Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 6

Results: 25

Design, Synthesis and Biological Evaluation of Trimethine Cyanine Dyes as Fluorescent Probes for the Detection of Tau Fibrils in Alzheimer's Disease Brain and Olfactory Epithelium.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 891, doi. 10.1002/cmdc.201300090

By:

Gu, Jiamin;
Anumala, Upendra Rao;
Heyny‐von Haußen, Roland;
Hölzer, Jana;
Goetschy‐Meyer, Valérie;
Mall, Gerhard;
Hilger, Ingrid;
Czech, Christian;
Schmidt, Boris

Publication type:

Article

Synthesis, Antitumor Evaluation and Docking Study of Novel 4-Anilinoquinazoline Derivatives as Potential Epidermal Growth Factor Receptor (EGFR) Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 928, doi. 10.1002/cmdc.201300120

By:

Rao, Guo‐Wu;
Xu, Geng‐Jie;
Wang, Jian;
Jiang, Xu‐Liang;
Li, Hai‐Bo

Publication type:

Article

Structure-Activity Relationships of Quinoxaline-Based 5-HT3A and 5-HT3AB Receptor-Selective Ligands.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 946, doi. 10.1002/cmdc.201300032

By:

Thompson, Andrew J.;
Verheij, Mark H. P.;
van Muijlwijk‐Koezen, Jacqueline E.;
Lummis, Sarah C. R.;
Leurs, Rob;
de Esch, Iwan J. P.

Publication type:

Article

Discovery and Characterization of ACT-335827, an Orally Available, Brain Penetrant Orexin Receptor Type 1 Selective Antagonist.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 898, doi. 10.1002/cmdc.201300003

By:

Steiner, Michel A.;
Gatfield, John;
Brisbare‐Roch, Catherine;
Dietrich, Hendrik;
Treiber, Alexander;
Jenck, Francois;
Boss, Christoph

Publication type:

Article

Bioisosteres in Medicinal Chemistry. Edited by Nathan Brown.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 1012, doi. 10.1002/cmdc.201300117

By:

Bunch, Lennart

Publication type:

Article

Inside Cover: Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria (ChemMedChem 6/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 866, doi. 10.1002/cmdc.201390021

By:

Chang, Jun;
Zhang, Si‐Ji;
Jiang, Yong‐Wei;
Xu, Liang;
Yu, Jian‐Ming;
Zhou, Wen‐Jiang;
Sun, Xun

Publication type:

Article

Synthesis and Anti-herpetic Activity of Phosphoramidate ProTides.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 985, doi. 10.1002/cmdc.201300035

By:

Maiti, Munmun;
Persoons, Leentje;
Andrei, Graciela;
Snoeck, Robert;
Balzarini, Jan;
Herdewijn, Piet

Publication type:

Article

Potent Inhibitors of Phosphatidylinositol 3 (PI3) Kinase that have Antiproliferative Activity Only When Delivered as Prodrug Forms.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 914, doi. 10.1002/cmdc.201200583

By:

O'Brien, Nathan J.;
Amran, Syazwani;
Medan, Jelena;
Cleary, Ben;
Deady, Leslie W.;
Jennings, Ian G.;
Thompson, Philip E.;
Abbott, Belinda M.

Publication type:

Article

Cancer Epigenetics: Biomolecular Therapeutics for Human Cancer. Edited by Antonio Giordano and Marcella Macaluso.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 1014, doi. 10.1002/cmdc.201300152

By:

Blagg, Julian

Publication type:

Article

An Efficient Bioorthogonal Strategy Using CuAAC Click Chemistry for Radiofluorinations of SNEW Peptides and the Role of Copper Depletion.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 935, doi. 10.1002/cmdc.201300053

By:

Pretze, Marc;
Kuchar, Manuela;
Bergmann, Ralf;
Steinbach, Jörg;
Pietzsch, Jens;
Mamat, Constantin

Publication type:

Article

Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure-Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human Cathepsin L.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 967, doi. 10.1002/cmdc.201300112

By:

Ehmke, Veronika;
Winkler, Edwin;
Banner, David W.;
Haap, Wolfgang;
Schweizer, W. Bernd;
Rottmann, Matthias;
Kaiser, Marcel;
Freymond, Céline;
Schirmeister, Tanja;
Diederich, François

Publication type:

Article

From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 919, doi. 10.1002/cmdc.201300057

By:

Buscató, Estel.la;
Büttner, Dominik;
Brüggerhoff, Astrid;
Klingler, Franca‐Maria;
Weber, Julia;
Scholz, Bastian;
Živković, Aleksandra;
Marschalek, Rolf;
Stark, Holger;
Steinhilber, Dieter;
Bode, Helge B.;
Proschak, Ewgenij

Publication type:

Article

Rhenium Complexes with Visible-Light-Induced Anticancer Activity.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 924, doi. 10.1002/cmdc.201300060

By:

Kastl, Anja;
Dieckmann, Sandra;
Wähler, Kathrin;
Völker, Timo;
Kastl, Lena;
Merkel, Anna Lena;
Vultur, Adina;
Shannan, Batool;
Harms, Klaus;
Ocker, Matthias;
Parak, Wolfgang J.;
Herlyn, Meenhard;
Meggers, Eric

Publication type:

Article

Selective Bisubstrate Inhibitors with Sub-nanomolar Affinity for Protein Kinase Pim-1.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 909, doi. 10.1002/cmdc.201300042

By:

Ekambaram, Ramesh;
Enkvist, Erki;
Vaasa, Angela;
Kasari, Marje;
Raidaru, Gerda;
Knapp, Stefan;
Uri, Asko

Publication type:

Article

Cover Picture: From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties (ChemMedChem 6/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 865, doi. 10.1002/cmdc.201390020

By:

Buscató, Estel.la;
Büttner, Dominik;
Brüggerhoff, Astrid;
Klingler, Franca‐Maria;
Weber, Julia;
Scholz, Bastian;
Živković, Aleksandra;
Marschalek, Rolf;
Stark, Holger;
Steinhilber, Dieter;
Bode, Helge B.;
Proschak, Ewgenij

Publication type:

Article

A Facile Hydroxyindole Carboxylic Acid Based Focused Library Approach for Potent and Selective Inhibitors of Mycobacterium Protein Tyrosine Phosphatase B.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 904, doi. 10.1002/cmdc.201300115

By:

Zeng, Li‐Fan;
Xu, Jie;
He, Yantao;
He, Rongjun;
Wu, Li;
Gunawan, Andrea M.;
Zhang, Zhong‐Yin

Publication type:

Article

Radiolabeled Heterobivalent Peptidic Ligands: an Approach with High Future Potential for in vivo Imaging and Therapy of Malignant Diseases.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 883, doi. 10.1002/cmdc.201300081

By:

Fischer, Gabriel;
Schirrmacher, Ralf;
Wängler, Björn;
Wängler, Carmen

Publication type:

Article

Innovations in Biomolecular Modeling and Simulations. Edited by Tamar Schlick.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 1012, doi. 10.1002/cmdc.201300052

By:

Orozco, Modesto

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 6/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 6, p. 878, doi. 10.1002/cmdc.201390023
Publication type:: Article

Back Cover: Structure-Activity Relationships of Quinoxaline-Based 5-HT3A and 5-HT3AB Receptor-Selective Ligands (ChemMedChem 6/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 1020, doi. 10.1002/cmdc.201390024

By:

Thompson, Andrew J.;
Verheij, Mark H. P.;
van Muijlwijk‐Koezen, Jacqueline E.;
Lummis, Sarah C. R.;
Leurs, Rob;
de Esch, Iwan J. P.

Publication type:

Article

Synthesis and in vitro Evaluation of West Nile Virus Protease Inhibitors Based on the 2-{6-[2-(5-Phenyl-4 H-{1,2,4]triazol-3-ylsulfanyl)acetylamino]benzothiazol-2-ylsulfanyl}acetamide Scaffold.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 994, doi. 10.1002/cmdc.201300114

By:

Samanta, Sanjay;
Lim, Ting Liang;
Lam, Yulin

Publication type:

Article

MAO Inhibitory Activity of 2-Arylbenzofurans versus 3-Arylcoumarins: Synthesis, in vitro Study, and Docking Calculations.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 956, doi. 10.1002/cmdc.201300048

By:

Ferino, Giulio;
Cadoni, Enzo;
Matos, Maria João;
Quezada, Elias;
Uriarte, Eugenio;
Santana, Lourdes;
Vilar, Santiago;
Tatonetti, Nicholas P.;
Yáñez, Matilde;
Viña, Dolores;
Picciau, Carmen;
Serra, Silvia;
Delogu, Giovanna

Publication type:

Article

Synthesis and Evaluation of Water-Soluble Prodrugs of Ursodeoxycholic Acid (UDCA), an Anti-apoptotic Bile Acid.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 1002, doi. 10.1002/cmdc.201300059

By:

Dosa, Peter I.;
Ward, Tim;
Castro, Rui E.;
Rodrigues, Cecília M. P.;
Steer, Clifford J.

Publication type:

Article

Graphical Abstract: ChemMedChem 6/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 6, p. 867, doi. 10.1002/cmdc.201390022
Publication type:: Article

Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria.

Published in:

ChemMedChem, 2013, v. 8, n. 6, p. 976, doi. 10.1002/cmdc.201300011

By:

Chang, Jun;
Zhang, Si‐Ji;
Jiang, Yong‐Wei;
Xu, Liang;
Yu, Jian‐Ming;
Zhou, Wen‐Jiang;
Sun, Xun

Publication type:

Article

Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 6

Design, Synthesis and Biological Evaluation of Trimethine Cyanine Dyes as Fluorescent Probes for the Detection of Tau Fibrils in Alzheimer's Disease Brain and Olfactory Epithelium.

Synthesis, Antitumor Evaluation and Docking Study of Novel 4-Anilinoquinazoline Derivatives as Potential Epidermal Growth Factor Receptor (EGFR) Inhibitors.

Structure-Activity Relationships of Quinoxaline-Based 5-HT<sub>3</sub>A and 5-HT<sub>3</sub>AB Receptor-Selective Ligands.

Discovery and Characterization of ACT-335827, an Orally Available, Brain Penetrant Orexin Receptor Type 1 Selective Antagonist.

Bioisosteres in Medicinal Chemistry. Edited by Nathan Brown.

Inside Cover: Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria (ChemMedChem 6/2013).

Synthesis and Anti-herpetic Activity of Phosphoramidate ProTides.

Potent Inhibitors of Phosphatidylinositol 3 (PI3) Kinase that have Antiproliferative Activity Only When Delivered as Prodrug Forms.

Cancer Epigenetics: Biomolecular Therapeutics for Human Cancer. Edited by Antonio Giordano and Marcella Macaluso.

An Efficient Bioorthogonal Strategy Using CuAAC Click Chemistry for Radiofluorinations of SNEW Peptides and the Role of Copper Depletion.

Optimization of Triazine Nitriles as Rhodesain Inhibitors: Structure-Activity Relationships, Bioisosteric Imidazopyridine Nitriles, and X-ray Crystal Structure Analysis with Human Cathepsin L.

From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties.

Rhenium Complexes with Visible-Light-Induced Anticancer Activity.

Selective Bisubstrate Inhibitors with Sub-nanomolar Affinity for Protein Kinase Pim-1.

Cover Picture: From a Multipotent Stilbene to Soluble Epoxide Hydrolase Inhibitors with Antiproliferative Properties (ChemMedChem 6/2013).

A Facile Hydroxyindole Carboxylic Acid Based Focused Library Approach for Potent and Selective Inhibitors of Mycobacterium Protein Tyrosine Phosphatase B.

Radiolabeled Heterobivalent Peptidic Ligands: an Approach with High Future Potential for in vivo Imaging and Therapy of Malignant Diseases.

Innovations in Biomolecular Modeling and Simulations. Edited by Tamar Schlick.

Spotlights on our sister journals: ChemMedChem 6/2013.

Back Cover: Structure-Activity Relationships of Quinoxaline-Based 5-HT<sub>3</sub>A and 5-HT<sub>3</sub>AB Receptor-Selective Ligands (ChemMedChem 6/2013).

Synthesis and in vitro Evaluation of West Nile Virus Protease Inhibitors Based on the 2-{6-[2-(5-Phenyl-4 H-{1,2,4]triazol-3-ylsulfanyl)acetylamino]benzothiazol-2-ylsulfanyl}acetamide Scaffold.

MAO Inhibitory Activity of 2-Arylbenzofurans versus 3-Arylcoumarins: Synthesis, in vitro Study, and Docking Calculations.

Synthesis and Evaluation of Water-Soluble Prodrugs of Ursodeoxycholic Acid (UDCA), an Anti-apoptotic Bile Acid.

Graphical Abstract: ChemMedChem 6/2013.

Design, Synthesis, and Antibacterial Activity of Demethylvancomycin Analogues against Drug-Resistant Bacteria.