publication type:

Article

Synthesis of 2-[18F]Fluoro-2-deoxyisosorbide 5-mononitrate and Assessment of Its in vivo Biodistribution as Determined by Dynamic Positron Emission Tomography (PET).

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1724, doi. 10.1002/cmdc.201500275

By:

Santschi, Nico;
Wagner, Stefan;
Daniliuc, Constantin;
Hermann, Sven;
Schäfers, Michael;
Gilmour, Ryan

Publication type:

Article

Enzymatically Cleavable siRNA Prodrugs: a New Paradigm for the Intracellular Delivery of RNA-Based Therapeutics.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1625, doi. 10.1002/cmdc.201500279

By:

Ducho, Christian

Publication type:

Article

Lipopeptide Nanoparticles: Development of Vaccines against Hookworm Parasite.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1647, doi. 10.1002/cmdc.201500227

By:

Fuaad, Abdullah A. H. Ahmad;
Pearson, Mark S.;
Pickering, Darren A.;
Becker, Luke;
Zhao, Guangzu;
Loukas, Alex C.;
Skwarczynski, Mariusz;
Toth, Istvan

Publication type:

Article

Innovative Disulfide Esters of Dithiocarbamic Acid as Women-Controlled Contraceptive Microbicides: A Bioisosterism Approach.

Published in:

ChemMedChem, 2015, v. 10, n. 10, p. 1739, doi. 10.1002/cmdc.201500291

By:

Mandalapu, Dhanaraju;
Lal, Nand;
Kumar, Lokesh;
Kushwaha, Bhavana;
Gupta, Sonal;
Kumar, Lalit;
Bala, Veenu;
Yadav, Santosh K.;
Singh, Pratiksha;
Singh, Nidhi;
Maikhuri, Jagdamba P.;
Sankhwar, Satya N.;
Shukla, Praveen K.;
Siddiqi, Imran;
Gupta, Gopal;
Sharma, Vishnu L.

Publication type:

Article

Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 10

Investigating the Selectivity of Metalloenzyme Inhibitors in the Presence of Competing Metalloproteins.

Membrane-Active Small Molecules: Designs Inspired by Antimicrobial Peptides.

Thermodynamics and Kinetics of Drug Binding. Edited by György M. Keseru and David C. Swinney.

Discovery of Novel, Potent, and Specific Cell-Death Inducers in the Jurkat Acute Lymphoblastic Leukemia Cell Line.

(−)-Tarchonanthuslactone: Design of New Analogues, Evaluation of their Antiproliferative Activity on Cancer Cell Lines, and Preliminary Mechanistic Studies.

A Bisbenzamidine Phosphonate as a Janus-faced Inhibitor for Trypsin-like Serine Proteases.

Cover Picture: Synthesis and Evaluation of Novel Acyclic Nucleoside Phosphonates as Inhibitors of Plasmodium falciparum and Human 6-Oxopurine Phosphoribosyltransferases (ChemMedChem 10/2015).

Inside Cover: Synthesis of 2-[<sup>18</sup>F]Fluoro-2-deoxyisosorbide 5-mononitrate and Assessment of Its in vivo Biodistribution as Determined by Dynamic Positron Emission Tomography (PET) (ChemMedChem 10/2015).

Phage Selection of Bicyclic Peptide Ligands of the Notch1 Receptor.

Graphical Abstract: ChemMedChem 10/2015.

Spotlights on our sister journals: ChemMedChem 10/2015.

Discovery, Synthesis, and Optimization of Diarylisoxazole-3-carboxamides as Potent Inhibitors of the Mitochondrial Permeability Transition Pore.

Design, Synthesis, and Evaluation of an <sup>18</sup>F-Labeled Radiotracer Based on Celecoxib-NBD for Positron Emission Tomography (PET) Imaging of Cyclooxygenase-2 (COX-2).

Successful Drug Discovery. Edited by Janos Fischer.

Pyrazolopyrimidines: Potent Inhibitors Targeting the Capsid of Rhino- and Enteroviruses.

Synthesis and Evaluation of Novel Acyclic Nucleoside Phosphonates as Inhibitors of Plasmodium falciparum and Human 6-Oxopurine Phosphoribosyltransferases.

Antitargets and Drug Safety. Edited by László Urbán, Vinod F. Patel, and Roy J. Vaz.

Back Cover: Lipopeptide Nanoparticles: Development of Vaccines against Hookworm Parasite (ChemMedChem 10/2015).

Potent Synergy between Spirocyclic Pyrrolidinoindolinones and Fluconazole against Candida albicans.

Synthesis of 2-[<sup>18</sup>F]Fluoro-2-deoxyisosorbide 5-mononitrate and Assessment of Its in vivo Biodistribution as Determined by Dynamic Positron Emission Tomography (PET).

Enzymatically Cleavable siRNA Prodrugs: a New Paradigm for the Intracellular Delivery of RNA-Based Therapeutics.

Lipopeptide Nanoparticles: Development of Vaccines against Hookworm Parasite.

Innovative Disulfide Esters of Dithiocarbamic Acid as Women-Controlled Contraceptive Microbicides: A Bioisosterism Approach.