Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 1

Results: 28

Identification of Green Tea Catechins as Potent Inhibitors of the Polo-Box Domain of Polo-Like kinase 1.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 158, doi. 10.1002/cmdc.201402284

By:

Shan, Hong‐Mei;
Shi, Yanxia;
Quan, Junmin

Publication type:

Article

Conjugation of Cisplatin Analogues and Cyclooxygenase Inhibitors to Overcome Cisplatin Resistance.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 183, doi. 10.1002/cmdc.201402353

By:

Neumann, Wilma;
Crews, Brenda C.;
Sárosi, Menyhárt B.;
Daniel, Cristina M.;
Ghebreselasie, Kebreab;
Scholz, Matthias S.;
Marnett, Lawrence J.;
Hey‐Hawkins, Evamarie

Publication type:

Article

Targeting a Dynamic Protein-Protein Interaction: Fragment Screening against the Malaria Myosin A Motor Complex.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 134, doi. 10.1002/cmdc.201402357

By:

Douse, Christopher H.;
Vrielink, Nina;
Wenlin, Zhang;
Cota, Ernesto;
Tate, Edward W.

Publication type:

Article

Design of gem-Difluoro- bis-Tetrahydrofuran as P2 Ligand for HIV-1 Protease Inhibitors to Improve Brain Penetration: Synthesis, X-ray Studies, and Biological Evaluation.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 107, doi. 10.1002/cmdc.201402358

By:

Ghosh, Arun K.;
Yashchuk, Sofiya;
Mizuno, Akira;
Chakraborty, Nilanjana;
Agniswamy, Johnson;
Wang, Yuan‐Fang;
Aoki, Manabu;
Gomez, Pedro Miguel Salcedo;
Amano, Masayuki;
Weber, Irene T.;
Mitsuya, Hiroaki

Publication type:

Article

Evaluating p97 Inhibitor Analogues for Their Domain Selectivity and Potency against the p97-p47 Complex.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 52, doi. 10.1002/cmdc.201402420

By:

Fang, Chen‐Jie;
Gui, Lin;
Zhang, Xiaoyi;
Moen, Derek R.;
Li, Kelin;
Frankowski, Kevin J.;
Lin, Henry J.;
Schoenen, Frank J.;
Chou, Tsui‐Fen

Publication type:

Article

Cover Picture: ChemMedChem has reached...︁ The Big TEN! (ChemMedChem 1/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 1, doi. 10.1002/cmdc.201490048

By:

Williams, Scott D.;
Ortúzar, Natalia

Publication type:

Article

Concise Notice to Authors.

Published in:: ChemMedChem, 2015, v. 10, n. 1, p. 22, doi. 10.1002/cmdc.201490049
Publication type:: Article

ChemMedChem has reached...︁ The Big TEN!

Published in:

2015

By:

Williams, Scott D.;
Ortúzar, Natalia

Publication type:

Editorial

Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 144, doi. 10.1002/cmdc.201402371

By:

Castellano, Sabrina;
Milite, Ciro;
Feoli, Alessandra;
Viviano, Monica;
Mai, Antonello;
Novellino, Ettore;
Tosco, Alessandra;
Sbardella, Gianluca

Publication type:

Article

[3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 83, doi. 10.1002/cmdc.201402344

By:

Baumeister, Paul;
Erdmann, Daniela;
Biselli, Sabrina;
Kagermeier, Nicole;
Elz, Sigurd;
Bernhardt, Günther;
Buschauer, Armin

Publication type:

Article

Stimuli-Responsive Polymeric Nanoparticles for Nanomedicine.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 24, doi. 10.1002/cmdc.201402290

By:

Crucho, Carina I. C.

Publication type:

Article

Nucleoside Mono- and Diphosphate Prodrugs of 2′,3′-Dideoxyuridine and 2′,3′-Dideoxy-2′,3′-didehydrouridine.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 94, doi. 10.1002/cmdc.201402295

By:

Pertenbreiter, Florian;
Balzarini, Jan;
Meier, Chris

Publication type:

Article

Design and Structural Analysis of Aromatic Inhibitors of Type II Dehydroquinase from Mycobacterium tuberculosis.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 116, doi. 10.1002/cmdc.201402298

By:

Howard, Nigel I.;
Dias, Marcio V. B.;
Peyrot, Fabienne;
Chen, Liuhong;
Schmidt, Marco F.;
Blundell, Tom L.;
Abell, Chris

Publication type:

Article

Discovery and Characterization of 2-(Cyclopropanesulfonamido)- N-(2-ethoxyphenyl)benzamide, ML382: a Potent and Selective Positive Allosteric Modulator of MrgX1.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 57, doi. 10.1002/cmdc.201402277

By:

Wen, Wandong;
Wang, Yan;
Li, Zhe;
Tseng, Pang‐Yen;
McManus, Owen B.;
Wu, Meng;
Li, Min;
Lindsley, Craig W.;
Dong, Xinzhong;
Hopkins, Corey R.

Publication type:

Article

Drug Delivery to the Malaria Parasite Using an Arterolane-Like Scaffold.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 47, doi. 10.1002/cmdc.201402362

By:

Fontaine, Shaun D.;
Spangler, Benjamin;
Gut, Jiri;
Lauterwasser, Erica M. W.;
Rosenthal, Philip J.;
Renslo, Adam R.

Publication type:

Article

Receptor-Mediated Uptake of Boron-Rich Neuropeptide Y Analogues for Boron Neutron Capture Therapy.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 164, doi. 10.1002/cmdc.201402368

By:

Ahrens, Verena M.;
Frank, René;
Boehnke, Solveig;
Schütz, Christian L.;
Hampel, Gabriele;
Iffland, Dorothée S.;
Bings, Nicolas H.;
Hey‐Hawkins, Evamarie;
Beck‐Sickinger, Annette G.

Publication type:

Article

Carborane-Derived Local Anesthetics are Isomer Dependent.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 62, doi. 10.1002/cmdc.201402369

By:

Kracke, George R.;
VanGordon, Monika R.;
Sevryugina, Yulia V.;
Kueffer, Peter J.;
Kabytaev, Kuanysh;
Jalisatgi, Satish S.;
Hawthorne, M. Frederick

Publication type:

Article

The Discovery of a Highly Selective 5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3- d]pyrimidin-4(3 H)-one SIRT2 Inhibitor that is Neuroprotective in an in vitro Parkinson's Disease Model.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 69, doi. 10.1002/cmdc.201402431

By:

Di Fruscia, Paolo;
Zacharioudakis, Emmanouil;
Liu, Chang;
Moniot, Sébastien;
Laohasinnarong, Sasiwan;
Khongkow, Mattaka;
Harrison, Ian F.;
Koltsida, Konstantina;
Reynolds, Christopher R.;
Schmidtkunz, Karin;
Jung, Manfred;
Chapman, Kathryn L.;
Steegborn, Clemens;
Dexter, David T.;
Sternberg, Michael J. E.;
Lam, Eric W.‐F.;
Fuchter, Matthew J.

Publication type:

Article

Nucleic Acid Aptamer-Mediated Drug Delivery for Targeted Cancer Therapy.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 39, doi. 10.1002/cmdc.201402312

By:

Zhu, Huijie;
Li, Jin;
Zhang, Xiao‐Bing;
Ye, Mao;
Tan, Weihong

Publication type:

Article

3-Deazaneplanocin A and Neplanocin A Analogues and Their Effects on Apoptotic Cell Death.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 173, doi. 10.1002/cmdc.201402315

By:

Tam, Eric K. W.;
Nguyen, Tuan Minh;
Lim, Cheryl Z. H.;
Lee, Puay Leng;
Li, Zhimei;
Jiang, Xia;
Santhanakrishnan, Sridhar;
Tan, Tiong Wei;
Goh, Yi Ling;
Wong, Sze Yue;
Yang, Haiyan;
Ong, Esther H. Q.;
Hill, Jeffrey;
Yu, Qiang;
Chai, Christina L. L.

Publication type:

Article

Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 2, doi. 10.1002/cmdc.201490050

By:

Castellano, Sabrina;
Milite, Ciro;
Feoli, Alessandra;
Viviano, Monica;
Mai, Antonello;
Novellino, Ettore;
Tosco, Alessandra;
Sbardella, Gianluca

Publication type:

Article

Graphical Abstract: ChemMedChem 1/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 1, p. 3, doi. 10.1002/cmdc.201490051
Publication type:: Article

Back Cover: [3H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H2 Receptor Antagonist (ChemMedChem 1/2015).

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 212, doi. 10.1002/cmdc.201490052

By:

Baumeister, Paul;
Erdmann, Daniela;
Biselli, Sabrina;
Kagermeier, Nicole;
Elz, Sigurd;
Bernhardt, Günther;
Buschauer, Armin

Publication type:

Article

Development of Second-Generation Small-Molecule RhoA Inhibitors with Enhanced Water Solubility, Tissue Potency, and Significant in vivo Efficacy.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 193, doi. 10.1002/cmdc.201402386

By:

Ma, Sheng;
Deng, Jing;
Li, Baoli;
Li, Xiujiang;
Yan, Zhaowei;
Zhu, Jin;
Chen, Gang;
Wang, Zhong;
Jiang, Hualiang;
Miao, Liyan;
Li, Jian

Publication type:

Article

Advanced Drug Delivery. Edited by Ashim K. Mitra, Chi H. Lee, Kun Chen.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 209, doi. 10.1002/cmdc.201402388

By:

Barbu, Eugen

Publication type:

Article

Scaffold Hopping in Medicinal Chemistry. Edited by Nathan Brown.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 207, doi. 10.1002/cmdc.201402450

By:

Holliday, John

Publication type:

Article

In vivo Models for Drug Discovery. Edited by Jose Miguel Vela, Rafael Maldonado, and Michel Hamon.

Published in:

ChemMedChem, 2015, v. 10, n. 1, p. 208, doi. 10.1002/cmdc.201402451

By:

Vogt, Andreas

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 1/2015.

Published in:: ChemMedChem, 2015, v. 10, n. 1, p. 18, doi. 10.1002/cmdc.201580113
Publication type:: Article

Works matching IS 18607179 AND DT 2015 AND VI 10 AND IP 1

Identification of Green Tea Catechins as Potent Inhibitors of the Polo-Box Domain of Polo-Like kinase 1.

Conjugation of Cisplatin Analogues and Cyclooxygenase Inhibitors to Overcome Cisplatin Resistance.

Targeting a Dynamic Protein-Protein Interaction: Fragment Screening against the Malaria Myosin A Motor Complex.

Design of gem-Difluoro- bis-Tetrahydrofuran as P2 Ligand for HIV-1 Protease Inhibitors to Improve Brain Penetration: Synthesis, X-ray Studies, and Biological Evaluation.

Evaluating p97 Inhibitor Analogues for Their Domain Selectivity and Potency against the p97-p47 Complex.

Cover Picture: ChemMedChem has reached...︁ The Big TEN! (ChemMedChem 1/2015).

Concise Notice to Authors.

ChemMedChem has reached...︁ The Big TEN!

Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF.

[<sup>3</sup>H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H<sub>2</sub> Receptor Antagonist.

Stimuli-Responsive Polymeric Nanoparticles for Nanomedicine.

Nucleoside Mono- and Diphosphate Prodrugs of 2′,3′-Dideoxyuridine and 2′,3′-Dideoxy-2′,3′-didehydrouridine.

Design and Structural Analysis of Aromatic Inhibitors of Type II Dehydroquinase from Mycobacterium tuberculosis.

Discovery and Characterization of 2-(Cyclopropanesulfonamido)- N-(2-ethoxyphenyl)benzamide, ML382: a Potent and Selective Positive Allosteric Modulator of MrgX1.

Drug Delivery to the Malaria Parasite Using an Arterolane-Like Scaffold.

Receptor-Mediated Uptake of Boron-Rich Neuropeptide Y Analogues for Boron Neutron Capture Therapy.

Carborane-Derived Local Anesthetics are Isomer Dependent.

The Discovery of a Highly Selective 5,6,7,8-Tetrahydrobenzo[4,5]thieno[2,3- d]pyrimidin-4(3 H)-one SIRT2 Inhibitor that is Neuroprotective in an in vitro Parkinson's Disease Model.

Nucleic Acid Aptamer-Mediated Drug Delivery for Targeted Cancer Therapy.

3-Deazaneplanocin A and Neplanocin A Analogues and Their Effects on Apoptotic Cell Death.

Inside Cover: Identification of Structural Features of 2-Alkylidene-1,3-Dicarbonyl Derivatives that Induce Inhibition and/or Activation of Histone Acetyltransferases KAT3B/p300 and KAT2B/PCAF (ChemMedChem 1/2015).

Graphical Abstract: ChemMedChem 1/2015.

Back Cover: [<sup>3</sup>H]UR-DE257: Development of a Tritium-Labeled Squaramide-Type Selective Histamine H<sub>2</sub> Receptor Antagonist (ChemMedChem 1/2015).

Development of Second-Generation Small-Molecule RhoA Inhibitors with Enhanced Water Solubility, Tissue Potency, and Significant in vivo Efficacy.

Advanced Drug Delivery. Edited by Ashim K. Mitra, Chi H. Lee, Kun Chen.

Scaffold Hopping in Medicinal Chemistry. Edited by Nathan Brown.

In vivo Models for Drug Discovery. Edited by Jose Miguel Vela, Rafael Maldonado, and Michel Hamon.

Spotlights on our sister journals: ChemMedChem 1/2015.