Works matching IS 18607179 AND DT 2012 AND VI 7 AND IP 5

Results: 23

Synthesis of Simplified Tedanolide Analogues-Connecting Tedanolide to Myriaporone and Gephyronic Acid.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 771, doi. 10.1002/cmdc.201100576

By:

Diaz, Nina;
Naini, Arun;
Muthukumar, Yazh;
Sasse, Florenz;
Kalesse, Markus

Publication type:

Article

Spotlights on our sister journals: ChemMedChem 5/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 5, p. 758, doi. 10.1002/cmdc.201290021
Publication type:: Article

Characterization of Plasmodium Liver Stage Inhibition by Halofuginone.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 844, doi. 10.1002/cmdc.201200045

By:

Derbyshire, Emily R.;
Mazitschek, Ralph;
Clardy, Jon

Publication type:

Article

Cover Picture: Characterization of Plasmodium Liver Stage Inhibition by Halofuginone (ChemMedChem 5/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 745, doi. 10.1002/cmdc.201290018

By:

Derbyshire, Emily R.;
Mazitschek, Ralph;
Clardy, Jon

Publication type:

Article

Effects of Cyclic Lipodepsipeptide Structural Modulation on Stability, Antibacterial Activity, and Human Cell Toxicity.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 871, doi. 10.1002/cmdc.201200016

By:

Bionda, Nina;
Stawikowski, Maciej;
Stawikowska, Roma;
Cudic, Maré;
López-Vallejo, Fabian;
Treitl, Daniela;
Medina-Franco, José;
Cudic, Predrag

Publication type:

Article

Investigations on the 4-Quinolone-3-Carboxylic Acid Motif Part 5: Modulation of the Physicochemical Profile of a Set of Potent and Selective Cannabinoid-2 Receptor Ligands through a Bioisosteric Approach.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 920, doi. 10.1002/cmdc.201100573

By:

Mugnaini, Claudia;
Nocerino, Stefania;
Pedani, Valentina;
Pasquini, Serena;
Tafi, Andrea;
De Chiaro, Maria;
Bellucci, Luca;
Valoti, Massimo;
Guida, Francesca;
Luongo, Livio;
Dragoni, Stefania;
Ligresti, Alessia;
Rosenberg, Avraham;
Bolognini, Daniele;
Cascio, Maria Grazia;
Pertwee, Roger G.;
Moaddel, Ruin;
Maione, Sabatino;
Di Marzo, Vincenzo;
Corelli, Federico

Publication type:

Article

Graphical Abstract: ChemMedChem 5/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 5, p. 747, doi. 10.1002/cmdc.201290020
Publication type:: Article

Structure-Activity Relationships of Organofluorine Inhibitors of β-Amyloid Self-Assembly.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 910, doi. 10.1002/cmdc.201100569

By:

Török, Béla;
Sood, Abha;
Bag, Seema;
Kulkarni, Aditya;
Borkin, Dmitry;
Lawler, Elizabeth;
Dasgupta, Sujaya;
Landge, Shainaz;
Abid, Mohammed;
Zhou, Weihong;
Foster, Michelle;
LeVine, Harry;
Török, Marianna

Publication type:

Article

Synthesis of Small Molecules Targeting Multiple DNA Structures using Click Chemistry.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 792, doi. 10.1002/cmdc.201200060

By:

Howell, Lesley A.;
Bowater, Richard A.;
O'Connell, Maria A.;
Reszka, Anthony P.;
Neidle, Stephen;
Searcey, Mark

Publication type:

Article

Heme Oxygenase Inhibition by α-(1 H-Imidazol-1-yl)-ω-phenylalkanes: Effect of Introduction of Heteroatoms in the Alkyl Linker.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 897, doi. 10.1002/cmdc.201100602

By:

Vlahakis, Jason Z.;
Lazar, Carmen;
Roman, Gheorghe;
Vukomanovic, Dragic;
Nakatsu, Kanji;
Szarek, Walter A.

Publication type:

Article

Synthesis, Biological Activity, and ADME Properties of Novel S-DABOs/ N-DABOs as HIV Reverse Transcriptase Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 883, doi. 10.1002/cmdc.201200056

By:

Radi, Marco;
Pagano, Mafalda;
Franchi, Luigi;
Castagnolo, Daniele;
Schenone, Silvia;
Casaluce, Gianni;
Zamperini, Claudio;
Dreassi, Elena;
Maga, Giovanni;
Samuele, Alberta;
Gonzalo, Encarna;
Clotet, Bonaventura;
Esté, José A.;
Botta, Maurizio

Publication type:

Article

Structural Determination of NSC 670224, Synthesis of Analogues and Biological Evaluation.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 761, doi. 10.1002/cmdc.201200038

By:

Zuckerman, Nathaniel B.;
Myers, Andrew S.;
Quan, Tiffani K.;
Bray, Walter M.;
Lokey, R. Scott;
Hartzog, Grant A.;
Konopelski, Joseph P.

Publication type:

Article

Structure-Based Design of Novel Pyrimido[4,5- c]pyridazine Derivatives as Dihydropteroate Synthase Inhibitors with Increased Affinity.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 861, doi. 10.1002/cmdc.201200049

By:

Zhao, Ying;
Hammoudeh, Dalia;
Yun, Mi-Kyung;
Qi, Jianjun;
White, Stephen W.;
Lee, Richard E.

Publication type:

Article

Synthesis and Evaluation of Anticancer Natural Product Analogues Based on Angelmarin: Targeting the Tolerance towards Nutrient Deprivation.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 766, doi. 10.1002/cmdc.201100564

By:

Magolan, Jakob;
Adams, Nathan B. P.;
Onozuka, Hiroko;
Hungerford, Natasha L.;
Esumi, Hiroyasu;
Coster, Mark J.

Publication type:

Article

Anticancer Activity of Silver- N-Heterocyclic Carbene Complexes: Caspase-Independent Induction of Apoptosis via Mitochondrial Apoptosis-Inducing Factor (AIF).

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 805, doi. 10.1002/cmdc.201200055

By:

Eloy, Laure;
Jarrousse, Anne-Sophie;
Teyssot, Marie-Laure;
Gautier, Arnaud;
Morel, Laurent;
Jolivalt, Claude;
Cresteil, Thierry;
Roland, Sylvain

Publication type:

Article

Comparative Binding Energy (COMBINE) Analysis Supports a Proposal for the Binding Mode of Epothilones to β-Tubulin.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 836, doi. 10.1002/cmdc.201200065

By:

Coderch, Claire;
Klett, Javier;
Morreale, Antonio;
Díaz, J. Fernando;
Gago, Federico

Publication type:

Article

Generating Orally Active Galanin Analogues with Analgesic Activities.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 903, doi. 10.1002/cmdc.201100574

By:

Robertson, Charles R.;
Pruess, Timothy H.;
Grussendorf, Erin;
White, H. Steve;
Bulaj, Grzegorz

Publication type:

Article

Preview: ChemMedChem 6/2012.

Published in:: ChemMedChem, 2012, v. 7, n. 5, p. 935, doi. 10.1002/cmdc.201290022
Publication type:: Article

Inside Cover: Effects of Cyclic Lipodepsipeptide Structural Modulation on Stability, Antibacterial Activity, and Human Cell Toxicity (ChemMedChem 5/2012).

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 746, doi. 10.1002/cmdc.201290019

By:

Bionda, Nina;
Stawikowski, Maciej;
Stawikowska, Roma;
Cudic, Maré;
López-Vallejo, Fabian;
Treitl, Daniela;
Medina-Franco, José;
Cudic, Predrag

Publication type:

Article

An Efficient Synthesis of Quinoxalinone Derivatives as Potent Inhibitors of Aldose Reductase.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 823, doi. 10.1002/cmdc.201200054

By:

Yang, Yanchun;
Zhang, Shuzhen;
Wu, Bobin;
Ma, Mingming;
Chen, Xin;
Qin, Xiangyu;
He, Minlan;
Hussain, Saghir;
Jing, Chaojun;
Ma, Bing;
Zhu, Changjin

Publication type:

Article

Bulbispermine: A Crinine-Type Amaryllidaceae Alkaloid Exhibiting Cytostatic Activity toward Apoptosis-Resistant Glioma Cells.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 815, doi. 10.1002/cmdc.201100608

By:

Luchetti, Giovanni;
Johnston, Robert;
Mathieu, Véronique;
Lefranc, Florence;
Hayden, Kathryn;
Andolfi, Anna;
Lamoral-Theys, Delphine;
Reisenauer, Mary R.;
Champion, Cody;
Pelly, Stephen C.;
van Otterlo, Willem A. L.;
Magedov, Igor V.;
Kiss, Robert;
Evidente, Antonio;
Rogelj, Snezna;
Kornienko, Alexander

Publication type:

Article

Exploring the Anticancer Activity of Functionalized Isoindigos: Synthesis, Drug-like Potential, Mode of Action and Effect on Tumor-Induced Xenografts.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 777, doi. 10.1002/cmdc.201200018

By:

Wee, Xi Kai;
Yang, Tianming;
Go, Mei Lin

Publication type:

Article

Discovery of N-Arylalkyl-3-hydroxy-4-oxo-3,4-dihydroquinazolin-2-carboxamide Derivatives as HCV NS5B Polymerase Inhibitors.

Published in:

ChemMedChem, 2012, v. 7, n. 5, p. 850, doi. 10.1002/cmdc.201200058

By:

Deore, Ravindra Ramesh;
Chen, Grace Shiahuy;
Chang, Pei-Teh;
Chern, Ting-Rong;
Lai, Shin-Yu;
Chuang, Ming-Hsieh;
Lin, Jung-Hsin;
Kung, Fan-Lu;
Chen, Chien-Shu;
Chiou, Chun-Tang;
Chern, Ji-Wang

Publication type:

Article