Works matching IS 18607179 AND DT 2014 AND VI 9 AND IP 11

Results: 20

Natural Products in Medicinal Chemistry.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2602, doi. 10.1002/cmdc.201402297
By:
- Sarker, Satyajit D.
Publication type:
Article
Synthesis and Structure-Activity Relationship Studies of 2-(1,3,4-Oxadiazole-2(3H)-thione)-3-amino-5-arylthieno[2,3-b]pyridines as Inhibitors of DRAK2.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2587, doi. 10.1002/cmdc.201402234
By:
- Leonczak, Piotr;
- Gao, Ling‐Jie;
- Ramadori, Anna Teresa;
- Lescrinier, Eveline;
- Rozenski, Jef;
- De Jonghe, Steven;
- Herdewijn, Piet
Publication type:
Article
Molecular Mechanism of Action of 2-Ferrocenyl-1,1-diphenylbut-1-ene on HL-60 Leukemia Cells.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2580, doi. 10.1002/cmdc.201402219
By:
- de Oliveira, Alane Cabral;
- da Silva, Emanuella Gomes;
- Rocha, Danilo Damasceno;
- Hillard, Elizabeth A.;
- Pigeon, Pascal;
- Jaouen, Gérard;
- Rodrigues, Felipe A. R.;
- de Abreu, Fabiane C.;
- da Rocha Ferreira, Fabrícia;
- Goulart, Marilia O. F.;
- Costa‐Lotufo, Letícia V.
Publication type:
Article
Design and Synthesis of Aminostilbene-Arylpropenones as Tubulin Polymerization Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2565, doi. 10.1002/cmdc.201402256
By:
- Kamal, Ahmed;
- Kumar, G. Bharath;
- Polepalli, Sowjanya;
- Shaik, Anver Basha;
- Reddy, Vangala Santhosh;
- Reddy, M. Kashi;
- Reddy, Ch. Ratna;
- Mahesh, Rasala;
- Kapure, Jeevak Sopanrao;
- Jain, Nishant
Publication type:
Article
α-Keto Phenylamides as P1'-Extended Proteasome Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2557, doi. 10.1002/cmdc.201402244
By:
- Voss, Constantin;
- Scholz, Christoph;
- Knorr, Sabine;
- Beck, Philipp;
- Stein, Martin L.;
- Zall, Andrea;
- Kuckelkorn, Ulrike;
- Kloetzel, Peter‐Michael;
- Groll, Michael;
- Hamacher, Kay;
- Schmidt, Boris
Publication type:
Article
Non-natural Acetogenin Analogues as Potent Trypanosoma brucei Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2548, doi. 10.1002/cmdc.201402272
By:
- Florence, Gordon J.;
- Fraser, Andrew L.;
- Gould, Eoin R.;
- King, Elizabeth F. B.;
- Menzies, Stefanie K.;
- Morris, Joanne C.;
- Tulloch, Lindsay B.;
- Smith, Terry K.
Publication type:
Article
Structure-Guided Design of Thiazolidine Derivatives as Mycobacterium tuberculosis Pantothenate Synthetase Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2538, doi. 10.1002/cmdc.201402171
By:
- Devi, Parthiban Brindha;
- Samala, Ganesh;
- Sridevi, Jonnalagadda Padma;
- Saxena, Shalini;
- Alvala, Mallika;
- Salina, Elena G.;
- Sriram, Dharmarajan;
- Yogeeswari, Perumal
Publication type:
Article
Biological Evaluation of Potent Triclosan-Derived Inhibitors of the Enoyl-Acyl Carrier Protein Reductase InhA in Drug-Sensitive and Drug-Resistant Strains of Mycobacterium tuberculosis.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2528, doi. 10.1002/cmdc.201402255
By:
- Stec, Jozef;
- Vilchèze, Catherine;
- Lun, Shichun;
- Perryman, Alexander L.;
- Wang, Xin;
- Freundlich, Joel S.;
- Bishai, William;
- Jacobs, William R.;
- Kozikowski, Alan P.
Publication type:
Article
Novel Hinge-Binding Motifs for Janus Kinase 3 Inhibitors: A Comprehensive Structure-Activity Relationship Study on Tofacitinib Bioisosteres.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2516, doi. 10.1002/cmdc.201402252
By:
- Gehringer, Matthias;
- Forster, Michael;
- Pfaffenrot, Ellen;
- Bauer, Silke M.;
- Laufer, Stefan A.
Publication type:
Article
Drug Screening Boosted by Hyperpolarized Long-Lived States in NMR.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2509, doi. 10.1002/cmdc.201402214
By:
- Buratto, Roberto;
- Bornet, Aurélien;
- Milani, Jonas;
- Mammoli, Daniele;
- Vuichoud, Basile;
- Salvi, Nicola;
- Singh, Maninder;
- Laguerre, Aurélien;
- Passemard, Solène;
- Gerber‐Lemaire, Sandrine;
- Jannin, Sami;
- Bodenhausen , Geoffrey
Publication type:
Article
Are 1,4- and 1,5-Disubstituted 1,2,3-Triazoles Good Pharmacophoric Groups?
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2497, doi. 10.1002/cmdc.201402233
By:
- Massarotti, Alberto;
- Aprile, Silvio;
- Mercalli, Valentina;
- Del Grosso, Erika;
- Grosa, Giorgio;
- Sorba, Giovanni;
- Tron, Gian Cesare
Publication type:
Article
Structure-Activity Relationship, Biological, and Pharmacological Characterization of the Proline Sulfonamide ACT-462206: a Potent, Brain-Penetrant Dual Orexin 1/Orexin 2 Receptor Antagonist.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2486, doi. 10.1002/cmdc.201402258
By:
- Boss, Christoph;
- Roch‐Brisbare, Catherine;
- Steiner, Michel A.;
- Treiber, Alexander;
- Dietrich, Hendrik;
- Jenck, Francois;
- von Raumer, Markus;
- Sifferlen, Thierry;
- Brotschi, Christine;
- Heidmann, Bibia;
- Williams, Jodi T.;
- Aissaoui, Hamed;
- Siegrist, Romain;
- Gatfield, John
Publication type:
Article
5-(Piperidin-4-yl)-3-Hydroxypyrazole: A Novel Scaffold for Probing the Orthosteric γ-Aminobutyric Acid Type A Receptor Binding Site.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2475, doi. 10.1002/cmdc.201402248
By:
- Krall, Jacob;
- Kongstad, Kenneth T.;
- Nielsen, Birgitte;
- Sørensen, Troels E.;
- Balle, Thomas;
- Jensen, Anders A.;
- Frølund, Bente
Publication type:
Article
Position and Length of Fatty Acids Strongly Affect Receptor Selectivity Pattern of Human Pancreatic Polypeptide Analogues.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2463, doi. 10.1002/cmdc.201402235
By:
- Mäde, Veronika;
- Bellmann‐Sickert, Kathrin;
- Kaiser, Anette;
- Meiler, Jens;
- Beck‐Sickinger, Annette G.
Publication type:
Article
Small Molecules that Target the Toxic RNA in Myotonic Dystrophy Type 2.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2455, doi. 10.1002/cmdc.201402095
By:
- Nguyen, Lien;
- Lee, JuYeon;
- Wong, Chun‐Ho;
- Zimmerman, Steven C.
Publication type:
Article
Amphiphilic Bicyclic Peptides as Cellular Delivery Agents.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2449, doi. 10.1002/cmdc.201402230
By:
- Oh, Donghoon;
- Darwish, Shaban Anwar;
- Shirazi, Amir Nasrolahi;
- Tiwari, Rakesh Kumar;
- Parang, Keykavous
Publication type:
Article
Diaryl-Substituted Azolylthioacetamides: Inhibitor Discovery of New Delhi Metallo-β-Lactamase-1 (NDM-1).
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2445, doi. 10.1002/cmdc.201402249
By:
- Zhang, Yi‐Lin;
- Yang, Ke‐Wu;
- Zhou, Ya‐Jun;
- LaCuran, Alecander E.;
- Oelschlaeger, Peter;
- Crowder, Michael W.
Publication type:
Article
In Vitro Antiamoebic Activity Evaluation and Docking Studies of Metronidazole-Triazole Hybrids.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2439, doi. 10.1002/cmdc.201402240
By:
- Negi, Beena;
- Raj, K. Kranthi;
- Siddiqui, Shadab Miyan;
- Ramachandran, Dittakavi;
- Azam, Amir;
- Rawat, Diwan S.
Publication type:
Article
Recent Advances in The Discovery of N-Myristoyltransferase Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2425, doi. 10.1002/cmdc.201402174
By:
- Zhao, Can;
- Ma, Shutao
Publication type:
Article
Therapeutic Strategies for Metabolic Diseases: Small-Molecule Diacylglycerol Acyltransferase (DGAT) Inhibitors.
Published in:
ChemMedChem, 2014, v. 9, n. 11, p. 2410, doi. 10.1002/cmdc.201402069
By:
- Naik, Ravi;
- Obiang‐Obounou, Brice W.;
- Kim, Minkyoung;
- Choi, Yongseok;
- Lee, Hyun Sun;
- Lee, Kyeong
Publication type:
Article