Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 1

Results: 28

Highly Ligand Efficient and Selective N-2-(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 149, doi. 10.1002/cmdc.201200450

By:

Baud, Matthias G. J.;
Haus, Patricia;
Leiser, Thomas;
Meyer‐Almes, Franz‐Josef;
Fuchter, Matthew J.

Publication type:

Article

Editorial: Premature Publishing and Over-fragmentation.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 6, doi. 10.1002/cmdc.201200494

By:

Tarzia, Giorgio

Publication type:

Article

C3′/C4′-Stereochemical Effects of Digitoxigenin α- L-/α- D-Glycoside in Cancer Cytotoxicity.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 63, doi. 10.1002/cmdc.201200465

By:

Hinds, John W.;
McKenna, Sean B.;
Sharif, Ehesan U.;
Wang, Hua‐Yu L.;
Akhmedov, Novruz G.;
O'Doherty, George A.

Publication type:

Article

Thiadiazole-a Promising Structure in Medicinal Chemistry.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 27, doi. 10.1002/cmdc.201200355

By:

Li, Yijing;
Geng, Jingkun;
Liu, Yang;
Yu, Shenghui;
Zhao, Guisen

Publication type:

Article

Inside Cover: From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography (ChemMedChem 1/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 2, doi. 10.1002/cmdc.201290066

By:

Mocharla, Vani P.;
Walsh, Joseph C.;
Padgett, Henry C.;
Su, Helen;
Fueger, Barbara;
Weber, Wolfgang A.;
Czernin, Johannes;
Kolb, Hartmuth C.

Publication type:

Article

Synthesis and Quantitative Structure-Activity Relationships of Selective BCRP Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 125, doi. 10.1002/cmdc.201200377

By:

Marighetti, Federico;
Steggemann, Kerstin;
Hanl, Markus;
Wiese, Michael

Publication type:

Article

Designing Multi-Target Drugs. Edited by J. Richard Morphy and C. John Harris.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 166, doi. 10.1002/cmdc.201200420

By:

Peters, Jens‐Uwe

Publication type:

Article

Nanoparticles in Biology and Medicine: Methods and Protocols. Edited by Mikhail Soloviev.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 167, doi. 10.1002/cmdc.201200430

By:

Fröhlich, Eleonore

Publication type:

Article

How is 68Ga Labeling of Macrocyclic Chelators Influenced by Metal Ion Contaminants in 68Ge/68Ga Generator Eluates?

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 95, doi. 10.1002/cmdc.201200471

By:

Šimeček, Jakub;
Hermann, Petr;
Wester, Hans‐Jürgen;
Notni, Johannes

Publication type:

Article

Low-Molecular-Weight CXCR4 Ligands with Variable Spacers.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 118, doi. 10.1002/cmdc.201200390

By:

Narumi, Tetsuo;
Aikawa, Haruo;
Tanaka, Tomohiro;
Hashimoto, Chie;
Ohashi, Nami;
Nomura, Wataru;
Kobayakawa, Takuya;
Takano, Hikaru;
Hirota, Yuki;
Murakami, Tsutomu;
Yamamoto, Naoki;
Tamamura, Hirokazu

Publication type:

Article

Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 104, doi. 10.1002/cmdc.201200417

By:

Lacotte, Pierre;
Puente, Celine;
Ambroise, Yves

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 1/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 1, p. 20, doi. 10.1002/cmdc.201290065
Publication type:: Article

Reduction of Helical Content by Insertion of a Disulfide Bond Leads to an Antimicrobial Peptide with Decreased Hemolytic Activity.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 59, doi. 10.1002/cmdc.201200463

By:

Hwang, Heeyong;
Hyun, Soonsil;
Kim, Yangsoo;
Yu, Jaehoon

Publication type:

Article

3D-QSAR-Assisted Drug Design: Identification of a Potent Quinazoline-Based Aurora Kinase Inhibitor.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 136, doi. 10.1002/cmdc.201200464

By:

Ke, Yi‐Yu;
Shiao, Hui‐Yi;
Hsu, Yung Chang;
Chu, Chang‐Ying;
Wang, Wen‐Chieh;
Lee, Yen‐Chun;
Lin, Wen‐Hsing;
Chen, Chun‐Hwa;
Hsu, John T. A.;
Chang, Chun‐Wei;
Lin, Cheng‐Wei;
Yeh, Teng‐Kuang;
Chao, Yu‐Sheng;
Coumar, Mohane Selvaraj;
Hsieh, Hsing‐Pang

Publication type:

Article

Exploring the Polyamine Regulatory Site of the NMDA Receptor: a Parallel Synthesis Approach.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 82, doi. 10.1002/cmdc.201200470

By:

Berger, Michael L.;
Pöhler, Thomas;
Schadt, Oliver;
Stanger, Maximilian;
Rebernik, Patrick;
Scholze, Petra;
Noe, Christian R.

Publication type:

Article

Drug Discovery in Infectious Diseases, Volume 3: Parasitic Helminths: Targets, Screens, Drugs and Vaccines. Edited by Conor R. Caffrey.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 164, doi. 10.1002/cmdc.201200515

By:

Davioud‐Charvet, Elisabeth

Publication type:

Article

Combining Quantum Mechanical Ligand Conformation Analysis and Protein Modeling to Elucidate GPCR-Ligand Binding Modes.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 49, doi. 10.1002/cmdc.201200412

By:

Schultes, Sabine;
Engelhardt, Harald;
Roumen, Luc;
Zuiderveld, Obbe P.;
Haaksma, Eric E. J.;
de Esch, Iwan J. P.;
Leurs, Rob;
de Graaf, Chris

Publication type:

Article

Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 75, doi. 10.1002/cmdc.201200376

By:

Held, Cornelia;
Plomer, Manuel;
Hübner, Harald;
Meltretter, Jasmin;
Pischetsrieder, Monika;
Gmeiner, Peter

Publication type:

Article

Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 112, doi. 10.1002/cmdc.201200411

By:

Olson, Margaret E.;
Li, Ming;
Harris, Reuben S.;
Harki, Daniel A.

Publication type:

Article

Editorial: Lucky Number 8!

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 3, doi. 10.1002/cmdc.201200495

By:

Williams, Scott D.;
Ortúzar, Natalia

Publication type:

Article

Cover Picture: Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors (ChemMedChem 1/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 1, doi. 10.1002/cmdc.201290064

By:

Lacotte, Pierre;
Puente, Celine;
Ambroise, Yves

Publication type:

Article

Back Cover: Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold (ChemMedChem 1/2013).

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 172, doi. 10.1002/cmdc.201290068

By:

Olson, Margaret E.;
Li, Ming;
Harris, Reuben S.;
Harki, Daniel A.

Publication type:

Article

Introduction to Strategies for Organic Synthesis. By Laurie S. Starkey.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 164, doi. 10.1002/cmdc.201200440

By:

Moloney, Mark G.

Publication type:

Article

Discovery of Schaeffer's Acid Analogues as Lead Structures of Mycobacterium tuberculosis Type II Dehydroquinase Using a Rational Drug Design Approach.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 54, doi. 10.1002/cmdc.201200508

By:

Schmidt, Marco F.;
Korb, Oliver;
Howard, Nigel I.;
Dias, Marcio V. B.;
Blundell, Tom L.;
Abell, Chris

Publication type:

Article

Identification of LasR Ligands through a Virtual Screening Approach.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 157, doi. 10.1002/cmdc.201200434

By:

Skovstrup, Søren;
Le Quement, Sebastian Thordal;
Hansen, Thomas;
Jakobsen, Tim Holm;
Harmsen, Morten;
Tolker‐Nielsen, Tim;
Nielsen, Thomas E.;
Givskov, Michael;
Taboureau, Olivier

Publication type:

Article

From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 43, doi. 10.1002/cmdc.201200466

By:

Mocharla, Vani P.;
Walsh, Joseph C.;
Padgett, Henry C.;
Su, Helen;
Fueger, Barbara;
Weber, Wolfgang A.;
Czernin, Johannes;
Kolb, Hartmuth C.

Publication type:

Article

Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT6 Receptor Ligands.

Published in:

ChemMedChem, 2013, v. 8, n. 1, p. 70, doi. 10.1002/cmdc.201200396

By:

Szalata, Claude;
Szymoniak, Jan;
Fabis, Frédéric;
Butt‐Gueulle, Sabrina;
Rault, Sylvain;
Bertus, Philippe;
Gérard, Stéphane;
Sapi, Janos

Publication type:

Article

Graphical Abstract: ChemMedChem 1/2013.

Published in:: ChemMedChem, 2013, v. 8, n. 1, p. 9, doi. 10.1002/cmdc.201290067
Publication type:: Article

Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 1

Highly Ligand Efficient and Selective N-2-(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A.

Editorial: Premature Publishing and Over-fragmentation.

C3′/C4′-Stereochemical Effects of Digitoxigenin α- L-/α- D-Glycoside in Cancer Cytotoxicity.

Thiadiazole-a Promising Structure in Medicinal Chemistry.

Inside Cover: From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography (ChemMedChem 1/2013).

Synthesis and Quantitative Structure-Activity Relationships of Selective BCRP Inhibitors.

Designing Multi-Target Drugs. Edited by J. Richard Morphy and C. John Harris.

Nanoparticles in Biology and Medicine: Methods and Protocols. Edited by Mikhail Soloviev.

How is <sup>68</sup>Ga Labeling of Macrocyclic Chelators Influenced by Metal Ion Contaminants in <sup>68</sup>Ge/<sup>68</sup>Ga Generator Eluates?

Low-Molecular-Weight CXCR4 Ligands with Variable Spacers.

Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors.

Spotlights on our sister journals: ChemMedChem 1/2013.

Reduction of Helical Content by Insertion of a Disulfide Bond Leads to an Antimicrobial Peptide with Decreased Hemolytic Activity.

3D-QSAR-Assisted Drug Design: Identification of a Potent Quinazoline-Based Aurora Kinase Inhibitor.

Exploring the Polyamine Regulatory Site of the NMDA Receptor: a Parallel Synthesis Approach.

Drug Discovery in Infectious Diseases, Volume 3: Parasitic Helminths: Targets, Screens, Drugs and Vaccines. Edited by Conor R. Caffrey.

Combining Quantum Mechanical Ligand Conformation Analysis and Protein Modeling to Elucidate GPCR-Ligand Binding Modes.

Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand.

Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold.

Editorial: Lucky Number 8!

Cover Picture: Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors (ChemMedChem 1/2013).

Back Cover: Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold (ChemMedChem 1/2013).

Introduction to Strategies for Organic Synthesis. By Laurie S. Starkey.

Discovery of Schaeffer's Acid Analogues as Lead Structures of Mycobacterium tuberculosis Type II Dehydroquinase Using a Rational Drug Design Approach.

Identification of LasR Ligands through a Virtual Screening Approach.

From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography.

Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT<sub>6</sub> Receptor Ligands.

Graphical Abstract: ChemMedChem 1/2013.