Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 9

Results: 22

cis-[Pt<sup>II</sup>(1 R,2 R-DACH)(3-acetoxy-1,1-cyclobutanedicarboxylato)], a Water-Soluble, Oxalate-Free and Stable Analogue of Oxaliplatin: Synthesis, Characterization, and Biological Evaluations.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1465, doi. 10.1002/cmdc.201300249

By:

Liu, Weiping;
Ye, Qingsong;
Jiang, Jing;
Lou, Liguang;
Xu, Yongping;
Xie, Chengying;
Xie, Mingjin

Publication type:

Article

6-Aryl and Heterocycle Quinazoline Derivatives as Potent EGFR Inhibitors with Improved Activity toward Gefitinib-Sensitive and -Resistant Tumor Cell Lines.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1495, doi. 10.1002/cmdc.201300147

By:

Hamed, Mostafa M.;
Abou El Ella, Dalal A.;
Keeton, Adam B.;
Piazza, Gary A.;
Abadi, Ashraf H.;
Hartmann, Rolf W.;
Engel, Matthias

Publication type:

Article

Graphical Abstract: ChemMedChem 9/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 9, p. 1423, doi. 10.1002/cmdc.201390037
Publication type:: Article

Strategic Targeting of Multiple Water-Mediated Interactions: A Concise and Rational Structure-Based Design Approach to Potent and Selective MMP-13 Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1457, doi. 10.1002/cmdc.201300278

By:

Fischer, Thomas;
Riedl, Rainer

Publication type:

Article

Overcoming the Limitations of Fragment Merging: Rescuing a Strained Merged Fragment Series Targeting Mycobacterium tuberculosis CYP121.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1451, doi. 10.1002/cmdc.201300219

By:

Hudson, Sean A.;
Surade, Sachin;
Coyne, Anthony G.;
McLean, Kirsty J.;
Leys, David;
Munro, Andrew W.;
Abell, Chris

Publication type:

Article

The Cell's Nucleolus: an Emerging Target for Chemotherapeutic Intervention.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1441, doi. 10.1002/cmdc.201300262

By:

Pickard, Amanda J.;
Bierbach, Ulrich

Publication type:

Article

Inside Cover: A Parallel Semisynthetic Approach for Structure-Activity Relationship Studies of Peptide YY (ChemMedChem 9/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1422, doi. 10.1002/cmdc.201390036

By:

Albertsen, Louise;
Østergaard, Søren;
Paulsson, Johan F.;
Norrild, Jens Chr.;
Strømgaard, Kristian

Publication type:

Article

Synthesis and in vitro Evaluation of West Nile Virus Protease Inhibitors Based on the 1,3,4,5-Tetrasubstituted 1 H-Pyrrol-2(5 H)-one Scaffold.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1554, doi. 10.1002/cmdc.201300244

By:

Gao, Yaojun;
Samanta, Sanjay;
Cui, Taian;
Lam, Yulin

Publication type:

Article

Thiuram Disulfides as Pseudo-irreversible Inhibitors of Lymphoid Tyrosine Phosphatase.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1561, doi. 10.1002/cmdc.201300215

By:

Kulkarni, Rhushikesh A.;
Stanford, Stephanie M.;
Vellore, Nadeem A.;
Krishnamurthy, Divya;
Bliss, Matthew R.;
Baron, Riccardo;
Bottini, Nunzio;
Barrios, Amy M.

Publication type:

Article

Probing the S1′ Site for the Identification of Non-Zinc-Binding MMP-2 Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1475, doi. 10.1002/cmdc.201300186

By:

Di Pizio, Antonella;
Laghezza, Antonio;
Tortorella, Paolo;
Agamennone, Mariangela

Publication type:

Article

A Parallel Semisynthetic Approach for Structure-Activity Relationship Studies of Peptide YY.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1505, doi. 10.1002/cmdc.201300290

By:

Albertsen, Louise;
Østergaard, Søren;
Paulsson, Johan F.;
Norrild, Jens Chr.;
Strømgaard, Kristian

Publication type:

Article

Synthesis and Biological Evaluation of 2-Arylamino-5- (3′-Indolyl)-1,3,4-Oxadiazoles as Potent Cytotoxic Agents.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1468, doi. 10.1002/cmdc.201300221

By:

Tantak, Mukund P;
Kumar, Anil;
Noel, Brett;
Shah, Kavita;
Kumar, Dalip

Publication type:

Article

Cover Picture: Probing the S1′ Site for the Identification of Non-Zinc-Binding MMP-2 Inhibitors (ChemMedChem 9/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1421, doi. 10.1002/cmdc.201390035

By:

Pizio, Antonella Di;
Laghezza, Antonio;
Tortorella, Paolo;
Agamennone, Mariangela

Publication type:

Article

Zopolrestat as a Human Glyoxalase I Inhibitor and Its Structural Basis.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1462, doi. 10.1002/cmdc.201300243

By:

Zhai, Jing;
Zhang, Hong;
Zhang, Ligping;
Zhao, Yining;
Chen, Sangke;
Chen, Yunyun;
Peng, Xinyu;
Li, Qing;
Yuan, Minggui;
Hu, Xiaopeng

Publication type:

Article

Back Cover: Strategic Targeting of Multiple Water-Mediated Interactions: A Concise and Rational Structure-Based Design Approach to Potent and Selective MMP-13 Inhibitors (ChemMedChem 9/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1572, doi. 10.1002/cmdc.201390039

By:

Fischer, Thomas;
Riedl, Rainer

Publication type:

Article

Chemical, Pharmacological, and in vitro Metabolic Stability Studies on Enantiomerically Pure RC-33 Compounds: Promising Neuroprotective Agents Acting as σ<sub>1</sub> Receptor Agonists.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1514, doi. 10.1002/cmdc.201300218

By:

Rossi, Daniela;
Pedrali, Alice;
Gaggeri, Raffaella;
Marra, Annamaria;
Pignataro, Luca;
Laurini, Erik;
Dal Col, Valentina;
Fermeglia, Maurizio;
Pricl, Sabrina;
Schepmann, Dirk;
Wünsch, Bernhard;
Peviani, Marco;
Curti, Daniela;
Collina, Simona

Publication type:

Article

Structure-Activity Relationship Studies of Pyrrolone Antimalarial Agents.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1537, doi. 10.1002/cmdc.201300177

By:

Murugesan, Dinakaran;
Kaiser, Marcel;
White, Karen L.;
Norval, Suzanne;
Riley, Jennifer;
Wyatt, Paul G.;
Charman, Susan A.;
Read, Kevin D.;
Yeates, Clive;
Gilbert, Ian H.

Publication type:

Article

Rise of the Selective Inhibitors of Anti-Apoptotic Bcl-2 Family Proteins.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1437, doi. 10.1002/cmdc.201300301

By:

Han, Li;
Wang, Renxiao

Publication type:

Article

Rational Design of Resorcylic Acid Lactone Analogues as Covalent MNK1/2 Kinase Inhibitors by Tuning the Reactivity of an Enamide Michael Acceptor.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1483, doi. 10.1002/cmdc.201300231

By:

Xu, Jin;
Chen, Anqi;
Joy, Joma;
Xavier, Vanessa Joanne;
Ong, Esther H. Q.;
Hill, Jeffrey;
Chai, Christina L. L.

Publication type:

Article

An Endoperoxide-Based Hybrid Approach to Deliver Falcipain Inhibitors Inside Malaria Parasites.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1528, doi. 10.1002/cmdc.201300202

By:

Oliveira, Rudi;
Newton, Ana S.;
Guedes, Rita C.;
Miranda, Daniela;
Amewu, Richard K.;
Srivastava, Abhishek;
Gut, Jiri;
Rosenthal, Philip J.;
O'Neill, Paul M.;
Ward, Stephen A.;
Lopes, Francisca;
Moreira, Rui

Publication type:

Article

Synthesis and Biological Evaluation of N-Substituted Sophocarpinic Acid Derivatives as Coxsackievirus B3 Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 9, p. 1545, doi. 10.1002/cmdc.201300224

By:

Gao, Li‐Mei;
Tang, Sheng;
Wang, Yan‐Xiang;
Gao, Rong‐Mei;
Zhang, Xin;
Peng, Zong‐Gen;
Li, Jian‐Rui;
Jiang, Jian‐Dong;
Li, Yu‐Huan;
Song, Dan‐Qing

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 9/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 9, p. 1432, doi. 10.1002/cmdc.201390038
Publication type:: Article