Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 9

Results: 24

Back Cover: Cinnamic Acid/Chloroquinoline Conjugates as Potent Agents against Chloroquine-Resistant Plasmodium falciparum (ChemMedChem 9/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1692, doi. 10.1002/cmdc.201290046

By:

Pérez, Bianca;
Teixeira, Cátia;
Gut, Jiri;
Rosenthal, Philip J.;
Gomes, José R. B.;
Gomes, Paula

Publication type:

Article

Graphical Abstract: ChemMedChem 9/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 9, p. 1511, doi. 10.1002/cmdc.201290043
Publication type:: Article

Dipeptidyl Peptidase IV-Activated Prodrugs of Anti-Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1612, doi. 10.1002/cmdc.201200295

By:

Diez-Torrubia, Alberto;
Cabrera, Silvia;
De Meester, Ingrid;
Camarasa, María-José;
Balzarini, Jan;
Velázquez, Sonsoles

Publication type:

Article

Anti-influenza Drug Discovery: Identification of an Orally Bioavailable Quinoline Derivative through Activity- and Property-Guided Lead Optimization.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1546, doi. 10.1002/cmdc.201200259

By:

Yeh, Jiann-Yih;
Coumar, Mohane Selvaraj;
Shiao, Hui-Yi;
Lin, Ta-Jen;
Lee, Yen-Chun;
Hung, Hui-Chen;
Ko, Shengkai;
Kuo, Fu-Ming;
Fang, Ming-Yu;
Huang, Yu-Lin;
Hsu, John T. A.;
Yeh, Teng-Kuang;
Shih, Shin-Ru;
Chao, Yu-Sheng;
Horng, Jim-Tong;
Hsieh, Hsing-Pang

Publication type:

Article

Inside Cover: Modeling, Synthesis and Biological Evaluation of Potential Retinoid X Receptor-Selective Agonists: Novel Halogenated Analogues of 4-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic Acid (Bexarotene) (ChemMedChem 9/2012)

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1510, doi. 10.1002/cmdc.201290042

By:

Furmick, Julie K.;
Kaneko, Ichiro;
Walsh, Angela N.;
Yang, Joanna;
Bhogal, Jaskaran S.;
Gray, Geoffrey M.;
Baso, Juan C.;
Browder, Drew O.;
Prentice, Jessica L. S.;
Montano, Luis A.;
Huynh, Chanh C.;
Marcus, Lisa M.;
Tsosie, Dorian G.;
Kwon, Jungeun S.;
Quezada, Alexis;
Reyes, Nicole M.;
Lemming, Brittney;
Saini, Puneet;
van der Vaart, Arjan;
Groy, Thomas L.

Publication type:

Article

Designing Multitarget Anti-inflammatory Agents: Chemical Modulation of the Lumiracoxib Structure toward Dual Thromboxane Antagonists-COX-2 Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1647, doi. 10.1002/cmdc.201200272

By:

Bertinaria, Massimo;
Shaikh, Mohammed Abrar Abdul Gaffar;
Buccellati, Carola;
Cena, Clara;
Rolando, Barbara;
Lazzarato, Loretta;
Fruttero, Roberta;
Gasco, Alberto;
Hoxha, Malvina;
Capra, Valérie;
Sala, Angelo;
Rovati, G. Enrico

Publication type:

Article

M. Jung.

Published in:: ChemMedChem, 2012, v. 7, n. 9, p. 1525, doi. 10.1002/cmdc.201200280
Publication type:: Article

Synthesis and Antimicrobial Activities of Oximes Derived from O-Benzylhydroxylamine as FabH Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1587, doi. 10.1002/cmdc.201200225

By:

Luo, Yin;
Zhang, Li-Rong;
Hu, Yang;
Zhang, Shuai;
Fu, Jie;
Wang, Xiao-Ming;
Zhu, Hai-Liang

Publication type:

Article

Synthesis of Stable Genipin Derivatives and Studies of Their Neuroprotective Activity in PC12 Cells.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1661, doi. 10.1002/cmdc.201200258

By:

Luo, Jun;
Wang, Rikang;
Huang, Zhao;
Yang, Jian;
Yao, Xinsheng;
Chen, Heru;
Zheng, Wenhua

Publication type:

Article

Recent Advances in Neuraminidase Inhibitor Development as Anti-influenza Drugs.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1527, doi. 10.1002/cmdc.201200155

By:

Feng, Enguang;
Ye, Deju;
Li, Jian;
Zhang, Dengyou;
Wang, Jinfang;
Zhao, Fei;
Hilgenfeld, Rolf;
Zheng, Mingyue;
Jiang, Hualiang;
Liu, Hong

Publication type:

Article

Cover Picture: Dipeptidyl Peptidase IV-Activated Prodrugs of Anti-Varicella Zoster Virus Bicyclic Nucleoside Analogues Containing Different Self-Cleavage Spacer Systems (ChemMedChem 9/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1509, doi. 10.1002/cmdc.201290041

By:

Diez-Torrubia, Alberto;
Cabrera, Silvia;
De Meester, Ingrid;
Camarasa, María-José;
Balzarini, Jan;
Velázquez, Sonsoles

Publication type:

Article

An Efficient Synthesis of a Hydroxyethylamine (HEA) Isostere and Its α-Aminophosphonate and Phosphoramidate Derivatives as Potential Anti-HIV Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1601, doi. 10.1002/cmdc.201200271

By:

Bhattacharya, Asish K.;
Rana, Kalpeshkumar C.;
Pannecouque, Christophe;
De Clercq, Eric

Publication type:

Article

Preview: ChemMedChem 10/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 9, p. 1691, doi. 10.1002/cmdc.201290045
Publication type:: Article

Semisynthetic Ursolic Acid Fluorolactone Derivatives Inhibit Growth with Induction of p21<sup>waf1</sup> and Induce Apoptosis with Upregulation of NOXA and Downregulation of c-FLIP in Cancer Cells.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1635, doi. 10.1002/cmdc.201200282

By:

Leal, Ana S.;
Wang, Rui;
Salvador, Jorge A. R.;
Jing, Yongkui

Publication type:

Article

Evaluation of Flavonoid and Resveratrol Chemical Libraries Reveals Abyssinone II as a Promising Antibacterial Lead.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1541, doi. 10.1002/cmdc.201200253

By:

Sun, Dianqing;
Hurdle, Julian G.;
Lee, Robin;
Lee, Richard;
Cushman, Mark;
Pezzuto, John M.

Publication type:

Article

Curcumin Analogues with Potent and Selective Anti-proliferative Activity on Acute Promyelocytic Leukemia: Involvement of Accumulated Misfolded Nuclear Receptor Co-repressor (N-CoR) Protein as a Basis for Selective Activity.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1567, doi. 10.1002/cmdc.201200293

By:

Tan, Kheng-Lin;
Koh, Siang-Boon;
Ee, Rachel Pui-Lai;
Khan, Matiullah;
Go, Mei-Lin

Publication type:

Article

β- D-Glucosyl Conjugates of Highly Potent Inhibitors of Blood Coagulation Factor Xa Bearing 2-Chorothiophene as a P1 Motif.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1669, doi. 10.1002/cmdc.201200224

By:

Lopopolo, Gianfranco;
de Candia, Modesto;
Panza, Luigi;
Romano, Maria Rosaria;
Lograno, Marcello Diego;
Campagna, Francesco;
Altomare, Cosimo

Publication type:

Article

Differentiating between Models of Epothilone Binding to Microtubules Using Tubulin Mutagenesis, Cytotoxicity, and Molecular Modeling.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1580, doi. 10.1002/cmdc.201200286

By:

Entwistle, Ruth A.;
Rizk, Rania S.;
Cheng, Daniel M.;
Lushington, Gerald H.;
Himes, Richard H.;
Gupta, Mohan L.

Publication type:

Article

Cinnamic Acid/Chloroquinoline Conjugates as Potent Agents against Chloroquine-Resistant Plasmodium falciparum.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1537, doi. 10.1002/cmdc.201200257

By:

Pérez, Bianca;
Teixeira, Cátia;
Gut, Jiri;
Rosenthal, Philip J.;
Gomes, José R. B.;
Gomes, Paula

Publication type:

Article

Synthesis and Biological Evaluation of CTP Synthetase Inhibitors as Potential Agents for the Treatment of African Trypanosomiasis.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1623, doi. 10.1002/cmdc.201200304

By:

Tamborini, Lucia;
Pinto, Andrea;
Smith, Terry K.;
Major, Louise L.;
Iannuzzi, Maria C.;
Cosconati, Sandro;
Marinelli, Luciana;
Novellino, Ettore;
Lo Presti, Leonardo;
Wong, Pui E.;
Barrett, Michael P.;
De Micheli, Carlo;
Conti, Paola

Publication type:

Article

Library Screening by Means of Mass Spectrometry (MS) Binding Assays-Exemplarily Demonstrated for a Pseudostatic Library Addressing γ-Aminobutyric Acid (GABA) Transporter 1 (GAT1).

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1678, doi. 10.1002/cmdc.201200201

By:

Sindelar, Miriam;
Wanner, Klaus T.

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 9/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 9, p. 1522, doi. 10.1002/cmdc.201290044
Publication type:: Article

Synthesis and Molecular Modeling Studies of Derivatives of a Highly Potent Peptidomimetic Vinyl Ester as Falcipain-2 Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1594, doi. 10.1002/cmdc.201200274

By:

Ettari, Roberta;
Micale, Nicola;
Grazioso, Giovanni;
Bova, Floriana;
Schirmeister, Tanja;
Grasso, Silvana;
Zappalà, Maria

Publication type:

Article

Modeling, Synthesis and Biological Evaluation of Potential Retinoid X Receptor-Selective Agonists: Novel Halogenated Analogues of 4-[1-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic Acid (Bexarotene).

Published in:

ChemMedChem, 2012, v. 7, n. 9, p. 1551, doi. 10.1002/cmdc.201290042

By:

Furmick, Julie K.;
Kaneko, Ichiro;
Walsh, Angela N.;
Yang, Joanna;
Bhogal, Jaskaran S.;
Gray, Geoffrey M.;
Baso, Juan C.;
Browder, Drew O.;
Prentice, Jessica L. S.;
Montano, Luis A.;
Huynh, Chanh C.;
Marcus, Lisa M.;
Tsosie, Dorian G.;
Kwon, Jungeun S.;
Quezada, Alexis;
Reyes, Nicole M.;
Lemming, Brittney;
Saini, Puneet;
van der Vaart, Arjan;
Groy, Thomas L.

Publication type:

Article