Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 12

Results: 21

De Novo Design, Synthesis and Evaluation of Benzylpiperazine Derivatives as Highly Selective Binders of Mcl-1.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1986, doi. 10.1002/cmdc.201300316

By:

Ding, Xiao;
Li, Yan;
Lv, Li;
Zhou, Mi;
Han, Li;
Zhang, Zhengxi;
Ba, Qian;
Li, Jingquan;
Wang, Hui;
Liu, Hong;
Wang, Renxiao

Publication type:

Article

Effect of Linker Length and Composition on Heterobivalent Ligand-Mediated Receptor Cross-Talk between the A1 Adenosine and β2 Adrenergic Receptors.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2036, doi. 10.1002/cmdc.201300286

By:

Barlow, Nicholas;
Baker, Stephen P.;
Scammells, Peter J.

Publication type:

Article

Probing Binding and Cellular Activity of Pyrrolidinone and Piperidinone Small Molecules Targeting the Urokinase Receptor.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1963, doi. 10.1002/cmdc.201300340

By:

Mani, Timmy;
Liu, Degang;
Zhou, Donghui;
Li, Liwei;
Knabe, William Eric;
Wang, Fang;
Oh, Kyungsoo;
Meroueh, Samy O.

Publication type:

Article

Design and Generation of Highly Diverse Fluorinated Fragment Libraries and their Efficient Screening with Improved 19F NMR Methodology.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2057, doi. 10.1002/cmdc.201300351

By:

Vulpetti, Anna;
Dalvit, Claudio

Publication type:

Article

Inside Cover: Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity (ChemMedChem 12/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1898, doi. 10.1002/cmdc.201390051

By:

Niso, Mauro;
Abate, Carmen;
Contino, Marialessandra;
Ferorelli, Savina;
Azzariti, Amalia;
Perrone, Roberto;
Colabufo, Nicola Antonio;
Berardi, Francesco

Publication type:

Article

Synthesis, Characterization, and Metabolism Studies of Fluspidine Enantiomers.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2047, doi. 10.1002/cmdc.201300322

By:

Holl, Katharina;
Falck, Evamaria;
Köhler, Jens;
Schepmann, Dirk;
Humpf, Hans‐Ulrich;
Brust, Peter;
Wünsch, Bernhard

Publication type:

Article

para-Substituted 2-Phenyl-3,4-dihydroquinazolin-4-ones As Potent and Selective Tankyrase Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1978, doi. 10.1002/cmdc.201300337

By:

Haikarainen, Teemu;
Koivunen, Jarkko;
Narwal, Mohit;
Venkannagari, Harikanth;
Obaji, Ezeogo;
Joensuu, Päivi;
Pihlajaniemi, Taina;
Lehtiö, Lari

Publication type:

Article

Synthesis and Biological Evaluation of Imidazopyridine-Oxindole Conjugates as Microtubule-Targeting Agents.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2015, doi. 10.1002/cmdc.201300308

By:

Kamal, Ahmed;
Reddy, Vangala Santhosh;
Karnewar, Santosh;
Chourasiya, Sumit S.;
Shaik, Anver Basha;
Kumar, G. Bharath;
Kishor, Chandan;
Reddy, M. Kashi;
Narasimha Rao, M. P.;
Nagabhushana, Ananthamurthy;
Ramakrishna, Kallaganti V. S.;
Addlagatta, Anthony;
Kotamraju, Srigiridhar

Publication type:

Article

Chromophore-Linked Substrate (CLS405): Probing Metallo-β-Lactamase Activity and Inhibition.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1923, doi. 10.1002/cmdc.201300350

By:

Makena, Anne;
van Berkel, Sander S.;
Lejeune, Clarisse;
Owens, Raymond J.;
Verma, Anil;
Salimraj, Ramya;
Spencer, James;
Brem, Jürgen;
Schofield, Christopher J.

Publication type:

Article

Corrigendum: Small-Molecule Modulators for Epigenetics Targets.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1904, doi. 10.1002/cmdc.201300464

By:

Knapp, Stefan;
Weinmann, Hilmar

Publication type:

Article

Development of Rhodesain Inhibitors with a 3-Bromoisoxazoline Warhead.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2070, doi. 10.1002/cmdc.201300390

By:

Ettari, Roberta;
Tamborini, Lucia;
Angelo, Ilenia C.;
Grasso, Silvana;
Schirmeister, Tanja;
Lo Presti, Leonardo;
De Micheli, Carlo;
Pinto, Andrea;
Conti, Paola

Publication type:

Article

Cover Picture: Chromophore-Linked Substrate (CLS405): Probing Metallo-β-Lactamase Activity and Inhibition (ChemMedChem 12/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1897, doi. 10.1002/cmdc.201390050

By:

Makena, Anne;
van Berkel, Sander S.;
Lejeune, Clarisse;
Owens, Raymond J.;
Verma, Anil;
Salimraj, Ramya;
Spencer, James;
Brem, Jürgen;
Schofield, Christopher J.

Publication type:

Article

Discovery of MK-8742: An HCV NS5A Inhibitor with Broad Genotype Activity.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1930, doi. 10.1002/cmdc.201300343

By:

Coburn, Craig A.;
Meinke, Peter T.;
Chang, Wei;
Fandozzi, Christine M.;
Graham, Donald J.;
Hu, Bin;
Huang, Qian;
Kargman, Stacia;
Kozlowski, Joseph;
Liu, Rong;
McCauley, John A.;
Nomeir, Amin A.;
Soll, Richard M.;
Vacca, Joseph P.;
Wang, Dahai;
Wu, Hao;
Zhong, Bin;
Olsen, David B.;
Ludmerer, Steven W.

Publication type:

Article

Back Cover: Synthesis and Biological Evaluation of Imidazopyridine-Oxindole Conjugates as Microtubule-Targeting Agents (ChemMedChem 12/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2080, doi. 10.1002/cmdc.201390054

By:

Kamal, Ahmed;
Reddy, Vangala Santhosh;
Karnewar, Santosh;
Chourasiya, Sumit S.;
Shaik, Anver Basha;
Kumar, G. Bharath;
Kishor, Chandan;
Reddy, M. Kashi;
Narasimha Rao, M. P.;
Nagabhushana, Ananthamurthy;
Ramakrishna, Kallaganti V. S.;
Addlagatta, Anthony;
Kotamraju, Srigiridhar

Publication type:

Article

Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 2026, doi. 10.1002/cmdc.201300291

By:

Niso, Mauro;
Abate, Carmen;
Contino, Marialessandra;
Ferorelli, Savina;
Azzariti, Amalia;
Perrone, Roberto;
Colabufo, Nicola Antonio;
Berardi, Francesco

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 12/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 12, p. 1908, doi. 10.1002/cmdc.201390053
Publication type:: Article

Synthesis and Structure-Activity Relationship Studies of Quinoxaline Derivatives as Aldose Reductase Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1913, doi. 10.1002/cmdc.201300324

By:

Wu, Bobin;
Yang, Yanchun;
Qin, Xiangyu;
Zhang, Shuzhen;
Jing, Chaojun;
Zhu, Changjin;
Ma, Bing

Publication type:

Article

Graphical Abstract: ChemMedChem 12/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 12, p. 1899, doi. 10.1002/cmdc.201390052
Publication type:: Article

A Template-Based Approach to Inhibitors of Calpain 2, 20S Proteasome, and HIV-1 Protease.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1918, doi. 10.1002/cmdc.201300387

By:

Jones, Seth A.;
Neilsen, Paul M.;
Siew, Limei;
Callen, David F.;
Goldfarb, Nathan E.;
Dunn, Ben M.;
Abell, Andrew D.

Publication type:

Article

Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1941, doi. 10.1002/cmdc.201300287

By:

Sancineto, Luca;
Iraci, Nunzio;
Massari, Serena;
Attanasio, Vanessa;
Corazza, Gianmarco;
Barreca, Maria Letizia;
Sabatini, Stefano;
Manfroni, Giuseppe;
Avanzi, Nilla Roberta;
Cecchetti, Violetta;
Pannecouque, Christophe;
Marcello, Alessandro;
Tabarrini, Oriana

Publication type:

Article

Amythiamicin D and Related Thiopeptides as Inhibitors of the Bacterial Elongation Factor EF-Tu: Modification of the Amino Acid at Carbon Atom C2 of Ring C Dramatically Influences Activity.

Published in:

ChemMedChem, 2013, v. 8, n. 12, p. 1954, doi. 10.1002/cmdc.201300323

By:

Gross, Stefan;
Nguyen, Fabian;
Bierschenk, Matthias;
Sohmen, Daniel;
Menzel, Thomas;
Antes, Iris;
Wilson, Daniel N.;
Bach, Thorsten

Publication type:

Article

Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 12

De Novo Design, Synthesis and Evaluation of Benzylpiperazine Derivatives as Highly Selective Binders of Mcl-1.

Effect of Linker Length and Composition on Heterobivalent Ligand-Mediated Receptor Cross-Talk between the A<sub>1</sub> Adenosine and β<sub>2</sub> Adrenergic Receptors.

Probing Binding and Cellular Activity of Pyrrolidinone and Piperidinone Small Molecules Targeting the Urokinase Receptor.

Design and Generation of Highly Diverse Fluorinated Fragment Libraries and their Efficient Screening with Improved <sup>19</sup>F NMR Methodology.

Inside Cover: Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity (ChemMedChem 12/2013).

Synthesis, Characterization, and Metabolism Studies of Fluspidine Enantiomers.

para-Substituted 2-Phenyl-3,4-dihydroquinazolin-4-ones As Potent and Selective Tankyrase Inhibitors.

Synthesis and Biological Evaluation of Imidazopyridine-Oxindole Conjugates as Microtubule-Targeting Agents.

Chromophore-Linked Substrate (CLS405): Probing Metallo-β-Lactamase Activity and Inhibition.

Corrigendum: Small-Molecule Modulators for Epigenetics Targets.

Development of Rhodesain Inhibitors with a 3-Bromoisoxazoline Warhead.

Cover Picture: Chromophore-Linked Substrate (CLS405): Probing Metallo-β-Lactamase Activity and Inhibition (ChemMedChem 12/2013).

Discovery of MK-8742: An HCV NS5A Inhibitor with Broad Genotype Activity.

Back Cover: Synthesis and Biological Evaluation of Imidazopyridine-Oxindole Conjugates as Microtubule-Targeting Agents (ChemMedChem 12/2013).

Sigma-2 Receptor Agonists as Possible Antitumor Agents in Resistant Tumors: Hints for Collateral Sensitivity.

Spotlights on our sister journals: ChemMedChem 12/2013.

Synthesis and Structure-Activity Relationship Studies of Quinoxaline Derivatives as Aldose Reductase Inhibitors.

Graphical Abstract: ChemMedChem 12/2013.

A Template-Based Approach to Inhibitors of Calpain 2, 20S Proteasome, and HIV-1 Protease.

Computer-Aided Design, Synthesis and Validation of 2-Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti-HIV-1 Tat-Mediated Transcription Activity.

Amythiamicin D and Related Thiopeptides as Inhibitors of the Bacterial Elongation Factor EF-Tu: Modification of the Amino Acid at Carbon Atom C2 of Ring C Dramatically Influences Activity.