Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 7

Results: 27

Activity-Based Probes for the Study of Proteases: Recent Advances and Developments.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1146, doi. 10.1002/cmdc.201200057

By:

Serim, Sevnur;
Haedke, Ute;
Verhelst, Steven H. L.

Publication type:

Article

Inside Cover: Structural Characterization and Computer-Aided Optimization of a Small-Molecule Inhibitor of the Arp2/3 Complex, a Key Regulator of the Actin Cytoskeleton (ChemMedChem 7/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1130, doi. 10.1002/cmdc.201290030

By:

Baggett, Andrew W.;
Cournia, Zoe;
Han, Min Suk;
Patargias, George;
Glass, Adam C.;
Liu, Shih-Yuan;
Nolen, Brad J.

Publication type:

Article

Back Cover: Design, Synthesis, and in vitro Antibacterial Activity of Fluoroquinolone Derivatives Containing a Chiral 3-(Alkoxyimino)-2-(aminomethyl)azetidine Moiety (ChemMedChem 7/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1300, doi. 10.1002/cmdc.201290034

By:

Lv, Kai;
Sun, Yexin;
Sun, Lanyin;
Wei, Zengquan;
Guo, Huiyuan;
Wu, Jinwei;
Liu, Mingliang

Publication type:

Article

Selectively Guanidinylated Aminoglycosides as Antibiotics.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1237, doi. 10.1002/cmdc.201200150

By:

Fair, Richard J.;
Hensler, Mary E.;
Thienphrapa, Wdee;
Dam, Quang N.;
Nizet, Victor;
Tor, Yitzhak

Publication type:

Article

Discovery, Synthesis, and in vitro Evaluation of West Nile Virus Protease Inhibitors Based on the 9,10-Dihydro-3 H,4a H-1,3,9,10a-tetraazaphenanthren-4-one Scaffold.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1210, doi. 10.1002/cmdc.201200136

By:

Samanta, Sanjay;
Cui, Taian;
Lam, Yulin

Publication type:

Article

Identification of a 17β-Hydroxysteroid Dehydrogenase Type 10 Steroidal Inhibitor: A Tool to Investigate the Role of Type 10 in Alzheimer's Disease and Prostate Cancer.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1181, doi. 10.1002/cmdc.201200129

By:

Ayan, Diana;
Maltais, René;
Poirier, Donald

Publication type:

Article

Preview: ChemMedChem 8/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 7, p. 1299, doi. 10.1002/cmdc.201290033
Publication type:: Article

Predicting Drug Metabolism by Cytochrome P450 2C9: Comparison with the 2D6 and 3A4 Isoforms.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1202, doi. 10.1002/cmdc.201200160

By:

Rydberg, Patrik;
Olsen, Lars

Publication type:

Article

6-Halogenochromones Bearing Tryptamine: One-Step Access to Potent and Highly Selective Inhibitors of Breast Cancer Resistance Protein.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1177, doi. 10.1002/cmdc.201200154

By:

Valdameri, Glaucio;
Genoux-Bastide, Estelle;
Gauthier, Charlotte;
Peres, Basile;
Terreux, Raphaël;
Winnischofer, Sheila M. B.;
Rocha, Maria E. M.;
Di Pietro, Attilio;
Boumendjel, Ahcène

Publication type:

Article

Synthesis, Structure-Activity Relationship and Docking Studies of Substituted Aryl Thiazolyl Phenylsulfonamides as Potential Protein Tyrosine Phosphatase 1B Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1185, doi. 10.1002/cmdc.201200197

By:

Varshney, Kanika;
Gupta, Swati;
Rahuja, Neha;
Rawat, Arun K.;
Singh, Nagendra;
Tamarkar, Akhilesh K.;
Srivastava, Arvind K.;
Saxena, Anil K.

Publication type:

Article

Drug Design Strategies: Quantitative Approaches. Edited by David J. Livingstone and Andrew M. Davis.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1295, doi. 10.1002/cmdc.201200168

By:

Matter, Hans

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 7/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 7, p. 1142, doi. 10.1002/cmdc.201290032
Publication type:: Article

Chemical Genomics and Proteomics: Reviews and Protocols. Edited by Edward D. Zanders.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1297, doi. 10.1002/cmdc.201200170

By:

Brunsveld, Luc

Publication type:

Article

Design, Synthesis, and Biological Evaluation of 2-Aminobenzanilide Derivatives as Potent and Selective HDAC Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1256, doi. 10.1002/cmdc.201200193

By:

Stolfa, Diana A.;
Stefanachi, Angela;
Gajer, Julia M.;
Nebbioso, Angela;
Altucci, Lucia;
Cellamare, Saverio;
Jung, Manfred;
Carotti, Angelo

Publication type:

Article

Synthesis and Biological Evaluation of Adenosines with Heterobicyclic and Polycyclic N<sup>6</sup>-Substituents as Adenosine A<sub>1</sub> Receptor Agonists.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1191, doi. 10.1002/cmdc.201200208

By:

Gosling, Joshua I.;
Baker, Stephen P.;
Haynes, John M.;
Kassiou, Michael;
Pouton, Colin W.;
Warfe, Lyndon;
White, Paul J.;
Scammells, Peter J.

Publication type:

Article

O-Linked Triazolotriazines: Potent and Selective c-Met Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1276, doi. 10.1002/cmdc.201200145

By:

Chen, Fang;
Wang, Ying;
Ai, Jing;
Zhan, Zhengsheng;
Lv, Yongcong;
Liang, Zhongjie;
Luo, Cheng;
Mei, Desheng;
Geng, Meiyu;
Duan, Wenhu

Publication type:

Article

Bicyclic Peptides with Optimized Ring Size Inhibit Human Plasma Kallikrein and its Orthologues While Sparing Paralogous Proteases.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1173, doi. 10.1002/cmdc.201200071

By:

Baeriswyl, Vanessa;
Rapley, Helen;
Pollaro, Lisa;
Stace, Catherine;
Teufel, Dan;
Walker, Edward;
Chen, Shiyu;
Winter, Greg;
Tite, John;
Heinis, Christian

Publication type:

Article

The Development of FtsZ Inhibitors as Potential Antibacterial Agents.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1161, doi. 10.1002/cmdc.201200156

By:

Ma, Siti;
Ma, Shutao

Publication type:

Article

Cover Picture: Bicyclic Peptides with Optimized Ring Size Inhibit Human Plasma Kallikrein and its Orthologues While Sparing Paralogous Proteases (ChemMedChem 7/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1129, doi. 10.1002/cmdc.201290029

By:

Baeriswyl, Vanessa;
Rapley, Helen;
Pollaro, Lisa;
Stace, Catherine;
Teufel, Dan;
Walker, Edward;
Chen, Shiyu;
Winter, Greg;
Tite, John;
Heinis, Christian

Publication type:

Article

Synthesis and Structure-Activity Relationship Studies of HIV-1 Virion Infectivity Factor (Vif) Inhibitors that Block Viral Replication.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1217, doi. 10.1002/cmdc.201200079

By:

Ali, Akbar;
Wang, Jinhua;
Nathans, Robin S.;
Cao, Hong;
Sharova, Natalia;
Stevenson, Mario;
Rana, Tariq M.

Publication type:

Article

Graphical Abstract: ChemMedChem 7/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 7, p. 1131, doi. 10.1002/cmdc.201290031
Publication type:: Article

Design, Synthesis, and in vitro Antibacterial Activity of Fluoroquinolone Derivatives Containing a Chiral 3-(Alkoxyimino)-2-(aminomethyl)azetidine Moiety.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1230, doi. 10.1002/cmdc.201200210

By:

Lv, Kai;
Sun, Yexin;
Sun, Lanyin;
Wei, Zengquan;
Guo, Huiyuan;
Wu, Jinwei;
Liu, Mingliang

Publication type:

Article

Synthesis of a Heparan Sulfate Mimetic Library Targeting FGF and VEGF via Click Chemistry on a Monosaccharide Template.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1267, doi. 10.1002/cmdc.201200151

By:

Liu, Ligong;
Li, Caiping;
Cochran, Siska;
Jimmink, Shane;
Ferro, Vito

Publication type:

Article

Structural Characterization and Computer-Aided Optimization of a Small-Molecule Inhibitor of the Arp2/3 Complex, a Key Regulator of the Actin Cytoskeleton.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1286, doi. 10.1002/cmdc.201200104

By:

Baggett, Andrew W.;
Cournia, Zoe;
Han, Min Suk;
Patargias, George;
Glass, Adam C.;
Liu, Shih-Yuan;
Nolen, Brad J.

Publication type:

Article

Joaquín M. Campos.

Published in:: ChemMedChem, 2012, v. 7, n. 7, p. 1145, doi. 10.1002/cmdc.201200218
Publication type:: Article

Development of an ( S)-1-{2-[Tris(4-methoxyphenyl)methoxy]ethyl}piperidine-3-carboxylic acid [( S)-SNAP-5114] Carba Analogue Inhibitor for Murine γ-Aminobutyric Acid Transporter Type 4.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1245, doi. 10.1002/cmdc.201200126

By:

Pabel, Jörg;
Faust, Mark;
Prehn, Cornelia;
Wörlein, Babette;
Allmendinger, Lars;
Höfner, Georg;
Wanner, Klaus T.

Publication type:

Article

New Synthetic Technologies in Medicinal Chemistry. Edited by Elizabeth Farrant.

Published in:

ChemMedChem, 2012, v. 7, n. 7, p. 1296, doi. 10.1002/cmdc.201200177

By:

Kirschning, Andreas

Publication type:

Article