Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 1

Results: 28

Highly Ligand Efficient and Selective N-2-(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 149, doi. 10.1002/cmdc.201200450
By:
- Baud, Matthias G. J.;
- Haus, Patricia;
- Leiser, Thomas;
- Meyer‐Almes, Franz‐Josef;
- Fuchter, Matthew J.
Publication type:
Article
Editorial: Premature Publishing and Over-fragmentation.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 6, doi. 10.1002/cmdc.201200494
By:
- Tarzia, Giorgio
Publication type:
Article
C3′/C4′-Stereochemical Effects of Digitoxigenin α- L-/α- D-Glycoside in Cancer Cytotoxicity.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 63, doi. 10.1002/cmdc.201200465
By:
- Hinds, John W.;
- McKenna, Sean B.;
- Sharif, Ehesan U.;
- Wang, Hua‐Yu L.;
- Akhmedov, Novruz G.;
- O'Doherty, George A.
Publication type:
Article
Thiadiazole-a Promising Structure in Medicinal Chemistry.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 27, doi. 10.1002/cmdc.201200355
By:
- Li, Yijing;
- Geng, Jingkun;
- Liu, Yang;
- Yu, Shenghui;
- Zhao, Guisen
Publication type:
Article
Inside Cover: From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography (ChemMedChem 1/2013).
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 2, doi. 10.1002/cmdc.201290066
By:
- Mocharla, Vani P.;
- Walsh, Joseph C.;
- Padgett, Henry C.;
- Su, Helen;
- Fueger, Barbara;
- Weber, Wolfgang A.;
- Czernin, Johannes;
- Kolb, Hartmuth C.
Publication type:
Article
Synthesis and Quantitative Structure-Activity Relationships of Selective BCRP Inhibitors.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 125, doi. 10.1002/cmdc.201200377
By:
- Marighetti, Federico;
- Steggemann, Kerstin;
- Hanl, Markus;
- Wiese, Michael
Publication type:
Article
Designing Multi-Target Drugs. Edited by J. Richard Morphy and C. John Harris.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 166, doi. 10.1002/cmdc.201200420
By:
- Peters, Jens‐Uwe
Publication type:
Article
How is 68Ga Labeling of Macrocyclic Chelators Influenced by Metal Ion Contaminants in 68Ge/68Ga Generator Eluates?
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 95, doi. 10.1002/cmdc.201200471
By:
- Šimeček, Jakub;
- Hermann, Petr;
- Wester, Hans‐Jürgen;
- Notni, Johannes
Publication type:
Article
Nanoparticles in Biology and Medicine: Methods and Protocols. Edited by Mikhail Soloviev.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 167, doi. 10.1002/cmdc.201200430
By:
- Fröhlich, Eleonore
Publication type:
Article
Low-Molecular-Weight CXCR4 Ligands with Variable Spacers.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 118, doi. 10.1002/cmdc.201200390
By:
- Narumi, Tetsuo;
- Aikawa, Haruo;
- Tanaka, Tomohiro;
- Hashimoto, Chie;
- Ohashi, Nami;
- Nomura, Wataru;
- Kobayakawa, Takuya;
- Takano, Hikaru;
- Hirota, Yuki;
- Murakami, Tsutomu;
- Yamamoto, Naoki;
- Tamamura, Hirokazu
Publication type:
Article
Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 104, doi. 10.1002/cmdc.201200417
By:
- Lacotte, Pierre;
- Puente, Celine;
- Ambroise, Yves
Publication type:
Article
Spotlights on our sister journals: ChemMedChem 1/2013.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 20, doi. 10.1002/cmdc.201290065
Publication type:
Article
Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 75, doi. 10.1002/cmdc.201200376
By:
- Held, Cornelia;
- Plomer, Manuel;
- Hübner, Harald;
- Meltretter, Jasmin;
- Pischetsrieder, Monika;
- Gmeiner, Peter
Publication type:
Article
3D-QSAR-Assisted Drug Design: Identification of a Potent Quinazoline-Based Aurora Kinase Inhibitor.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 136, doi. 10.1002/cmdc.201200464
By:
- Ke, Yi‐Yu;
- Shiao, Hui‐Yi;
- Hsu, Yung Chang;
- Chu, Chang‐Ying;
- Wang, Wen‐Chieh;
- Lee, Yen‐Chun;
- Lin, Wen‐Hsing;
- Chen, Chun‐Hwa;
- Hsu, John T. A.;
- Chang, Chun‐Wei;
- Lin, Cheng‐Wei;
- Yeh, Teng‐Kuang;
- Chao, Yu‐Sheng;
- Coumar, Mohane Selvaraj;
- Hsieh, Hsing‐Pang
Publication type:
Article
Exploring the Polyamine Regulatory Site of the NMDA Receptor: a Parallel Synthesis Approach.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 82, doi. 10.1002/cmdc.201200470
By:
- Berger, Michael L.;
- Pöhler, Thomas;
- Schadt, Oliver;
- Stanger, Maximilian;
- Rebernik, Patrick;
- Scholze, Petra;
- Noe, Christian R.
Publication type:
Article
Drug Discovery in Infectious Diseases, Volume 3: Parasitic Helminths: Targets, Screens, Drugs and Vaccines. Edited by Conor R. Caffrey.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 164, doi. 10.1002/cmdc.201200515
By:
- Davioud‐Charvet, Elisabeth
Publication type:
Article
Combining Quantum Mechanical Ligand Conformation Analysis and Protein Modeling to Elucidate GPCR-Ligand Binding Modes.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 49, doi. 10.1002/cmdc.201200412
By:
- Schultes, Sabine;
- Engelhardt, Harald;
- Roumen, Luc;
- Zuiderveld, Obbe P.;
- Haaksma, Eric E. J.;
- de Esch, Iwan J. P.;
- Leurs, Rob;
- de Graaf, Chris
Publication type:
Article
Reduction of Helical Content by Insertion of a Disulfide Bond Leads to an Antimicrobial Peptide with Decreased Hemolytic Activity.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 59, doi. 10.1002/cmdc.201200463
By:
- Hwang, Heeyong;
- Hyun, Soonsil;
- Kim, Yangsoo;
- Yu, Jaehoon
Publication type:
Article
Discovery of Schaeffer's Acid Analogues as Lead Structures of Mycobacterium tuberculosis Type II Dehydroquinase Using a Rational Drug Design Approach.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 54, doi. 10.1002/cmdc.201200508
By:
- Schmidt, Marco F.;
- Korb, Oliver;
- Howard, Nigel I.;
- Dias, Marcio V. B.;
- Blundell, Tom L.;
- Abell, Chris
Publication type:
Article
Identification of LasR Ligands through a Virtual Screening Approach.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 157, doi. 10.1002/cmdc.201200434
By:
- Skovstrup, Søren;
- Le Quement, Sebastian Thordal;
- Hansen, Thomas;
- Jakobsen, Tim Holm;
- Harmsen, Morten;
- Tolker‐Nielsen, Tim;
- Nielsen, Thomas E.;
- Givskov, Michael;
- Taboureau, Olivier
Publication type:
Article
Cover Picture: Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors (ChemMedChem 1/2013).
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 1, doi. 10.1002/cmdc.201290064
By:
- Lacotte, Pierre;
- Puente, Celine;
- Ambroise, Yves
Publication type:
Article
Back Cover: Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold (ChemMedChem 1/2013).
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 172, doi. 10.1002/cmdc.201290068
By:
- Olson, Margaret E.;
- Li, Ming;
- Harris, Reuben S.;
- Harki, Daniel A.
Publication type:
Article
Introduction to Strategies for Organic Synthesis. By Laurie S. Starkey.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 164, doi. 10.1002/cmdc.201200440
By:
- Moloney, Mark G.
Publication type:
Article
Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 112, doi. 10.1002/cmdc.201200411
By:
- Olson, Margaret E.;
- Li, Ming;
- Harris, Reuben S.;
- Harki, Daniel A.
Publication type:
Article
From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 43, doi. 10.1002/cmdc.201200466
By:
- Mocharla, Vani P.;
- Walsh, Joseph C.;
- Padgett, Henry C.;
- Su, Helen;
- Fueger, Barbara;
- Weber, Wolfgang A.;
- Czernin, Johannes;
- Kolb, Hartmuth C.
Publication type:
Article
Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT6 Receptor Ligands.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 70, doi. 10.1002/cmdc.201200396
By:
- Szalata, Claude;
- Szymoniak, Jan;
- Fabis, Frédéric;
- Butt‐Gueulle, Sabrina;
- Rault, Sylvain;
- Bertus, Philippe;
- Gérard, Stéphane;
- Sapi, Janos
Publication type:
Article
Editorial: Lucky Number 8!
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 3, doi. 10.1002/cmdc.201200495
By:
- Williams, Scott D.;
- Ortúzar, Natalia
Publication type:
Article
Graphical Abstract: ChemMedChem 1/2013.
Published in:
ChemMedChem, 2013, v. 8, n. 1, p. 9, doi. 10.1002/cmdc.201290067
Publication type:
Article

Works matching IS 18607179 AND DT 2013 AND VI 8 AND IP 1

Highly Ligand Efficient and Selective N-2-(Thioethyl)picolinamide Histone Deacetylase Inhibitors Inspired by the Natural Product Psammaplin A.

Editorial: Premature Publishing and Over-fragmentation.

C3′/C4′-Stereochemical Effects of Digitoxigenin α- L-/α- D-Glycoside in Cancer Cytotoxicity.

Thiadiazole-a Promising Structure in Medicinal Chemistry.

Inside Cover: From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography (ChemMedChem 1/2013).

Synthesis and Quantitative Structure-Activity Relationships of Selective BCRP Inhibitors.

Designing Multi-Target Drugs. Edited by J. Richard Morphy and C. John Harris.

How is <sup>68</sup>Ga Labeling of Macrocyclic Chelators Influenced by Metal Ion Contaminants in <sup>68</sup>Ge/<sup>68</sup>Ga Generator Eluates?

Nanoparticles in Biology and Medicine: Methods and Protocols. Edited by Mikhail Soloviev.

Low-Molecular-Weight CXCR4 Ligands with Variable Spacers.

Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors.

Spotlights on our sister journals: ChemMedChem 1/2013.

Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand.

3D-QSAR-Assisted Drug Design: Identification of a Potent Quinazoline-Based Aurora Kinase Inhibitor.

Exploring the Polyamine Regulatory Site of the NMDA Receptor: a Parallel Synthesis Approach.

Drug Discovery in Infectious Diseases, Volume 3: Parasitic Helminths: Targets, Screens, Drugs and Vaccines. Edited by Conor R. Caffrey.

Combining Quantum Mechanical Ligand Conformation Analysis and Protein Modeling to Elucidate GPCR-Ligand Binding Modes.

Reduction of Helical Content by Insertion of a Disulfide Bond Leads to an Antimicrobial Peptide with Decreased Hemolytic Activity.

Discovery of Schaeffer's Acid Analogues as Lead Structures of Mycobacterium tuberculosis Type II Dehydroquinase Using a Rational Drug Design Approach.

Identification of LasR Ligands through a Virtual Screening Approach.

Cover Picture: Synthesis and Evaluation of 3,4-Dihydropyrimidin-2(1 H)-ones as Sodium Iodide Symporter Inhibitors (ChemMedChem 1/2013).

Back Cover: Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold (ChemMedChem 1/2013).

Introduction to Strategies for Organic Synthesis. By Laurie S. Starkey.

Small-Molecule APOBEC3G DNA Cytosine Deaminase Inhibitors Based on a 4-Amino-1,2,4-triazole-3-thiol Scaffold.

From In Situ to In Vivo: An In Situ Click-Chemistry-Derived Carbonic Anhydrase II Imaging Agent for Positron Emission Tomography.

Cyclopropyl-tryptamine Analogues: Synthesis and Biological Evaluation as 5-HT<sub>6</sub> Receptor Ligands.

Editorial: Lucky Number 8!

Graphical Abstract: ChemMedChem 1/2013.