Works matching IS 18607179 AND DT 2014 AND VI 9 AND IP 7

Results: 34

Anti-Dengue-Virus Activity and Structure-Activity Relationship Studies of Lycorine Derivatives.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1522, doi. 10.1002/cmdc.201300505

By:

Wang, Peng;
Li, Lin‐Feng;
Wang, Qing‐Yin;
Shang, Lu‐Qing;
Shi, Pei‐Yong;
Yin, Zheng

Publication type:

Article

Retracted: Synthesis and Cytotoxic Activity of 2-Anilinopyridine-3-Acrylamides as Tubulin Polymerization Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1615, doi. 10.1002/cmdc.201400036

By:

Kamal, Ahmed;
Ashraf, Md.;
Khan, M. Naseer Ahmed;
Nimbarte, Vijaykumar D.;
Faazil, Shaikh;
Subba Reddy, N. V.;
Taj, Shaik

Publication type:

Article

Development and Screening of a Series of Antibody-Conjugated and Silica-Coated Iron Oxide Nanoparticles for Targeting the Prostate-Specific Membrane Antigen.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1356, doi. 10.1002/cmdc.201300549

By:

Mukherjee, Amarnath;
Darlington, Thomas;
Baldwin, Richard;
Holz, Charles;
Olson, Sage;
Kulkarni, Prakash;
DeWeese, Theodore L.;
Getzenberg, Robert H.;
Ivkov, Robert;
Lupold, Shawn E.

Publication type:

Article

Cytotoxic Triosmium Carbonyl Clusters: A Structure-Activity Relationship Study.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1453, doi. 10.1002/cmdc.201300394

By:

Lee, Hui Zhi Shirley;
Leong, Weng Kee;
Top, Siden;
Vessières, Anne

Publication type:

Article

Anticancer Potential of (Pentamethylcyclopentadienyl)chloridoiridium(III) Complexes Bearing κ P and κ P,κ S-Coordinated Ph2PCH2CH2CH2S(O) xPh ( x=0-2) Ligands.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1586, doi. 10.1002/cmdc.201300479

By:

Ludwig, Gerd;
Ranđelović, Ivan;
Maksimović‐Ivanić, Danijela;
Mijatović, Sanja;
Bulatović, Mirna Z.;
Miljković, Djordje;
Korb, Marcus;
Lang, Heinrich;
Steinborn, Dirk;
Kaluđerović, Goran N.

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 7/2014.

Published in:: ChemMedChem, 2014, v. 9, n. 7, p. 1346, doi. 10.1002/cmdc.201490026
Publication type:: Article

Targeting Cystalysin, a Virulence Factor of Treponema denticola-Supported Periodontitis.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1501, doi. 10.1002/cmdc.201300527

By:

Spyrakis, Francesca;
Cellini, Barbara;
Bruno, Stefano;
Benedetti, Paolo;
Carosati, Emanuele;
Cruciani, Gabriele;
Micheli, Fabrizio;
Felici, Antonio;
Cozzini, Pietro;
Kellogg, Glen E.;
Voltattorni, Carla Borri;
Mozzarelli, Andrea

Publication type:

Article

Development of 3-Phenyl- N-(2-(3-phenylureido)ethyl)-thiophene-2-sulfonamide Compounds as Inhibitors of Antiapoptotic Bcl-2 Family Proteins.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1436, doi. 10.1002/cmdc.201400058

By:

Yang, Chengwen;
Chen, Sha;
Zhou, Mi;
Li, Yan;
Li, Yangfeng;
Zhang, Zhengxi;
Liu, Zhen;
Ba, Qian;
Li, Jingquan;
Wang, Hui;
Yan, Xiaomei;
Ma, Dawei;
Wang, Renxiao

Publication type:

Article

Bis(dipyridophenazine)(2-(2′-pyridyl)pyrimidine-4-carboxylic acid)ruthenium(II) Hexafluorophosphate: A Lesson in Stubbornness.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1419, doi. 10.1002/cmdc.201400029

By:

Joshi, Tanmaya;
Pierroz, Vanessa;
Ferrari, Stefano;
Gasser, Gilles

Publication type:

Article

Synthesis and Biological Evaluation of Imidazo[2,1- b][1,3,4]thiadiazole-Linked Oxindoles as Potent Tubulin Polymerization Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1463, doi. 10.1002/cmdc.201400069

By:

Kamal, Ahmed;
Rao, M. P. Narasimha;
Das, Pompi;
Swapna, P.;
Polepalli, Sowjanya;
Nimbarte, Vijaykumar D.;
Mullagiri, Kishore;
Kovvuri, Jeshma;
Jain, Nishant

Publication type:

Article

Fluorine-Containing 6,7-Dialkoxybiaryl-Based Inhibitors for Phosphodiesterase 10 A: Synthesis and in vitro Evaluation of Inhibitory Potency, Selectivity, and Metabolism.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1476, doi. 10.1002/cmdc.201300522

By:

Schwan, Gregor;
Barbar Asskar, Ghadir;
Höfgen, Norbert;
Kubicova, Lenka;
Funke, Uta;
Egerland, Ute;
Zahn, Michael;
Nieber, Karen;
Scheunemann, Matthias;
Sträter, Norbert;
Brust, Peter;
Briel, Detlef

Publication type:

Article

Insight into the Functional and Structural Properties of 3-Arylcoumarin as an Interesting Scaffold in Monoamine Oxidase B Inhibition.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1488, doi. 10.1002/cmdc.201300533

By:

Matos, Maria João;
Vilar, Santiago;
García‐Morales, Verónica;
Tatonetti, Nicholas P.;
Uriarte, Eugenio;
Santana, Lourdes;
Viña, Dolores

Publication type:

Article

Computational and Experimental Insight into the Molecular Mechanism of Carboxamide Inhibitors of Succinate-Ubquinone Oxidoreductase.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1512, doi. 10.1002/cmdc.201300456

By:

Zhu, Xiao‐Lei;
Xiong, Li;
Li, Hui;
Song, Xin‐Ya;
Liu, Jing‐Jing;
Yang, Guang‐Fu

Publication type:

Article

Graphical Abstract: ChemMedChem 7/2014.

Published in:: ChemMedChem, 2014, v. 9, n. 7, p. 1335, doi. 10.1002/cmdc.201490025
Publication type:: Article

Efficiently Detecting Metallodrug-Protein Adducts: Ion Trap versus Time-of-Flight Mass Analyzers.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1351, doi. 10.1002/cmdc.201400020

By:

Meier, Samuel M.;
Babak, Maria V.;
Keppler, Bernhard K.;
Hartinger, Christian G.

Publication type:

Article

1-(1 H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1534, doi. 10.1002/cmdc.201400042

By:

Hequet, Arnaud;
Burchak, Olga N.;
Jeanty, Matthieu;
Guinchard, Xavier;
Le Pihive, Emmanuelle;
Maigre, Laure;
Bouhours, Pascale;
Schneider, Dominique;
Maurin, Max;
Paris, Jean‐Marc;
Denis, Jean‐Noël;
Jolivalt, Claude

Publication type:

Article

Simplified Silvestrol Analogues with Potent Cytotoxic Activity.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1556, doi. 10.1002/cmdc.201400024

By:

Hawkins, Bill C.;
Lindqvist, Lisa M.;
Nhu, Duong;
Sharp, Phillip P.;
Segal, David;
Powell, Andrew K.;
Campbell, Michael;
Ryan, Eileen;
Chambers, Jennifer M.;
White, Jonathan M.;
Rizzacasa, Mark A.;
Lessene, Guillaume;
Huang, David C. S.;
Burns, Christopher J.

Publication type:

Article

Optimization of the Antiviral Potency and Lipophilicity of Halogenated 2,6-Diarylpyridinamines as a Novel Class of HIV-1 NNRTIS.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1546, doi. 10.1002/cmdc.201400075

By:

Wu, Zhi‐Yuan;
Liu, Na;
Qin, Bingjie;
Huang, Li;
Yu, Fei;
Qian, Keduo;
Morris‐Natschke, Susan L.;
Jiang, Shibo;
Chen, Chin Ho;
Lee, Kuo‐Hsiung;
Xie, Lan

Publication type:

Article

The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 2.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1387, doi. 10.1002/cmdc.201400046

By:

Wakenhut, Florian;
Tran, Thien Duc;
Pickford, Chris;
Shaw, Stephen;
Westby, Mike;
Smith‐Burchnell, Caroline;
Watson, Lesa;
Paradowski, Michael;
Milbank, Jared;
Stonehouse, David;
Cheung, Kathy;
Wybrow, Robert;
Daverio, Felice;
Crook, Samuel;
Statham, Keith;
Leese, David;
Stead, Darren;
Adam, Fiona;
Hay, Duncan;
Roberts, Lee R.

Publication type:

Article

Synthetic and Biological Studies of Tubulin Targeting C2-Substituted 7-Deazahypoxanthines Derived from Marine Alkaloid Rigidins.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1428, doi. 10.1002/cmdc.201300532

By:

Scott, Robert;
Karki, Menuka;
Reisenauer, Mary R.;
Rodrigues, Roberta;
Dasari, Ramesh;
Smith, W. Ross;
Pelly, Stephen C.;
van Otterlo, Willem A. L.;
Shuster, Charles B.;
Rogelj, Snezna;
Magedov, Igor V.;
Frolova, Liliya V.;
Kornienko, Alexander

Publication type:

Article

Xanthones from Swertia mussotii as Multitarget-Directed Antidiabetic Agents.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1374, doi. 10.1002/cmdc.201300507

By:

Zheng, Huan‐Huan;
Luo, Cui‐Ting;
Chen, Heru;
Lin, Juan‐Na;
Ye, Chun‐Ling;
Mao, Shuang‐Shuang;
Li, Yu‐Lin

Publication type:

Article

Efficient Acid-Catalyzed 18F/19F Fluoride Exchange of BODIPY Dyes.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1368, doi. 10.1002/cmdc.201300506

By:

Keliher, Edmund J.;
Klubnick, Jenna A.;
Reiner, Thomas;
Mazitschek, Ralph;
Weissleder, Ralph

Publication type:

Article

Cover Picture: Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery System (ChemMedChem 7/2014).

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1333, doi. 10.1002/cmdc.201490024

By:

Barile, Elisa;
Wang, Si;
Das, Swadesh K.;
Noberini, Roberta;
Dahl, Russell;
Stebbins, John L.;
Pasquale, Elena B.;
Fisher, Paul B.;
Pellecchia, Maurizio

Publication type:

Article

Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery System.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1403, doi. 10.1002/cmdc.201400067

By:

Barile, Elisa;
Wang, Si;
Das, Swadesh K.;
Noberini, Roberta;
Dahl, Russell;
Stebbins, John L.;
Pasquale, Elena B.;
Fisher, Paul B.;
Pellecchia, Maurizio

Publication type:

Article

The Integrin Ligand c(RGDf( NMe)Nal) Reduces Neointimal Hyperplasia in a Polymer-Free Drug-Eluting Stent System.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1413, doi. 10.1002/cmdc.201400078

By:

Rechenmacher, Florian;
Steigerwald, Kristin;
Laufer, Burkhardt;
Neubauer, Stefanie;
Kapp, Tobias G.;
Li, Liang;
Mas‐Moruno, Carlos;
Joner, Michael;
Kessler, Horst

Publication type:

Article

Small-Molecule Inhibitors of AF6 PDZ-Mediated Protein-Protein Interactions.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1458, doi. 10.1002/cmdc.201300553

By:

Vargas, Carolyn;
Radziwill, Gerald;
Krause, Gerd;
Diehl, Anne;
Keller, Sandro;
Kamdem, Nestor;
Czekelius, Constantin;
Kreuchwig, Annika;
Schmieder, Peter;
Doyle, Declan;
Moelling, Karin;
Hagen, Volker;
Schade, Markus;
Oschkinat, Hartmut

Publication type:

Article

'À la Carte' Peptide Shuttles: Tools to Increase Their Passage across the Blood-Brain Barrier.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1594, doi. 10.1002/cmdc.201300575

By:

Malakoutikhah, Morteza;
Guixer, Bernat;
Arranz‐Gibert, Pol;
Teixidó, Meritxell;
Giralt, Ernest

Publication type:

Article

The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 1.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1378, doi. 10.1002/cmdc.201400045

By:

Tran, Thien Duc;
Wakenhut, Florian;
Pickford, Chris;
Shaw, Stephen;
Westby, Mike;
Smith‐Burchnell, Caroline;
Watson, Lesa;
Paradowski, Michael;
Milbank, Jared;
Brimage, Rebecca A.;
Halstead, Rebecca;
Glen, Rebecca;
Wilson, Craig P.;
Adam, Fiona;
Hay, Duncan;
Chiva, Jean‐Yves;
Nichols, Carly;
Blakemore, David C.;
Gardner, Iain;
Dayal, Satish

Publication type:

Article

3-Aminoazetidin-2-one Derivatives as N-Acylethanolamine Acid Amidase (NAAA) Inhibitors Suitable for Systemic Administration.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1602, doi. 10.1002/cmdc.201300546

By:

Fiasella, Annalisa;
Nuzzi, Andrea;
Summa, Maria;
Armirotti, Andrea;
Tarozzo, Glauco;
Tarzia, Giorgio;
Mor, Marco;
Bertozzi, Fabio;
Bandiera, Tiziano;
Piomelli, Daniele

Publication type:

Article

Novel Heterobimetallic Radiotheranostic: Preparation, Activity, and Biodistribution.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1567, doi. 10.1002/cmdc.201300494

By:

Adriaenssens, Louis;
Liu, Qiang;
Chaux‐Picquet, Fanny;
Tasan, Semra;
Picquet, Michel;
Denat, Franck;
Le Gendre, Pierre;
Marques, Fernanda;
Fernandes, Célia;
Mendes, Filipa;
Gano, Lurdes;
Campello, Maria Paula Cabral;
Bodio, Ewen

Publication type:

Article

Back Cover: The Integrin Ligand c(RGDf( NMe)Nal) Reduces Neointimal Hyperplasia in a Polymer-Free Drug-Eluting Stent System (ChemMedChem 7/2014).

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1620, doi. 10.1002/cmdc.201490027

By:

Rechenmacher, Florian;
Steigerwald, Kristin;
Laufer, Burkhardt;
Neubauer, Stefanie;
Kapp, Tobias G.;
Li, Liang;
Mas‐Moruno, Carlos;
Joner, Michael;
Kessler, Horst

Publication type:

Article

Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2-Amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6 H-quinazolin-5-one Oxime.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1574, doi. 10.1002/cmdc.201400037

By:

Amici, Raffaella;
Bigogno, Chiara;
Boggio, Roberto;
Colombo, Andrea;
Courtney, Stephen M.;
Dal Zuffo, Roberto;
Dondio, Giulio;
Fusar, Fulvia;
Gagliardi, Stefania;
Minucci, Saverio;
Molteni, Marco;
Montalbetti, Christian A. G. N.;
Mortoni, Annalisa;
Varasi, Mario;
Vultaggio, Stefania;
Mercurio, Ciro

Publication type:

Article

Structural Optimization and Biological Screening of a Steroidal Scaffold Possessing Cucurbitacin-Like Functionalities as B-Raf Inhibitors.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1361, doi. 10.1002/cmdc.201300523

By:

Ahmed, Mahmoud S.;
Kopel, Lucas C.;
Halaweish, Fathi T.

Publication type:

Article

Stereoselective Reduction of 1- O-Isopropyloxygenipin Enhances Its Neuroprotective Activity in Neuronal Cells from Apoptosis Induced by Sodium Nitroprusside.

Published in:

ChemMedChem, 2014, v. 9, n. 7, p. 1397, doi. 10.1002/cmdc.201400051

By:

Wang, Rikang;
Yang, Jian;
Liao, Sufen;
Xiao, Gaokeng;
Luo, Jun;
Zhang, Lang;
Little, Peter J.;
Chen, Heru;
Zheng, Wenhua

Publication type:

Article

Works matching IS 18607179 AND DT 2014 AND VI 9 AND IP 7

Anti-Dengue-Virus Activity and Structure-Activity Relationship Studies of Lycorine Derivatives.

Retracted: Synthesis and Cytotoxic Activity of 2-Anilinopyridine-3-Acrylamides as Tubulin Polymerization Inhibitors.

Development and Screening of a Series of Antibody-Conjugated and Silica-Coated Iron Oxide Nanoparticles for Targeting the Prostate-Specific Membrane Antigen.

Cytotoxic Triosmium Carbonyl Clusters: A Structure-Activity Relationship Study.

Anticancer Potential of (Pentamethylcyclopentadienyl)chloridoiridium(III) Complexes Bearing κ P and κ P,κ S-Coordinated Ph<sub>2</sub>PCH<sub>2</sub>CH<sub>2</sub>CH<sub>2</sub>S(O)<sub> x</sub>Ph ( x=0-2) Ligands.

Spotlights on our sister journals: ChemMedChem 7/2014.

Targeting Cystalysin, a Virulence Factor of Treponema denticola-Supported Periodontitis.

Development of 3-Phenyl- N-(2-(3-phenylureido)ethyl)-thiophene-2-sulfonamide Compounds as Inhibitors of Antiapoptotic Bcl-2 Family Proteins.

Bis(dipyridophenazine)(2-(2′-pyridyl)pyrimidine-4-carboxylic acid)ruthenium(II) Hexafluorophosphate: A Lesson in Stubbornness.

Synthesis and Biological Evaluation of Imidazo[2,1- b][1,3,4]thiadiazole-Linked Oxindoles as Potent Tubulin Polymerization Inhibitors.

Fluorine-Containing 6,7-Dialkoxybiaryl-Based Inhibitors for Phosphodiesterase 10 A: Synthesis and in vitro Evaluation of Inhibitory Potency, Selectivity, and Metabolism.

Insight into the Functional and Structural Properties of 3-Arylcoumarin as an Interesting Scaffold in Monoamine Oxidase B Inhibition.

Computational and Experimental Insight into the Molecular Mechanism of Carboxamide Inhibitors of Succinate-Ubquinone Oxidoreductase.

Graphical Abstract: ChemMedChem 7/2014.

Efficiently Detecting Metallodrug-Protein Adducts: Ion Trap versus Time-of-Flight Mass Analyzers.

1-(1 H-Indol-3-yl)ethanamine Derivatives as Potent Staphylococcus aureus NorA Efflux Pump Inhibitors.

Simplified Silvestrol Analogues with Potent Cytotoxic Activity.

Optimization of the Antiviral Potency and Lipophilicity of Halogenated 2,6-Diarylpyridinamines as a Novel Class of HIV-1 NNRTIS.

The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 2.

Synthetic and Biological Studies of Tubulin Targeting C2-Substituted 7-Deazahypoxanthines Derived from Marine Alkaloid Rigidins.

Xanthones from Swertia mussotii as Multitarget-Directed Antidiabetic Agents.

Efficient Acid-Catalyzed <sup>18</sup>F/<sup>19</sup>F Fluoride Exchange of BODIPY Dyes.

Cover Picture: Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery System (ChemMedChem 7/2014).

Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery System.

The Integrin Ligand c(RGDf( NMe)Nal) Reduces Neointimal Hyperplasia in a Polymer-Free Drug-Eluting Stent System.

Small-Molecule Inhibitors of AF6 PDZ-Mediated Protein-Protein Interactions.

'À la Carte' Peptide Shuttles: Tools to Increase Their Passage across the Blood-Brain Barrier.

The Discovery of Potent Nonstructural Protein 5A (NS5A) Inhibitors with a Unique Resistance Profile-Part 1.

3-Aminoazetidin-2-one Derivatives as N-Acylethanolamine Acid Amidase (NAAA) Inhibitors Suitable for Systemic Administration.

Novel Heterobimetallic Radiotheranostic: Preparation, Activity, and Biodistribution.

Back Cover: The Integrin Ligand c(RGDf( NMe)Nal) Reduces Neointimal Hyperplasia in a Polymer-Free Drug-Eluting Stent System (ChemMedChem 7/2014).

Chiral Resolution and Pharmacological Characterization of the Enantiomers of the Hsp90 Inhibitor 2-Amino-7-[4-fluoro-2-(3-pyridyl)phenyl]-4-methyl-7,8-dihydro-6 H-quinazolin-5-one Oxime.

Structural Optimization and Biological Screening of a Steroidal Scaffold Possessing Cucurbitacin-Like Functionalities as B-Raf Inhibitors.

Stereoselective Reduction of 1- O-Isopropyloxygenipin Enhances Its Neuroprotective Activity in Neuronal Cells from Apoptosis Induced by Sodium Nitroprusside.